Page last updated: 2024-09-03

deltorphin ii, ala(2)- and estrone

deltorphin ii, ala(2)- has been researched along with estrone in 2 studies

Compound Research Comparison

Studies (deltorphin ii, ala(2)-)	Trials (deltorphin ii, ala(2)-)	Recent Studies (post-2010) (deltorphin ii, ala(2)-)	Studies (estrone)	Trials (estrone)	Recent Studies (post-2010) (estrone)
233	0	20	10,266	432	1,372

Protein Interaction Comparison

Protein	Taxonomy	estrone (IC50)
Estrogen receptor	Homo sapiens (human)	0.1261
Polyunsaturated fatty acid lipoxygenase ALOX15	Oryctolagus cuniculus (rabbit)	6.589
17-beta-hydroxysteroid dehydrogenase type 1	Homo sapiens (human)	0.4134
Sodium-dependent serotonin transporter	Homo sapiens (human)	5.301
Estrogen receptor beta	Homo sapiens (human)	0.3743
Broad substrate specificity ATP-binding cassette transporter ABCG2	Homo sapiens (human)	3

Research

Studies (2)

Timeframe	Studies, this research(%)	All Research%
pre-1990	0 (0.00)	18.7374
1990's	0 (0.00)	18.2507
2000's	2 (100.00)	29.6817
2010's	0 (0.00)	24.3611
2020's	0 (0.00)	2.80

Authors

Authors	Studies
Gervasini, G; Glaeser, H; Kim, RB; Leake, BF; Lee, W; Moeckel, GW; Roberts, RL; Smith, LH	1
Brun, ME; Funk, C; Grimm, HP; Kansy, M; Lavé, T; Poirier, A; Portmann, R; Senner, F	1

Other Studies

2 other study(ies) available for deltorphin ii, ala(2)- and estrone

Article	Year
Polymorphisms in human organic anion-transporting polypeptide 1A2 (OATP1A2): implications for altered drug disposition and central nervous system drug entry. The Journal of biological chemistry, 2005, Mar-11, Volume: 280, Issue:10 Topics: Amino Acid Sequence; Amino Acid Substitution; Brain; Enkephalin, D-Penicillamine (2,5)-; Estrone; Humans; Kidney; Kinetics; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Molecular Sequence Data; Oligopeptides; Organ Specificity; Polymorphism, Genetic; Polymorphism, Single Nucleotide; Protein Conformation; Protein Structure, Secondary	2005
Design, data analysis, and simulation of in vitro drug transport kinetic experiments using a mechanistic in vitro model. Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:12 Topics: Algorithms; Animals; Biological Transport, Active; CHO Cells; Computer Simulation; Cricetinae; Cricetulus; Diffusion; Estrone; Fatty Acids, Monounsaturated; Fluvastatin; Hepatocytes; Indoles; Kinetics; Male; Membranes, Artificial; Models, Biological; Naphthalenes; Oligopeptides; Organic Anion Transporters; Permeability; Pharmaceutical Preparations; Pharmacokinetics; Piperidines; Quinolines; Rats; Rats, Wistar; Sincalide; Temperature; Terfenadine	2008

Article

Year

Polymorphisms in human organic anion-transporting polypeptide 1A2 (OATP1A2): implications for altered drug disposition and central nervous system drug entry.

The Journal of biological chemistry, 2005, Mar-11, Volume: 280, Issue:10

Topics: Amino Acid Sequence; Amino Acid Substitution; Brain; Enkephalin, D-Penicillamine (2,5)-; Estrone; Humans; Kidney; Kinetics; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Molecular Sequence Data; Oligopeptides; Organ Specificity; Polymorphism, Genetic; Polymorphism, Single Nucleotide; Protein Conformation; Protein Structure, Secondary

2005

Design, data analysis, and simulation of in vitro drug transport kinetic experiments using a mechanistic in vitro model.

Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:12

Topics: Algorithms; Animals; Biological Transport, Active; CHO Cells; Computer Simulation; Cricetinae; Cricetulus; Diffusion; Estrone; Fatty Acids, Monounsaturated; Fluvastatin; Hepatocytes; Indoles; Kinetics; Male; Membranes, Artificial; Models, Biological; Naphthalenes; Oligopeptides; Organic Anion Transporters; Permeability; Pharmaceutical Preparations; Pharmacokinetics; Piperidines; Quinolines; Rats; Rats, Wistar; Sincalide; Temperature; Terfenadine

2008