deltorphin i, ala(2)- has been researched along with etorphine in 7 studies
| Studies (deltorphin i, ala(2)-) | Trials (deltorphin i, ala(2)-) | Recent Studies (post-2010) (deltorphin i, ala(2)-) | Studies (etorphine) | Trials (etorphine) | Recent Studies (post-2010) (etorphine) |
|---|---|---|---|---|---|
| 122 | 0 | 4 | 798 | 23 | 63 |
| 122 | 0 | 4 | 12 | 0 | 1 |
| Protein | Taxonomy | deltorphin i, ala(2)- (IC50) | etorphine (IC50) |
|---|---|---|---|
| Delta-type opioid receptor | Rattus norvegicus (Norway rat) | 0.0074 | |
| Mu-type opioid receptor | Rattus norvegicus (Norway rat) | 0.0001 | |
| Kappa-type opioid receptor | Cavia porcellus (domestic guinea pig) | 0.0018 |
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 2 (28.57) | 18.2507 |
| 2000's | 4 (57.14) | 29.6817 |
| 2010's | 1 (14.29) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Allouche, S; Jauzac, P; Marie, N; Roussel, M | 1 |
| Allouche, S; Hasbi, A; Homburger, V; Jauzac, P; Polastron, J | 1 |
| Allouche, S; Jauzac, P; Lecoq, I; Marie, N | 1 |
| Aguila, B; Allouche, S; Davis, A; Hasbi, A; Jauzac, P; Marie, N | 1 |
| Benaderet, TS; Bishop-Mathis, K; Dersch, CM; Partilla, JS; Prisinzano, TE; Rothman, RB; Simpson, DS; Wang, X; Xu, H | 1 |
| Aguila, B; Allouche, S; Borsodi, A; Coulbault, L; Davis, A; Gurevich, VV; Hasbi, A; Jauzac, P; Le bras, F; Marie, N; Tóth, G | 1 |
| Bernard, D; Coop, A; MacKerell, AD | 1 |
7 other study(ies) available for deltorphin i, ala(2)- and etorphine
| Article | Year |
|---|---|
Differential desensitization of human delta-opioid receptors by peptide and alkaloid agonists.
Topics: Adenylyl Cyclase Inhibitors; Alkaloids; Analgesics; Analgesics, Opioid; Cyclic AMP; Drug Interactions; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Etorphine; Humans; Naloxone; Neuroblastoma; Oligopeptides; Peptides; Receptors, Opioid, delta; Tumor Cells, Cultured | 1999 |
Differential G-protein activation by alkaloid and peptide opioid agonists in the human neuroblastoma cell line SK-N-BE.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Alkaloids; Animals; Azides; Cell Membrane; Colforsin; Cyclic AMP; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Etorphine; GTP-Binding Proteins; Guanosine Triphosphate; Humans; Isoelectric Point; Neuroblastoma; Neurons; Oligodeoxyribonucleotides, Antisense; Oligopeptides; Peptides; Pertussis Toxin; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta; Tumor Cells, Cultured; Virulence Factors, Bordetella | 1999 |
Differential sorting of human delta-opioid receptors after internalization by peptide and alkaloid agonists.
Topics: Alkaloids; Analgesics, Opioid; Down-Regulation; Endosomes; Enkephalin, D-Penicillamine (2,5)-; Etorphine; Humans; Kinetics; Oligopeptides; Peptides; Receptors, Opioid, delta; Recombinant Proteins; Transfection | 2003 |
Different kinases desensitize the human delta-opioid receptor (hDOP-R) in the neuroblastoma cell line SK-N-BE upon peptidic and alkaloid agonists.
Topics: Analgesics, Opioid; Cell Line, Tumor; Cyclic AMP-Dependent Protein Kinases; Enkephalin, D-Penicillamine (2,5)-; Etorphine; G-Protein-Coupled Receptor Kinase 2; Humans; Mutation; Neuroblastoma; Oligopeptides; Protein Kinase C; Protein Kinase Inhibitors; Protein Kinases; Protein-Tyrosine Kinases; Receptors, Opioid, delta | 2008 |
Differential effects of opioid agonists on G protein expression in CHO cells expressing cloned human opioid receptors.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Opioid; Animals; Benzamides; Blotting, Western; CHO Cells; Cricetinae; Cricetulus; Diterpenes, Clerodane; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Etorphine; Female; Furans; Gene Expression; GTP-Binding Protein alpha Subunits, G12-G13; GTP-Binding Protein alpha Subunits, Gi-Go; Humans; Morphine; Oligopeptides; Piperazines; Pyrones; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu | 2008 |
ßarrestin1-biased agonism at human δ-opioid receptor by peptidic and alkaloid ligands.
Topics: Arrestins; beta-Arrestins; Cell Line; Endocytosis; Enkephalin, D-Penicillamine (2,5)-; Etorphine; Humans; Ligands; Oligopeptides; Receptors, Opioid, delta; RNA Interference; RNA, Small Interfering; Signal Transduction | 2012 |
Quantitative conformationally sampled pharmacophore for delta opioid ligands: reevaluation of hydrophobic moieties essential for biological activity.
Topics: Animals; Cell Line, Tumor; Enkephalin, Leucine; Hydrophobic and Hydrophilic Interactions; Ligands; Models, Molecular; Molecular Conformation; Phenylalanine; Quantitative Structure-Activity Relationship; Rats; Receptors, Opioid, delta | 2007 |