Page last updated: 2024-09-03

des-enkephalin-gamma-endorphin and naloxone

des-enkephalin-gamma-endorphin has been researched along with naloxone in 4 studies

Compound Research Comparison

Studies
(des-enkephalin-gamma-endorphin)
Trials
(des-enkephalin-gamma-endorphin)
Recent Studies (post-2010)
(des-enkephalin-gamma-endorphin)
Studies
(naloxone)
Trials
(naloxone)
Recent Studies (post-2010) (naloxone)
416020,1341,2573,321

Protein Interaction Comparison

ProteinTaxonomydes-enkephalin-gamma-endorphin (IC50)naloxone (IC50)
Cytochrome P450 2D6Homo sapiens (human)2
Delta-type opioid receptorMus musculus (house mouse)0.043
Delta-type opioid receptorRattus norvegicus (Norway rat)0.0219
Mu-type opioid receptorRattus norvegicus (Norway rat)0.0019
Kappa-type opioid receptorRattus norvegicus (Norway rat)0.0019
Mu-type opioid receptorHomo sapiens (human)0.0397
Delta-type opioid receptorHomo sapiens (human)0.1896
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)0.05
Kappa-type opioid receptorHomo sapiens (human)0.0795
Mu-type opioid receptorMus musculus (house mouse)0.0154
Mu-type opioid receptorCavia porcellus (domestic guinea pig)0.0089
Beta-2 adrenergic receptorCavia porcellus (domestic guinea pig)0.0055

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19902 (50.00)18.7374
1990's1 (25.00)18.2507
2000's1 (25.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Andringa-Bakker, EA; de Rotte, AA; de Wied, D; van de Buuse, M; van Wimersma Greidanus, TB1
Kay, N; Morley, JE; van Ree, JM1
Di Giannuario, A; Loizzo, A; Luzi, M; Pieretti, S1
Capasso, A1

Other Studies

4 other study(ies) available for des-enkephalin-gamma-endorphin and naloxone

ArticleYear
The effect of gamma-type endorphins on alpha-MSH release in the rat.
    Life sciences, 1985, Jul-22, Volume: 37, Issue:3

    Topics: Animals; Antipsychotic Agents; Apomorphine; beta-Endorphin; Dose-Response Relationship, Drug; Endorphins; gamma-Endorphin; Haloperidol; Injections, Intraventricular; Male; Melanocyte-Stimulating Hormones; Naloxone; Pituitary Gland, Anterior; Rats; Rats, Inbred Strains

1985
Enhancement of human lymphocyte natural killing function by non-opioid fragments of beta-endorphin.
    Life sciences, 1987, Mar-16, Volume: 40, Issue:11

    Topics: beta-Endorphin; Endorphins; gamma-Endorphin; Humans; Killer Cells, Natural; Naloxone; Peptide Fragments

1987
Subchronic treatment with fragments of beta-endorphin prevents electroencephalographic seizures and behavioral alterations induced by centrally administered beta-endorphin in the rabbit.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 268, Issue:2

    Topics: Animals; Behavior, Animal; beta-Endorphin; Electroencephalography; Endorphins; Haloperidol; Injections, Intraventricular; Male; Naloxone; Peptide Fragments; Rabbits; Seizures

1994
Beta-endorphin fragments DTgammaE and DEgammaE reduced morphine inhibition of electrically-induced contractions and opiate withdrawal.
    Medicinal chemistry (Shariqah (United Arab Emirates)), 2009, Volume: 5, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Acetylcholine; Animals; beta-Endorphin; Electric Stimulation; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Guinea Pigs; Ileum; In Vitro Techniques; Jejunum; Male; Morphine; Muscle Contraction; Muscle, Smooth; Naloxone; Oligopeptides; Peptide Fragments; Rabbits; Substance Withdrawal Syndrome

2009