Page last updated: 2024-08-23

daunorubicin and ly335979

daunorubicin has been researched along with ly335979 in 8 studies

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (12.50)18.2507
2000's6 (75.00)29.6817
2010's1 (12.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Castanys, S; Chávez Orellana, H; Estévez-Braun, A; Gamarro, F; Jiménez-Alonso, S; López, M; Muñoz Martinez, F; Pérez-Lomas, AL; Ravelo, AG1
De Angelis, P; den Boer, M; Lehne, G; Rugstad, HE1
den Boer, M; Lehne, G; Mørkrid, L; Rugstad, HE1
Green, LJ; Marder, P; Slapak, CA1
Aarons, L; Burgess, M; Callies, S; de Alwis, DP; Mehta, A1
Baker, RJ; Burgess, M; Ethell, M; Ganeshaguru, K; Gerrard, G; Jones, DT; McCullough, H; Mehta, AB; Payne, E; Potter, M; Prentice, HG1
Baer, MR; Duran, GE; Fielding, R; Lancet, JE; List, AF; Marcelletti, JF; Multani, PS; Sikic, BI1
Bennett, JM; Cripe, LD; Ketterling, RP; Lazarus, HM; Litzow, MR; Luger, S; Paietta, EM; Rowe, JM; Tallman, MS; Uno, H1

Trials

4 trial(s) available for daunorubicin and ly335979

ArticleYear
Population pharmacokinetic model for daunorubicin and daunorubicinol coadministered with zosuquidar.3HCl (LY335979).
    Cancer chemotherapy and pharmacology, 2004, Volume: 54, Issue:1

    Topics: Antibiotics, Antineoplastic; Antineoplastic Combined Chemotherapy Protocols; ATP Binding Cassette Transporter, Subfamily B, Member 1; Bile Canaliculi; Daunorubicin; Dibenzocycloheptenes; Dose-Response Relationship, Drug; Drug Interactions; Drug Resistance, Multiple; Humans; Models, Theoretical; Quinolines

2004
Clinical effects and P-glycoprotein inhibition in patients with acute myeloid leukemia treated with zosuquidar trihydrochloride, daunorubicin and cytarabine.
    Haematologica, 2004, Volume: 89, Issue:7

    Topics: Abdominal Pain; Adult; Aged; Antineoplastic Combined Chemotherapy Protocols; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cytarabine; Daunorubicin; Diarrhea; Dibenzocycloheptenes; Drug Resistance; Drug Screening Assays, Antitumor; Female; Flow Cytometry; Humans; Leukemia, Promyelocytic, Acute; Male; Middle Aged; Nausea; Quinolines; Remission Induction

2004
A phase I trial of continuous infusion of the multidrug resistance inhibitor zosuquidar with daunorubicin and cytarabine in acute myeloid leukemia.
    Leukemia research, 2009, Volume: 33, Issue:8

    Topics: Aged; Antineoplastic Combined Chemotherapy Protocols; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cytarabine; Daunorubicin; Dibenzocycloheptenes; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Female; Humans; Leukemia, Myeloid, Acute; Male; Middle Aged; Quinolines; Time Factors

2009
Zosuquidar, a novel modulator of P-glycoprotein, does not improve the outcome of older patients with newly diagnosed acute myeloid leukemia: a randomized, placebo-controlled trial of the Eastern Cooperative Oncology Group 3999.
    Blood, 2010, Nov-18, Volume: 116, Issue:20

    Topics: Aged; Aged, 80 and over; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Daunorubicin; Dibenzocycloheptenes; Female; Humans; Leukemia, Myeloid, Acute; Male; Multivariate Analysis; Placebos; Prognosis; Quinolines; Remission Induction; Survival Analysis; Treatment Outcome

2010

Other Studies

4 other study(ies) available for daunorubicin and ly335979

ArticleYear
Bis-pyranobenzoquinones as a new family of reversal agents of the multidrug resistance phenotype mediated by P-glycoprotein in mammalian cells and the protozoan parasite Leishmania.
    Journal of medicinal chemistry, 2008, Nov-27, Volume: 51, Issue:22

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzoquinones; Crystallography, X-Ray; Daunorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Leishmania tropica; Mice; Models, Molecular; Molecular Structure; NIH 3T3 Cells; Parasitic Sensitivity Tests; Phenotype; Stereoisomerism; Structure-Activity Relationship

2008
Growth inhibition, cytokinesis failure and apoptosis of multidrug-resistant leukemia cells after treatment with P-glycoprotein inhibitory agents.
    Leukemia, 1999, Volume: 13, Issue:5

    Topics: Antineoplastic Agents; Apoptosis; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cyclosporins; Daunorubicin; Dibenzocycloheptenes; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; Leukemia; Peptides, Cyclic; Phenotype; Quinolines; Tumor Cells, Cultured

1999
Diverse effects of P-glycoprotein inhibitory agents on human leukemia cells expressing the multidrug resistance protein (MRP).
    International journal of clinical pharmacology and therapeutics, 2000, Volume: 38, Issue:4

    Topics: Antibiotics, Antineoplastic; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; Cyclosporins; Daunorubicin; Dibenzocycloheptenes; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Flow Cytometry; Fluorescence; Humans; Leukemia, Myeloid; Peptides, Cyclic; Quinolines; Tumor Cells, Cultured

2000
Modulation by LY335979 of P-glycoprotein function in multidrug-resistant cell lines and human natural killer cells.
    Biochemical pharmacology, 2001, Jun-01, Volume: 61, Issue:11

    Topics: Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Daunorubicin; Dibenzocycloheptenes; Dose-Response Relationship, Drug; Drug Interactions; Drug Resistance, Multiple; Fluorescent Dyes; HL-60 Cells; Humans; Killer Cells, Natural; Quinolines; Rhodamine 123

2001