Page last updated: 2024-08-23

darodipine and isradipine

darodipine has been researched along with isradipine in 15 studies

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-199010 (66.67)18.7374
1990's5 (33.33)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Colombo, G; Fadda, F; Garau, B; Gessa, GL1
Holck, M; Osterrieder, W1
Chaumet-Riffaud, P; Lemaire, M; Pinquier, JL; Tillement, JP; Urien, S1
Chaumet-Riffaud, P; Pinquier, JL; Tillement, JP; Urien, S1
Al-Mahmood, HA; el-Khatim, MS; Gumaa, KA; Thulesius, O1
Handley, DA; Melden, MK; Saunders, RN; Van Valen, RG1
Chaumet-Riffaud, P; Kiechel, JR; Paquette, B; Pinquier, JL; Tillement, JP; Urien, S1
Barrès, C; Cerutti, C; Morin, B; Sassard, J1
Jie, K; Timmermans, PB; van Brummelen, P; van Zwieten, PA; Vermey, P1
Karobath, M; Supavilai, P1
Cortés, R; Karobath, M; Palacios, JM; Supavilai, P1
Dall'Olio, R; Gaggi, R; Gianni, AM; Roncada, P1
Brée, F; Carrupt, PA; Giroud, Y; Testa, B; Tillement, JP; Tsai, RS; Urien, S1
Brauns, T; Glossmann, H; Haugland, RP; Kimball, SD; Prinz, H; Striessnig, J1
D'Allolio, R; Gaggi, R; Roncada, P; Santangelo, M1

Trials

1 trial(s) available for darodipine and isradipine

ArticleYear
Influence of calcium entry blockade on alpha 1- and alpha 2-adrenoceptor mediated vasoconstriction in the forearm of hypertensive patients.
    European journal of clinical pharmacology, 1987, Volume: 32, Issue:2

    Topics: Adult; Azepines; Calcium Channel Blockers; Female; Forearm; Hemodynamics; Humans; Hypertension; Isradipine; Male; Methoxamine; Middle Aged; Nifedipine; Oxadiazoles; Receptors, Adrenergic, alpha; Regional Blood Flow; Vascular Resistance; Vasoconstriction

1987

Other Studies

14 other study(ies) available for darodipine and isradipine

ArticleYear
Isradipine and other calcium channel antagonists attenuate ethanol consumption in ethanol-preferring rats.
    Alcoholism, clinical and experimental research, 1992, Volume: 16, Issue:3

    Topics: Alcohol Drinking; Animals; Calcium Channel Blockers; Dihydropyridines; Dose-Response Relationship, Drug; Ethanol; Isradipine; Male; Nifedipine; Rats; Rats, Inbred Strains; Verapamil

1992
Inhibition of myocardial Ca2+ channels by three dihydropyridines with different structural features: potential-dependent blockade by Ro 18-3981.
    British journal of pharmacology, 1987, Volume: 91, Issue:1

    Topics: Animals; Calcium Channel Blockers; Dihydropyridines; Female; Guinea Pigs; Heart; In Vitro Techniques; Ion Channels; Isradipine; Male; Membrane Potentials; Myocardial Contraction; Myocardium; Nifedipine; Oxadiazoles; Potassium; Pyridines

1987
Comparative binding of two closely related dihydropyridines (isradipine and darodipine) to serum proteins and erythrocytes.
    Pharmacology, 1988, Volume: 36, Issue:5

    Topics: Binding, Competitive; Blood Proteins; Calcium Channel Blockers; Dihydropyridines; Erythrocytes; gamma-Globulins; Humans; Isradipine; Lipoproteins; Nifedipine; Pyridines

1988
Differences in the serum binding determinants of isradipine and darodipine--consequences for serum protein binding in various diseases.
    British journal of clinical pharmacology, 1989, Volume: 28, Issue:5

    Topics: Adult; Blood Proteins; Calcium Channel Blockers; Fatty Acids, Nonesterified; Female; Humans; Hydrogen-Ion Concentration; Inflammation; Isradipine; Liver Diseases; Male; Middle Aged; Nifedipine; Orosomucoid; Protein Binding; Pyridines; Serum Albumin

1989
The effect of calcium-blockers nicardipine, darodipine, PN-200-110 and nifedipine on insulin release from isolated rat pancreatic islets.
    Acta physiologica Scandinavica, 1986, Volume: 126, Issue:2

    Topics: Animals; Calcium Channel Blockers; Cells, Cultured; Glucose; Insulin; Insulin Secretion; Islets of Langerhans; Isradipine; Male; Nicardipine; Nifedipine; Oxadiazoles; Rats; Rats, Inbred Strains

1986
Suppression of rat carotid lesion development by the calcium channel blocker PN 200-110.
    The American journal of pathology, 1986, Volume: 124, Issue:1

    Topics: Angioplasty, Balloon; Animals; Arteriosclerosis; Blood Platelets; Blood Pressure; Carotid Arteries; Hypotension; Isradipine; Male; Muscle, Smooth, Vascular; Nifedipine; Oxadiazoles; Rats; Rats, Inbred Strains

1986
Effect of the binding of isradipine and darodipine to different plasma proteins on their transfer through the rat blood-brain barrier. Drug binding to lipoproteins does not limit the transfer of drug.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 242, Issue:1

    Topics: Animals; Biological Transport; Blood Proteins; Blood-Brain Barrier; Brain; Humans; Isradipine; Lipoproteins; Liver; Male; Nifedipine; Orosomucoid; Pyridines; Rats; Rats, Inbred Strains; Serum Albumin

1987
Cardiovascular effects of two new calcium antagonists, PY 108-068 and PN 200-110, in conscious spontaneously hypertensive rats.
    British journal of pharmacology, 1988, Volume: 93, Issue:1

    Topics: Animals; Blood Pressure; Calcium Channel Blockers; Dose-Response Relationship, Drug; Heart Rate; Hemodynamics; Isradipine; Male; Nifedipine; Nitroglycerin; Oxadiazoles; Phenylephrine; Pressoreceptors; Rats; Rats, Inbred SHR; Reflex

1988
The interaction of [3H]PY 108-068 and of [3H]PN 200-110 with calcium channel binding sites in rat brain.
    Journal of neural transmission, 1984, Volume: 60, Issue:3-4

    Topics: Animals; Brain; In Vitro Techniques; Ion Channels; Isradipine; Kinetics; Male; Membranes; Molecular Conformation; Nifedipine; Oxadiazoles; Rats; Rats, Inbred Strains; Structure-Activity Relationship

1984
Calcium antagonist binding sites in the rat brain: quantitative autoradiographic mapping using the 1,4-dihydropyridines [3H]PN 200-110 and [3H]PY 108-068.
    Journal of neural transmission, 1984, Volume: 60, Issue:3-4

    Topics: Animals; Autoradiography; Binding Sites; Brain; Calcium Channel Blockers; Isradipine; Male; Nifedipine; Oxadiazoles; Rats; Rats, Inbred Strains

1984
Peculiar effects of isradipine and darodipine on the rat brain dopaminergic system.
    General pharmacology, 1995, Volume: 26, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Calcium Channel Blockers; Corpus Striatum; Dopamine; Haloperidol; Homovanillic Acid; Injections, Intraperitoneal; Isradipine; Male; Motor Activity; Nifedipine; Nimodipine; Parietal Lobe; Rats; Rats, Sprague-Dawley

1995
Mechanism of ligand binding to alpha 1-acid glycoprotein (orosomucoid): correlated thermodynamic factors and molecular parameters of polarity.
    The Biochemical journal, 1995, Mar-01, Volume: 306 ( Pt 2)

    Topics: Binding Sites; Chemical Phenomena; Chemistry, Physical; Hydrogen Bonding; Indoles; Isradipine; Ligands; Nifedipine; Orosomucoid; Progesterone; Propanolamines; Propranolol; Temperature; Thermodynamics; Warfarin

1995
L-type calcium channels: binding domains for dihydropyridines and benzothiazepines are located in close proximity to each other.
    Biochemistry, 1997, Mar-25, Volume: 36, Issue:12

    Topics: Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Dihydropyridines; Diltiazem; Fluorescent Dyes; Isomerism; Isradipine; Kinetics; Nicotinic Acids; Nifedipine; Nitrendipine; Oxadiazoles; Rabbits

1997
Interactions between darodipine or isradipine and the 5-HT1A receptor agonist 8-OHDPAT in rat brain.
    Pharmacology, biochemistry, and behavior, 1997, Volume: 58, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Brain; Calcium Channel Blockers; Dose-Response Relationship, Drug; Drug Interactions; Isradipine; Male; Nifedipine; Rats; Rats, Sprague-Dawley; Serotonin Receptor Agonists

1997