deltorphin ii, ala(2)- has been researched along with deltorphin in 8 studies
Studies (deltorphin ii, ala(2)-) | Trials (deltorphin ii, ala(2)-) | Recent Studies (post-2010) (deltorphin ii, ala(2)-) | Studies (deltorphin) | Trials (deltorphin) | Recent Studies (post-2010) (deltorphin) |
---|---|---|---|---|---|
233 | 0 | 20 | 174 | 1 | 18 |
Protein | Taxonomy | deltorphin ii, ala(2)- (IC50) | deltorphin (IC50) |
---|---|---|---|
Delta-type opioid receptor | Mus musculus (house mouse) | 0.0495 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 4 (50.00) | 18.2507 |
2000's | 1 (12.50) | 29.6817 |
2010's | 2 (25.00) | 24.3611 |
2020's | 1 (12.50) | 2.80 |
Authors | Studies |
---|---|
Davis, P; Horvath, R; Hruby, VJ; Kramer, TH; Lipkowski, AW; Misicka, A; Yamamura, HI | 1 |
Angelucci, F; Negri, L; Noviello, V | 1 |
Balboni, G; Borea, PA; Marastoni, M; Morari, M; Salvadori, S; Tomatis, R | 1 |
Borsodi, A; Darula, Z; Spetea, M; Tóth, G | 1 |
Chocyk, A; Labuz, D; Przewlocka, B; Toth, G; Wedzony, K | 1 |
Fairbanks, CA; Kitto, KF; Messing, RO; Metcalf, MD; Schuster, DJ; Wilcox, GL | 1 |
Hu, N; Li, Y; Shu, R; Wang, C; Wang, G; Wang, H; Xie, K; Yu, Y; Zhang, L | 1 |
Bhutia, YD; Ganapathy, V; Higuchi, K; Sato, T | 1 |
8 other study(ies) available for deltorphin ii, ala(2)- and deltorphin
Article | Year |
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Topographical requirements for delta opioid ligands: common structural features of dermenkephalin and deltorphin.
Topics: Amino Acid Sequence; Animals; Aspartic Acid; Guinea Pigs; In Vitro Techniques; Male; Mice; Mice, Inbred ICR; Models, Chemical; Molecular Sequence Data; Oligopeptides; Protein Conformation; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta | 1992 |
Behavioural effects of deltorphins in rats.
Topics: Analgesics; Animals; Behavior, Animal; Indoles; Injections, Intraventricular; Male; Morphinans; Motor Activity; Naloxone; Naltrexone; Oligopeptides; Pain Measurement; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Social Behavior; Stereotyped Behavior | 1991 |
Synthesis and structure-activity relationships of deltorphin analogues.
Topics: Amino Acid Sequence; Animals; Binding, Competitive; Chemical Phenomena; Chemistry; Guinea Pigs; Male; Mice; Molecular Sequence Data; Muscle, Smooth; Oligopeptides; Rats; Rats, Inbred Strains; Receptors, Opioid; Structure-Activity Relationship | 1991 |
Synthesis and binding characteristics of the highly selective radiolabelled deltorphin analogues containing 2-aminotetralin-2-carboxylic acid in position 3.
Topics: 2-Naphthylamine; Amino Acids; Animals; Brain; Membranes; Oligopeptides; Protein Conformation; Radioligand Assay; Rats; Rats, Wistar; Receptors, Opioid, delta; Tritium | 1997 |
Endomorphin-2, deltorphin II and their analogs suppress formalin-induced nociception and c-Fos expression in the rat spinal cord.
Topics: Analgesics, Opioid; Animals; Behavior, Animal; Dose-Response Relationship, Drug; Formaldehyde; Inflammation; Male; Morphine; Nociceptors; Oligopeptides; Proto-Oncogene Proteins c-fos; Rats; Rats, Wistar; Receptors, Opioid, delta; Receptors, Opioid, mu; Spinal Cord; Time Factors | 2003 |
Ligand requirements for involvement of PKCε in synergistic analgesic interactions between spinal μ and δ opioid receptors.
Topics: Analgesics, Opioid; Animals; Behavior, Animal; Drug Therapy, Combination; Female; Hot Temperature; Ligands; Male; Mice, Knockout; Morphine; Morpholines; Oligopeptides; Pain; Protein Kinase C-epsilon; Protein Multimerization; Receptors, Opioid, delta; Receptors, Opioid, mu; Spinal Cord | 2015 |
Inhibition of DOR prevents remifentanil induced postoperative hyperalgesia through regulating the trafficking and function of spinal NMDA receptors in vivo and in vitro.
Topics: Anesthetics, Intravenous; Animals; Disease Models, Animal; Hot Temperature; Hyperalgesia; Lumbar Vertebrae; Male; Naltrexone; Narcotic Antagonists; Oligopeptides; Pain Threshold; Pain, Postoperative; Piperidines; Posterior Horn Cells; Random Allocation; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid, delta; Remifentanil; Spinal Cord; Tissue Culture Techniques; Touch | 2015 |
Involvement of a Na
Topics: Amyloid beta-Peptides; Animals; Biological Transport; Blood-Brain Barrier; Cell Line; Endothelial Cells; Humans; Kinetics; Membrane Transport Modulators; Membrane Transport Proteins; Mice; Models, Biological; Oligopeptides; Peptide Fragments; Sodium | 2020 |