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des-enkephalin-gamma-endorphin and apomorphine

des-enkephalin-gamma-endorphin has been researched along with apomorphine in 11 studies

Compound Research Comparison

Studies
(des-enkephalin-gamma-endorphin)
Trials
(des-enkephalin-gamma-endorphin)
Recent Studies (post-2010)
(des-enkephalin-gamma-endorphin)
Studies
(apomorphine)
Trials
(apomorphine)
Recent Studies (post-2010) (apomorphine)
41609,205287780

Protein Interaction Comparison

ProteinTaxonomydes-enkephalin-gamma-endorphin (IC50)apomorphine (IC50)
Tryptophan 5-hydroxylase 1Rattus norvegicus (Norway rat)0.22
D(2) dopamine receptorHomo sapiens (human)0.0146
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)7.75
DRattus norvegicus (Norway rat)0.4744
D(3) dopamine receptorRattus norvegicus (Norway rat)0.1432
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)0.063
D(2) dopamine receptorBos taurus (cattle)0.3385
D(1A) dopamine receptorHomo sapiens (human)0.025
D(4) dopamine receptorHomo sapiens (human)0.025
D(1B) dopamine receptorHomo sapiens (human)0.025
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)0.063
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)0.063
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)7.75
D(1B) dopamine receptorRattus norvegicus (Norway rat)0.1432
D(4) dopamine receptorRattus norvegicus (Norway rat)0.1432
D(3) dopamine receptorHomo sapiens (human)0.025
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)7.75
D(2) dopamine receptorRattus norvegicus (Norway rat)0.0813
E3 ubiquitin-protein ligase Mdm2Homo sapiens (human)0.205
5-hydroxytryptamine receptor 4 Rattus norvegicus (Norway rat)1.35
DBos taurus (cattle)0.3385

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19909 (81.82)18.7374
1990's2 (18.18)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Elands, J; Kiraly, I; van Ree, JM; Wolterink, G2
Andringa-Bakker, EA; de Rotte, AA; de Wied, D; van de Buuse, M; van Wimersma Greidanus, TB1
Costall, B; Domeney, AM; Naylor, RJ1
Radhakishun, FS; van Ree, JM; Westerink, BH1
Mulder, AH; Radhakishun, FS; Stoof, JC; van Ree, JM; Versteeg, DH1
Radhakishun, FS; Van Ree, JM1
De Wied, D; Drago, F; Van Ree, JM1
Király, I; Van Ree, JM1
Codd, EE; Scholtens, H; Van Ree, JM; Verhoef, JC; Witter, A; Wolterink, G1
Radhakishun, FS; Stoof, JC; van Ree, JM; Westerink, BH; Wolterink, G1

Other Studies

11 other study(ies) available for des-enkephalin-gamma-endorphin and apomorphine

ArticleYear
Gamma-type endorphins and brain dopaminergic systems.
    Progress in clinical and biological research, 1990, Volume: 328

    Topics: Animals; Antipsychotic Agents; Apomorphine; Behavior, Animal; beta-Endorphin; Brain; Caudate Nucleus; Cerebral Cortex; Dopamine; Nucleus Accumbens; Rats; Receptors, Dopamine

1990
The effect of gamma-type endorphins on alpha-MSH release in the rat.
    Life sciences, 1985, Jul-22, Volume: 37, Issue:3

    Topics: Animals; Antipsychotic Agents; Apomorphine; beta-Endorphin; Dose-Response Relationship, Drug; Endorphins; gamma-Endorphin; Haloperidol; Injections, Intraventricular; Male; Melanocyte-Stimulating Hormones; Naloxone; Pituitary Gland, Anterior; Rats; Rats, Inbred Strains

1985
Antipsychotic substances and dopamine in the rat brain; behavioral studies reveal distinct dopamine receptor systems.
    European journal of pharmacology, 1989, Aug-03, Volume: 166, Issue:3

    Topics: Animals; Antipsychotic Agents; Apomorphine; Behavior, Animal; beta-Endorphin; Brain Chemistry; Cerebral Cortex; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Injections; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Dopamine; Substantia Nigra; Sulpiride

1989
Desenkephalin-gamma-endorphin is an antagonist of the hyperactivity response induced by infusion of dopamine into the nucleus accumbens of rat and ventral striatum of marmoset.
    Neuropharmacology, 1989, Volume: 28, Issue:11

    Topics: Animals; Apomorphine; beta-Endorphin; Callitrichinae; Corpus Striatum; Dopamine; Dopamine Agents; Dopamine Antagonists; Female; Fluphenazine; Haloperidol; Injections; Male; Motor Activity; Nucleus Accumbens; Rats; Rats, Inbred Strains; Septal Nuclei

1989
Dopamine release in the nucleus accumbens of freely moving rats determined by on-line dialysis: effects of apomorphine and the neuroleptic-like peptide desenkephalin-gamma-endorphin.
    Neuroscience letters, 1988, Jul-08, Volume: 89, Issue:3

    Topics: Animals; Antipsychotic Agents; Apomorphine; beta-Endorphin; Computers; Dialysis; Dopamine; Male; Motor Activity; Nucleus Accumbens; Peptides; Rats; Rats, Inbred Strains; Septal Nuclei

1988
The neuroleptic-like peptide desenkephalin-gamma-endorphin does not antagonize the dopamine receptor agonist-induced inhibition of the release of [3H]dopamine from rat nucleus accumbens slices in vitro.
    Brain research, 1987, Nov-24, Volume: 426, Issue:2

    Topics: Animals; Apomorphine; beta-Endorphin; Dopamine; Ergolines; In Vitro Techniques; Male; Nucleus Accumbens; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Septal Nuclei; Tritium

1987
The hypomotility elicited by small doses of apomorphine seems exclusively mediated by dopaminergic systems in the nucleus accumbens.
    European journal of pharmacology, 1987, May-07, Volume: 137, Issue:1

    Topics: Analysis of Variance; Animals; Apomorphine; beta-Endorphin; Endorphins; Haloperidol; Male; Motor Activity; Nucleus Accumbens; Rats; Rats, Inbred Strains; Receptors, Dopamine; Septal Nuclei; Stereotyped Behavior; Sulpiride

1987
Desenkephalin-gamma-endorphin restores the impaired sensitivity of hypophysectomized rats to small doses of apomorphine.
    European journal of pharmacology, 1986, Sep-09, Volume: 128, Issue:3

    Topics: Animals; Apomorphine; beta-Endorphin; Endorphins; Hypophysectomy; Male; Motor Activity; Prolactin; Rats; Rats, Inbred Strains; Stereotyped Behavior

1986
Non-opiate beta-endorphin fragments and dopamine--VI. Behavioural analysis of the interaction between gamma-type endorphins and dopaminergic systems in the nucleus accumbens of rats.
    Neuropharmacology, 1984, Volume: 23, Issue:5

    Topics: Amphetamine; Animals; Apomorphine; Behavior, Animal; beta-Endorphin; Bromocriptine; Dopamine; Endorphins; Ergolines; Fluphenazine; gamma-Endorphin; Haloperidol; Male; Motor Activity; Nucleus Accumbens; Rats; Rats, Inbred Strains; Septal Nuclei; Sulpiride

1984
In vivo interaction of gamma-type endorphins with dopaminergic ligands in rat brain.
    European journal of pharmacology, 1983, Apr-08, Volume: 88, Issue:4

    Topics: Animals; Apomorphine; beta-Endorphin; Brain; Endorphins; Motor Activity; Peptide Fragments; Rats; Receptors, Dopamine; Spiperone

1983
Subchronic treatment with the neuroleptic-like peptide desenkephalin-gamma-endorphin may decrease dopaminergic neurotransmission in the nucleus accumbens of rats.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 1994, Volume: 4, Issue:2

    Topics: Animals; Antipsychotic Agents; Apomorphine; beta-Endorphin; Depression, Chemical; Dopamine; Dopamine Agents; In Vitro Techniques; Injections; Injections, Subcutaneous; Male; Nucleus Accumbens; Rats; Rats, Wistar; Synaptic Transmission

1994