Page last updated: 2024-09-03

dermorphin, arg(2)- and morphine

dermorphin, arg(2)- has been researched along with morphine in 2 studies

Compound Research Comparison

Studies
(dermorphin, arg(2)-)
Trials
(dermorphin, arg(2)-)
Recent Studies (post-2010)
(dermorphin, arg(2)-)
Studies
(morphine)
Trials
(morphine)
Recent Studies (post-2010) (morphine)
120144,2705,2008,695

Protein Interaction Comparison

ProteinTaxonomydermorphin, arg(2)- (IC50)morphine (IC50)
Delta-type opioid receptorMus musculus (house mouse)0.2939
Delta-type opioid receptorRattus norvegicus (Norway rat)0.2278
Kappa-type opioid receptorMus musculus (house mouse)0.0828
Mu-type opioid receptorRattus norvegicus (Norway rat)0.0385
Kappa-type opioid receptorRattus norvegicus (Norway rat)0.0545
Mu-type opioid receptorHomo sapiens (human)0.122
Delta-type opioid receptorHomo sapiens (human)0.1199
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)0.9308
Kappa-type opioid receptorHomo sapiens (human)0.655
Mu-type opioid receptorMus musculus (house mouse)0.3305
Mu-type opioid receptorCavia porcellus (domestic guinea pig)0.202
Beta-2 adrenergic receptorCavia porcellus (domestic guinea pig)0.25

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (50.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's1 (50.00)2.80

Authors

AuthorsStudies
Imam, MZ; Kong, D; Kuo, A; Smith, MT; Williams, CM1
Chaki, K; Kawamura, S; Kisara, K; Nakata, N; Sakurada, S; Sakurada, T; Suzuki, K1

Other Studies

2 other study(ies) available for dermorphin, arg(2)- and morphine

ArticleYear
Analgesic Opioid Ligand Discovery Based on Nonmorphinan Scaffolds Derived from Natural Sources.
    Journal of medicinal chemistry, 2022, 02-10, Volume: 65, Issue:3

    Topics: Analgesics, Opioid; Animals; Biological Products; Cell Line, Tumor; Chemistry, Pharmaceutical; Drug Discovery; Humans; Ligands; Pain; Peptides; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu

2022
Tolerance and cross-tolerance to the antinociceptive effects of [D-Arg2]-dermorphin tetrapeptide analogue and morphine.
    Neuropharmacology, 1993, Volume: 32, Issue:7

    Topics: Amino Acid Sequence; Analgesics; Animals; Drug Tolerance; Male; Molecular Sequence Data; Morphine; Nociceptors; Oligopeptides; Pain Measurement; Rats; Rats, Wistar

1993