Page last updated: 2024-09-05

dabigatran and rifampin

dabigatran has been researched along with rifampin in 3 studies

Compound Research Comparison

Studies
(dabigatran)
Trials
(dabigatran)
Recent Studies (post-2010)
(dabigatran)
Studies
(rifampin)
Trials
(rifampin)
Recent Studies (post-2010) (rifampin)
3,8872613,49020,4681,4996,552

Protein Interaction Comparison

ProteinTaxonomydabigatran (IC50)rifampin (IC50)
Polyunsaturated fatty acid lipoxygenase ALOX15Oryctolagus cuniculus (rabbit)2.949
Caspase-1Homo sapiens (human)8.319
Alpha-synucleinHomo sapiens (human)7.1
Enoyl-[acyl-carrier-protein] reductase [NADH]Mycobacterium tuberculosis H37Rv0.03
DNA-directed RNA polymerase subunit betaMycobacterium tuberculosis H37Rv0.01
Solute carrier organic anion transporter family member 1B3Homo sapiens (human)1.5
Solute carrier organic anion transporter family member 1B1Homo sapiens (human)1.5

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's3 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Härtter, S; Koenen-Bergmann, M; Lemke, U; Nehmiz, G; Reilly, PA; Sharma, A; Timmer, W1
Costales, C; Eatemadpour, S; Kimoto, E; Lazzaro, S; Varma, MV; Yamazaki, S1
Bairlein, M; Denner, K; Fricke, R; Gieschen, H; Graudenz, K; Korjamo, T; Koskinen, M; Prien, O; von Bühler, CJ; Wilkinson, G; Zurth, C1

Trials

2 trial(s) available for dabigatran and rifampin

ArticleYear
Decrease in the oral bioavailability of dabigatran etexilate after co-medication with rifampicin.
    British journal of clinical pharmacology, 2012, Volume: 74, Issue:3

    Topics: Administration, Oral; Adult; Area Under Curve; Benzimidazoles; Biological Availability; Dabigatran; Drug Interactions; Enzyme Inhibitors; Female; Glucuronides; Half-Life; Humans; Male; Prodrugs; Pyridines; Rifampin; Young Adult

2012
Drug-Drug Interaction Potential of Darolutamide: In Vitro and Clinical Studies.
    European journal of drug metabolism and pharmacokinetics, 2019, Volume: 44, Issue:6

    Topics: Aged; Cells, Cultured; Cytochrome P-450 CYP3A Inducers; Cytochrome P-450 CYP3A Inhibitors; Cytochrome P-450 Enzyme System; Dabigatran; Drug Interactions; Enzyme Induction; Female; Humans; Itraconazole; Male; Membrane Transport Proteins; Microsomes, Liver; Midazolam; Middle Aged; Pyrazoles; Rifampin; Rosuvastatin Calcium

2019

Other Studies

1 other study(ies) available for dabigatran and rifampin

ArticleYear
Physiologically-Based Pharmacokinetic Modeling Approach to Predict Rifampin-Mediated Intestinal P-Glycoprotein Induction.
    CPT: pharmacometrics & systems pharmacology, 2019, Volume: 8, Issue:9

    Topics: Administration, Oral; ATP Binding Cassette Transporter, Subfamily B, Member 1; Dabigatran; Digoxin; Drug Interactions; Female; Gene Expression Regulation; Healthy Volunteers; Humans; Intestinal Mucosa; Male; Models, Biological; Propanolamines; Quinidine; Rifampin

2019