Page last updated: 2024-09-03

deramciclane and tiagabine

deramciclane has been researched along with tiagabine in 2 studies

Compound Research Comparison

Studies
(deramciclane)
Trials
(deramciclane)
Recent Studies (post-2010)
(deramciclane)
Studies
(tiagabine)
Trials
(tiagabine)
Recent Studies (post-2010) (tiagabine)
40102571102111

Protein Interaction Comparison

ProteinTaxonomyderamciclane (IC50)tiagabine (IC50)
Sodium- and chloride-dependent GABA transporter 1Rattus norvegicus (Norway rat)2.2107
Sodium- and chloride-dependent GABA transporter 1Homo sapiens (human)0.2213
Sodium- and chloride-dependent GABA transporter 1Mus musculus (house mouse)0.1968
Sodium- and chloride-dependent betaine transporterMus musculus (house mouse)0.27

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (50.00)18.2507
2000's0 (0.00)29.6817
2010's1 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kardos, J; Kovács, I; Nyitrai, G; Skuban, N1
Hiramatsu, M1

Reviews

1 review(s) available for deramciclane and tiagabine

ArticleYear
[Functional role for GABA transporters in the CNS].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 2014, Volume: 143, Issue:4

    Topics: Animals; Brain; Camphanes; Carbazoles; Carrier Proteins; Central Nervous System Diseases; Drug Discovery; GABA Plasma Membrane Transport Proteins; GABA Uptake Inhibitors; Humans; Isoxazoles; Mental Disorders; Molecular Targeted Therapy; Nipecotic Acids; Piperidines; Tiagabine

2014

Other Studies

1 other study(ies) available for deramciclane and tiagabine

ArticleYear
Inhibition of [3H]D-aspartate release by deramciclane.
    European journal of pharmacology, 1999, Sep-24, Volume: 381, Issue:2-3

    Topics: 4-Aminopyridine; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Anxiety Agents; Aspartic Acid; Camphanes; Cell Membrane; Cerebral Cortex; Depression, Chemical; Excitatory Amino Acid Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Male; Nerve Endings; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Rats; Rats, Wistar; Receptors, GABA-A; Tiagabine

1999