Page last updated: 2024-08-21

cyproterone acetate and nilutamide

cyproterone acetate has been researched along with nilutamide in 29 studies

Research

Studies (29)

TimeframeStudies, this research(%)All Research%
pre-199011 (37.93)18.7374
1990's9 (31.03)18.2507
2000's7 (24.14)29.6817
2010's2 (6.90)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Schröder, FH2
Bolt, J; Mulder, E; Schuurmans, AL; Veldscholte, J1
Namer, M1
Furr, BJ2
Daricello, G; Pavone, C; Pavone-Macaluso, M; Romano, C; Serretta, V1
de Jong, FH; Lamberts, SW; Uitterlinden, P1
Ayub, M; Levell, MJ1
Dupront, A; Meyer, BH; Pottier, J; Tremblay, D1
Bouman, FG; de Voogt, HJ; Geldof, AA; Gooren, LJ; Rao, BR1
Bruchovsky, N; Fletcher, T; Foekens, JA; Goldenberg, SL; Lawson, D; Rennie, PS1
Abreu, LC; Hayashi, H; Picarelli, ZP; Porto, CS1
Brown, TR; Migeon, CJ; Rothwell, SW; Sultan, C1
Govindan, MV; Koutsilieris, M; Pagé, N; Warriar, N2
McLeod, DG1
Matzkin, H; Soloway, MS1
Benassayag, E1
Bonnet, P1
Candas, B; Labrie, F1
Collette, L; Denis, LJ; Schröder, FH; Studer, UE; Sylvester, RJ1
Cardi, A; Di Silverio, F; Sciarra, A1
Baltogiannis, D; Charalabopoulos, K; Giannakopoulos, X; Sofikitis, N1
Debré, B; Delongchamps, NB; Peyromaure, M; Zerbib, M1
Hara, S; Hyochi, N; Isaacs, JT; Ishioka, J; Kageyama, Y; Kihara, K; Singh, P; Urushibara, M1
Bastide, C; Bruyère, F; Guy, L; Karsenty, G; Rozet, F1

Reviews

9 review(s) available for cyproterone acetate and nilutamide

ArticleYear
Pure antiandrogens as monotherapy in prospective studies of prostatic carcinoma.
    Progress in clinical and biological research, 1990, Volume: 359

    Topics: Androgen Antagonists; Anilides; Animals; Cyproterone; Cyproterone Acetate; Flutamide; Humans; Imidazoles; Imidazolidines; Male; Nitriles; Prospective Studies; Prostatic Neoplasms; Tosyl Compounds

1990
Clinical applications of antiandrogens.
    Journal of steroid biochemistry, 1988, Volume: 31, Issue:4B

    Topics: Androgen Antagonists; Breast Neoplasms; Cyproterone; Cyproterone Acetate; Female; Flutamide; Humans; Imidazoles; Imidazolidines; Male; Prostatic Hyperplasia; Prostatic Neoplasms; Puberty, Precocious; Skin Diseases; Spironolactone

1988
Antiandrogenic drugs.
    Cancer, 1993, Feb-01, Volume: 71, Issue:3 Suppl

    Topics: Androgen Receptor Antagonists; Anilides; Cyproterone Acetate; Diethylstilbestrol; Drug Administration Schedule; Flutamide; Humans; Imidazoles; Imidazolidines; Male; Megestrol; Megestrol Acetate; Nitriles; Prostatic Neoplasms; Randomized Controlled Trials as Topic; Tosyl Compounds

1993
Antiandrogenic agents as monotherapy in advanced prostatic carcinoma.
    Cancer, 1993, Feb-01, Volume: 71, Issue:3 Suppl

    Topics: Androgen Antagonists; Anilides; Antineoplastic Agents; Cyproterone Acetate; Flutamide; Humans; Imidazoles; Imidazolidines; Male; Neoplasm Staging; Nitriles; Prognosis; Prostatic Neoplasms; Testosterone; Tosyl Compounds

1993
The place and the results of monotherapy.
    Acta urologica Belgica, 1998, Volume: 66, Issue:2

    Topics: Androgen Antagonists; Anilides; Antineoplastic Agents; Antineoplastic Agents, Hormonal; Cyproterone Acetate; Flutamide; Humans; Imidazoles; Imidazolidines; Male; Nitriles; Prostatic Neoplasms; Tosyl Compounds

1998
Antiandrogens as monotherapy for prostate cancer.
    European urology, 1998, Volume: 34 Suppl 3

    Topics: Androgen Antagonists; Anilides; Antineoplastic Agents; Antineoplastic Agents, Hormonal; Cyproterone Acetate; Flutamide; Humans; Imidazoles; Imidazolidines; Male; Nitriles; Prostatic Neoplasms; Tosyl Compounds

1998
Antiandrogen monotherapy: recommendations for the treatment of prostate cancer.
    Urologia internationalis, 2004, Volume: 72, Issue:2

    Topics: Androgen Antagonists; Anilides; Chemotherapy, Adjuvant; Cyproterone Acetate; Flutamide; Humans; Imidazoles; Imidazolidines; Male; Nitriles; Orchiectomy; Prostatic Neoplasms; Quality of Life; Randomized Controlled Trials as Topic; Tosyl Compounds

2004
Monotherapy in advanced prostate cancer: an overview.
    Experimental oncology, 2004, Volume: 26, Issue:3

    Topics: Adenocarcinoma; Androgen Antagonists; Anilides; Antineoplastic Agents, Hormonal; Combined Modality Therapy; Cyproterone Acetate; Dihydrotestosterone; Estrogens; Flutamide; Gonadotropin-Releasing Hormone; Humans; Imidazolidines; Male; Nitriles; Orchiectomy; Palliative Care; Progesterone Congeners; Prostatic Neoplasms; Randomized Controlled Trials as Topic; Testosterone; Tosyl Compounds

2004
[Hormonal treatment in prostate cancer].
    Progres en urologie : journal de l'Association francaise d'urologie et de la Societe francaise d'urologie, 2013, Volume: 23, Issue:15

    Topics: Androgen Antagonists; Androgen Receptor Antagonists; Antineoplastic Agents, Hormonal; Benzamides; Combined Modality Therapy; Cyproterone Acetate; Diethylstilbestrol; Estramustine; Estrogens, Non-Steroidal; Flutamide; Gonadotropin-Releasing Hormone; Humans; Imidazolidines; Male; Neoplasm Metastasis; Neoplasms, Hormone-Dependent; Nitriles; Oligopeptides; Phenylthiohydantoin; Prostatectomy; Prostatic Neoplasms

2013

Trials

2 trial(s) available for cyproterone acetate and nilutamide

ArticleYear
Pure antiandrogens as monotherapy in prospective studies of prostatic carcinoma.
    Progress in clinical and biological research, 1990, Volume: 359

    Topics: Androgen Antagonists; Anilides; Animals; Cyproterone; Cyproterone Acetate; Flutamide; Humans; Imidazoles; Imidazolidines; Male; Nitriles; Prospective Studies; Prostatic Neoplasms; Tosyl Compounds

1990
[Indications of antiandrogens in benign hyperplasia of the prostate].
    Journal d'urologie, 1995, Volume: 101, Issue:2

    Topics: Aged; Aged, 80 and over; Androgen Antagonists; Cyproterone Acetate; Flutamide; Humans; Imidazoles; Imidazolidines; Male; Middle Aged; Prostatic Hyperplasia

1995

Other Studies

19 other study(ies) available for cyproterone acetate and nilutamide

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Stimulatory effects of antiandrogens on LNCaP human prostate tumor cell growth, EGF-receptor level and acid phosphatase secretion.
    The Journal of steroid biochemistry and molecular biology, 1990, Dec-20, Volume: 37, Issue:6

    Topics: Acid Phosphatase; Androgen Antagonists; Antineoplastic Agents; Cyproterone; Cyproterone Acetate; ErbB Receptors; Estradiol; Humans; Imidazoles; Imidazolidines; Male; Prostatic Neoplasms; Tumor Cells, Cultured

1990
"Casodex" (ICI 176,334)--a new, pure, peripherally-selective anti-androgen: preclinical studies.
    Hormone research, 1989, Volume: 32 Suppl 1

    Topics: Androgen Antagonists; Anilides; Animals; Cyproterone; Cyproterone Acetate; Dogs; Flutamide; Imidazoles; Imidazolidines; Male; Nitriles; Prostatic Neoplasms; Rats; Tosyl Compounds

1989
[Antiandrogens in monotherapy or combined therapy for treatment of advanced cancer of the prostate].
    Archivos espanoles de urologia, 1989, Volume: 42 Suppl 2

    Topics: Aged; Aged, 80 and over; Androgen Antagonists; Anilides; Antineoplastic Agents; Combined Modality Therapy; Cyproterone; Cyproterone Acetate; Flutamide; Follow-Up Studies; Humans; Imidazoles; Imidazolidines; Male; Middle Aged; Neoplasm Staging; Nitriles; Orchiectomy; Prostatic Neoplasms; Tosyl Compounds

1989
Rat prostatic weight regression in reaction to ketoconazole, cyproterone acetate, and RU 23908 as adjuncts to a depot formulation of gonadotropin-releasing hormone analogue.
    Cancer research, 1988, Nov-01, Volume: 48, Issue:21

    Topics: Adrenocorticotropic Hormone; Animals; Buserelin; Cyproterone; Cyproterone Acetate; Delayed-Action Preparations; Goserelin; Imidazoles; Imidazolidines; Ketoconazole; Luteinizing Hormone; Male; Orchiectomy; Organ Size; Prostate; Prostatic Neoplasms; Rats; Rats, Inbred Strains

1988
Inhibition of rat testicular 17 alpha-hydroxylase and 17,20-lyase activities by anti-androgens (flutamide, hydroxyflutamide, RU23908, cyproterone acetate) in vitro.
    Journal of steroid biochemistry, 1987, Volume: 28, Issue:1

    Topics: Aldehyde-Lyases; Androgen Antagonists; Animals; Cyproterone; Cyproterone Acetate; Cytochrome P-450 Enzyme System; Flutamide; Imidazoles; Imidazolidines; Kinetics; Male; Microsomes; Rats; Rats, Inbred Strains; Steroid 17-alpha-Hydroxylase; Steroid Hydroxylases; Testis

1987
The kinetics of antiandrogens in humans.
    Progress in clinical and biological research, 1987, Volume: 243A

    Topics: Androgen Antagonists; Anilides; Cyproterone; Cyproterone Acetate; Flutamide; Humans; Imidazoles; Imidazolidines; Male; Prostatic Neoplasms

1987
Androgen action blockade does not result in reduction in size but changes histology of the normal human prostate.
    The Prostate, 1987, Volume: 11, Issue:4

    Topics: Adult; Androgen Antagonists; Cyproterone; Cyproterone Acetate; Ethinyl Estradiol; Follicle Stimulating Hormone; Humans; Imidazoles; Imidazolidines; Luteinizing Hormone; Male; Prolactin; Prostate; Testosterone

1987
ICI 176,334: a novel non-steroidal, peripherally-selective antiandrogen.
    Progress in clinical and biological research, 1988, Volume: 260

    Topics: Androgen Antagonists; Anilides; Animals; Cyproterone; Cyproterone Acetate; Dogs; Flutamide; Imidazoles; Imidazolidines; Male; Nitriles; Prostate; Radioligand Assay; Rats; Receptors, Androgen; Seminal Vesicles; Testosterone; Tosyl Compounds

1988
Relative effectiveness of alternative androgen withdrawal therapies in initiating regression of rat prostate.
    The Journal of urology, 1988, Volume: 139, Issue:6

    Topics: Anilides; Animals; Cyproterone; Cyproterone Acetate; Diethylstilbestrol; Dihydrotestosterone; Flutamide; Gonadotropin-Releasing Hormone; Imidazoles; Imidazolidines; Leuprolide; Male; Megestrol; Megestrol Acetate; Orchiectomy; Prostate; Rats; Rats, Inbred Strains; Receptors, Androgen

1988
Effects of castration and antiandrogens (RU 23908 and cyproterone acetate) on glandulain activity and on the secretory epithelium of the rat submandibular gland.
    Brazilian journal of medical and biological research = Revista brasileira de pesquisas medicas e biologicas, 1988, Volume: 21, Issue:3

    Topics: Aminopeptidases; Androgen Antagonists; Animals; Cyproterone; Cyproterone Acetate; Imidazoles; Imidazolidines; Male; Orchiectomy; Rats; Sex Characteristics; Submandibular Gland

1988
Inhibition of androgen binding in human foreskin fibroblasts by antiandrogens.
    Steroids, 1981, Volume: 37, Issue:6

    Topics: Androgen Antagonists; Androgens; Binding, Competitive; Cyproterone; Cyproterone Acetate; Dihydrotestosterone; Estrenes; Fibroblasts; Humans; Imidazoles; Imidazolidines; Infant, Newborn; Male; Metribolone; Penis; Receptors, Androgen; Receptors, Steroid; Subcellular Fractions; Testosterone

1981
Antiandrogens inhibit human androgen receptor-dependent gene transcription activation in the human prostate cancer cells LNCaP.
    The Prostate, 1994, Volume: 24, Issue:4

    Topics: Amino Acid Sequence; Androgen Antagonists; Binding, Competitive; Blotting, Western; Chloramphenicol O-Acetyltransferase; Cyproterone Acetate; Dihydrotestosterone; Dose-Response Relationship, Drug; Flutamide; Gene Expression Regulation, Viral; Humans; Imidazoles; Imidazolidines; Male; Mammary Tumor Virus, Mouse; Molecular Sequence Data; Promoter Regions, Genetic; Prostatic Neoplasms; Receptors, Androgen; Transcription, Genetic; Transfection; Tumor Cells, Cultured

1994
Interaction of antiandrogen-androgen receptor complexes with DNA and transcription activation.
    The Journal of steroid biochemistry and molecular biology, 1993, Volume: 46, Issue:6

    Topics: Androgen Antagonists; Animals; Binding, Competitive; Blotting, Western; Cell Line; Chloramphenicol O-Acetyltransferase; Chlorocebus aethiops; Cyproterone Acetate; Dihydrotestosterone; DNA; Flutamide; Gene Expression Regulation; Humans; Imidazoles; Imidazolidines; Kidney; Kinetics; Mammary Tumor Virus, Mouse; Metribolone; Receptors, Androgen; Recombinant Proteins; Transcription Factors; Transcription, Genetic; Transcriptional Activation; Transfection

1993
Androgen blockade in prostate cancer.
    Lancet (London, England), 2000, Jul-22, Volume: 356, Issue:9226

    Topics: Androgen Antagonists; Cyproterone Acetate; Flutamide; Humans; Imidazoles; Imidazolidines; Male; Meta-Analysis as Topic; Orchiectomy; Prostatic Neoplasms

2000
Why phase III trials of maximal androgen blockade versus castration in M1 prostate cancer rarely show statistically significant differences.
    The Prostate, 2001, Jun-15, Volume: 48, Issue:1

    Topics: Androgen Antagonists; Anilides; Clinical Trials, Phase III as Topic; Cyproterone Acetate; Factor Analysis, Statistical; Flutamide; Gonadotropin-Releasing Hormone; Goserelin; Humans; Imidazoles; Imidazolidines; Leuprolide; Male; Meta-Analysis as Topic; Nitriles; Orchiectomy; Prognosis; Prostatic Neoplasms; Research Design; Survival Analysis; Tosyl Compounds; Treatment Outcome

2001
Intermittent androgen deprivation for biologic recurrence after radical prostatectomy: long-term experience.
    Urology, 2005, Volume: 65, Issue:4

    Topics: Aged; Androgen Antagonists; Cyproterone Acetate; Follow-Up Studies; Humans; Imidazolidines; Male; Middle Aged; Neoplasm Recurrence, Local; Prostatectomy; Prostatic Neoplasms; Time Factors

2005
Effects of steroidal and non-steroidal antiandrogens on wild-type and mutant androgen receptors.
    The Prostate, 2007, Jun-01, Volume: 67, Issue:8

    Topics: Allylestrenol; Androgen Antagonists; Androgen Receptor Antagonists; Androgens; Anilides; Cyproterone Acetate; Flutamide; Humans; Imidazolidines; Male; Models, Molecular; Mutagenesis, Site-Directed; Neoplasms, Hormone-Dependent; Nitriles; Plasmids; Prostate-Specific Antigen; Prostatic Neoplasms; Receptors, Androgen; Reverse Transcriptase Polymerase Chain Reaction; RNA, Neoplasm; Testosterone; Tosyl Compounds; Transcription, Genetic; Transfection

2007