dapsone and diazepam

dapsone has been researched along with diazepam in 17 studies

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-19906 (35.29)18.7374
1990's0 (0.00)18.2507
2000's4 (23.53)29.6817
2010's7 (41.18)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chang, TK; Ensom, MH; Kiang, TK1
Andricopulo, AD; Moda, TL; Montanari, CA1
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Brodersen, R; Honoré, B1
Karp, W; Robertson, A1
Ho, CK; Karp, WB; Robertson, AF1
Brodersen, R1
Bwibo, NO1
Andersen, S; Brodersen, R; Cashore, WJ; Ebbesen, F; Jacobsen, C; Larsen, S; Sønderskov, O1
Baron-Flores, V; Caballero-Chacón, S; Díaz-Ruiz, A; Farfán-Briseño, AC; Franco-Pérez, J; Manjarrez-Marmolejo, J; Méndez-Armenta, M; Nava-Ruiz, C; Ríos, C; Ruiz-Diaz, A1

Reviews

2 review(s) available for dapsone and diazepam

ArticleYear
UDP-glucuronosyltransferases and clinical drug-drug interactions.
    Pharmacology & therapeutics, 2005, Volume: 106, Issue:1

    Topics: Clinical Trials as Topic; Drug Interactions; Enzyme Activation; Enzyme Induction; Glucuronides; Glucuronosyltransferase; Humans; Pharmaceutical Preparations; Pharmacogenetics; Polymorphism, Genetic

2005
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

15 other study(ies) available for dapsone and diazepam

ArticleYear
Hologram QSAR model for the prediction of human oral bioavailability.
    Bioorganic & medicinal chemistry, 2007, Dec-15, Volume: 15, Issue:24

    Topics: Administration, Oral; Biological Availability; Holography; Humans; Models, Biological; Models, Molecular; Molecular Structure; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2007
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Drug binding properties of neonatal albumin.
    Acta paediatrica Scandinavica, 1989, Volume: 78, Issue:3

    Topics: Adult; Age Factors; Dapsone; Diazepam; Fetal Blood; Humans; Infant, Newborn; Receptors, Albumin; Receptors, Cell Surface; Serum Albumin; Sulfamethizole; Warfarin

1989
Albumin binding of bumetanide.
    Developmental pharmacology and therapeutics, 1986, Volume: 9, Issue:4

    Topics: Adult; Binding, Competitive; Bumetanide; Dapsone; Diazepam; Diuretics; Fetal Blood; Furosemide; Humans; In Vitro Techniques; Infant, Newborn; Kinetics; Protein Binding; Serum Albumin

1986
Hematin and bilirubin binding to human serum albumin and newborn serum.
    Acta paediatrica Scandinavica, 1985, Volume: 74, Issue:3

    Topics: Bilirubin; Dapsone; Dialysis; Diazepam; Heme; Hemin; Horseradish Peroxidase; Humans; Infant, Newborn; Light; Methods; Serum Albumin; Sulfamethizole

1985
Fusidic acid binding to serum albumin and interaction with binding of bilirubin.
    Acta paediatrica Scandinavica, 1985, Volume: 74, Issue:6

    Topics: Adult; Bilirubin; Binding, Competitive; Dapsone; Diazepam; Fusidic Acid; Humans; Methods; Oxidation-Reduction; Serum Albumin; Warfarin

1985
Accidental poisoning in children in Uganda.
    British medical journal, 1969, Dec-06, Volume: 4, Issue:5683

    Topics: Amitriptyline; Aspirin; Barbiturates; Child; Child, Preschool; Chloroquine; Codeine; Dapsone; Diazepam; Ethanol; Female; Humans; Infant; Iron; Kerosene; Male; Pesticides; Poisoning; Quinine; Tetrachloroethylene; Uganda

1969
Determination of reserve albumin-equivalent for ligand binding, probing two distinct binding functions of the protein.
    Analytical biochemistry, 1982, Volume: 121, Issue:2

    Topics: Bilirubin; Chemical Phenomena; Chemistry; Dapsone; Diazepam; Humans; Hydrogen-Ion Concentration; Ligands; Mathematics; Models, Chemical; Protein Binding; Serum Albumin; Temperature; Thermodynamics

1982
Efficacy of dapsone administered alone or in combination with diazepam to inhibit status epilepticus in rats.
    Brain research, 2019, 04-01, Volume: 1708

    Topics: Animals; Anticonvulsants; Dapsone; Diazepam; Electroencephalography; Hippocampus; Kainic Acid; Male; Neurons; Neuroprotective Agents; Pyramidal Cells; Rats; Rats, Wistar; Seizures; Status Epilepticus

2019