Page last updated: 2024-09-02

deoxyglucose and verapamil

deoxyglucose has been researched along with verapamil in 18 studies

Compound Research Comparison

Studies
(deoxyglucose)
Trials
(deoxyglucose)
Recent Studies (post-2010)
(deoxyglucose)
Studies
(verapamil)
Trials
(verapamil)
Recent Studies (post-2010) (verapamil)
11,4261711,37517,6211,5272,067

Protein Interaction Comparison

ProteinTaxonomydeoxyglucose (IC50)verapamil (IC50)
Solute carrier family 22 member 1 Homo sapiens (human)6.8
Voltage-dependent L-type calcium channel subunit alpha-1FHomo sapiens (human)0.2
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.297
ATP-dependent translocase ABCB1Mus musculus (house mouse)2
ATP-dependent translocase ABCB1Homo sapiens (human)2.2346
Cytochrome P450 3A4Homo sapiens (human)3.8008
Alpha-2A adrenergic receptorHomo sapiens (human)0.579
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)3.02
ATP-dependent translocase ABCB1Mus musculus (house mouse)10
Catechol O-methyltransferaseHomo sapiens (human)0.2
Potassium voltage-gated channel subfamily A member 3Homo sapiens (human)8
Histamine H2 receptorHomo sapiens (human)2.59
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.442
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.297
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)3.02
Sodium-dependent serotonin transporterHomo sapiens (human)0.24
Multidrug resistance-associated protein 1 Homo sapiens (human)5.598
D(3) dopamine receptorHomo sapiens (human)0.186
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.165
5-hydroxytryptamine receptor 7Cavia porcellus (domestic guinea pig)6.8
Voltage-dependent L-type calcium channel subunit alpha-1D Homo sapiens (human)0.2
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)0.3945
Voltage-dependent L-type calcium channel subunit alpha-1SHomo sapiens (human)0.2
Voltage-dependent L-type calcium channel subunit alpha-1CHomo sapiens (human)0.175
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)1.1934

Research

Studies (18)

TimeframeStudies, this research(%)All Research%
pre-19905 (27.78)18.7374
1990's9 (50.00)18.2507
2000's3 (16.67)29.6817
2010's1 (5.56)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Baum, SG; Fleischer, N; Kaneko, Y; Shapiro, S1
Daniel, JC; Lecerf, JM; Levy, SB; Slapak, CA1
Briggs, JP; Brosius, FC; Furspan, PB; Lorenz, JN; Schnermann, J1
Gibson, IF; Martin, W; Weir, CJ1
Castillo, GR; Rosen, OM; Vera, JC1
Byers, DM; Cook, HW; George, TP; Palmer, FB; Spence, MW1
Segal, J1
Draznin, B; Kao, M; Sherman, N; Sussman, KE1
Breitbart, H; Rubinstein, S; Zarca, A1
Draznin, B; Eckel, RH; Kao, M; Sherman, NA; Sussman, KE; Yost, T1
Gimeno, AL; Gimeno, MF; Goldraij, A; Sterin, AB1
Kopsidas, G; MacPhee, DG1
Bright, RT; Rubin, LJ; Salvaterra, CG; Yuan, XJ1
Leist, M; Nicotera, P; Volbracht, C1
Borchard, G; de Boer, AG; Deryckere, K; Florea, BI; Junginger, HE; Kooiman, K; Schrier, SM; van der Sandt, IC1
Lerch, R; Montessuit, C; Papageorgiou, I; Rosenblatt-Velin, N1
Achilles, J; Harms, H; Müller, S1
Cok, A; Holstege, CP; Louters, LL; Rekman, J; Stehouwer, N; Tidball, A1

Other Studies

18 other study(ies) available for deoxyglucose and verapamil

ArticleYear
The role of calcium in insulin release from hamster insulinoma cells.
    Endocrinology, 1977, Volume: 101, Issue:2

    Topics: Adenoma, Islet Cell; Animals; Calcium; Cricetinae; Cyclic AMP; Deoxyglucose; Female; Glucagon; Glucose; Insulin; Insulin Secretion; Islets of Langerhans; Mesocricetus; Ouabain; Potassium; Rats; Somatostatin; Verapamil

1977
Energy-dependent accumulation of daunorubicin into subcellular compartments of human leukemia cells and cytoplasts.
    The Journal of biological chemistry, 1992, May-25, Volume: 267, Issue:15

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Cell Compartmentation; Chloroquine; Daunorubicin; Deoxyglucose; Dinitrophenols; Drug Interactions; Drug Resistance; Energy Metabolism; Ethylmaleimide; Humans; Leukemia; Membrane Glycoproteins; Methylamines; Microscopy, Fluorescence; Monensin; Ouabain; Sodium Azide; Tumor Cells, Cultured; Vanadates; Verapamil

1992
Intracellular ATP can regulate afferent arteriolar tone via ATP-sensitive K+ channels in the rabbit.
    The Journal of clinical investigation, 1992, Volume: 90, Issue:3

    Topics: Adenosine Triphosphate; Animals; Arterioles; Deoxyglucose; Diazoxide; Glyburide; In Vitro Techniques; Perfusion; Potassium Channels; Rabbits; Vasoconstriction; Verapamil

1992
Effects of metabolic inhibitors on endothelium-dependent and endothelium-independent vasodilatation of rat and rabbit aorta.
    British journal of pharmacology, 1991, Volume: 102, Issue:1

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Acetylcholine; Animals; Antimetabolites; Aorta, Thoracic; Bucladesine; Deoxyglucose; Endothelium, Vascular; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle Relaxation; Muscle Tonus; Muscle, Smooth, Vascular; Nitric Oxide; Nitroglycerin; Rabbits; Rats; Rats, Inbred Strains; Rotenone; Vasodilation; Verapamil

1991
A possible role for a mammalian facilitative hexose transporter in the development of resistance to drugs.
    Molecular and cellular biology, 1991, Volume: 11, Issue:7

    Topics: Amino Acid Sequence; Animals; Antibodies; ATP Binding Cassette Transporter, Subfamily B, Member 1; Brain; Cell Line; Cytochalasin B; Cytochalasins; Deoxyglucose; Drug Resistance; Glucose; Hexoses; Kinetics; Membrane Glycoproteins; Mice; Molecular Sequence Data; Monosaccharide Transport Proteins; Oocytes; Phloretin; Rats; Verapamil; Vinblastine; Xenopus laevis

1991
Inhibition of phosphatidylcholine and phosphatidylethanolamine biosynthesis by cytochalasin B in cultured glioma cells: potential regulation of biosynthesis by Ca(2+)-dependent mechanisms.
    Biochimica et biophysica acta, 1991, Jul-09, Volume: 1084, Issue:2

    Topics: Animals; Biological Transport, Active; Calcium; Carbon Radioisotopes; Cell Line; Choline; Cytochalasin B; Deoxyglucose; Ethanolamine; Ethanolamines; Glioma; Glucose; Kinetics; Phosphates; Phosphatidylcholines; Phosphatidylethanolamines; Phosphorus Radioisotopes; Rats; Tritium; Verapamil

1991
In vivo effect of 3,5,3'-triiodothyronine on calcium uptake in several tissues in the rat: evidence for a physiological role for calcium as the first messenger for the prompt action of thyroid hormone at the level of the plasma membrane.
    Endocrinology, 1990, Volume: 127, Issue:1

    Topics: Adipose Tissue; Animals; Cadmium; Calcium; Calcium Radioisotopes; Deoxyglucose; Diaphragm; Female; Heart; Kinetics; Lanthanum; Liver; Male; Manganese; Myocardium; Rats; Triiodothyronine; Verapamil

1990
Relationship between cytosolic free calcium concentration and 2-deoxyglucose uptake in adipocytes isolated from 2- and 12-month-old rats.
    Endocrinology, 1988, Volume: 122, Issue:6

    Topics: Adipose Tissue; Aging; Animals; Calcium; Cytosol; Deoxy Sugars; Deoxyglucose; Glyburide; Insulin; Ion Channels; Kinetics; Male; Nitrendipine; Potassium; Rats; Rats, Inbred Strains; Verapamil

1988
Transport mechanism for calcium and phosphate in ram spermatozoa.
    Biochimica et biophysica acta, 1988, Oct-20, Volume: 944, Issue:3

    Topics: Animals; Biological Transport; Calcium; Calcium-Binding Proteins; Cell Membrane; Deoxyglucose; Male; Mersalyl; Oligomycins; Oxygen Consumption; Phosphates; Ruthenium Red; Sheep; Sperm Motility; Spermatozoa; Verapamil

1988
Possible role of cytosolic free calcium concentrations in mediating insulin resistance of obesity and hyperinsulinemia.
    The Journal of clinical investigation, 1988, Volume: 82, Issue:6

    Topics: Adipose Tissue; Adult; Biopsy; Calcium; Cytosol; Deoxyglucose; Female; Glyburide; Humans; Hyperinsulinism; In Vitro Techniques; Insulin; Insulin Resistance; Obesity; Verapamil

1988
Modification by insulin of the effects of anoxia, substrate deprivation, metabolic inhibitors and verapamil on contractions of isolated rat uterine smooth muscle.
    Pharmacological research communications, 1982, Volume: 14, Issue:3

    Topics: Animals; Antimetabolites; Deoxyglucose; Female; In Vitro Techniques; Insulin; Iodoacetates; Iodoacetic Acid; Oxytocin; Rats; Rats, Inbred Strains; Uterine Contraction; Uterus; Verapamil

1982
Mutagenesis by 9-aminoacridine in Salmonella typhimurium: inhibition by glucose and other PTS class A carbon sources.
    Mutation research, 1994, Apr-15, Volume: 306, Issue:2

    Topics: Aminacrine; Arabinose; Deoxyglucose; Glucose; Glycerol; Lactates; Lactic Acid; Methylglucosides; Mutagenesis; Phosphoenolpyruvate Sugar Phosphotransferase System; Salmonella typhimurium; Verapamil

1994
Inhibition of glycolysis by 2-DG increases [Ca2+]i in pulmonary arterial smooth muscle cells.
    The American journal of physiology, 1995, Volume: 269, Issue:2 Pt 1

    Topics: Animals; Calcium; Calcium-Transporting ATPases; Cells, Cultured; Deoxyglucose; Extracellular Space; Glycolysis; Indoles; Intracellular Membranes; Muscle, Smooth, Vascular; Osmolar Concentration; Pulmonary Artery; Rats; Verapamil

1995
ATP controls neuronal apoptosis triggered by microtubule breakdown or potassium deprivation.
    Molecular medicine (Cambridge, Mass.), 1999, Volume: 5, Issue:7

    Topics: Adenosine Triphosphate; Amino Acid Chloromethyl Ketones; Animals; Apoptosis; Carrier Proteins; Caspase 3; Caspase Inhibitors; Caspases; Cerebellum; Colchicine; Cyclosporine; Cysteine Proteinase Inhibitors; Deoxyglucose; Dizocilpine Maleate; Energy Metabolism; Enzyme Activation; Enzyme Inhibitors; Glutathione; Mice; Mice, Inbred BALB C; Microfilament Proteins; Microtubules; Neurons; Neuroprotective Agents; Nitroso Compounds; Nocodazole; Oligopeptides; Paclitaxel; Potassium; Protein Biosynthesis; S-Nitrosoglutathione; Tacrolimus; Verapamil

1999
Evidence of P-glycoprotein mediated apical to basolateral transport of flunisolide in human broncho-tracheal epithelial cells (Calu-3).
    British journal of pharmacology, 2001, Volume: 134, Issue:7

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Bronchi; Cell Line; Cell Polarity; Cell Survival; Cyclosporins; Deoxyglucose; Dibenzocycloheptenes; Epithelial Cells; Fluocinolone Acetonide; Humans; Immunoblotting; Mass Spectrometry; Microscopy, Confocal; Quinolines; Sodium Azide; Temperature; Time Factors; Trachea; Verapamil

2001
Insulin resistance in adult cardiomyocytes undergoing dedifferentiation: role of GLUT4 expression and translocation.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 2004, Volume: 18, Issue:7

    Topics: Animals; Atrial Natriuretic Factor; Biological Transport, Active; Calcium Channel Blockers; Cell Differentiation; Cell Size; Cells, Cultured; Deoxyglucose; Diacetyl; Enzyme Activation; Gene Expression Regulation; Glucose Transporter Type 1; Glucose Transporter Type 4; Insulin; Insulin Resistance; Monosaccharide Transport Proteins; Muscle Proteins; Myocardial Contraction; Myocytes, Cardiac; Phosphatidylinositol 3-Kinases; Phosphorylation; Protein Processing, Post-Translational; Protein Serine-Threonine Kinases; Protein Transport; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Proto-Oncogene Proteins c-cbl; Rats; RNA, Messenger; Sarcolemma; Ubiquitin-Protein Ligases; Verapamil

2004
Analysis of living S. cerevisiae cell states--a three color approach.
    Cytometry. Part A : the journal of the International Society for Analytical Cytology, 2006, Volume: 69, Issue:3

    Topics: 4-Chloro-7-nitrobenzofurazan; Benzimidazoles; Calcium Channel Blockers; Cell Division; Cell Respiration; Deoxyglucose; DNA, Fungal; Flow Cytometry; Fluorescent Dyes; Indoles; Microscopy, Fluorescence; Propidium; Saccharomyces cerevisiae; Staining and Labeling; Verapamil

2006
Verapamil inhibits the glucose transport activity of GLUT1.
    Journal of medical toxicology : official journal of the American College of Medical Toxicology, 2010, Volume: 6, Issue:2

    Topics: Animals; Antimetabolites; Calcium Channel Blockers; Calcium Chloride; Chelating Agents; Deoxyglucose; Dose-Response Relationship, Drug; Edetic Acid; Fibroblasts; Glucose; Glucose Transporter Type 1; Hyperglycemia; Mice; Verapamil

2010