Page last updated: 2024-09-03

deltorphin ii, ala(2)- and dynorphins

deltorphin ii, ala(2)- has been researched along with dynorphins in 6 studies

Compound Research Comparison

Studies
(deltorphin ii, ala(2)-)
Trials
(deltorphin ii, ala(2)-)
Recent Studies (post-2010)
(deltorphin ii, ala(2)-)
Studies
(dynorphins)
Trials
(dynorphins)
Recent Studies (post-2010) (dynorphins)
703368415
602368415
2330203,09624514

Protein Interaction Comparison

ProteinTaxonomydeltorphin ii, ala(2)- (IC50)dynorphins (IC50)
Delta-type opioid receptorMus musculus (house mouse)0.0077
Kappa-type opioid receptorHomo sapiens (human)0.0001

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (33.33)18.2507
2000's3 (50.00)29.6817
2010's1 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Davis, P; Hruby, VJ; Lai, J; Lee, YS; Liu, L; Ma, SW; Petrov, RR; Porreca, F; Vanderah, TW; Vardanyan, RS1
Adapa, ID; Auh, JS; Berzetei-Gurske, IP; Brandt, SR; Craymer, K; Farrington, L; Haggart, D; Kennedy, JM; O'Brien, A; Polgar, WE; Rodriguez, L; Schwartz, RW; Toll, L; White, A1
Camargo, AC; Fernandes, BL; Ferro, ES; Gomes, MD; Juliano, L; Ribeiro, MJ; Sasaki, Y; Suzuki, K; Toffoletto, O1
Lunzer, MM; Portoghese, PS1
Chavkin, C; Gendron, L; Pintar, JE1
Capasso, A1

Other Studies

6 other study(ies) available for deltorphin ii, ala(2)- and dynorphins

ArticleYear
Effect of anchoring 4-anilidopiperidines to opioid peptides.
    Bioorganic & medicinal chemistry letters, 2013, Jun-01, Volume: 23, Issue:11

    Topics: Animals; Cell Line; Fentanyl; Humans; Kinetics; Mice; Opioid Peptides; Piperidines; Protein Binding; Receptors, Opioid, delta; Receptors, Opioid, mu; Structure-Activity Relationship

2013
Standard binding and functional assays related to medications development division testing for potential cocaine and opiate narcotic treatment medications.
    NIDA research monograph, 1998, Volume: 178

    Topics: Animals; Aorta, Thoracic; Cocaine; Cyclic AMP; Electric Stimulation; Guinea Pigs; Humans; Ileum; In Vitro Techniques; Male; Mice; Muscle, Smooth; Opioid-Related Disorders; Rats; Receptors, Dopamine; Receptors, Opioid; Receptors, Serotonin; Substance-Related Disorders

1998
Structural requirements of bioactive peptides for interaction with endopeptidase 22.19.
    Neuropeptides, 1994, Volume: 26, Issue:4

    Topics: Amino Acid Sequence; Animals; beta-Lipotropin; Bradykinin; Brain; Dynorphins; Metalloendopeptidases; Molecular Sequence Data; Neuropeptides; Oligopeptides; Rabbits; Structure-Activity Relationship; Substrate Specificity

1994
Identity of the putative delta1-opioid receptor as a delta-kappa heteromer in the mouse spinal cord.
    European journal of pharmacology, 2003, Apr-25, Volume: 467, Issue:1-3

    Topics: Animals; Benzylidene Compounds; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Immune Sera; Mice; Naltrexone; Oligopeptides; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Somatostatin; Spinal Cord

2003
Essential role of mu opioid receptor in the regulation of delta opioid receptor-mediated antihyperalgesia.
    Neuroscience, 2007, Dec-19, Volume: 150, Issue:4

    Topics: Animals; beta-Endorphin; Dose-Response Relationship, Drug; Dynorphins; Enkephalins; Freund's Adjuvant; Hyperalgesia; Inflammation; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Motor Activity; Naltrexone; Narcotic Antagonists; Oligopeptides; Pain Measurement; Protein Precursors; Reaction Time; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Somatostatin

2007
Comparison with naloxone of two dynorphin A analogues with K- and delta-opioid antagonist activity.
    Medicinal chemistry (Shariqah (United Arab Emirates)), 2009, Volume: 5, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Dose-Response Relationship, Drug; Dynorphins; Guinea Pigs; Ileum; Jejunum; Male; Muscle Contraction; Naloxone; Oligopeptides; Peptides; Rabbits; Receptors, Opioid, delta; Receptors, Opioid, kappa; Structure-Activity Relationship

2009