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deltorphin i, ala(2)- and naltrexone

deltorphin i, ala(2)- has been researched along with naltrexone in 11 studies

Compound Research Comparison

Studies
(deltorphin i, ala(2)-)
Trials
(deltorphin i, ala(2)-)
Recent Studies (post-2010)
(deltorphin i, ala(2)-)
Studies
(naltrexone)
Trials
(naltrexone)
Recent Studies (post-2010) (naltrexone)
122048,7451,2282,642

Protein Interaction Comparison

ProteinTaxonomydeltorphin i, ala(2)- (IC50)naltrexone (IC50)
Cytochrome P450 2D6Homo sapiens (human)1
Delta-type opioid receptorMus musculus (house mouse)0.0051
Delta-type opioid receptorRattus norvegicus (Norway rat)0.0063
Kappa-type opioid receptorMus musculus (house mouse)0.006
Mu-type opioid receptorRattus norvegicus (Norway rat)0.0005
Kappa-type opioid receptorRattus norvegicus (Norway rat)0.0005
Mu-type opioid receptorHomo sapiens (human)0.006
Delta-type opioid receptorHomo sapiens (human)0.0319
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)0.0093
Kappa-type opioid receptorHomo sapiens (human)0.0377
Mu-type opioid receptorMus musculus (house mouse)0.0076
Mu-type opioid receptorCavia porcellus (domestic guinea pig)0.0004

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's8 (72.73)18.2507
2000's3 (27.27)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Crook, TJ; Hill, RG; Kitchen, I1
Angelucci, F; Negri, L; Noviello, V1
Crook, TJ; Hill, RG; Kitchen, I; Muhammad, BY1
Iwamoto, Y; Kamei, J; Kasuya, Y; Misawa, M; Nagase, H1
Mokhtari, M; Tafani, JA; Zajac, JM1
Capobianchi, MR; Negri, L; Noviello, L; Papadia, S1
Desprat, C; Zajac, JM1
Borsodi, A; Hill, RG; Kelly, MD; Kitchen, I; Toth, G1
Kieffer, BL; Maldonado, R; Matthes, HW; Melchiorri, P; Negri, L; Severini, C1
Barlow, M; Caffrey, JL; Davis, S; Deo, SH; Farias, M; Yoshishige, D1
Balboni, G; Jinsmaa, Y; Lazarus, LH; Marczak, ED; Salvadori, S1

Other Studies

11 other study(ies) available for deltorphin i, ala(2)- and naltrexone

ArticleYear
Effects of the delta-opioid receptor antagonist naltrindole on antinociceptive responses to selective delta-agonists in post-weanling rats.
    British journal of pharmacology, 1992, Volume: 107, Issue:2

    Topics: Analgesics; Animals; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine; Enkephalins; Indoles; Male; Morphinans; Naloxone; Naltrexone; Narcotic Antagonists; Oligopeptides; Pain Measurement; Rats; Rats, Wistar; Receptors, Opioid, delta

1992
Behavioural effects of deltorphins in rats.
    European journal of pharmacology, 1991, Dec-17, Volume: 209, Issue:3

    Topics: Analgesics; Animals; Behavior, Animal; Indoles; Injections, Intraventricular; Male; Morphinans; Motor Activity; Naloxone; Naltrexone; Oligopeptides; Pain Measurement; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Social Behavior; Stereotyped Behavior

1991
Evidence that weaning stimulates the developmental expression of a delta-opioid receptor subtype in the rat.
    Brain research. Developmental brain research, 1994, Mar-18, Volume: 78, Issue:1

    Topics: Analgesics; Animals; Dose-Response Relationship, Drug; Enkephalin, Leucine; Female; Male; Naltrexone; Narcotic Antagonists; Oligopeptides; Rats; Rats, Wistar; Receptors, Opioid, delta; Weaning

1994
Streptozotocin-induced diabetes selectively enhances antinociception mediated by delta 1- but not delta 2-opioid receptors.
    Life sciences, 1994, Volume: 55, Issue:6

    Topics: Analgesia; Animals; Benzylidene Compounds; Diabetes Mellitus, Experimental; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Male; Mice; Mice, Inbred ICR; Naltrexone; Oligopeptides; Receptors, Opioid, delta; Receptors, Opioid, mu; Streptozocin

1994
Binding in vivo of selective mu and delta opioid agonists: localization by autoradiography.
    Neuropeptides, 1993, Volume: 25, Issue:3

    Topics: Amino Acid Sequence; Analgesics; Animals; Autoradiography; Binding, Competitive; Brain; D-Ala(2),MePhe(4),Met(0)-ol-enkephalin; Diffusion; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Injections, Intraventricular; Male; Mice; Molecular Sequence Data; Naltrexone; Oligopeptides; Pain Measurement; Protein Binding; Receptors, Opioid, delta; Receptors, Opioid, mu

1993
Immunomodulatory responses to delta-opioid receptor ligands in human lymphocytes.
    European journal of pharmacology, 1997, Aug-06, Volume: 332, Issue:2

    Topics: Analgesics, Opioid; Humans; Interferon-gamma; Leukocytes, Mononuclear; Ligands; Lymphocyte Activation; Naltrexone; Narcotic Antagonists; Oligopeptides; Phytohemagglutinins; Receptors, Opioid, delta; Thymidine

1997
Differential modulation of mu- and delta-opioid antinociception by neuropeptide FF receptors in young mice.
    Neuropeptides, 1997, Volume: 31, Issue:1

    Topics: Age Factors; Analgesics, Opioid; Animals; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Male; Mice; Mice, Inbred Strains; Morphine; Naltrexone; Narcotic Antagonists; Neuropeptides; Nociceptors; Oligopeptides; Receptors, Neuropeptide; Receptors, Opioid, delta; Receptors, Opioid, mu

1997
Weaning-induced development of delta-opioid receptors in rat brain: differential effects of guanine nucleotides and sodium upon ligand-receptor recognition.
    British journal of pharmacology, 1998, Volume: 125, Issue:5

    Topics: Animals; Brain; Guanylyl Imidodiphosphate; In Vitro Techniques; Ligands; Naltrexone; Oligopeptides; Rats; Rats, Wistar; Receptors, Opioid, delta; Sodium; Weaning

1998
Activity of mu- and delta-opioid agonists in vas deferens from mice deficient in MOR gene.
    British journal of pharmacology, 2001, Volume: 132, Issue:7

    Topics: Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Female; Genotype; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Mice, Inbred Strains; Mice, Mutant Strains; Morphine; Muscle Contraction; Naltrexone; Narcotic Antagonists; Oligopeptides; Receptors, Opioid, delta; Receptors, Opioid, mu; Vas Deferens

2001
The monosialosyl ganglioside GM-1 reduces the vagolytic efficacy of delta2-opioid receptor stimulation.
    American journal of physiology. Heart and circulatory physiology, 2006, Volume: 291, Issue:5

    Topics: Analgesics, Opioid; Animals; Benzylidene Compounds; Bradycardia; Dogs; Dose-Response Relationship, Drug; Enkephalin, Methionine; Female; G(M1) Ganglioside; Male; Naltrexone; Narcotic Antagonists; Oligopeptides; Receptors, Opioid, delta; Sinoatrial Node; Stimulation, Chemical; Vagus Nerve

2006
Inhibition of the development of morphine tolerance by a potent dual mu-delta-opioid antagonist, H-Dmt-Tic-Lys-NH-CH2-Ph.
    Pharmacology, biochemistry, and behavior, 2008, Volume: 90, Issue:4

    Topics: Analgesics, Opioid; Animals; Area Under Curve; Dose-Response Relationship, Drug; Drug Tolerance; Injections, Intraventricular; Injections, Subcutaneous; Ligands; Male; Mice; Morphine; Naltrexone; Narcotic Antagonists; Oligopeptides; Reaction Time; Receptors, Opioid, delta; Receptors, Opioid, mu; Somatostatin

2008