dapsone and sulfadiazine

dapsone has been researched along with sulfadiazine in 36 studies

Research

Studies (36)

TimeframeStudies, this research(%)All Research%
pre-199020 (55.56)18.7374
1990's3 (8.33)18.2507
2000's6 (16.67)29.6817
2010's7 (19.44)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Genther, CS; Smith, CS1
Doman, TN; McGovern, SL; Seidler, J; Shoichet, BK1
Ayscue, R; Gannett, PM; Locuson, CW; Tracy, TS1
Lombardo, F; Obach, RS; Waters, NJ1
González-Díaz, H; Orallo, F; Quezada, E; Santana, L; Uriarte, E; Viña, D; Yáñez, M1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Davidson, DE; Hickman, RL; Johnsen, DO; Kinnamon, KE; Tanticharoenyos, P1
Kovacs, JA; Masur, H1
Cushion, MT; Foy, JM; Kim, CK; Linke, MJ; Walzer, PD1
Catterall, JR; Potasman, I; Remington, JS1
Piening, E; Schirren, C1
Desai, SC; Nair, GM1
Maren, TH; McCullough, JL1
Gregory, KG; Peters, W1
Garg, LC; Maren, TH1
Schneider, MD1
Peters, W4
Reba, RC; Sheehy, TW1
Bayles, A; Olszewski, B; Thompson, PE; Waitz, JA1
Ganpule, M1
Dankert, W; Hartman, PG; Mehlhorn, H; Then, RL1
Aboulker, JP; Azihary, M; Carbon, C; Charreau, I; Oksenhendler, E; Tournerie, C1
Allegra, CJ; Kovacs, JA; Martinez, A1
JACOBS, L; KAUFMAN, HE; MELTON, ML1
Födinger, D; Karlhofer, FM; Kopp, T; Pieczkowski, F; Schneeberger, A; Sitaru, C; Stingl, G; Zillikens, D1
Brandão, MAF; Ferreira, AO; Patrício, FB; Polonini, HC; Raposo, NRB; Silva, SL1

Reviews

2 review(s) available for dapsone and sulfadiazine

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Pneumocystis carinii pneumonia: therapy and prophylaxis.
    The Journal of infectious diseases, 1988, Volume: 158, Issue:1

    Topics: Acquired Immunodeficiency Syndrome; Anti-Bacterial Agents; Dapsone; Drug Combinations; Drug Therapy, Combination; Humans; Pentamidine; Pneumonia, Pneumocystis; Pyrimethamine; Quinazolines; Recurrence; Sulfadiazine; Sulfamethoxazole; Trimethoprim; Trimethoprim, Sulfamethoxazole Drug Combination; Trimetrexate

1988

Trials

1 trial(s) available for dapsone and sulfadiazine

ArticleYear
Pneumocystis carinii pneumonia in the patient with AIDS.
    Chest, 1985, Volume: 88, Issue:5

    Topics: Acquired Immunodeficiency Syndrome; Animals; Bronchoscopy; Clinical Trials as Topic; Dapsone; Drug Combinations; Drug Therapy, Combination; Eflornithine; Humans; Male; Ornithine; Pentamidine; Pneumocystis; Pneumonia, Pneumocystis; Pyrimethamine; Sulfadiazine; Sulfamethoxazole; Therapeutic Irrigation; Trimethoprim; Trimethoprim, Sulfamethoxazole Drug Combination

1985

Other Studies

33 other study(ies) available for dapsone and sulfadiazine

ArticleYear
Antifolate studies. Activities of 40 potential antimalarial compounds against sensitive and chlorguanide triazine resistant strains of folate-requiring bacteria and Escherichia coli.
    Journal of medicinal chemistry, 1977, Volume: 20, Issue:2

    Topics: Animals; Antimalarials; Bacteria; Drug Resistance, Microbial; Escherichia coli; Folic Acid; Folic Acid Antagonists; Malaria; Mice; Plasmodium berghei; Triazines

1977
Identification and prediction of promiscuous aggregating inhibitors among known drugs.
    Journal of medicinal chemistry, 2003, Oct-09, Volume: 46, Issue:21

    Topics: Antifungal Agents; beta-Lactamase Inhibitors; Chemical Phenomena; Chemistry, Physical; Chymotrypsin; Enzyme Inhibitors; Kinetics; Light; Malate Dehydrogenase; Models, Molecular; Molecular Conformation; Scattering, Radiation; Structure-Activity Relationship

2003
Use of simple docking methods to screen a virtual library for heteroactivators of cytochrome P450 2C9.
    Journal of medicinal chemistry, 2007, Mar-22, Volume: 50, Issue:6

    Topics: Animals; Aryl Hydrocarbon Hydroxylases; Cytochrome P-450 CYP2C9; Dapsone; Databases, Factual; Enzyme Activators; Enzyme Inhibitors; Flurbiprofen; Humans; Models, Molecular; Molecular Structure; NADPH-Ferrihemoprotein Reductase; Quantitative Structure-Activity Relationship; Rats

2007
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Quantitative structure-activity relationship and complex network approach to monoamine oxidase A and B inhibitors.
    Journal of medicinal chemistry, 2008, Nov-13, Volume: 51, Issue:21

    Topics: Computational Biology; Drug Design; Humans; Isoenzymes; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Quantitative Structure-Activity Relationship

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Evaluating new antimalarial drugs against trophozoite induced Plasmodium cynomolgi malaria in rhesus monkeys.
    The American journal of tropical medicine and hygiene, 1976, Volume: 25, Issue:1

    Topics: Amodiaquine; Animals; Antimalarials; Dapsone; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Drug Tolerance; Haplorhini; Macaca mulatta; Malaria; Phenanthrenes; Primaquine; Prodigiosin; Pyrimethamine; Quinine; Sulfadiazine; Sulfadimethoxine; Sulfalene; Trimethoprim

1976
Inhibitors of folic acid synthesis in the treatment of experimental Pneumocystis carinii pneumonia.
    Antimicrobial agents and chemotherapy, 1988, Volume: 32, Issue:1

    Topics: Animals; Dapsone; Drug Therapy, Combination; Folic Acid Antagonists; Immunosuppression Therapy; Male; Pneumonia, Pneumocystis; Pyrimethamine; Pyrimidines; Rats; Rats, Inbred Strains; Sulfadiazine; Sulfadoxine; Sulfamethoxazole; Trimethoprim

1988
[Chemotherapy of leprosy].
    Archiv fur klinische und experimentelle Dermatologie, 1970, Volume: 237, Issue:1

    Topics: Dapsone; Female; Humans; Isoniazid; Leprosy; Male; Sulfadiazine; Sulfones; Thioacetazone; Urea; Vitamin D

1970
Chemotherapeutic sensitivity and viability of Nocardia asteroides and Nocardia brasiliensis in drugs.
    Mycopathologia et mycologia applicata, 1973, Aug-31, Volume: 50, Issue:4

    Topics: Agar; Chloramphenicol; Culture Media; Dapsone; Microbial Sensitivity Tests; Nocardia; Nocardia asteroides; Penicillin Resistance; Penicillins; Streptomycin; Sulfadiazine; Tetracycline

1973
Dihydropteroate synthetase from Plasmodium berghei: isolation, properties, and inhibition by dapsone and sulfadiazine.
    Molecular pharmacology, 1974, Volume: 10, Issue:1

    Topics: Aminobenzoates; Animals; Buffers; Carbon Radioisotopes; Chromatography, Paper; Dapsone; Hydro-Lyases; Hydrogen-Ion Concentration; Kinetics; Magnesium; Methanol; Plasmodium berghei; Proteins; Pteridines; Sulfadiazine; Sulfones

1974
Mycetoma due to Nocardia.
    Archives of dermatology, 1970, Volume: 102, Issue:3

    Topics: Anti-Bacterial Agents; Dapsone; Foot Diseases; Humans; Male; Middle Aged; Mycetoma; Nocardia; Sulfadiazine; Sulfisoxazole; Sulfonamides

1970
The chemotherapy of rodent malaria. IX. Causal prophylaxis. I. A method for demonstrating drug action on exo-erythrocytic stages.
    Annals of tropical medicine and parasitology, 1970, Volume: 64, Issue:1

    Topics: Animals; Antimalarials; Chloroquine; Dapsone; Malaria; Male; Mice; Plasmodium; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Sulfadiazine; Triazines

1970
Determination of arylamines in urine without the interference of indican.
    The Journal of laboratory and clinical medicine, 1971, Volume: 77, Issue:3

    Topics: Amines; Dapsone; Humans; Hydrogen-Ion Concentration; Hydrolysis; Indican; Indicators and Reagents; Methods; Spectrophotometry; Sulfadiazine; Trichloroacetic Acid

1971
Characteristics and cross-resistance patterns of chloroquine-resistant Plasmodium berghei infections in mice.
    Experimental parasitology, 1968, Volume: 23, Issue:1

    Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; Dapsone; Drug Resistance, Microbial; Female; Hematocrit; Isoenzymes; L-Lactate Dehydrogenase; Malaria; Mice; Organ Size; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Rodent Diseases; Serum Albumin; Serum Globulins; Spleen; Splenomegaly; Sulfadiazine

1968
Drug resistance in Plasmodium berghei Vincke and Lips, 1948. I. Chloroquine resistance.
    Experimental parasitology, 1965, Volume: 17, Issue:1

    Topics: Amodiaquine; Animals; Chloroquine; Dapsone; Malaria; Mice; Plasmodium; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Sulfadiazine; Triazines

1965
Drug resistance in Plasmodium berghei Vincke and Lips, 1948. II. Triazine resistance.
    Experimental parasitology, 1965, Volume: 17, Issue:1

    Topics: Animals; Dapsone; In Vitro Techniques; Malaria; Mice; Plasmodium; Primaquine; Proguanil; Pyrimethamine; Sulfadiazine; Triazines

1965
Drug resistance in Plasmodium berghei Vincke and Lips, 1948. 3. Multiple drug resistance.
    Experimental parasitology, 1965, Volume: 17, Issue:1

    Topics: Animals; Antimalarials; Dapsone; In Vitro Techniques; Malaria; Mice; Plasmodium; Quinacrine; Sulfadiazine; Triazines

1965
Drug responses of mepacrine- and primaquine-resistant strains of Plasmodium berghei Vincke and Lips, 1948.
    Annals of tropical medicine and parasitology, 1966, Volume: 60, Issue:1

    Topics: Animals; Antimalarials; Chloroquine; Dapsone; Mice; Plasmodium; Primaquine; Pyrimethamine; Quinine; Sulfadiazine

1966
Treatment of chloroquine-resistant Plasmodium falciparum infections in Vietnam.
    Annals of internal medicine, 1967, Volume: 66, Issue:3

    Topics: Chloroquine; Dapsone; Humans; Malaria; Military Medicine; Pyrimethamine; Quinacrine; Quinine; Sulfadiazine; Sulfonamides; Vietnam

1967
Relations among antimalarial drugs: results of studies with cycloguanil-, sulfone-, or chloroquine-resistant Plasmodium berghei in mice.
    The American journal of tropical medicine and hygiene, 1967, Volume: 16, Issue:2

    Topics: Acridines; Amodiaquine; Animals; Antimalarials; Arsenicals; Chloroquine; Dapsone; Drug Resistance, Microbial; In Vitro Techniques; Injections, Subcutaneous; Mice; Plasmodium; Sulfadiazine

1967
Juvenile dermatitis herpetiformis. Case reports of six children from Birmingham.
    The British journal of dermatology, 1967, Volume: 79, Issue:4

    Topics: Child, Preschool; Dapsone; Dermatitis Herpetiformis; Female; Humans; Infant; Male; Psychosomatic Medicine; Sulfadiazine

1967
A pilot study on the efficacy of epiroprim against developmental stages of Toxoplasma gondii and Pneumocystis carinii in animal models.
    Parasitology research, 1995, Volume: 81, Issue:4

    Topics: Animals; Anti-Bacterial Agents; Anti-Infective Agents; Dapsone; Drug Therapy, Combination; Female; Folic Acid Antagonists; Male; Mice; Mice, Inbred Strains; Mice, Nude; Mice, SCID; Pilot Projects; Pneumocystis; Pneumocystis Infections; Pyrimethamine; Rats; Rats, Nude; Sodium Chloride; Sulfadiazine; Toxoplasma; Toxoplasmosis, Animal; Trimethoprim

1995
Toxoplasma gondii infection in advanced HIV infection.
    AIDS (London, England), 1994, Volume: 8, Issue:4

    Topics: Adult; AIDS-Related Opportunistic Infections; Dapsone; Encephalitis; Female; Humans; Male; Middle Aged; Pyrimethamine; Sulfadiazine; Sulfadoxine; Survival Rate; Toxoplasmosis; Toxoplasmosis, Cerebral; Trimethoprim, Sulfamethoxazole Drug Combination

1994
Efficacy of epiroprim (Ro11-8958), a new dihydrofolate reductase inhibitor, in the treatment of acute Toxoplasma infection in mice.
    The American journal of tropical medicine and hygiene, 1996, Volume: 54, Issue:3

    Topics: Acute Disease; Administration, Oral; Animals; Anti-Infective Agents; Antiprotozoal Agents; Dapsone; Drug Therapy, Combination; Folic Acid Antagonists; Half-Life; Humans; Injections, Intraperitoneal; Injections, Subcutaneous; Mice; Mice, Inbred BALB C; Sulfadiazine; Toxoplasmosis, Animal; Trimethoprim

1996
TREATMENT OF EXPERIMENTAL OCULAR TOXOPLASMOSIS.
    Archives of ophthalmology (Chicago, Ill. : 1960), 1964, Volume: 71

    Topics: Animals; Dapsone; Eye; Guinea Pigs; Head; Pyrimethamine; Rabbits; Research; Sulfadiazine; Toxoplasmosis, Ocular; Triazines; Uveitis

1964
IgA pemphigus--occurrence of anti-desmocollin 1 and anti-desmoglein 1 antibody reactivity in an individual patient.
    Journal der Deutschen Dermatologischen Gesellschaft = Journal of the German Society of Dermatology : JDDG, 2006, Volume: 4, Issue:12

    Topics: Anti-Bacterial Agents; Anti-Infective Agents; Anti-Inflammatory Agents; Autoantibodies; Autoantigens; Cefamandole; Dapsone; Desmocollins; Desmoglein 1; Enzyme-Linked Immunosorbent Assay; Fluorescent Antibody Technique; Humans; Immunoglobulin A; Male; Middle Aged; Ointments; Pemphigus; Skin; Sulfadiazine; Time Factors; Treatment Outcome

2006
Feasibility of amlodipine besylate, chloroquine phosphate, dapsone, phenytoin, pyridoxine hydrochloride, sulfadiazine, sulfasalazine, tetracycline hydrochloride, trimethoprim and zonisamide in SyrSpend(®) SF PH4 oral suspensions.
    Journal of pharmaceutical and biomedical analysis, 2016, Jan-25, Volume: 118

    Topics: Administration, Oral; Amlodipine; Chloroquine; Chromatography, High Pressure Liquid; Dapsone; Drug Stability; Drug Storage; Feasibility Studies; Hydrogen-Ion Concentration; Isoxazoles; Phenytoin; Pyridoxine; Sulfadiazine; Sulfasalazine; Suspensions; Tetracycline; Trimethoprim; Zonisamide

2016