Page last updated: 2024-09-03

deltorphin ii, ala(2)- and endomorphin 1

deltorphin ii, ala(2)- has been researched along with endomorphin 1 in 4 studies

Compound Research Comparison

Studies
(deltorphin ii, ala(2)-)
Trials
(deltorphin ii, ala(2)-)
Recent Studies (post-2010)
(deltorphin ii, ala(2)-)
Studies
(endomorphin 1)
Trials
(endomorphin 1)
Recent Studies (post-2010) (endomorphin 1)
7034482109
2330204482109

Protein Interaction Comparison

ProteinTaxonomydeltorphin ii, ala(2)- (IC50)endomorphin 1 (IC50)
Delta-type opioid receptorMus musculus (house mouse)0.026
Mu-type opioid receptorRattus norvegicus (Norway rat)0.0005
Mu-type opioid receptorHomo sapiens (human)0.0275
Mu-type opioid receptorMus musculus (house mouse)0.0363

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (25.00)18.2507
2000's1 (25.00)29.6817
2010's2 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Davis, P; Hruby, VJ; Lai, J; Lee, YS; Liu, L; Ma, SW; Petrov, RR; Porreca, F; Vanderah, TW; Vardanyan, RS1
Mizoguchi, H; Narita, M; Sora, I; Tseng, LF; Uhl, GR1
Gyires, K; Zádori, Z1
Bonnet, JJ; Costentin, J; Cravezic, A; do Rego, JC; Fichna, J; Gach, K; Janecka, A; Perlikowska, R; Wyrebska, A1

Other Studies

4 other study(ies) available for deltorphin ii, ala(2)- and endomorphin 1

ArticleYear
Effect of anchoring 4-anilidopiperidines to opioid peptides.
    Bioorganic & medicinal chemistry letters, 2013, Jun-01, Volume: 23, Issue:11

    Topics: Animals; Cell Line; Fentanyl; Humans; Kinetics; Mice; Opioid Peptides; Piperidines; Protein Binding; Receptors, Opioid, delta; Receptors, Opioid, mu; Structure-Activity Relationship

2013
Absence of G-protein activation by mu-opioid receptor agonists in the spinal cord of mu-opioid receptor knockout mice.
    British journal of pharmacology, 1999, Volume: 126, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Opioid; Animals; Binding, Competitive; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Membranes; Mice; Mice, Inbred C57BL; Mice, Inbred Strains; Mice, Knockout; Mice, Transgenic; Morphine; Oligopeptides; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Spinal Cord; Sulfur Radioisotopes; Tritium

1999
[Analysis of central mechanisms involved in gastric mucosal integrity].
    Neuropsychopharmacologia Hungarica : a Magyar Pszichofarmakologiai Egyesulet lapja = official journal of the Hungarian Association of Psychopharmacology, 2008, Volume: 10, Issue:3

    Topics: Animals; Arachidonic Acids; beta-Endorphin; Clonidine; Endocannabinoids; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Ethanol; Excitatory Amino Acids; Gastric Mucosa; Injections, Intraventricular; Male; Naloxone; Naltrexone; Narcotic Antagonists; Neurotransmitter Agents; Nociceptin; Oligopeptides; Opioid Peptides; Oxazoles; Polyunsaturated Alkamides; Rats; Rats, Wistar; Receptors, Opioid; Rilmenidine; Stomach Ulcer

2008
Effect of potent endomorphin degradation blockers on analgesic and antidepressant-like responses in mice.
    Neuropharmacology, 2011, Volume: 61, Issue:8

    Topics: Analgesics, Opioid; Analysis of Variance; Animals; Antidepressive Agents; Brain; Depression; Dipeptidyl Peptidase 4; Disease Models, Animal; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Hyperalgesia; Injections, Intraventricular; Male; Mice; Motor Activity; Oligopeptides; Pain Measurement; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu; Swimming; Tritium

2011