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deltorphin ii, ala(2)- and clonidine

deltorphin ii, ala(2)- has been researched along with clonidine in 5 studies

Compound Research Comparison

Studies
(deltorphin ii, ala(2)-)
Trials
(deltorphin ii, ala(2)-)
Recent Studies (post-2010)
(deltorphin ii, ala(2)-)
Studies
(clonidine)
Trials
(clonidine)
Recent Studies (post-2010) (clonidine)
23302013,6922,0441,394

Protein Interaction Comparison

ProteinTaxonomydeltorphin ii, ala(2)- (IC50)clonidine (IC50)
Alpha-2A adrenergic receptorHomo sapiens (human)0.101
Alpha-2B adrenergic receptorHomo sapiens (human)0.0353
Alpha-2C adrenergic receptorHomo sapiens (human)0.0115
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)5.365
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)0.0173
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)0.0173
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)0.0173
Alpha-1D adrenergic receptorHomo sapiens (human)1.21
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)5.365
Alpha-2A adrenergic receptorBos taurus (cattle)0.002
NischarinRattus norvegicus (Norway rat)0.3662

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's4 (80.00)29.6817
2010's1 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fairbanks, CA; Kitto, KF; Nguyen, HO; Posthumus, IJ; Stone, LS; Wilcox, GL1
Borys, D; Hosohata, K; Navratilova, E; Nylen, A; Porreca, F; Roeske, WR; Vanderah, TW; Varga, EV; Yamamura, HI1
Gyires, K; Zádori, Z1
Chabot-Doré, AJ; Fairbanks, CA; Kitto, KF; Overland, AC; Rothwell, PE; Stone, LS; Wilcox, GL1
Fairbanks, CA; Kitto, KF; Messing, RO; Overland, AC; Schuster, DJ; Stone, LS; Wilcox, GL1

Other Studies

5 other study(ies) available for deltorphin ii, ala(2)- and clonidine

ArticleYear
alpha(2C)-Adrenergic receptors mediate spinal analgesia and adrenergic-opioid synergy.
    The Journal of pharmacology and experimental therapeutics, 2002, Volume: 300, Issue:1

    Topics: Adrenergic alpha-Agonists; Analgesics; Analgesics, Opioid; Animals; Clonidine; Drug Synergism; Immunohistochemistry; Male; Mice; Mice, Inbred ICR; Mice, Knockout; Oligonucleotides, Antisense; Oligopeptides; Pain Measurement; Receptors, Adrenergic, alpha-2; Receptors, Opioid; Spinal Cord; Substance P; Sympathetic Nervous System

2002
Antinociception depends on the presence of G protein gamma2-subunits in brain.
    European journal of pharmacology, 2005, Jan-31, Volume: 508, Issue:1-3

    Topics: Analgesics; Analgesics, Opioid; Animals; Benzoxazines; Brain; Clonidine; GTP-Binding Proteins; Injections, Intraventricular; Male; Mice; Mice, Inbred ICR; Morphine; Morpholines; Naphthalenes; Oligonucleotides, Antisense; Oligopeptides; Pain; Pain Measurement; Time Factors

2005
[Analysis of central mechanisms involved in gastric mucosal integrity].
    Neuropsychopharmacologia Hungarica : a Magyar Pszichofarmakologiai Egyesulet lapja = official journal of the Hungarian Association of Psychopharmacology, 2008, Volume: 10, Issue:3

    Topics: Animals; Arachidonic Acids; beta-Endorphin; Clonidine; Endocannabinoids; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Ethanol; Excitatory Amino Acids; Gastric Mucosa; Injections, Intraventricular; Male; Naloxone; Naltrexone; Narcotic Antagonists; Neurotransmitter Agents; Nociceptin; Oligopeptides; Opioid Peptides; Oxazoles; Polyunsaturated Alkamides; Rats; Rats, Wistar; Receptors, Opioid; Rilmenidine; Stomach Ulcer

2008
Protein kinase C mediates the synergistic interaction between agonists acting at alpha2-adrenergic and delta-opioid receptors in spinal cord.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2009, Oct-21, Volume: 29, Issue:42

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Anesthetics, Local; Animals; Calcitonin Gene-Related Peptide; Clonidine; Dose-Response Relationship, Drug; Drug Combinations; Drug Synergism; Enzyme Inhibitors; Evoked Potentials; Excitatory Postsynaptic Potentials; Female; Hyperalgesia; In Vitro Techniques; Injections, Spinal; Male; Mice; Mice, Inbred C57BL; Mice, Inbred ICR; Oligopeptides; Patch-Clamp Techniques; Posterior Horn Cells; Potassium; Protein Kinase C; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Receptors, Opioid, delta; Signal Transduction; Spinal Cord; Substance P; Tetrodotoxin

2009
Protein kinase Cε is required for spinal analgesic synergy between delta opioid and alpha-2A adrenergic receptor agonist pairs.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2013, Aug-14, Volume: 33, Issue:33

    Topics: Adrenergic alpha-2 Receptor Agonists; Analgesics; Anesthesia, Spinal; Animals; Brimonidine Tartrate; Clonidine; Drug Synergism; Enzyme Inhibitors; Female; Immunohistochemistry; Isoenzymes; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Oligopeptides; Protein Kinase C-epsilon; Quinoxalines; Receptors, Adrenergic, alpha-2; Receptors, Opioid, delta; Spinal Cord

2013