Page last updated: 2024-08-16

delavirdine and amprenavir

delavirdine has been researched along with amprenavir in 14 studies

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (14.29)18.2507
2000's9 (64.29)29.6817
2010's1 (7.14)24.3611
2020's2 (14.29)2.80

Authors

AuthorsStudies
Dansette, PM; Fontana, E; Poli, SM1
Chou, KC; González-Díaz, H; Martinez de la Vega, O; Prado-Prado, FJ; Ubeira, FM; Uriarte, E1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Delabio, LC; Dutra, JP; Hembecker, M; Kita, DH; Moure, VR; Pereira, GDS; Scheiffer, G; Valdameri, G; Zattoni, IF1
Dranchak, PK; Huang, R; Inglese, J; Lamy, L; Oliphant, E; Queme, B; Tao, D; Wang, Y; Xia, M1
Temesgen, Z; Wright, AJ1
Belohradsky, BH; Engelhorn, C; Hoffmann, F; Kurowski, M; Notheis, G; Wintergerst, U1
Bartoli, A; Feroggio, M; Gianelli, L; Maserati, R; Montagna, M; Regazzi, MB; Villani, P1
Alexander, C; Harris, M; Montaner, JS; O'Shaughnessy, M1
Garrett, M; Hee, B; Kerr, BM; Petersen, C; Tran, JQ1
Brosen, K; Justesen, US; Klitgaard, NA; Pedersen, C2
Belohradsky, BH; Engelhorn, C; Hoffmann, F; Kruse, G; Kurowski, M; Notheis, G; Stocker, H; Wintergerst, U1

Reviews

4 review(s) available for delavirdine and amprenavir

ArticleYear
Cytochrome p450 enzymes mechanism based inhibitors: common sub-structures and reactivity.
    Current drug metabolism, 2005, Volume: 6, Issue:5

    Topics: Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Drug Interactions; Enzyme Inhibitors; Humans; Isoenzymes; Structure-Activity Relationship; Terminology as Topic

2005
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Targeting breast cancer resistance protein (BCRP/ABCG2): Functional inhibitors and expression modulators.
    European journal of medicinal chemistry, 2022, Jul-05, Volume: 237

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily G, Member 2; Breast Neoplasms; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Female; Humans; Neoplasm Proteins; Neoplastic Stem Cells

2022
Antiretrovirals.
    Mayo Clinic proceedings, 1999, Volume: 74, Issue:12

    Topics: Adolescent; Adult; Alkynes; Anti-HIV Agents; Benzoxazines; Carbamates; Cyclopropanes; Delavirdine; Didanosine; Dideoxynucleosides; Female; Furans; HIV Infections; Humans; Indinavir; Lamivudine; Nelfinavir; Nevirapine; Oxazines; Pregnancy; Pregnancy Complications, Infectious; Protease Inhibitors; Reverse Transcriptase Inhibitors; Ritonavir; Saquinavir; Stavudine; Sulfonamides; Zalcitabine; Zidovudine

1999

Trials

3 trial(s) available for delavirdine and amprenavir

ArticleYear
Pharmacokinetic interaction between amprenavir and delavirdine: evidence of induced clearance by amprenavir.
    Clinical pharmacology and therapeutics, 2002, Volume: 72, Issue:6

    Topics: Administration, Oral; Adult; Anti-HIV Agents; Antiretroviral Therapy, Highly Active; Area Under Curve; Carbamates; Delavirdine; Drug Administration Schedule; Drug Interactions; Female; Furans; Humans; Longitudinal Studies; Male; Middle Aged; Reference Values; Sulfonamides

2002
Pharmacokinetic interaction between amprenavir and delavirdine after multiple-dose administration in healthy volunteers.
    British journal of clinical pharmacology, 2003, Volume: 55, Issue:1

    Topics: Anti-HIV Agents; Carbamates; Delavirdine; Drug Interactions; Furans; Humans; Male; Prospective Studies; Sulfonamides

2003
Dose-dependent pharmacokinetics of delavirdine in combination with amprenavir in healthy volunteers.
    The Journal of antimicrobial chemotherapy, 2004, Volume: 54, Issue:1

    Topics: Adult; Anti-HIV Agents; Area Under Curve; Carbamates; Chromatography, High Pressure Liquid; Delavirdine; Dose-Response Relationship, Drug; Drug Combinations; Furans; Humans; Male; Prospective Studies; Spectrophotometry, Ultraviolet; Sulfonamides

2004

Other Studies

7 other study(ies) available for delavirdine and amprenavir

ArticleYear
Unified QSAR approach to antimicrobials. 4. Multi-target QSAR modeling and comparative multi-distance study of the giant components of antiviral drug-drug complex networks.
    Bioorganic & medicinal chemistry, 2009, Jan-15, Volume: 17, Issue:2

    Topics: Anti-Infective Agents; Antiviral Agents; Artificial Intelligence; Computer Simulation; Drug Evaluation, Preclinical; Molecular Structure; Quantitative Structure-Activity Relationship

2009
In vivo quantitative high-throughput screening for drug discovery and comparative toxicology.
    Disease models & mechanisms, 2023, 03-01, Volume: 16, Issue:3

    Topics: Animals; Caenorhabditis elegans; Drug Discovery; High-Throughput Screening Assays; Humans; Proteomics; Small Molecule Libraries

2023
Pharmacokinetic interaction of amprenavir in combination with efavirenz or delavirdine in HIV-infected children.
    AIDS (London, England), 2000, Aug-18, Volume: 14, Issue:12

    Topics: Adolescent; Alkynes; Anti-HIV Agents; Benzoxazines; Carbamates; Child; Child, Preschool; Cyclopropanes; Delavirdine; Drug Interactions; Drug Therapy, Combination; Furans; HIV Infections; Humans; Oxazines; Reverse Transcriptase Inhibitors; Sulfonamides; Time Factors

2000
Antivirals update.
    Project Inform perspective, 1998, Issue:26

    Topics: Anti-HIV Agents; Carbamates; Delavirdine; Dideoxynucleosides; Drug Resistance, Microbial; Drug Therapy, Combination; Drugs, Investigational; Furans; HIV Infections; HIV Protease Inhibitors; Humans; Indinavir; Nevirapine; Reverse Transcriptase Inhibitors; Salvage Therapy; Sulfonamides

1998
Antiretrovirals: simultaneous determination of five protease inhibitors and three nonnucleoside transcriptase inhibitors in human plasma by a rapid high-performance liquid chromatography--mass spectrometry assay.
    Therapeutic drug monitoring, 2001, Volume: 23, Issue:4

    Topics: Alkynes; Benzoxazines; Carbamates; Chromatography, Liquid; Cyclopropanes; Delavirdine; Drug Monitoring; Furans; HIV Protease Inhibitors; Humans; Indinavir; Mass Spectrometry; Nelfinavir; Nevirapine; Oxazines; Reproducibility of Results; Reverse Transcriptase Inhibitors; Ritonavir; Saquinavir; Sensitivity and Specificity; Sulfonamides

2001
Delavirdine increases drug exposure of ritonavir-boosted protease inhibitors.
    AIDS (London, England), 2002, Mar-29, Volume: 16, Issue:5

    Topics: Anti-HIV Agents; Antiretroviral Therapy, Highly Active; Carbamates; Delavirdine; Drug Synergism; Furans; HIV Infections; HIV Protease Inhibitors; Humans; Lopinavir; Pyrimidinones; Reverse Transcriptase Inhibitors; Ritonavir; Sulfonamides

2002
Long-term pharmacokinetics of amprenavir in combination with delavirdine in HIV-infected children.
    AIDS (London, England), 2004, Jul-02, Volume: 18, Issue:10

    Topics: Adolescent; Anti-HIV Agents; Area Under Curve; Carbamates; Child; Delavirdine; Drug Combinations; Furans; HIV Infections; Humans; Reverse Transcriptase Inhibitors; Sulfonamides

2004