Page last updated: 2024-09-03

dermorphin, arg(2)- and dermorphin

dermorphin, arg(2)- has been researched along with dermorphin in 5 studies

Compound Research Comparison

Studies
(dermorphin, arg(2)-)
Trials
(dermorphin, arg(2)-)
Recent Studies (post-2010)
(dermorphin, arg(2)-)
Studies
(dermorphin)
Trials
(dermorphin)
Recent Studies (post-2010) (dermorphin)
1201401239

Protein Interaction Comparison

ProteinTaxonomydermorphin, arg(2)- (IC50)dermorphin (IC50)
Delta-type opioid receptorMus musculus (house mouse)0.0389
Mu-type opioid receptorRattus norvegicus (Norway rat)0.0043
Mu-type opioid receptorHomo sapiens (human)0.0018
Delta-type opioid receptorHomo sapiens (human)0.2492
Mu-type opioid receptorMus musculus (house mouse)0.0086
Mu-type opioid receptorCavia porcellus (domestic guinea pig)0.0026

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19903 (60.00)18.7374
1990's1 (20.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's1 (20.00)2.80

Authors

AuthorsStudies
Imam, MZ; Kong, D; Kuo, A; Smith, MT; Williams, CM1
Kisara, K; Sakurada, S; Sakurada, T; Sasaki, Y; Suzuki, K; Watanabe, H1
Fujita, H; Hosono, M; Kisara, K; Matsui, M; Sakurada, S; Sakurada, T; Sasaki, Y; Suzuki, K1
Kisara, K; Sakurada, S; Sakurada, T; Sasaki, Y; Sato, T; Suzuki, K; Watanabe, H1
Baturina, EIu; Deĭgin, VI; Iarova, EP; Kamenskiĭ, AA; Sarycheva, NIu1

Other Studies

5 other study(ies) available for dermorphin, arg(2)- and dermorphin

ArticleYear
Analgesic Opioid Ligand Discovery Based on Nonmorphinan Scaffolds Derived from Natural Sources.
    Journal of medicinal chemistry, 2022, 02-10, Volume: 65, Issue:3

    Topics: Analgesics, Opioid; Animals; Biological Products; Cell Line, Tumor; Chemistry, Pharmaceutical; Drug Discovery; Humans; Ligands; Pain; Peptides; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu

2022
Different effects of peptidase inhibitors on dermorphin- and on [D-Arg2]dermorphin-induced antinociceptive activity.
    European journal of pharmacology, 1992, Jan-28, Volume: 211, Issue:1

    Topics: Analgesics, Opioid; Animals; Anti-Bacterial Agents; Captopril; Male; Mice; Mice, Inbred Strains; Oligopeptides; Opioid Peptides; Pain Measurement; Peptides; Thiorphan

1992
On the degradation of dermorphin and D-Arg2-dermorphin analogs by a soluble rat brain extract.
    Biochemical and biophysical research communications, 1985, Aug-15, Volume: 130, Issue:3

    Topics: Amino Acids; Analgesics, Opioid; Animals; Anti-Bacterial Agents; Brain; Captopril; Chromatography, High Pressure Liquid; Cytosol; Kinetics; Oligopeptides; Opioid Peptides; Peptides; Rats; Rats, Inbred Strains; Structure-Activity Relationship

1985
Dermorphin analogues containing D-kyotorphin: structure-antinociceptive relationships in mice.
    British journal of pharmacology, 1986, Volume: 87, Issue:1

    Topics: Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Ileum; In Vitro Techniques; Male; Mice; Muscle Contraction; Oligopeptides; Opioid Peptides; Peptide Fragments; Structure-Activity Relationship

1986
[Paradoxical correlations of the effectiveness of the intranasal and intraperitoneal administration of dermorphins in rats].
    Biulleten' eksperimental'noi biologii i meditsiny, 1988, Volume: 105, Issue:2

    Topics: Administration, Intranasal; Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Injections, Intraperitoneal; Male; Oligopeptides; Opioid Peptides; Pain Measurement; Rats; Reaction Time; Time Factors

1988