deltorphin i, ala(2)- has been researched along with deltorphin ii, ala(2)- in 20 studies
Studies (deltorphin i, ala(2)-) | Trials (deltorphin i, ala(2)-) | Recent Studies (post-2010) (deltorphin i, ala(2)-) | Studies (deltorphin ii, ala(2)-) | Trials (deltorphin ii, ala(2)-) | Recent Studies (post-2010) (deltorphin ii, ala(2)-) |
---|---|---|---|---|---|
122 | 0 | 4 | 233 | 0 | 20 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 1 (5.00) | 18.7374 |
1990's | 15 (75.00) | 18.2507 |
2000's | 3 (15.00) | 29.6817 |
2010's | 1 (5.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Davis, P; Horvath, R; Hruby, VJ; Kramer, TH; Lipkowski, AW; Misicka, A; Yamamura, HI | 1 |
Burks, TF; Carr, DB; Davis, P; Fang, L; Hruby, VJ; Knapp, RJ; Kramer, T; Lipkowski, AW; Misicka, A; Yamamura, HI | 1 |
Angelucci, F; Negri, L; Noviello, V | 1 |
Jacobson, AE; Ni, Q; Rice, KC; Rothman, RB; Xu, H | 1 |
Burks, TF; Davis, P; Haaseth, RC; Hruby, VJ; Kramer, TH; Matsunaga, TO; Toth, G | 1 |
Balboni, G; Borea, PA; Marastoni, M; Morari, M; Salvadori, S; Tomatis, R | 1 |
Corsi, R; Egger, R; Kreil, G; Negri, L; Richter, K; Severini, C | 1 |
Barra, D; Corsi, R; Erspamer, V; Falconieri-Erspamer, G; Kreil, G; Melchiorri, P; Negri, L; Severini, C; Simmaco, M | 1 |
Bouzit, H; Hepp, AM; Heyl, DL; Johnson, TW; Kurtz, KR; Mousigian, C; Schmitter, SJ | 1 |
Böcskey, Z; Borsodi, A; Darula, Z; Fülöp, F; Jaspers, H; Péter, A; Tóth, G; Tóth, Z; Tourwé, D; Verheyden, P | 1 |
Lattanzi, R; Melchiorri, P; Negri, L; Potenza, RL; Severini, C | 1 |
Abbruscato, TJ; Davis, TP; Gillespie, TJ; Hau, VS; Hruby, VJ; Thomas, SA; Zsigo, J | 1 |
Borsodi, A; Darula, Z; Spetea, M; Tóth, G | 1 |
Escobar, S; Heyl, DL; Makhlouf, H; Marks, EL; Mohammedshah, T; Mousigian, C; Schullery, SE; Wilenkin, BS | 1 |
Borsodi, A; Hill, RG; Kelly, MD; Kitchen, I; Toth, G | 1 |
Borsodi, A; Labuz, D; Machelska, H; Przewlocka, B; Przewłocki, R; Toth, G | 1 |
Kieffer, BL; Maldonado, R; Matthes, HW; Melchiorri, P; Negri, L; Severini, C | 1 |
Aibak, H; Beaudet, A; Cahill, CM; Clarke, PB; Collier, B; Henry, JL; Hoffert, C; Mennicken, F; Morinville, A; O'Donnell, D; Pradhan, A; Rymar, VV; Sadikot, AF; Stroh, T; Vincent, JP | 1 |
Dettmer, K; Hammock, BD; Hanna, D; Hansen, R; Whetstone, P | 1 |
Fairbanks, CA; Kitto, KF; Messing, RO; Metcalf, MD; Schuster, DJ; Wilcox, GL | 1 |
20 other study(ies) available for deltorphin i, ala(2)- and deltorphin ii, ala(2)-
Article | Year |
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Topographical requirements for delta opioid ligands: common structural features of dermenkephalin and deltorphin.
Topics: Amino Acid Sequence; Animals; Aspartic Acid; Guinea Pigs; In Vitro Techniques; Male; Mice; Mice, Inbred ICR; Models, Chemical; Molecular Sequence Data; Oligopeptides; Protein Conformation; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta | 1992 |
Topographical requirements for delta opioid ligands: presence of a carboxyl group in position 4 is not critical for deltorphin high delta receptor affinity and analgesic activity.
Topics: Amino Acid Sequence; Analgesics; Animals; Binding, Competitive; Brain; Male; Models, Molecular; Molecular Sequence Data; Oligopeptides; Pain; Protein Conformation; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta | 1991 |
Behavioural effects of deltorphins in rats.
Topics: Analgesics; Animals; Behavior, Animal; Indoles; Injections, Intraventricular; Male; Morphinans; Motor Activity; Naloxone; Naltrexone; Oligopeptides; Pain Measurement; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Social Behavior; Stereotyped Behavior | 1991 |
Preliminary ligand binding data for subtypes of the delta opioid receptor in rat brain membranes.
Topics: Amino Acid Sequence; Animals; Binding Sites; Brain; Cell Membrane; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; Kinetics; Molecular Sequence Data; Oligopeptides; Radioligand Assay; Rats; Receptors, Opioid; Receptors, Opioid, delta; Somatostatin | 1991 |
Influence of peptidase inhibitors on the apparent agonist potency of delta selective opioid peptides in vitro.
Topics: Amino Acid Sequence; Analgesics; Animals; Dose-Response Relationship, Drug; Endorphins; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Male; Mice; Mice, Inbred Strains; Molecular Sequence Data; Oligopeptides; Protease Inhibitors; Receptors, Opioid; Receptors, Opioid, delta; Vas Deferens | 1991 |
Synthesis and structure-activity relationships of deltorphin analogues.
Topics: Amino Acid Sequence; Animals; Binding, Competitive; Chemical Phenomena; Chemistry; Guinea Pigs; Male; Mice; Molecular Sequence Data; Muscle, Smooth; Oligopeptides; Rats; Rats, Inbred Strains; Receptors, Opioid; Structure-Activity Relationship | 1991 |
cDNAs encoding [D-Ala2]deltorphin precursors from skin of Phyllomedusa bicolor also contain genetic information for three dermorphin-related opioid peptides.
Topics: Amino Acid Sequence; Animals; Anura; Base Sequence; Colon; DNA; Guinea Pigs; In Vitro Techniques; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth; Oligopeptides; Opioid Peptides; Protein Precursors; Sequence Homology, Nucleic Acid; Skin | 1990 |
Deltorphins: a family of naturally occurring peptides with high affinity and selectivity for delta opioid binding sites.
Topics: Amino Acid Sequence; Animals; Anura; Brain; Enkephalins; Guinea Pigs; In Vitro Techniques; Kinetics; Male; Membranes; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth; Oligopeptides; Rats; Receptors, Opioid; Receptors, Opioid, delta; Skin; Vas Deferens | 1989 |
Substitution of aromatic and nonaromatic amino acids for the Phe3 residue in the delta-selective opioid peptide deltorphin I: effects on binding affinity and selectivity.
Topics: Amino Acid Sequence; Analgesics; Enkephalins; Kinetics; Molecular Sequence Data; Oligopeptides; Phenylalanine; Protein Conformation; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Structure-Activity Relationship; Tritium | 1994 |
Conformationally constrained deltorphin analogs with 2-aminotetralin-2-carboxylic acid in position 3.
Topics: Analgesics, Opioid; Animals; Binding, Competitive; Brain; Guinea Pigs; Ileum; Magnetic Resonance Spectroscopy; Male; Mice; Muscle Contraction; Oligopeptides; Opioid Peptides; Protein Binding; Protein Conformation; Rats; Receptors, Opioid, delta; Vas Deferens | 1997 |
Postnatal development of delta-opioid receptor subtypes in mice.
Topics: Animals; Animals, Suckling; Brain; Electric Stimulation; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Female; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Oligopeptides; Receptors, Opioid, delta; Vas Deferens | 1997 |
Structure-activity relationships of a series of [D-Ala2]deltorphin I and II analogues; in vitro blood-brain barrier permeability and stability.
Topics: Analgesics, Opioid; Animals; Blood-Brain Barrier; Cattle; Half-Life; In Vitro Techniques; Male; Mice; Mice, Inbred ICR; Oligopeptides; Recurrence; Structure-Activity Relationship | 1997 |
Synthesis and binding characteristics of the highly selective radiolabelled deltorphin analogues containing 2-aminotetralin-2-carboxylic acid in position 3.
Topics: 2-Naphthylamine; Amino Acids; Animals; Brain; Membranes; Oligopeptides; Protein Conformation; Radioligand Assay; Rats; Rats, Wistar; Receptors, Opioid, delta; Tritium | 1997 |
Binding to delta and mu opioid receptors by deltorphin I/II analogues modified at the Phe3 and Asp4/Glu4 side chains: a report of 32 new analogues and a QSAR study.
Topics: Algorithms; Amino Acid Substitution; Analgesics, Opioid; Kinetics; Ligands; Oligopeptides; Receptors, Opioid, delta; Receptors, Opioid, mu; Regression Analysis; Structure-Activity Relationship | 1997 |
Weaning-induced development of delta-opioid receptors in rat brain: differential effects of guanine nucleotides and sodium upon ligand-receptor recognition.
Topics: Animals; Brain; Guanylyl Imidodiphosphate; In Vitro Techniques; Ligands; Naltrexone; Oligopeptides; Rats; Rats, Wistar; Receptors, Opioid, delta; Sodium; Weaning | 1998 |
Antinociceptive effects of isoleucine derivatives of deltorphin I and deltorphin II in rat spinal cord: a search for selectivity of delta receptor subtypes.
Topics: Analgesics, Opioid; Animals; Isoleucine; Male; Oligopeptides; Pain Measurement; Pain Threshold; Rats; Rats, Wistar; Receptors, Opioid, delta; Spinal Cord | 1998 |
Activity of mu- and delta-opioid agonists in vas deferens from mice deficient in MOR gene.
Topics: Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Female; Genotype; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Mice, Inbred Strains; Mice, Mutant Strains; Morphine; Muscle Contraction; Naltrexone; Narcotic Antagonists; Oligopeptides; Receptors, Opioid, delta; Receptors, Opioid, mu; Vas Deferens | 2001 |
Morphine-induced changes in delta opioid receptor trafficking are linked to somatosensory processing in the rat spinal cord.
Topics: Animals; Fluorescent Dyes; Guanosine 5'-O-(3-Thiotriphosphate); In Situ Hybridization; Lumbosacral Region; Male; Microscopy, Fluorescence; Morphine; Narcotics; Oligopeptides; Posterior Horn Cells; Protein Transport; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta; Receptors, Opioid, mu; Rhizotomy; Spinal Cord; Up-Regulation | 2004 |
Autism and urinary exogenous neuropeptides: development of an on-line SPE-HPLC-tandem mass spectrometry method to test the opioid excess theory.
Topics: Analgesics, Opioid; Autistic Disorder; Case-Control Studies; Child; Chromatography, High Pressure Liquid; Endorphins; Humans; Methods; Neuropeptides; Oligopeptides; Tandem Mass Spectrometry | 2007 |
Ligand requirements for involvement of PKCε in synergistic analgesic interactions between spinal μ and δ opioid receptors.
Topics: Analgesics, Opioid; Animals; Behavior, Animal; Drug Therapy, Combination; Female; Hot Temperature; Ligands; Male; Mice, Knockout; Morphine; Morpholines; Oligopeptides; Pain; Protein Kinase C-epsilon; Protein Multimerization; Receptors, Opioid, delta; Receptors, Opioid, mu; Spinal Cord | 2015 |