dapi has been researched along with pentamidine in 19 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 3 (15.79) | 18.7374 |
1990's | 8 (42.11) | 18.2507 |
2000's | 4 (21.05) | 29.6817 |
2010's | 4 (21.05) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Cory, M; Fairley, TA; Tidwell, RR | 1 |
Clercq, ED; Dann, O | 1 |
Bentley, JA; Cory, M; Donkor, I; Fairley, TA; Lombardy, RJ; Naiman, NA; Ohemeng, KA; Tidwell, RR | 1 |
Lombardy, RL; Ramachandran, K; Tanious, FA; Tidwell, RR; Wilson, WD | 1 |
Bakunov, SA; Bakunova, SM; Barszcz, T; Brun, R; Tidwell, RR; Wenzler, T; Werbovetz, KA | 1 |
Barghash, Ael-D; Boykin, DW; Brun, R; Eisa, HM; Farahat, AA; Goda, FE; Kumar, A; Liu, Y; Mickelson, L; Say, M; Wenzler, T; Wilson, WD | 1 |
Barghash, AE; Boykin, DW; Brun, R; Eisa, HM; Farahat, AA; Goda, FE; Kumar, A; Liu, Y; Paliakov, E; Wenzler, T; Wilson, WD | 1 |
Huang, TL; Mayence, A; Vanden Eynde, JJ | 1 |
Estler, CJ; Sippel, H; Steinmann, U | 1 |
Estler, CJ; Paulini, H; Sippel, H; Stauffert, I; Steinmann, U | 1 |
Balber, AE; Frommel, TO | 1 |
Estler, CJ; Pesch, HJ; Sippel, H; Steinmann, U | 1 |
Alvarez Bujidos, ML; Balaña Fouce, R; Cubria, JC; Ordoñez, D; Reguera, R | 1 |
Bell, A; Kittler, L; Lober, G; Matesoi, D; Unger, E | 1 |
Balaña-Fouce, R; García-Fernández, AJ; Johnson, RA; Navas, IM; Ordóñez, D; Reguera, RM | 1 |
Bryant, AR; Degtyareva, NN; Loo, KM; Petty, JT; Wallace, BD | 1 |
Brown, MH; Hassan, KA; Skurray, RA; Souhani, T | 1 |
Coelho, AC; Cotrim, PC; da Silveira, JF; Gentil, LG | 1 |
Chen, X; Dürrnagel, S; Li, M; MacDonald, JF; Orser, BA; Qiu, L; Xiong, ZG | 1 |
1 review(s) available for dapi and pentamidine
Article | Year |
---|---|
Some non-conventional biomolecular targets for diamidines. A short survey.
Topics: Amidines; Animals; Diabetes Mellitus, Type 2; DNA; Enzymes; Humans; Hypertension; Ion Channels; Myotonic Dystrophy; Neoplasms; Neurodegenerative Diseases; Proteins; RNA; Thrombosis | 2014 |
18 other study(ies) available for dapi and pentamidine
Article | Year |
---|---|
Structure and DNA binding activity of analogues of 1,5-bis(4-amidinophenoxy)pentane (pentamidine)
Topics: DNA; Models, Molecular; Pentamidine | 1992 |
Diaryl amidine derivatives as oncornaviral DNA polymerase inhibitors.
Topics: Amidines; Animals; Antineoplastic Agents; Kinetics; Leukemia, Experimental; Mice; Moloney murine leukemia virus; Retroviridae; Reverse Transcriptase Inhibitors; Structure-Activity Relationship; Tilorone | 1980 |
Structure, DNA minor groove binding, and base pair specificity of alkyl- and aryl-linked bis(amidinobenzimidazoles) and bis(amidinoindoles).
Topics: Amidines; Animals; Base Composition; Benzimidazoles; Binding Sites; Cattle; Chemical Phenomena; Chemistry, Physical; DNA; Electrochemistry; Hot Temperature; Hydrogen Bonding; Indoles; Molecular Structure; Poly dA-dT; Polydeoxyribonucleotides; Structure-Activity Relationship; Viscosity | 1993 |
Synthesis and DNA interactions of benzimidazole dications which have activity against opportunistic infections.
Topics: AIDS-Related Opportunistic Infections; Antifungal Agents; Base Sequence; Benzimidazoles; Binding Sites; Circular Dichroism; DNA; Drug Design; Ethidium; Humans; Kinetics; Magnetic Resonance Spectroscopy; Molecular Sequence Data; Molecular Structure; Nucleic Acid Conformation; Oligodeoxyribonucleotides; Pneumonia, Pneumocystis; Poly dA-dT; RNA; Spectrophotometry; Thermodynamics | 1996 |
Synthesis and antiprotozoal activity of cationic 2-phenylbenzofurans.
Topics: Animals; Antiprotozoal Agents; Benzofurans; Cations; Disease Models, Animal; Leishmania; Mice; Molecular Structure; Structure-Activity Relationship; Trypanosoma; Trypanosomiasis | 2008 |
Synthesis, DNA binding, fluorescence measurements and antiparasitic activity of DAPI related diamidines.
Topics: Animals; Apoptosis; Binding Sites; Cells, Cultured; DNA, Protozoan; Drug Evaluation, Preclinical; Fluorescence; Indoles; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Rats; Trypanosoma brucei rhodesiense | 2010 |
Exploration of larger central ring linkers in furamidine analogues: synthesis and evaluation of their DNA binding, antiparasitic and fluorescence properties.
Topics: Animals; Antiparasitic Agents; Antiprotozoal Agents; Benzamidines; Benzimidazoles; Circular Dichroism; Cross-Linking Reagents; DNA, Protozoan; Fluorescence; Humans; Mice; Models, Chemical; Molecular Structure; Plasmodium falciparum; Structure-Activity Relationship; Trypanosoma brucei rhodesiense | 2011 |
Influence of pentamidine and two new trypanocidal agents (DAPI, DIPI) on liver metabolism of mice.
Topics: Animals; Energy Metabolism; Fluorescent Dyes; Indoles; Lipid Metabolism; Liver; Male; Mice; Pentamidine; Trypanocidal Agents | 1991 |
Investigations on mutagenicity and genotoxicity of pentamidine and some related trypanocidal diamidines.
Topics: Amidines; Cells, Cultured; Humans; Indoles; Lymphocytes; Mutagenicity Tests; Mutagens; Pentamidine; Salmonella typhimurium; Sister Chromatid Exchange; Structure-Activity Relationship; Trypanocidal Agents | 1990 |
Flow cytofluorimetric analysis of drug accumulation by multidrug-resistant Trypanosoma brucei brucei and T. b. rhodesiense.
Topics: Acriflavine; Animals; Benzimidazoles; Diminazene; Drug Resistance; Ethidium; Flow Cytometry; Fluorescent Dyes; Humans; Indoles; Melarsoprol; Mice; Pentamidine; Suramin; Trypanocidal Agents; Trypanosoma brucei brucei | 1987 |
Changes in serum transaminases, SDH and liver morphology after treatment with trypanocidal diamidines in mice.
Topics: Alanine Transaminase; Animals; Aspartate Aminotransferases; Dose-Response Relationship, Drug; Indoles; L-Iditol 2-Dehydrogenase; Liver; Male; Mice; Pentamidine; Sugar Alcohol Dehydrogenases; Transaminases; Trypanocidal Agents | 1985 |
Putrescine uptake inhibition by aromatic diamidines in Leishmania infantum promastigotes.
Topics: Amidines; Animals; Diminazene; Indoles; Kinetics; Leishmania infantum; Pentamidine; Putrescine; Stilbamidines | 1994 |
Determination of microscopic binding constants at individual DNA base sequences for the minor groove binders Hoechst 33258, DAPI and pentamidine.
Topics: Base Sequence; Binding Sites; Bisbenzimidazole; Deoxyribonuclease I; DNA; DNA Footprinting; DNA Restriction Enzymes; Electrophoresis, Polyacrylamide Gel; Escherichia coli; Fluorescent Dyes; Indoles; Intercalating Agents; Molecular Sequence Data; Molecular Structure; Nucleic Acid Conformation; Pentamidine; Plasmids | 1996 |
Structural determinants of putrescine uptake inhibition produced by cationic diamidines in the model of trypanosomatid Crithidia fasciculata.
Topics: Animals; Benzamidines; Carbanilides; Crithidia; Indoles; Leishmania; Pentamidine; Putrescine; Stilbamidines; Structure-Activity Relationship; Trypanocidal Agents | 1996 |
Hydration changes accompanying the binding of minor groove ligands with DNA.
Topics: Binding Sites; DNA; Indoles; Netropsin; Nucleic Acid Conformation; Pentamidine; Water | 2007 |
Analysis of tryptophan residues in the staphylococcal multidrug transporter QacA reveals long-distance functional associations of residues on opposite sides of the membrane.
Topics: Alanine; Amino Acid Sequence; Bacterial Proteins; Benzalkonium Compounds; Biological Transport; Blotting, Western; Cell Membrane; Chlorhexidine; Dequalinium; Drug Resistance, Microbial; Electrophoresis, Polyacrylamide Gel; Ethidium; Fluoresceins; Indoles; Membrane Transport Proteins; Microbial Sensitivity Tests; Models, Biological; Molecular Sequence Data; Mutagenesis, Site-Directed; Mutation; Pentamidine; Phenylalanine; Protein Structure, Secondary; Pyronine; Rhodamines; Staphylococcus; Tryptophan | 2008 |
Characterization of Leishmania (Leishmania) amazonensis promastigotes resistant to pentamidine.
Topics: Animals; Antiprotozoal Agents; ATP-Binding Cassette Transporters; Blotting, Southern; DNA, Protozoan; Drug Resistance; Electrophoresis, Gel, Pulsed-Field; Fluorescent Dyes; Indoles; Inhibitory Concentration 50; Leishmania mexicana; Microscopy, Fluorescence; Mutation; Pentamidine; Phenotype; Protozoan Proteins | 2008 |
Diarylamidines: high potency inhibitors of acid-sensing ion channels.
Topics: Acid Sensing Ion Channels; Amidines; Animals; Cells, Cultured; CHO Cells; Cricetinae; Cricetulus; Diminazene; Epithelial Sodium Channel Blockers; Epithelial Sodium Channels; Hippocampus; Indoles; Mice; Nerve Tissue Proteins; Neurons; Neurotransmitter Agents; Oocytes; Pentamidine; Sodium Channels; Stilbamidines; Xenopus laevis | 2010 |