Page last updated: 2024-09-03

deltakephalin and morphine

deltakephalin has been researched along with morphine in 20 studies

Compound Research Comparison

Studies
(deltakephalin)
Trials
(deltakephalin)
Recent Studies (post-2010)
(deltakephalin)
Studies
(morphine)
Trials
(morphine)
Recent Studies (post-2010) (morphine)
790044,2705,2008,695

Protein Interaction Comparison

ProteinTaxonomydeltakephalin (IC50)morphine (IC50)
Delta-type opioid receptorMus musculus (house mouse)0.2939
Delta-type opioid receptorRattus norvegicus (Norway rat)0.2278
Kappa-type opioid receptorMus musculus (house mouse)0.0828
Mu-type opioid receptorRattus norvegicus (Norway rat)0.0385
Kappa-type opioid receptorRattus norvegicus (Norway rat)0.0545
Mu-type opioid receptorHomo sapiens (human)0.122
Delta-type opioid receptorHomo sapiens (human)0.1199
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)0.9308
Kappa-type opioid receptorHomo sapiens (human)0.655
Mu-type opioid receptorMus musculus (house mouse)0.3305
Mu-type opioid receptorCavia porcellus (domestic guinea pig)0.202
Beta-2 adrenergic receptorCavia porcellus (domestic guinea pig)0.25

Research

Studies (20)

TimeframeStudies, this research(%)All Research%
pre-19907 (35.00)18.7374
1990's10 (50.00)18.2507
2000's3 (15.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Besse, D; Besson, JM; Lombard, MC1
Bing, Z; Bouhassira, D; Le Bars, D; Villanueva, L1
Layer, RT; Uretsky, NJ; Wallace, LJ1
Kaneto, H; Shiigi, Y; Takahashi, M1
Cesselin, F; Hamon, M; Legrand, JC; Lutz, O; Mauborgne, A1
Delay-Goyet, P; Meucci, E; Roques, BP; Zajac, JM1
Farges, RC; Meunier, JC; Moisand, C; Puget, A1
Blanchard, JC; Böhme, GA; Roques, BP; Stutzmann, JM2
Heyman, JS; Mosberg, HI; Omnaas, JR; Porreca, F; Vaught, JL1
Burks, TF; Hruby, VJ; Hurst, R; Mosberg, HI; Porreca, F1
Jauzac, P; Polastron, J1
Benoliel, JJ; Bourgoin, S; Cesselin, F; Collin, E; Hamon, M; Mauborgne, A1
Benoliel, JJ; Bourgoin, S; Cesselin, F; Collin, E; Hamon, M; Legrand, JC; Mauborgne, A1
Bourgoin, S; Cesselin, F; Collin, E; Frechilla, D; Hamon, M; Le Bars, D; Pohl, M1
Dupouy, V; Zajac, JM1
Catheline, G; Guilbaud, G; Idänpään-Heikkilä, JJ; Kayser, V1
Kramer, HK; Simon, EJ1
Jinsmaa, Y; Takahashi, M; Yoshikawa, M1
Jinsmaa, Y; Lipkowski, AW; Nakamura, F; Takenaka, Y; Yoshikawa, M1

Other Studies

20 other study(ies) available for deltakephalin and morphine

ArticleYear
Up-regulation of [3H]DAMGO and [3H]DTLET opioid binding sites in laminae I-II of the spinal cord in intact and deafferented morphine-tolerant rats.
    Neuroscience letters, 1992, Mar-02, Volume: 136, Issue:2

    Topics: Animals; Autoradiography; Drug Tolerance; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Morphine; Neurons, Afferent; Oligopeptides; Rats; Receptors, Opioid; Spinal Cord; Up-Regulation

1992
Depressive effects of mu and delta opioid receptor agonists on activities of dorsal horn neurones are enhanced by dibencozide.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 257, Issue:3

    Topics: Amino Acid Sequence; Analgesics; Animals; Cobamides; Depression, Chemical; Drug Interactions; Male; Molecular Sequence Data; Morphine; Nerve Fibers; Neurons; Oligopeptides; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu; Spinal Cord

1991
Effects of morphine in the nucleus accumbens on stimulant-induced locomotion.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 40, Issue:1

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amphetamine; Animals; Caffeine; Central Nervous System Stimulants; Dizocilpine Maleate; Dopamine Agents; Glutamine; Ibotenic Acid; Male; Morphine; Motor Activity; Neural Pathways; Nucleus Accumbens; Oligopeptides; Picrotoxin; Rats; Scopolamine; Synaptic Transmission

1991
Facilitation of memory retrieval by pretest morphine mediated by mu but not delta and kappa opioid receptors.
    Psychopharmacology, 1990, Volume: 102, Issue:3

    Topics: Analgesics; Animals; Avoidance Learning; Benzeneacetamides; Electroshock; Male; Memory; Mice; Mice, Inbred Strains; Morphine; Naloxone; Oligopeptides; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu

1990
Opposite effects of delta and mu opioid receptor agonists on the in vitro release of substance P-like material from the rat spinal cord.
    Journal of neurochemistry, 1987, Volume: 48, Issue:2

    Topics: Animals; D-Ala(2),MePhe(4),Met(0)-ol-enkephalin; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalins; In Vitro Techniques; Male; Morphine; Naloxone; Oligopeptides; Potassium; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu; Spinal Cord; Substance P; Tetrodotoxin; Veratridine

1987
Binding in vivo of selective mu and delta opioid receptor agonists: opioid receptor occupancy by endogenous enkephalins.
    European journal of pharmacology, 1989, Nov-21, Volume: 171, Issue:2-3

    Topics: Animals; Brain; Corpus Striatum; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Hydroxamic Acids; In Vitro Techniques; Injections; Kinetics; Male; Mice; Morphine; Oligopeptides; Phenylalanine; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu; Thiorphan

1989
Opioid receptor types in the brain of the Afghan pika (Ochotona rufescens), a species which is naturally tolerant to morphine.
    Life sciences, 1988, Volume: 43, Issue:8

    Topics: Animals; Binding, Competitive; Brain Chemistry; Diprenorphine; Drug Tolerance; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Guanylyl Imidodiphosphate; Lagomorpha; Membranes; Morphine; Oligopeptides; Rabbits; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Sodium

1988
Differential electrographic patterns for specific mu- and delta-opioid peptides in rats.
    European journal of pharmacology, 1986, Apr-09, Volume: 123, Issue:1

    Topics: Animals; Electroencephalography; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Epilepsy; Male; Morphine; Oligopeptides; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu

1986
Role of mu and delta receptors in the supraspinal and spinal analgesic effects of [D-Pen2, D-Pen5]enkephalin in the mouse.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:2

    Topics: Analgesia; Anesthesia, Spinal; Animals; Drug Synergism; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Male; Mice; Morphine; Oligopeptides; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu

1987
Effects of selective mu- and delta-opioid peptides on kindled amygdaloid seizures in rats.
    Neuroscience letters, 1987, Feb-24, Volume: 74, Issue:2

    Topics: Amygdala; Animals; Anticonvulsants; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Kindling, Neurologic; Male; Morphine; Oligopeptides; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu

1987
Roles of mu, delta and kappa opioid receptors in spinal and supraspinal mediation of gastrointestinal transit effects and hot-plate analgesia in the mouse.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 230, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesia; Animals; Digestive System Physiological Phenomena; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Hot Temperature; Injections, Intraventricular; Injections, Spinal; Male; Mice; Morphine; Narcotics; Oligopeptides; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Spinal Cord

1984
Different subtypes of opioid receptors have different affinities for G-proteins.
    Cellular and molecular biology (Noisy-le-Grand, France), 1994, Volume: 40, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adenylyl Cyclases; Amino Acid Sequence; Animals; Binding, Competitive; Cerebellum; Colforsin; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Etorphine; GTP-Binding Proteins; Guinea Pigs; Humans; Hybrid Cells; Molecular Sequence Data; Morphine; Naloxone; Neoplasm Proteins; Nerve Tissue Proteins; Neuroblastoma; Oligopeptides; Pyrrolidines; Rabbits; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu; Tumor Cells, Cultured

1994
Morphine reduces the release of met-enkephalin-like material from the rat spinal cord in vivo by acting at delta opioid receptors.
    Neuropeptides, 1994, Volume: 27, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Methionine; Enkephalins; Injections, Spinal; Male; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Oligopeptides; Pyrrolidines; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta; Spinal Cord

1994
Mu and delta opioid receptors mediate opposite modulations by morphine of the spinal release of cholecystokinin-like material.
    Brain research, 1994, Aug-08, Volume: 653, Issue:1-2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Cholecystokinin; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Male; Morphine; Narcotic Antagonists; Oligopeptides; Pyrrolidines; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu; Spinal Cord

1994
Opioid control of the release of calcitonin gene-related peptide-like material from the rat spinal cord in vivo.
    Brain research, 1993, Apr-23, Volume: 609, Issue:1-2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Calcitonin Gene-Related Peptide; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Injections, Spinal; Iodine Radioisotopes; Male; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Oligopeptides; Pyrrolidines; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Spinal Cord

1993
Effects of neuropeptide FF analogs on morphine analgesia in the nucleus raphe dorsalis.
    Regulatory peptides, 1995, Nov-10, Volume: 59, Issue:3

    Topics: Amino Acid Sequence; Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Male; Microinjections; Molecular Sequence Data; Morphine; Neuropeptides; Oligopeptides; Pain Measurement; Pain Threshold; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, Opioid

1995
The antinociceptive activity of kappa- but not delta-opioid receptor agonists is maintained in morphine-tolerant neuropathic rats.
    European journal of pharmacology, 1996, Dec-30, Volume: 318, Issue:2-3

    Topics: Analgesics, Opioid; Animals; Benzeneacetamides; Drug Tolerance; Male; Morphine; Oligopeptides; Pain; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta; Receptors, Opioid, kappa; Vocalization, Animal

1996
mu and delta-opioid receptor agonists induce mitogen-activated protein kinase (MAPK) activation in the absence of receptor internalization.
    Neuropharmacology, 2000, Jul-24, Volume: 39, Issue:10

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Binding, Competitive; CHO Cells; Concanavalin A; Cricetinae; Dose-Response Relationship, Drug; Endocytosis; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enzyme Activation; Hypertonic Solutions; Mitogen-Activated Protein Kinases; Morphine; Oligopeptides; Phosphorylation; Radioligand Assay; Receptors, Opioid, delta; Receptors, Opioid, mu; Sucrose; Time Factors

2000
Anti-analgesic and anti-amnesic effect of complement C3a.
    Life sciences, 2000, Sep-15, Volume: 67, Issue:17

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Avoidance Learning; Cerebral Ventricles; Complement C3a; Dose-Response Relationship, Drug; Electroshock; Humans; Injections, Intraventricular; Ischemia; Male; Mice; Mice, Inbred Strains; Morphine; Oligopeptides; Pain; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu

2000
Enterostatin (VPDPR) has anti-analgesic and anti-amnesic activities.
    Bioscience, biotechnology, and biochemistry, 2001, Volume: 65, Issue:1

    Topics: Adjuvants, Anesthesia; Amnesia; Analgesics, Opioid; Animals; Colipases; Enzyme Precursors; Male; Memory; Mice; Mice, Inbred Strains; Morphine; Oligopeptides; Protein Precursors; Scopolamine

2001