cysteine and monastrol

cysteine has been researched along with monastrol in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's6 (66.67)29.6817
2010's3 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Brier, S; Debonis, S; Forest, E; Kozielski, F; Lemaire, D2
Bernhardt, G; Buschauer, A; Gartner, M; Giannis, A; Gross, D; Müller, C; Sarli, V1
Kropf, DL; Peters, NT1
Filatova, IS; Planas-Silva, MD1
Chen, Y; Jiang, C; Wang, X; You, Q1
Kozielski, F; Skoufias, DA; Tcherniuk, S; van Lis, R1
Kim, S; Liu, J; Liu, L; Parameswaran, S; Wojcik, EJ1
Bolte, S; Buffin, E; Cladière, D; El Yakoubi, W; Leontiou, I; Vallot, A; Wassmann, K1

Other Studies

9 other study(ies) available for cysteine and monastrol

ArticleYear
Identification of the protein binding region of S-trityl-L-cysteine, a new potent inhibitor of the mitotic kinesin Eg5.
    Biochemistry, 2004, Oct-19, Volume: 43, Issue:41

    Topics: Adenosine Triphosphatases; Amino Acid Sequence; Antineoplastic Agents; Cysteine; Deuterium Exchange Measurement; Genetic Vectors; Growth Inhibitors; Humans; Kinesins; Mitosis; Molecular Motor Proteins; Molecular Sequence Data; Neurospora crassa; Peptide Fragments; Protein Binding; Protein Structure, Tertiary; Pyrimidines; Spectrometry, Mass, Electrospray Ionization; Thiones

2004
Inhibitors of kinesin Eg5: antiproliferative activity of monastrol analogues against human glioblastoma cells.
    Cancer chemotherapy and pharmacology, 2007, Volume: 59, Issue:2

    Topics: Acridines; Antineoplastic Agents, Phytogenic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line, Tumor; Cell Proliferation; Cell Survival; Cysteine; Dose-Response Relationship, Drug; Flow Cytometry; Fluoresceins; Glioblastoma; Humans; Insecticides; Kinesins; Molecular Structure; Paclitaxel; Pyrimidines; Quinazolines; Rotenone; Spindle Apparatus; Tetrahydroisoquinolines; Thiones; Time Factors; Tubulin; Tubulin Modulators; Vinblastine

2007
Molecular dissection of the inhibitor binding pocket of mitotic kinesin Eg5 reveals mutants that confer resistance to antimitotic agents.
    Journal of molecular biology, 2006, Jul-07, Volume: 360, Issue:2

    Topics: Amino Acid Sequence; Antimitotic Agents; Binding Sites; Cysteine; Drug Resistance; Kinesins; Kinetics; Mass Spectrometry; Mitosis; Models, Molecular; Molecular Sequence Data; Mutagenesis; Point Mutation; Protein Binding; Pyrimidines; Thiones

2006
Kinesin-5 motors are required for organization of spindle microtubules in Silvetia compressa zygotes.
    BMC plant biology, 2006, Aug-31, Volume: 6

    Topics: Cell Polarity; Cysteine; Cytokinesis; Dinitrobenzenes; Kinesins; Microtubules; Mitosis; Molecular Motor Proteins; Paclitaxel; Phaeophyceae; Pyrimidines; Spindle Apparatus; Sulfanilamides; Thiones; Zygote

2006
Estrogen-dependent regulation of Eg5 in breast cancer cells.
    Anti-cancer drugs, 2007, Volume: 18, Issue:7

    Topics: Blotting, Western; Breast Neoplasms; Cell Cycle; Cell Line, Tumor; Cysteine; Dose-Response Relationship, Drug; Down-Regulation; Estradiol; Estrogen Antagonists; Estrogens; Female; Flow Cytometry; Fulvestrant; Humans; Inhibitory Concentration 50; Kinesins; Mitosis; Pyrimidines; Receptors, Estrogen; Signal Transduction; Thiones; Up-Regulation

2007
Docking studies on kinesin spindle protein inhibitors: an important cooperative 'minor binding pocket' which increases the binding affinity significantly.
    Journal of molecular modeling, 2007, Volume: 13, Issue:9

    Topics: Amino Acid Sequence; Amino Acids; Cysteine; Diterpenes; Hydrogen Bonding; Indoles; Kinesins; Models, Molecular; Phenols; Protein Binding; Pyrimidines; Spindle Apparatus; Thiones

2007
Mutations in the human kinesin Eg5 that confer resistance to monastrol and S-trityl-L-cysteine in tumor derived cell lines.
    Biochemical pharmacology, 2010, Mar-15, Volume: 79, Issue:6

    Topics: Antineoplastic Agents; Binding Sites; Cysteine; Drug Resistance; Humans; Inhibitory Concentration 50; Kinesins; Models, Molecular; Mutation; Protein Binding; Pyrimidines; Thiones

2010
Loop 5-directed compounds inhibit chimeric kinesin-5 motors: implications for conserved allosteric mechanisms.
    The Journal of biological chemistry, 2011, Feb-25, Volume: 286, Issue:8

    Topics: Allosteric Regulation; Animals; Cysteine; Drosophila melanogaster; Drosophila Proteins; Humans; Kinesins; Microtubule-Associated Proteins; Protein Binding; Protein Structure, Secondary; Protein Structure, Tertiary; Pyrimidines; Recombinant Fusion Proteins; Thiones

2011
Tension-Induced Error Correction and Not Kinetochore Attachment Status Activates the SAC in an Aurora-B/C-Dependent Manner in Oocytes.
    Current biology : CB, 2018, 01-08, Volume: 28, Issue:1

    Topics: Animals; Cell Division; Cysteine; Female; Kinesins; Kinetochores; M Phase Cell Cycle Checkpoints; Meiosis; Mice; Oocytes; Paclitaxel; Pyrimidines; Thiones; Tubulin Modulators

2018