Page last updated: 2024-08-23

daunorubicin and hoe 33342

daunorubicin has been researched along with hoe 33342 in 24 studies

Research

Studies (24)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's8 (33.33)18.2507
2000's12 (50.00)29.6817
2010's4 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Burres, NS; Frigo, A; McAlpine, JB; Rasmussen, RR1
Huang, L; Humphreys, JE; Morgan, JB; Polli, JW; Serabjit-Singh, CS; Webster, LO; Wring, SA1
Balakrishnan, L; Janvilisri, T; Reuter, G; Shahi, S; van Veen, HW; Venter, H1
Casciano, CN; Clement, RP; Johnson, WW; Wang, EJ1
Borchardt, RT; Ouyang, H; Tang, F; Yang, JZ1
Globisch, C; Kassack, MU; Klinkhammer, W; Müller, H; Pajeva, IK; Wiese, M1
Belloc, F; Bernard, P; Boisseau, MR; Dumain, P; Lacombe, F; Lopez, F; Reifers, J1
Lizard, G; Lizard-Nacol, S; Maynadié, M; Poupon, MF; Roignot, P1
Buquen, JJ; Canitrot, D; Canitrot, Y; Lahmy, S; Lautier, D1
Bordes, M; Lizard, G; Lizard-Nacol, S; Maynadie, M; Poupon, MF; Roignot, P1
Ling, V; Shapiro, AB1
Fox, K; Lee, P; Ling, V; Shapiro, AB; Yang, YD1
Boezeman, J; de Witte, TM; Minderman, H; Pennings, AH; Raymakers, RA; Smeets, ME; Vierwinden, G1
Andreeff, M; Brenner, MK; Goodell, MA; Kuehnle, I; Marini, F; Wang, RY; Weidner, D; Wulf, GG1
Bibi, E; Lewinson, O1
Castanys, S; Cortés-Selva, F; Gamarro, F; Jiménez, IA; Lu, P; Muñoz-Martínez, F; Pérez-Victoria, JM; Ravelo, AG; Sharom, FJ1
Hamelik, RM; Krishan, A1
Brodbelt, JS; Keller, KM; Oehlers, L; Zhang, J1
Callaghan, R; Clark, R; Kerr, ID1
Agustiandari, H; Driessen, AJ; Madoori, PK; Thunnissen, AM1
Andrieu, T; Arnaud, O; Chang, G; Chaptal, V; Di Pietro, A; Doshi, R; Dussurgey, S; Falson, P; Henin, E; Martinez, L; Tao, H; Tod, M; Zhang, Q1
Imai, M; Shimada, I; Takahashi, H; Takeuchi, K; Tokunaga, Y1
Bloemberg, GV; Corradi, V; Hohl, M; Hürlimann, LM; Seeger, MA; Tieleman, DP1
Brown, K; Kaur, P; Li, W1

Other Studies

24 other study(ies) available for daunorubicin and hoe 33342

ArticleYear
A colorimetric microassay for the detection of agents that interact with DNA.
    Journal of natural products, 1992, Volume: 55, Issue:11

    Topics: Aminoglycosides; Anti-Bacterial Agents; Antibiotics, Antineoplastic; Colorimetry; DNA; Ethidium; Fermentation; Methyl Green; Spectrometry, Fluorescence

1992
Rational use of in vitro P-glycoprotein assays in drug discovery.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 299, Issue:2

    Topics: Adenosine Triphosphatases; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cells, Cultured; Chromatography, Liquid; Enzyme Inhibitors; Fluoresceins; Fluorescent Dyes; Humans; Mass Spectrometry; Pharmacology; Spodoptera

2001
Sterol transport by the human breast cancer resistance protein (ABCG2) expressed in Lactococcus lactis.
    The Journal of biological chemistry, 2003, Jun-06, Volume: 278, Issue:23

    Topics: Antineoplastic Agents, Hormonal; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Cholesterol; Estradiol; Gene Expression; Humans; Lactococcus lactis; Neoplasm Proteins; Progesterone; Sterols; Tamoxifen; Testosterone; Tritium

2003
Fluorescent substrates of sister-P-glycoprotein (BSEP) evaluated as markers of active transport and inhibition: evidence for contingent unequal binding sites.
    Pharmaceutical research, 2003, Volume: 20, Issue:4

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Binding Sites; Biological Transport, Active; Biomarkers; Cells, Cultured; Drug Interactions; Fluorescent Dyes; Humans

2003
Bidirectional transport of rhodamine 123 and Hoechst 33342, fluorescence probes of the binding sites on P-glycoprotein, across MDCK-MDR1 cell monolayers.
    Journal of pharmaceutical sciences, 2004, Volume: 93, Issue:5

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Binding Sites; Biological Transport; Cell Line; Cell Membrane; Dogs; Fluorescent Dyes; Humans; Rhodamine 123

2004
New functional assay of P-glycoprotein activity using Hoechst 33342.
    Bioorganic & medicinal chemistry, 2007, Dec-01, Volume: 15, Issue:23

    Topics: Adenosine Triphosphatases; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Cell Line, Tumor; Cell Proliferation; Dose-Response Relationship, Drug; Drug Resistance, Neoplasm; Fluoresceins; Humans; Microscopy, Fluorescence; Molecular Structure; Principal Component Analysis; Time Factors

2007
Intercalation of anthracyclines into living cell DNA analyzed by flow cytometry.
    Cytometry, 1992, Volume: 13, Issue:8

    Topics: Benzimidazoles; Daunorubicin; DNA; Energy Transfer; Flow Cytometry; Fluorescence; Humans; Idarubicin; Intercalating Agents; Leukemia, Promyelocytic, Acute; Tumor Cells, Cultured

1992
Evaluation of multidrug resistant phenotype by flow cytometry with monoclonal antibodies and functional tests.
    Bulletin du cancer, 1995, Volume: 82, Issue:3

    Topics: Antibodies, Monoclonal; Antimetabolites, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Daunorubicin; Drug Resistance, Multiple; Flow Cytometry; Fluorescent Antibody Technique; Fluorescent Dyes; Humans; Leukemia, Erythroblastic, Acute; Lymphoma, Non-Hodgkin; Phenotype; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Rhodamine 123; Rhodamines

1995
Functional study of multidrug resistance with fluorescent dyes. Limits of the assay for low levels of resistance and application in clinical samples.
    Cancer letters, 1996, Aug-23, Volume: 106, Issue:1

    Topics: Animals; Anthracyclines; Benzimidazoles; Cell Survival; Clone Cells; Daunorubicin; Drug Resistance, Multiple; Flow Cytometry; Fluorescent Dyes; Leukemia L1210; Mice; Phenotype; Quantum Theory; Reproducibility of Results; Rhodamine 123; Rhodamines; Sensitivity and Specificity; Tumor Cells, Cultured; Vinblastine

1996
Flow cytometry evaluation of the multidrug-resistant phenotype with functional tests involving uptake of daunorubicin, Hoechst 33342, or rhodamine 123: a comparative study.
    Cancer detection and prevention, 1995, Volume: 19, Issue:6

    Topics: Antibiotics, Antineoplastic; Antimetabolites, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Cell Death; Daunorubicin; Drug Resistance, Multiple; Flow Cytometry; Hot Temperature; Humans; Phenotype; Rhodamine 123; Rhodamines; Tumor Cells, Cultured

1995
Positively cooperative sites for drug transport by P-glycoprotein with distinct drug specificities.
    European journal of biochemistry, 1997, Nov-15, Volume: 250, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Binding Sites; Biological Transport; Cell Line; Cell Membrane; Colchicine; Cricetinae; Cricetulus; Dactinomycin; Daunorubicin; Doxorubicin; Etoposide; Fluorescence; Fluorescent Dyes; Kinetics; Liposomes; Protein Binding; Quercetin; Rhodamine 123; Rhodamines; Vinblastine

1997
Functional intracellular P-glycoprotein.
    International journal of cancer, 1998, Jun-10, Volume: 76, Issue:6

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Cell Line; Cyclosporine; Daunorubicin; Drug Resistance

1998
Idarubicin DNA intercalation is reduced by MRP1 and not Pgp.
    Leukemia, 1999, Volume: 13, Issue:9

    Topics: Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Base Pair Mismatch; Benzimidazoles; Daunorubicin; DNA-Binding Proteins; Energy Transfer; Flow Cytometry; Fluorescent Dyes; Humans; Idarubicin; Intercalating Agents; Multidrug Resistance-Associated Proteins; MutS Homolog 3 Protein; Rhodamines; Sensitivity and Specificity; Spectrometry, Fluorescence; Tumor Cells, Cultured

1999
A leukemic stem cell with intrinsic drug efflux capacity in acute myeloid leukemia.
    Blood, 2001, Aug-15, Volume: 98, Issue:4

    Topics: Acute Disease; Adolescent; Adult; Aged; Aged, 80 and over; Animals; Antibiotics, Antineoplastic; Antineoplastic Agents; Benzimidazoles; Cell Separation; Child; Child, Preschool; Daunorubicin; Drug Resistance; Female; Humans; Immunophenotyping; Infant; Leukemia, Myeloid; Leukocytes, Mononuclear; Male; Mice; Mice, Inbred NOD; Middle Aged; Mitoxantrone; Myelodysplastic Syndromes; Neoplasm Transplantation; Neoplasms, Second Primary; Stem Cell Transplantation; Stem Cells; Tumor Cells, Cultured

2001
Evidence for simultaneous binding of dissimilar substrates by the Escherichia coli multidrug transporter MdfA.
    Biochemistry, 2001, Oct-23, Volume: 40, Issue:42

    Topics: Bacterial Proteins; Benzalkonium Compounds; Benzimidazoles; Biological Transport; Chloramphenicol; Daunorubicin; Drug Resistance, Multiple, Bacterial; Escherichia coli; Escherichia coli Proteins; Ethidium; Membrane Transport Proteins; Onium Compounds; Organophosphorus Compounds; Protein Binding; Recombinant Proteins; Solubility; Tritium

2001
Celastraceae sesquiterpenes as a new class of modulators that bind specifically to human P-glycoprotein and reverse cellular multidrug resistance.
    Cancer research, 2004, Oct-01, Volume: 64, Issue:19

    Topics: Adenosine Triphosphatases; Adenosine Triphosphate; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Azides; Benzimidazoles; Binding, Competitive; Celastraceae; Cell Membrane; Daunorubicin; Dihydropyridines; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Fluoresceins; Humans; Kinetics; Liposomes; Membrane Transport Modulators; Membrane Transport Proteins; Mice; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; NIH 3T3 Cells; Photoaffinity Labels; Protein Binding; Sesquiterpenes; Substrate Specificity; Vinblastine

2004
Flow cytometric monitoring of fluorescent drug retention and efflux.
    Methods in molecular medicine, 2005, Volume: 111

    Topics: Antibiotics, Antineoplastic; Antineoplastic Agents; Benzimidazoles; Cell Line, Tumor; Daunorubicin; Drug Monitoring; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Flow Cytometry; Fluorescent Dyes; Humans; Hydrogen-Ion Concentration; Phenotype; Rhodamine 123

2005
Influence of initial charge state on fragmentation patterns for noncovalent drug/DNA duplex complexes.
    Journal of mass spectrometry : JMS, 2005, Volume: 40, Issue:10

    Topics: Benzimidazoles; Daunorubicin; Distamycins; DNA; Indoles; Netropsin; Nogalamycin; Oligodeoxyribonucleotides; Pharmaceutical Preparations; Spectrometry, Mass, Electrospray Ionization

2005
Multiple drugbinding sites on the R482G isoform of the ABCG2 transporter.
    British journal of pharmacology, 2006, Volume: 149, Issue:5

    Topics: Amino Acid Substitution; Animals; Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Benzimidazoles; Binding Sites; Biological Transport; Cell Line; Cell Membrane; Daunorubicin; Dose-Response Relationship, Drug; Kinetics; Mitoxantrone; Neoplasm Proteins; Polymorphism, Genetic; Prazosin; Protein Binding; Protein Isoforms; Radioligand Assay; Spodoptera; Temperature; Tritium

2006
Structure of the transcriptional regulator LmrR and its mechanism of multidrug recognition.
    The EMBO journal, 2009, Jan-21, Volume: 28, Issue:2

    Topics: Amino Acid Sequence; Bacterial Proteins; Benzimidazoles; Daunorubicin; Dimerization; Helix-Turn-Helix Motifs; Hydrogen Bonding; Lactococcus lactis; Models, Molecular; Molecular Sequence Data; Protein Binding; Protein Conformation; Transcription, Genetic

2009
Understanding polyspecificity within the substrate-binding cavity of the human multidrug resistance P-glycoprotein.
    The FEBS journal, 2014, Volume: 281, Issue:3

    Topics: Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Binding, Competitive; Biological Transport; Catalytic Domain; Daunorubicin; Drug Resistance, Multiple; Humans; Kinetics; Membrane Transport Modulators; Mice; Models, Molecular; Molecular Docking Simulation; NIH 3T3 Cells; Peptides, Cyclic; Protein Isoforms; Recombinant Proteins; Stereoisomerism

2014
Dynamic multidrug recognition by multidrug transcriptional repressor LmrR.
    Scientific reports, 2014, Nov-18, Volume: 4

    Topics: Base Sequence; Benzimidazoles; Binding Sites; Daunorubicin; Drug Resistance, Multiple, Bacterial; Ethidium; Gene Expression Regulation, Bacterial; Lactococcus lactis; Models, Molecular; Molecular Sequence Data; Multidrug Resistance-Associated Proteins; Promoter Regions, Genetic; Protein Binding; Protein Conformation; Repressor Proteins; Rhodamines; Transcription, Genetic

2014
The Heterodimeric ABC Transporter EfrCD Mediates Multidrug Efflux in Enterococcus faecalis.
    Antimicrobial agents and chemotherapy, 2016, Volume: 60, Issue:9

    Topics: Adenosine Triphosphate; Amino Acid Sequence; Anti-Bacterial Agents; ATP-Binding Cassette Transporters; Bacterial Proteins; Base Sequence; Benzimidazoles; Biological Transport; Chromosomes, Bacterial; Daunorubicin; Doxorubicin; Enterococcus faecalis; Ethidium; Fluoroquinolones; Gene Expression; Genetic Loci; Lactococcus lactis; Protein Binding; Protein Conformation, alpha-Helical; Protein Conformation, beta-Strand; Protein Interaction Domains and Motifs; Protein Multimerization; Proteolipids; Recombinant Proteins; Sequence Deletion; Transgenes

2016
Role of Aromatic and Negatively Charged Residues of DrrB in Multisubstrate Specificity Conferred by the DrrAB System of Streptomyces peucetius.
    Biochemistry, 2017, 04-04, Volume: 56, Issue:13

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Bacterial Proteins; Benzimidazoles; Daunorubicin; Doxorubicin; Drug Resistance, Multiple, Bacterial; Escherichia coli; Ethidium; Evolution, Molecular; Gene Expression; Models, Molecular; Multidrug Resistance-Associated Proteins; Mutation; Protein Binding; Protein Structure, Secondary; Recombinant Proteins; Static Electricity; Streptomyces; Structural Homology, Protein; Substrate Specificity; Verapamil

2017