cysteine and imatinib mesylate

cysteine has been researched along with imatinib mesylate in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (40.00)29.6817
2010's3 (60.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lagonigro, MS; Miselli, F; Negri, T; Pilotti, S; Pricl, S; Tamborini, E1
Angelo, LS; Kohanim, S; Kurzrock, R; Wu, JY; Yang, DJ1
Barluenga, S; Leproult, E; Moras, D; Winssinger, N; Wurtz, JM1
Dong, B; Huang, H; Qu, L; Weng, H; Zhao, P; Zhou, H1
Adam, T; Faber, E; Friedecký, D; Karlíková, R; Mičová, K; Najdekr, L; Vrobel, I1

Other Studies

5 other study(ies) available for cysteine and imatinib mesylate

ArticleYear
Re: Response of a KIT-positive extra-abdominal fibromatosis to imatinib mesylate and KIT genetic analysis.
    Journal of the National Cancer Institute, 2006, Nov-01, Volume: 98, Issue:21

    Topics: Alanine; Antineoplastic Agents; Benzamides; Biomarkers, Tumor; Cysteine; Fibroma; Humans; Imatinib Mesylate; Leucine; Methionine; Mutagenesis; Mutation; Piperazines; Polymorphism, Genetic; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-kit; Pyrimidines; Treatment Outcome

2006
Molecular imaging of Bcr-Abl phosphokinase in a xenograft model.
    Molecular cancer therapeutics, 2009, Volume: 8, Issue:3

    Topics: Animals; Antibodies; Benzamides; Cysteine; Female; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Indium Radioisotopes; K562 Cells; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Mice; Mice, Nude; Phosphotyrosine; Piperazines; Protein-Tyrosine Kinases; Pyrimidines; Radioimmunodetection; Tumor Burden; Xenograft Model Antitumor Assays

2009
Cysteine mapping in conformationally distinct kinase nucleotide binding sites: application to the design of selective covalent inhibitors.
    Journal of medicinal chemistry, 2011, Mar-10, Volume: 54, Issue:5

    Topics: Adenosine Triphosphate; Benzamides; Catalytic Domain; Cysteine; Drug Design; Humans; Imatinib Mesylate; Models, Molecular; Piperazines; Protein Conformation; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-abl; Proto-Oncogene Proteins c-kit; Pyrimidines; Receptor, Platelet-Derived Growth Factor alpha; Structure-Activity Relationship

2011
Oridonin Triggers Chaperon-mediated Proteasomal Degradation of BCR-ABL in Leukemia.
    Scientific reports, 2017, 01-27, Volume: 7

    Topics: Antineoplastic Agents; Apoptosis; Base Sequence; Cell Line, Tumor; Cell Proliferation; Cysteine; Diterpenes, Kaurane; Drug Resistance, Neoplasm; Fusion Proteins, bcr-abl; Gene Deletion; Heat Shock Transcription Factors; HL-60 Cells; HSP70 Heat-Shock Proteins; Humans; Imatinib Mesylate; K562 Cells; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Models, Biological; Molecular Chaperones; Oxidation-Reduction; Proteasome Endopeptidase Complex; Proteolysis; Ubiquitin

2017
Novel sulphur-containing imatinib metabolites found by untargeted LC-HRMS analysis.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2017, Jun-15, Volume: 104

    Topics: Antineoplastic Agents; Chromatography, Liquid; Cysteine; Cystine; Humans; Imatinib Mesylate; Protein Kinase Inhibitors; Sulfur; Tandem Mass Spectrometry

2017