dapsone and cycloguanil

dapsone has been researched along with cycloguanil in 14 studies

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19904 (28.57)18.7374
1990's5 (35.71)18.2507
2000's4 (28.57)29.6817
2010's1 (7.14)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Genther, CS; Smith, CS1
Queener, SF1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
González-Ruiz, A; Haworth, SJ; O'Neil, AB; Warhurst, DC1
Edstein, MD; Rieckmann, KH; Veenendaal, JR1
Berlin, OG; Bruckner, DA; Gonzalez, AH1
O'Sullivan, WJ; Rieckmann, KH; Scott, HV1
Rossan, RN; Schmidt, LH1
Edstein, MD; Rieckmann, KH; Shanks, GD; Teja-Isavadharm, P; Webster, HK1
Edstein, MD; Rieckmann, KH; Shanks, GD; Yeo, AE1
Peters, W; Robinson, BL; Stewart, LB1
Hunt, S; Kamau, EM; Nduati, E; Nzila, A1
Kamau, EM; Nduati, EW1
Aarons, L; Bojang, K; Edwards, G; Hughes, D; Manyando, C; Simpson, JA; Ward, S; Watkins, WA; Winstanley, P1

Reviews

1 review(s) available for dapsone and cycloguanil

ArticleYear
New drug developments for opportunistic infections in immunosuppressed patients: Pneumocystis carinii.
    Journal of medicinal chemistry, 1995, Nov-24, Volume: 38, Issue:24

    Topics: Animals; Drug Design; Humans; Immunosuppression Therapy; Molecular Structure; Opportunistic Infections; Pneumonia, Pneumocystis; Structure-Activity Relationship

1995

Other Studies

13 other study(ies) available for dapsone and cycloguanil

ArticleYear
Antifolate studies. Activities of 40 potential antimalarial compounds against sensitive and chlorguanide triazine resistant strains of folate-requiring bacteria and Escherichia coli.
    Journal of medicinal chemistry, 1977, Volume: 20, Issue:2

    Topics: Animals; Antimalarials; Bacteria; Drug Resistance, Microbial; Escherichia coli; Folic Acid; Folic Acid Antagonists; Malaria; Mice; Plasmodium berghei; Triazines

1977
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Dapsone in low doses prevents Pneumocystis carinii pneumonia in the rat model.
    The Journal of infection, 1991, Volume: 22, Issue:2

    Topics: Administration, Oral; Animals; Dapsone; Diet; Disease Models, Animal; Immune Tolerance; Male; Pneumonia, Pneumocystis; Proguanil; Random Allocation; Rats; Rats, Inbred Strains; Triazines

1991
Multiple-dose kinetics in healthy volunteers and in vitro antimalarial activity of proguanil plus dapsone.
    Chemotherapy, 1990, Volume: 36, Issue:3

    Topics: Adult; Animals; Anti-Infective Agents; Dapsone; Drug Administration Schedule; Drug Resistance; Drug Synergism; Drug Therapy, Combination; Half-Life; Humans; Male; Plasmodium falciparum; Proguanil; Time Factors; Triazines

1990
In-vitro activity of dapsone and two potentiators against Mycobacterium avium complex.
    The Journal of antimicrobial chemotherapy, 1989, Volume: 24, Issue:1

    Topics: Acquired Immunodeficiency Syndrome; Anti-Bacterial Agents; Dapsone; Drug Synergism; Humans; Microbial Sensitivity Tests; Mycobacterium avium Complex; Mycobacterium avium-intracellulare Infection; Proguanil; Sulfamethazine; Triazines

1989
Synergistic antimalarial activity of dapsone/dihydrofolate reductase inhibitors and the interaction of antifol, antipyrimidine and antipurine combinations against Plasmodium falciparum in vitro.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1987, Volume: 81, Issue:5

    Topics: Animals; Antimalarials; Antimetabolites; Dapsone; Drug Synergism; Plasmodium falciparum; Proguanil; Ribonucleosides; Triazines

1987
Activities of respository preparations of cycloguanil pamoate and 4,4'-diacetyldiaminodiphenylsulfone, alone and in combination, against infections with Plasmodium cynomolgi in rhesus monkeys.
    Antimicrobial agents and chemotherapy, 1984, Volume: 26, Issue:5

    Topics: Acedapsone; Animals; Antimalarials; Dapsone; Drug Combinations; Drug Resistance, Microbial; Macaca mulatta; Malaria; Particle Size; Plasmodium falciparum; Plasmodium vivax; Proguanil; Pyrimethamine; Time Factors; Triazines

1984
Oxidative activation of proguanil and dapsone acetylation in Thai soldiers.
    British journal of clinical pharmacology, 1994, Volume: 37, Issue:1

    Topics: Acetylation; Biotransformation; Chromatography, High Pressure Liquid; Dapsone; Humans; Malaria; Military Personnel; Oxidation-Reduction; Polymorphism, Genetic; Proguanil; Thailand; Triazines

1994
Ex vivo antimalarial activity of proguanil combined with dapsone against cycloguanil-resistant Plasmodium falciparum isolates.
    Acta tropica, 1997, Sep-10, Volume: 66, Issue:3

    Topics: Animals; Antimalarials; Dapsone; Drug Resistance; Drug Therapy, Combination; Humans; Malaria, Falciparum; Plasmodium falciparum; Proguanil; Triazines

1997
The chemotherapy of rodent malaria. LXII. Drug combinations to impede the selection of drug resistance, part 5: rates of development of resistance to some inhibitors of folate metabolism and to artesunate.
    Annals of tropical medicine and parasitology, 2004, Volume: 98, Issue:8

    Topics: Animals; Antimalarials; Artemisinins; Artesunate; Dapsone; Drug Resistance; Drug Therapy, Combination; Folic Acid Antagonists; Malaria, Falciparum; Male; Mice; Parasitemia; Plasmodium berghei; Plasmodium chabaudi; Plasmodium yoelii; Proguanil; Sesquiterpenes; Triazines

2004
2,4-diaminopteridine-based compounds as precursors for de novo synthesis of antifolates: a novel class of antimalarials.
    Antimicrobial agents and chemotherapy, 2005, Volume: 49, Issue:9

    Topics: Animals; Antimalarials; Dapsone; Dihydropteroate Synthase; Drug Combinations; Drug Synergism; Folic Acid Antagonists; Plasmodium; Proguanil; Pteridines; Saccharomyces cerevisiae; Tetrahydrofolate Dehydrogenase; Triazines

2005
Multiple synergistic interactions between atovaquone and antifolates against Plasmodium falciparum in vitro: a rational basis for combination therapy.
    Acta tropica, 2006, Volume: 97, Issue:3

    Topics: Animals; Antimalarials; Atovaquone; Dapsone; Drug Synergism; Drug Therapy, Combination; Folic Acid Antagonists; Naphthoquinones; Plasmodium falciparum; Proguanil; Triazines

2006
Population pharmacokinetic and pharmacodynamic modelling of the antimalarial chemotherapy chlorproguanil/dapsone.
    British journal of clinical pharmacology, 2006, Volume: 61, Issue:3

    Topics: Adolescent; Adult; Animals; Antimalarials; Child; Child, Preschool; Dapsone; Humans; Infant; Malaria, Falciparum; Middle Aged; Plasmodium falciparum; Proguanil; Prospective Studies; Triazines

2006