Page last updated: 2024-08-21

cytisine and varenicline

cytisine has been researched along with varenicline in 54 studies

Research

Studies (54)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's7 (12.96)29.6817
2010's32 (59.26)24.3611
2020's15 (27.78)2.80

Authors

AuthorsStudies
Arnold, EP; Bashore, CG; Bianco, KE; Brooks, PR; Coe, JW; Davis, TI; Fox, CB; Lebel, LA; Mansbach, RS; O'Neill, BT; Rollema, H; Sands, SB; Schulz, DW; Tingley, FD; Vetelino, MG; Wirtz, MC1
Benson, LR; Bhatti, BS; Breining, SR; Byrd, GD; Fedorov, NB; Hepler, CD; Hooker, DN; Kiser, MN; Lucero, LM; Lukas, RJ; Melvin, M; Mitchener, JP; Reynolds, LA; Sidach, SS; Whiteaker, P; Yohannes, D; Zhang, J1
Caldarone, BJ; Eaton, JB; Kozikowski, AP; Lukas, RJ; Yu, LF; Zhang, HK1
Cahill, K; Lancaster, T; Stead, LF5
Cahill, K; Lancaster, T; Stead, L1
Tutka, P1
Carroll, FI; Corrigall, WA; LeSage, MG; Ross, JT; Shelley, D1
Einarson, A; Riordan, S1
Papke, RL; Stitzel, JA; Wecker, L1
Bertrand, D; Bertrand, S; Coe, JW; Cremers, T; de Vries, M; Hurst, RS; Mather, RJ; O'Neill, BT; Rollema, H; Shrikhande, A; Tingley, FD; Tseng, E; Wang, EQ; Ward, KM; Williams, KE1
Cunningham, CS; McMahon, LR2
Al Rubaiy, SA; Bloom, SA; Guendisch, D; Papke, RL; Trocmé-Thibierge, C1
Gallagher, T; Haseler, CA; Hirschhäuser, C1
Cunningham, CS; Javors, MA; McMahon, LR1
Gallagher, T; Haseler, CA; Rucktooa, P; Sixma, TK; Smit, AB; van Elk, R1
Papke, RL; Stokes, C1
Busto, UE; Cassels, BK; Gysling, K; Quintanilla, ME; Sotomayor-Zárate, R; Tampier, L1
Milnerowicz, H; Sliwińska-Mossoń, M; Zieleń, I1
Cahill, K; Lancaster, T; Perera, R; Stevens, S1
Cahill, K; Hartmann-Boyce, J; Lancaster, T; Stead, LF1
Rahman, S; Sajja, RK1
Eibl, C; Guendisch, D; Mineur, YS; Papke, RL; Peng, C; Picciotto, MR; Stokes, C; Tian, C; Tomassoli, I1
Alexander, JC; Bruijnzeel, AW; Igari, M; Ji, Y; Papke, RL; Qi, X1
Cieślewicz, A; Jabłecka, A; Korzeniowska, K1
Cantrell, A; Everson-Hock, E; Leaviss, J; Ren, S; Stevens, JW; Stevenson, M; Strong, M; Sullivan, W1
Kuryatov, A; Ley, CK; Lindstrom, JM; Wang, J1
Benowitz, NL; Prochaska, JJ1
Bartlett, SE; Belmer, A; Holgate, J; Morgan, M; Patkar, OL; Quik, M; Shariff, M; Tam, V1
Cahill, K; Fanshawe, TR; Lancaster, T; Lindson-Hawley, N; Thomas, KH1
de Moura, FB; McMahon, LR2
Barnes, J; Bullen, C; Kurdziel, T; Parag, V; Pokhrel, S; Smith, B; Verbiest, M; Walker, N1
Absalom, NL; Ahring, PK; Balle, T; Chebib, M; Indurthi, DC; Lewis, TM; Liao, VW; Qudah, T1
Boland, VC; Courtney, RJ; Doran, CM; Farrell, M; Ferguson, SG; Gartner, C; Hall, W; Mattick, RP; McRobbie, H; Mendelsohn, CP; Paul, C; Petrie, D; Richmond, R; Shakeshaft, A; Siahpush, M; Thomas, D; Tutka, P; Walker, N; West, R; Zwar, N1
Filipponi, A; Giordano, P; Giulietti, F; Iacoacci, C; Rosettani, G; Sarzani, R; Spannella, F1
Barnes, J; Bullen, C; Cubillos Gutierrez, H; Jones, B; Lees, T; Parag, V; Pokhrel, S; Smith, B; Verbiest, M; Walker, N; Wharakura, MK1
Benowitz, N; Clarke, A; Jacobs, C; Nides, M; Rigotti, NA1
Boland, VC; Courtney, RJ; Doran, CM; Farrell, M; Ferguson, SG; Gartner, C; Hall, W; Kwan, BCH; Macdonald, C; Mattick, RP; McRobbie, H; Mendelsohn, CP; Paul, C; Petrie, D; Richmond, RL; Shakeshaft, A; Talukder, S; Thomas, D; Tutka, P; Walker, N; Weaver, NA; West, R; Zwar, NA1
Courtney, RJ; Farrell, M; Tutka, P1
Lang, AE1
Campagnari, S; Casari, R; Fusina, F; Lugoboni, F; Zamboni, L1
Apolone, G; Boeri, M; Boffi, R; Gallus, S; Ladisa, V; Ledda, RE; Marchianò, A; Milanese, G; Munarini, E; Pastorino, U; Rolli, L; Sabia, F; Sozzi, G; Suatoni, P; Trussardo, S; Valsecchi, C1
Bendiks, S; Blokhina, E; Bryant, K; Cheng, DM; Freiberg, MS; Gnatienko, N; Hahn, J; Krupitsky, E; Lioznov, D; Patts, G; Samet, JH; So-Armah, K; Stein, MD; Tindle, HA; Yaroslavtseva, T1
Boonsawat, W; Dilokthornsakul, P; Hansuri, N; Lertsinudom, S; Phusahat, P; Tawinkan, N; Theeranut, A; Zaeoue, U1
Chatkin, JM; Corrêa, PCRP1
Ashburner, JM; Klemenc Ketiš, Z; Oreskovic, S; Oreskovic, T; Percac-Lima, S; Rifel, J; Tiljak, H1
Budzyńska, B; Chałas, R; Maciąg, M; Rahnama-Hezavah, M; Stachurski, P; Świątkowska, A; Świątkowski, W; Tylżanowski, P1
Dennis, BB; Devereaux, PJ; Fairbairn, N; Lu, C; Mbuagbaw, L; Ofori, S; Olasupo, OO1
Barnes, J; Bullen, C; Calder, A; Laking, G; Parag, V; Walker, N1

Reviews

16 review(s) available for cytisine and varenicline

ArticleYear
Recent developments in novel antidepressants targeting α4β2-nicotinic acetylcholine receptors.
    Journal of medicinal chemistry, 2014, Oct-23, Volume: 57, Issue:20

    Topics: Alkaloids; Antidepressive Agents; Azetidines; Azocines; Depression; Humans; Ligands; Molecular Targeted Therapy; Nicotinic Agonists; Nicotinic Antagonists; Quinolizines; Receptors, Nicotinic

2014
Nicotine receptor partial agonists for smoking cessation.
    The Cochrane database of systematic reviews, 2007, Jan-24, Issue:1

    Topics: Alkaloids; Azocines; Benzazepines; Humans; Nicotine; Nicotinic Agonists; Quinolizines; Quinoxalines; Randomized Controlled Trials as Topic; Smoking Cessation; Varenicline

2007
An update on therapeutics for tobacco dependence.
    Expert opinion on pharmacotherapy, 2008, Volume: 9, Issue:1

    Topics: Alkaloids; Anti-Anxiety Agents; Azocines; Benzazepines; Bupropion; Clinical Trials as Topic; Databases, Bibliographic; Humans; Nicotine; Nicotinic Agonists; Piperidines; Pyrazoles; Quinolizines; Quinoxalines; Review Literature as Topic; Rimonabant; Smoking; Smoking Cessation; Varenicline

2008
Nicotine receptor partial agonists for smoking cessation.
    The Cochrane database of systematic reviews, 2008, Jul-16, Issue:3

    Topics: Alkaloids; Azocines; Benzazepines; Bupropion; Humans; Nicotine; Nicotinic Agonists; Quinolizines; Quinoxalines; Randomized Controlled Trials as Topic; Smoking; Smoking Cessation; Varenicline

2008
Nicotinic receptor partial agonists as novel compounds for the treatment of smoking cessation.
    Expert opinion on investigational drugs, 2008, Volume: 17, Issue:10

    Topics: Alkaloids; Animals; Azocines; Benzazepines; Clinical Trials as Topic; Dopamine; Humans; Nicotinic Agonists; Quinolizines; Quinoxalines; Smoking Cessation; Varenicline

2008
Smoking in pregnancy and lactation: a review of risks and cessation strategies.
    European journal of clinical pharmacology, 2009, Volume: 65, Issue:4

    Topics: Adult; Alkaloids; Antidepressive Agents; Azocines; Benzazepines; Breast Feeding; Bromocriptine; Cognitive Behavioral Therapy; Female; Humans; Lactation; Nicotine; Nicotinic Agonists; Pregnancy; Pregnancy Complications; Quinolizines; Quinoxalines; Risk Assessment; Risk Factors; Smoking; Smoking Cessation; Vaccines; Varenicline; Young Adult

2009
Nicotine receptor partial agonists for smoking cessation.
    The Cochrane database of systematic reviews, 2010, Dec-08, Issue:12

    Topics: Alkaloids; Azocines; Benzazepines; Bupropion; Humans; Nicotine; Nicotinic Agonists; Quinolizines; Quinoxalines; Randomized Controlled Trials as Topic; Smoking; Smoking Cessation; Substance Withdrawal Syndrome; Varenicline

2010
Nicotine receptor partial agonists for smoking cessation.
    The Cochrane database of systematic reviews, 2011, Feb-16, Issue:2

    Topics: Alkaloids; Azocines; Benzazepines; Bupropion; Humans; Nicotine; Nicotinic Agonists; Quinolizines; Quinoxalines; Randomized Controlled Trials as Topic; Smoking; Smoking Cessation; Substance Withdrawal Syndrome; Varenicline

2011
Nicotine receptor partial agonists for smoking cessation.
    The Cochrane database of systematic reviews, 2012, Apr-18, Issue:4

    Topics: Alkaloids; Azepines; Azocines; Benzazepines; Bupropion; Counseling; Heterocyclic Compounds, 4 or More Rings; Humans; Nicotine; Nicotinic Agonists; Quinolizines; Quinoxalines; Randomized Controlled Trials as Topic; Smoking; Smoking Cessation; Substance Withdrawal Syndrome; Varenicline

2012
[Drugs used to treat nicotine addiction].
    Przeglad lekarski, 2012, Volume: 69, Issue:10

    Topics: Adult; Age Distribution; Alkaloids; Azocines; Benzazepines; Bupropion; Causality; Comorbidity; Female; Humans; Male; Middle Aged; Nicotine; Nicotinic Agonists; Poland; Quinolizines; Quinoxalines; Sex Distribution; Smoking; Smoking Cessation; Smoking Prevention; Tobacco Use Disorder; Varenicline; Young Adult

2012
Pharmacological interventions for smoking cessation: an overview and network meta-analysis.
    The Cochrane database of systematic reviews, 2013, May-31, Issue:5

    Topics: Adult; Alkaloids; Antidepressive Agents, Second-Generation; Azocines; Benzazepines; Bupropion; Humans; Nicotinic Agonists; Nortriptyline; Quinolizines; Quinoxalines; Randomized Controlled Trials as Topic; Review Literature as Topic; Smoking; Smoking Cessation; Tobacco Use Cessation Devices; Varenicline

2013
What is the clinical effectiveness and cost-effectiveness of cytisine compared with varenicline for smoking cessation? A systematic review and economic evaluation.
    Health technology assessment (Winchester, England), 2014, Volume: 18, Issue:33

    Topics: Adult; Aged; Alkaloids; Azocines; Benzazepines; Cost-Benefit Analysis; Humans; Middle Aged; Nicotinic Agonists; Quality-Adjusted Life Years; Quinolizines; Quinoxalines; Randomized Controlled Trials as Topic; Smoking; Smoking Cessation; State Medicine; United Kingdom; Varenicline

2014
The Past, Present, and Future of Nicotine Addiction Therapy.
    Annual review of medicine, 2016, Volume: 67

    Topics: Alkaloids; Azocines; Bupropion; Directive Counseling; Dopamine Uptake Inhibitors; Drug Therapy, Combination; Health Policy; Humans; Nicotine; Nicotinic Agonists; Quinolizines; Smoking Cessation; Social Media; Text Messaging; Tobacco Use Cessation Devices; Tobacco Use Disorder; Varenicline

2016
Nicotine receptor partial agonists for smoking cessation.
    The Cochrane database of systematic reviews, 2016, May-09, Issue:5

    Topics: Alkaloids; Azepines; Azocines; Benzazepines; Bupropion; Counseling; Heterocyclic Compounds, 4 or More Rings; Humans; Nicotine; Nicotinic Agonists; Quinolizines; Randomized Controlled Trials as Topic; Smoking; Smoking Cessation; Substance Withdrawal Syndrome; Varenicline

2016
Pharmacological Approach to Smoking Cessation: An Updated Review for Daily Clinical Practice.
    High blood pressure & cardiovascular prevention : the official journal of the Italian Society of Hypertension, 2020, Volume: 27, Issue:5

    Topics: Alkaloids; Azocines; Bupropion; Clinical Decision-Making; Electronic Nicotine Delivery Systems; Humans; Quinolizines; Recurrence; Risk Factors; Smoking; Smoking Cessation; Smoking Cessation Agents; Tobacco Use Cessation Devices; Tobacco Use Disorder; Treatment Outcome; Varenicline

2020
Cytisine for smoking cessation: A systematic review and meta-analysis.
    Drug and alcohol dependence, 2023, 10-01, Volume: 251

    Topics: Adult; Alkaloids; Azocines; Benzazepines; Bupropion; Humans; Nicotine; Nicotinic Agonists; Quinolizines; Smoking Cessation; Varenicline

2023

Trials

10 trial(s) available for cytisine and varenicline

ArticleYear
Cytisine versus varenicline for smoking cessation for Māori (the indigenous people of New Zealand) and their extended family: protocol for a randomized non-inferiority trial.
    Addiction (Abingdon, England), 2019, Volume: 114, Issue:2

    Topics: Alkaloids; Azocines; Carbon Dioxide; Counseling; Equivalence Trials as Topic; Family; Humans; Native Hawaiian or Other Pacific Islander; New Zealand; Patient Safety; Quinolizines; Randomized Controlled Trials as Topic; Smoking Cessation; Smoking Cessation Agents; Varenicline

2019
The effectiveness, safety and cost-effectiveness of cytisine versus varenicline for smoking cessation in an Australian population: a study protocol for a randomized controlled non-inferiority trial.
    Addiction (Abingdon, England), 2019, Volume: 114, Issue:5

    Topics: Adult; Alkaloids; Australia; Azocines; Cost-Benefit Analysis; Double-Blind Method; Equivalence Trials as Topic; Female; Humans; Male; Quinolizines; Smoking Cessation; Treatment Outcome; Varenicline

2019
Cytisine versus varenicline for smoking cessation in New Zealand indigenous Māori: a randomized controlled trial.
    Addiction (Abingdon, England), 2021, Volume: 116, Issue:10

    Topics: Adult; Alkaloids; Azocines; Humans; New Zealand; Quality of Life; Quinolizines; Smoking Cessation; Treatment Outcome; Varenicline

2021
A Multicenter, Double-Blind, Randomized, Placebo-Controlled Phase 2b Trial of Cytisinicline in Adult Smokers (The ORCA-1 Trial).
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2021, 08-29, Volume: 23, Issue:10

    Topics: Adult; Alkaloids; Azocines; Benzazepines; Double-Blind Method; Humans; Quinolizines; Quinoxalines; Smokers; Treatment Outcome; Varenicline

2021
Effect of Cytisine vs Varenicline on Smoking Cessation: A Randomized Clinical Trial.
    JAMA, 2021, 07-06, Volume: 326, Issue:1

    Topics: Adult; Alkaloids; Azocines; Dreams; Female; Humans; Male; Middle Aged; Nausea; Quinolizines; Smoking Cessation; Smoking Cessation Agents; Treatment Outcome; Varenicline

2021
Cytisine Therapy Improved Smoking Cessation in the Randomized Screening and Multiple Intervention on Lung Epidemics Lung Cancer Screening Trial.
    Journal of thoracic oncology : official publication of the International Association for the Study of Lung Cancer, 2022, Volume: 17, Issue:11

    Topics: Alkaloids; Azocines; Early Detection of Cancer; Humans; Lung; Lung Neoplasms; Nicotine; Quinolizines; Smoking Cessation; Varenicline

2022
Effectiveness of Varenicline and Cytisine for Alcohol Use Reduction Among People With HIV and Substance Use: A Randomized Clinical Trial.
    JAMA network open, 2022, 08-01, Volume: 5, Issue:8

    Topics: Adult; Alcoholism; Alkaloids; Azocines; Benzazepines; Female; HIV Infections; Humans; Male; Nicotine; Nicotinic Agonists; Quinolizines; Smoking Cessation; Tobacco Use Cessation Devices; Varenicline

2022
Efficacy and Safety of Cytisine in Combination with a Community Pharmacists' Counselling for Smoking Cessation in Thailand: A Randomized Double-Blinded Placebo-Controlled Trial.
    International journal of environmental research and public health, 2022, 10-16, Volume: 19, Issue:20

    Topics: Adolescent; Benzazepines; Counseling; Female; Humans; Male; Nicotinic Agonists; Pharmacists; Prospective Studies; Smoking; Smoking Cessation; Thailand; Varenicline

2022
Cytisine Versus Varenicline for Smoking Cessation in a Primary Care Setting: A Randomized Non-inferiority Trial.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2023, 08-19, Volume: 25, Issue:9

    Topics: Alkaloids; Azocines; Benzazepines; Humans; Nicotine; Nicotinic Agonists; Primary Health Care; Quinolizines; Smoking Cessation; Treatment Outcome; Varenicline

2023
Effectiveness of nicotine salt vapes, cytisine, and a combination of these products, for smoking cessation in New Zealand: protocol for a three-arm, pragmatic, community-based randomised controlled trial.
    BMC public health, 2023, 09-11, Volume: 23, Issue:1

    Topics: Electronic Nicotine Delivery Systems; Humans; New Zealand; Nicotine; Quality of Life; Randomized Controlled Trials as Topic; Smoking Cessation; Sodium Chloride, Dietary; Tobacco Use Cessation Devices; Vaping; Varenicline

2023

Other Studies

28 other study(ies) available for cytisine and varenicline

ArticleYear
3,5-Bicyclic aryl piperidines: a novel class of alpha4beta2 neuronal nicotinic receptor partial agonists for smoking cessation.
    Bioorganic & medicinal chemistry letters, 2005, Nov-15, Volume: 15, Issue:22

    Topics: Animals; Cyclization; Molecular Structure; Piperidines; Rats; Receptors, Nicotinic; Smoking Cessation; Structure-Activity Relationship

2005
Structure-activity studies of 7-heteroaryl-3-azabicyclo[3.3.1]non-6-enes: a novel class of highly potent nicotinic receptor ligands.
    Journal of medicinal chemistry, 2012, Nov-26, Volume: 55, Issue:22

    Topics: Bridged Bicyclo Compounds, Heterocyclic; Calcium; Cells, Cultured; Electrophysiology; Humans; Kidney; Ligands; Molecular Structure; Neuroblastoma; Nicotine; Protein Subunits; Receptors, Nicotinic; Stereoisomerism; Structure-Activity Relationship

2012
Effects of the nicotinic receptor partial agonists varenicline and cytisine on the discriminative stimulus effects of nicotine in rats.
    Pharmacology, biochemistry, and behavior, 2009, Volume: 91, Issue:3

    Topics: Alkaloids; Animals; Azocines; Benzazepines; Conditioning, Operant; Data Interpretation, Statistical; Discrimination, Psychological; Dose-Response Relationship, Drug; Generalization, Stimulus; Male; Nicotine; Nicotinic Agonists; Quinolizines; Quinoxalines; Rats; Rats, Long-Evans; Receptors, Nicotinic; Varenicline

2009
Activation and inhibition of mouse muscle and neuronal nicotinic acetylcholine receptors expressed in Xenopus oocytes.
    The Journal of pharmacology and experimental therapeutics, 2010, Volume: 333, Issue:2

    Topics: Acetylcholine; Alkaloids; Animals; Azocines; Benzazepines; Decamethonium Compounds; Dihydro-beta-Erythroidine; Dose-Response Relationship, Drug; Electrophysiology; Gene Expression; Hexamethonium; Humans; Mecamylamine; Mice; Mice, Transgenic; Muscle, Skeletal; Nicotinic Antagonists; Oocytes; Quinolizines; Quinoxalines; Rats; Receptors, Nicotinic; Varenicline; Xenopus laevis

2010
Pre-clinical properties of the alpha4beta2 nicotinic acetylcholine receptor partial agonists varenicline, cytisine and dianicline translate to clinical efficacy for nicotine dependence.
    British journal of pharmacology, 2010, Volume: 160, Issue:2

    Topics: Alkaloids; Animals; ATP Binding Cassette Transporter, Subfamily B; ATP-Binding Cassette Sub-Family B Member 4; Azepines; Azocines; Benzazepines; Brain; Dopamine; Heterocyclic Compounds, 4 or More Rings; Humans; Limbic System; Male; Mice; Mice, Knockout; Nicotinic Agonists; Quinolizines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Smoking Cessation; Tissue Distribution; Tobacco Use Disorder; Varenicline; Xenopus laevis

2010
The effects of nicotine, varenicline, and cytisine on schedule-controlled responding in mice: differences in α4β2 nicotinic receptor activation.
    European journal of pharmacology, 2011, Mar-01, Volume: 654, Issue:1

    Topics: Alkaloids; Animals; Azocines; Benzazepines; Conditioning, Operant; Dihydro-beta-Erythroidine; Dose-Response Relationship, Drug; Injections, Intraperitoneal; Male; Mecamylamine; Mice; Mice, Inbred C57BL; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Quinolizines; Quinoxalines; Receptors, Nicotinic; Reinforcement Schedule; Smoking Cessation; Time Factors; Varenicline

2011
Electrophysiological perspectives on the therapeutic use of nicotinic acetylcholine receptor partial agonists.
    The Journal of pharmacology and experimental therapeutics, 2011, Volume: 337, Issue:2

    Topics: Acetylcholine; Alkaloids; alpha7 Nicotinic Acetylcholine Receptor; Animals; Azocines; Benzazepines; Bupropion; DNA, Complementary; Dopamine Uptake Inhibitors; Electrophysiological Phenomena; Humans; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Oocytes; Pyridinium Compounds; Quinolizines; Quinoxalines; Receptors, Nicotinic; Smoking Cessation; Varenicline; Xenopus

2011
Core modification of cytisine: a modular synthesis.
    Angewandte Chemie (International ed. in English), 2011, May-23, Volume: 50, Issue:22

    Topics: Alkaloids; Azocines; Benzazepines; Cyclization; Nicotinic Agonists; Pyridones; Quinolizines; Quinoxalines; Receptors, Nicotinic; Tin Compounds; Varenicline

2011
Pharmacologic characterization of a nicotine-discriminative stimulus in rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 2012, Volume: 341, Issue:3

    Topics: Alkaloids; Animals; Azocines; Benzazepines; Cocaine; Conditioning, Operant; Discrimination Learning; Dopamine Uptake Inhibitors; Drug Interactions; Female; Hypnotics and Sedatives; Macaca mulatta; Male; Mecamylamine; Midazolam; Nicotine; Nicotinic Agonists; Quinolizines; Quinoxalines; Receptors, Nicotinic; Varenicline

2012
Structural characterization of binding mode of smoking cessation drugs to nicotinic acetylcholine receptors through study of ligand complexes with acetylcholine-binding protein.
    The Journal of biological chemistry, 2012, Jul-06, Volume: 287, Issue:28

    Topics: Acetylcholine; Alkaloids; alpha7 Nicotinic Acetylcholine Receptor; Animals; Aplysia; Azocines; Benzazepines; Binding Sites; Binding, Competitive; Carrier Proteins; Cell Line; HEK293 Cells; Humans; Kinetics; Ligands; Models, Molecular; Mutation; Nicotine; Nicotinic Agonists; Protein Binding; Protein Structure, Secondary; Protein Structure, Tertiary; Quinolizines; Quinoxalines; Receptors, Nicotinic; Smoking Cessation; Varenicline

2012
Use of an α3β4 nicotinic acetylcholine receptor subunit concatamer to characterize ganglionic receptor subtypes with specific subunit composition reveals species-specific pharmacologic properties.
    Neuropharmacology, 2012, Volume: 63, Issue:4

    Topics: Acetylcholine; Alkaloids; Animals; Azocines; Benzazepines; Drug Partial Agonism; Evoked Potentials; Ganglia; Humans; Ligands; Mutagenesis, Site-Directed; Mutant Proteins; Nerve Tissue Proteins; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Oocytes; Protein Subunits; Quinolizines; Quinoxalines; Rats; Receptors, Nicotinic; Recombinant Fusion Proteins; Species Specificity; Varenicline; Xenopus laevis

2012
Varenicline and cytisine: two nicotinic acetylcholine receptor ligands reduce ethanol intake in University of Chile bibulous rats.
    Psychopharmacology, 2013, Volume: 227, Issue:2

    Topics: Alcohol Drinking; Alkaloids; Animals; Azocines; Benzazepines; Chile; Dose-Response Relationship, Drug; Drinking; Drug Administration Schedule; Ethanol; Male; Nicotinic Agonists; Quinolizines; Quinoxalines; Rats; Saccharin; Time Factors; Varenicline

2013
Multiple nicotine training doses in mice as a basis for differentiating the effects of smoking cessation aids.
    Psychopharmacology, 2013, Volume: 228, Issue:2

    Topics: Alkaloids; Animals; Azocines; Benzazepines; Dihydro-beta-Erythroidine; Discrimination Learning; Dose-Response Relationship, Drug; Male; Mecamylamine; Mice; Mice, Inbred C57BL; Midazolam; Morphine; Nicotine; Nicotinic Agonists; Quinolizines; Quinoxalines; Receptors, Nicotinic; Smoking Cessation; Tobacco Use Cessation Devices; Varenicline

2013
Efficacy of interventions to combat tobacco addiction: Cochrane update of 2012 reviews.
    Addiction (Abingdon, England), 2013, Volume: 108, Issue:10

    Topics: Alkaloids; Azocines; Behavior Therapy; Behavior, Addictive; Benzazepines; Humans; Meta-Analysis as Topic; Nicotinic Agonists; Quinolizines; Quinoxalines; Review Literature as Topic; Smoking; Smoking Cessation; Tobacco Use Disorder; Treatment Outcome; Varenicline

2013
Nicotinic receptor partial agonists modulate alcohol deprivation effect in C57BL/6J mice.
    Pharmacology, biochemistry, and behavior, 2013, Volume: 110

    Topics: Alcohol Drinking; Alkaloids; Animals; Azocines; Benzazepines; Male; Mice; Mice, Inbred C57BL; Nicotinic Agonists; Quinolizines; Quinoxalines; Varenicline

2013
Differential modulation of brain nicotinic acetylcholine receptor function by cytisine, varenicline, and two novel bispidine compounds: emergent properties of a hybrid molecule.
    The Journal of pharmacology and experimental therapeutics, 2013, Volume: 347, Issue:2

    Topics: Alkaloids; Animals; Azocines; Behavior, Animal; Benzazepines; Brain; Bridged Bicyclo Compounds, Heterocyclic; Dose-Response Relationship, Drug; Drug Partial Agonism; HEK293 Cells; Humans; Male; Membrane Potentials; Mice; Molecular Structure; Nicotinic Agonists; Oocytes; Patch-Clamp Techniques; Quinolizines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Tobacco Use Disorder; Varenicline; Xenopus laevis

2013
Varenicline and cytisine diminish the dysphoric-like state associated with spontaneous nicotine withdrawal in rats.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2014, Volume: 39, Issue:2

    Topics: Alkaloids; Animals; Azocines; Benzazepines; Infusion Pumps, Implantable; Male; Nicotine; Nicotinic Agonists; Quinolizines; Quinoxalines; Rats; Rats, Wistar; Substance Withdrawal Syndrome; Varenicline

2014
[Safety of nicotine addiction treatment].
    Przeglad lekarski, 2013, Volume: 70, Issue:10

    Topics: Abdominal Pain; Adult; Alkaloids; Azocines; Benzazepines; Boredom; Bupropion; Female; Headache; Humans; Male; Middle Aged; Nicotine; Patient Compliance; Quinolizines; Quinoxalines; Sleep Wake Disorders; Smoking Cessation; Tobacco Use Disorder; Varenicline; Xerostomia

2013
Efficient expression of functional (α6β2)2β3 AChRs in Xenopus oocytes from free subunits using slightly modified α6 subunits.
    PloS one, 2014, Volume: 9, Issue:7

    Topics: Acetylcholine; Alkaloids; Animals; Atropine; Azocines; Cholinergic Agonists; Female; Gene Expression; Humans; Membrane Potentials; Nicotine; Nicotinic Agonists; Oocytes; Patch-Clamp Techniques; Quinolizines; Receptors, Nicotinic; Recombinant Fusion Proteins; Varenicline; Xenopus laevis

2014
Neuronal Nicotinic Acetylcholine Receptor Modulators Reduce Sugar Intake.
    PloS one, 2016, Volume: 11, Issue:3

    Topics: Alkaloids; Animals; Azocines; Drug Evaluation, Preclinical; Food Preferences; Male; Mecamylamine; Nicotinic Agonists; Nicotinic Antagonists; Nucleus Accumbens; Quinolizines; Rats, Wistar; Receptors, Nicotinic; Sucrose; Varenicline

2016
The contribution of α4β2 and non-α4β2 nicotinic acetylcholine receptors to the discriminative stimulus effects of nicotine and varenicline in mice.
    Psychopharmacology, 2017, Volume: 234, Issue:5

    Topics: Aconitine; Alkaloids; alpha7 Nicotinic Acetylcholine Receptor; Animals; Azocines; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cocaine; Dihydro-beta-Erythroidine; Discrimination, Psychological; Dopamine Uptake Inhibitors; Hypnotics and Sedatives; Ibogaine; Male; Mecamylamine; Mice; Mice, Inbred C57BL; Midazolam; Nerve Tissue Proteins; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Pyridines; Quinolizines; Receptors, Nicotinic; Varenicline

2017
Differential cross-tolerance to the effects of nicotinic acetylcholine receptor drugs in C57BL/6J mice following chronic varenicline.
    Behavioural pharmacology, 2019, Volume: 30, Issue:5

    Topics: Alkaloids; Animals; Azocines; Bridged Bicyclo Compounds, Heterocyclic; Cocaine; Conditioning, Operant; Drug Tolerance; Female; Male; Mice; Mice, Inbred C57BL; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Pyridines; Quinolizines; Receptors, Nicotinic; Reinforcement, Psychology; Smoking Cessation; Varenicline

2019
Revisiting autosomal dominant nocturnal frontal lobe epilepsy (ADNFLE) mutations in the nicotinic acetylcholine receptor reveal an increase in efficacy regardless of stochiometry.
    Pharmacological research, 2019, Volume: 139

    Topics: Acetylcholine; Alkaloids; Animals; Azocines; Epilepsy, Frontal Lobe; Female; Mutation; Nicotine; Nicotinic Agonists; Oocytes; Quinolizines; Receptors, Nicotinic; Varenicline; Xenopus laevis

2019
The Effect of Cytisine vs Varenicline on Smoking Cessation-Reply.
    JAMA, 2021, 11-09, Volume: 326, Issue:18

    Topics: Alkaloids; Azocines; Quinolizines; Smoking Cessation; Varenicline

2021
The Effect of Cytisine vs Varenicline on Smoking Cessation.
    JAMA, 2021, 11-09, Volume: 326, Issue:18

    Topics: Alkaloids; Azocines; Quinolizines; Smoking Cessation; Varenicline

2021
Cytisine induced urticaria : a case report during a smoking cessation treatment.
    Acta bio-medica : Atenei Parmensis, 2022, 06-22, Volume: 93, Issue:S1

    Topics: Alkaloids; Azocines; Capsules; Female; Humans; Quinolizines; Smoking Cessation; Urticaria; Varenicline

2022
Could APO-varenicline and cytisine be solutions for the shortage of varenicline in Brazil?
    Jornal brasileiro de pneumologia : publicacao oficial da Sociedade Brasileira de Pneumologia e Tisilogia, 2023, 06-05, Volume: 49, Issue:3

    Topics: Alkaloids; Brazil; Humans; Smoking Cessation; Varenicline

2023
Nicotine and Cytisine Embryotoxicity in the Experimental Zebrafish Model.
    International journal of molecular sciences, 2023, Jul-28, Volume: 24, Issue:15

    Topics: Alkaloids; Animals; Azocines; Benzazepines; Humans; Nicotine; Nicotinic Agonists; Quinolizines; Quinoxalines; Receptors, Nicotinic; Varenicline; Zebrafish

2023
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