Page last updated: 2024-08-21

cyproterone acetate and mifepristone

cyproterone acetate has been researched along with mifepristone in 20 studies

Research

Studies (20)

TimeframeStudies, this research(%)All Research%
pre-19902 (10.00)18.7374
1990's6 (30.00)18.2507
2000's9 (45.00)29.6817
2010's2 (10.00)24.3611
2020's1 (5.00)2.80

Authors

AuthorsStudies
Edwards, JP; Farmer, LJ; Hamann, LG; Higuchi, RI; Jones, TK; Kong, JW; Marschke, KB; Wang, XN; Zhi, L1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Mercier, L; Miller, PA; Simons, SS1
Baulieu, EE; Jung-Testas, I1
Aso, T; Kubota, T; Taguchi, M1
Sar, M; Wilson, EM; Wong, CI; Zhou, ZX1
Gurpide, E; Markiewicz, L1
Chang, C; Miyamoto, H; Wilding, G; Yeh, S1
Rai, U1
Chatelain, RE; Cornell, W; Fink, C; Honer, C; Ksander, G; Marshall, P; Nam, K; Schumacher, C; Schweitzer, R; Steele, R1
Berrevoets, CA; Brinkmann, AO; Trapman, J; Umar, A1
Bass, AH; Remage-Healey, L1
Jänne, OA; Kang, Z; Palvimo, JJ1
MacBride, MM; Muddana, SS; Peterson, BR; Price, AM1
Chang, CY; Elbi, C; Hager, GL; Hendarwanto, A; Klokk, TI; Kurys, P; Nagaich, AK; Saatcioglu, F; Slagsvold, T1
De Rosier, T; Eliason, HC; Ervin, KM; Gowda, K; Kupcho, KR; Marks, BD; Ozers, MS; Qadir, N; Riddle, SM; Shekhani, MS1
Buijs, JT; Culig, Z; Grimm, S; Hemmer, DM; Hwang, MS; Kroon, J; Marijt, KA; Masood, M; Meijer, OC; Metselaar, JM; Puhr, M; Storm, G; van der Horst, G; van der Pluijm, G1
Kang, C; Kim, S; Kwon, Y; Lee, DY; Lee, E; Lee, M; Park, S; Ryu, J1

Other Studies

20 other study(ies) available for cyproterone acetate and mifepristone

ArticleYear
Synthesis and biological activity of a novel series of nonsteroidal, peripherally selective androgen receptor antagonists derived from 1,2-dihydropyridono[5,6-g]quinolines.
    Journal of medicinal chemistry, 1998, Feb-12, Volume: 41, Issue:4

    Topics: Androgen Antagonists; Androgen Receptor Antagonists; Animals; Cell Line; COS Cells; Dihydropyridines; Dihydrotestosterone; Gonadotropins; Heterocyclic Compounds; Humans; Indicators and Reagents; Male; Molecular Structure; Orchiectomy; Prostate; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Androgen; Receptors, Progesterone; Recombinant Proteins; Seminal Vesicles; Structure-Activity Relationship; Testosterone; Transfection

1998
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Antiglucocorticoid steroids have increased agonist activity in those hepatoma cell lines that are more sensitive to glucocorticoids.
    Journal of steroid biochemistry, 1986, Volume: 25, Issue:1

    Topics: Animals; Cell Line; Cyproterone; Cyproterone Acetate; Dexamethasone; Enzyme Induction; Estrenes; Glucocorticoids; Glutamate-Ammonia Ligase; Liver Neoplasms, Experimental; Mifepristone; Rats; Receptors, Glucocorticoid; Tyrosine Transaminase

1986
Effects of steroid hormones and antihormones in cultured cells.
    Experimental and clinical endocrinology, 1985, Volume: 86, Issue:2

    Topics: Animals; Cell Division; Cells, Cultured; Cyproterone; Cyproterone Acetate; Dexamethasone; Diethylstilbestrol; Dihydrotestosterone; Estradiol; Estrenes; Glucocorticoids; Gonadal Steroid Hormones; L Cells; Mammary Neoplasms, Experimental; Mice; Mifepristone; Receptors, Androgen; Receptors, Estrogen; Receptors, Glucocorticoid; Tamoxifen; Thymoma

1985
Direct effect of danazol on the DNA synthesis and ultrastructure of human cultured endometrial stromal cells.
    Gynecologic and obstetric investigation, 1995, Volume: 39, Issue:3

    Topics: Cells, Cultured; Cyproterone Acetate; Cytoplasm; Cytoskeleton; Danazol; DNA; Endometrium; Female; Humans; Microscopy, Electron; Mifepristone; Organelles; Stromal Cells; Time Factors

1995
Steroid requirement for androgen receptor dimerization and DNA binding. Modulation by intramolecular interactions between the NH2-terminal and steroid-binding domains.
    The Journal of biological chemistry, 1993, Sep-05, Volume: 268, Issue:25

    Topics: Androgens; Animals; Baculoviridae; Base Sequence; Binding Sites; Cell Line; Cyproterone Acetate; DNA; Flutamide; Genetic Vectors; Humans; Macromolecular Substances; Mifepristone; Molecular Sequence Data; Moths; Receptors, Androgen; Recombinant Proteins; Transfection

1993
Estrogenic and progestagenic activities of physiologic and synthetic androgens, as measured by in vitro bioassays.
    Methods and findings in experimental and clinical pharmacology, 1997, Volume: 19, Issue:4

    Topics: Adenocarcinoma; Alkaline Phosphatase; Androgen Antagonists; Androgens; Breast Neoplasms; Cyproterone Acetate; Endometrial Neoplasms; Estradiol; Estrogen Antagonists; Female; Flutamide; Gonanes; Humans; Mifepristone; Polyunsaturated Alkamides; Progestins; Tamoxifen; Testosterone; Testosterone Congeners; Tumor Cells, Cultured

1997
Promotion of agonist activity of antiandrogens by the androgen receptor coactivator, ARA70, in human prostate cancer DU145 cells.
    Proceedings of the National Academy of Sciences of the United States of America, 1998, Jun-23, Volume: 95, Issue:13

    Topics: Androgen Antagonists; Androgens; Anilides; Cyproterone Acetate; Drug Interactions; Flutamide; Humans; Imidazoles; Male; Mifepristone; Nitriles; Nuclear Receptor Coactivators; Oncogene Proteins; Prostatic Neoplasms; Protein Binding; Protein Conformation; Tosyl Compounds; Trans-Activators; Transcription Factors; Transcriptional Activation; Tumor Cells, Cultured

1998
Sex steroid hormones modulate the activation of murine peritoneal macrophages: receptor mediated modulation.
    Comparative biochemistry and physiology. Part C, Pharmacology, toxicology & endocrinology, 1998, Volume: 119, Issue:2

    Topics: Animals; Castration; Cyproterone Acetate; Estradiol; Female; Flutamide; Gonadal Steroid Hormones; Lipopolysaccharides; Macrophage Activation; Macrophages, Peritoneal; Male; Mice; Mice, Inbred BALB C; Mifepristone; Nitrites; Progesterone; Receptors, Steroid; Tamoxifen; Testosterone

1998
Glucocorticoid receptor antagonism by cyproterone acetate and RU486.
    Molecular pharmacology, 2003, Volume: 63, Issue:5

    Topics: Androgen Antagonists; Animals; Cyproterone Acetate; Drug Delivery Systems; Humans; Ligands; Male; Mifepristone; Rats; Rats, Sprague-Dawley; Receptors, Glucocorticoid; Receptors, Progesterone

2003
Differential modulation of androgen receptor transcriptional activity by the nuclear receptor co-repressor (N-CoR).
    The Biochemical journal, 2004, May-01, Volume: 379, Issue:Pt 3

    Topics: Androgen Antagonists; Androgen Receptor Antagonists; Animals; Binding, Competitive; Cell Line, Tumor; CHO Cells; Cricetinae; Cyproterone Acetate; Down-Regulation; Gene Expression Regulation; Ligands; Male; Metribolone; Mice; Mifepristone; Mutation; Nuclear Proteins; Nuclear Receptor Co-Repressor 1; Nuclear Receptor Coactivator 2; Promoter Regions, Genetic; Prostatic Neoplasms; Receptors, Androgen; Repressor Proteins; Transcription Factors; Transcription, Genetic; Transfection

2004
Rapid, hierarchical modulation of vocal patterning by steroid hormones.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2004, Jun-30, Volume: 24, Issue:26

    Topics: Animals; Batrachoidiformes; Cyproterone Acetate; Estradiol; Gonadal Steroid Hormones; Hormone Antagonists; Hydrocortisone; Male; Mesencephalon; Mifepristone; Receptors, Steroid; Rhombencephalon; Spinal Cord; Testosterone; Vocalization, Animal

2004
Coregulator recruitment and histone modifications in transcriptional regulation by the androgen receptor.
    Molecular endocrinology (Baltimore, Md.), 2004, Volume: 18, Issue:11

    Topics: Acetylation; Androgen Receptor Antagonists; Anilides; Cell Line, Tumor; Chromatin Immunoprecipitation; Cyproterone Acetate; DNA Polymerase II; Enhancer Elements, Genetic; Gene Expression Regulation; Histones; Humans; Male; Methylation; Mifepristone; Nitriles; Nuclear Proteins; Nuclear Receptor Coactivator 2; Promoter Regions, Genetic; Prostate-Specific Antigen; Prostatic Neoplasms; Protein-Arginine N-Methyltransferases; Receptors, Androgen; Tissue Kallikreins; Tosyl Compounds; Trans-Activators; Transcription Factors; Transcription, Genetic

2004
11beta-alkyl-Delta9-19-nortestosterone derivatives: high-affinity ligands and potent partial agonists of the androgen receptor.
    Journal of medicinal chemistry, 2004, Oct-07, Volume: 47, Issue:21

    Topics: Androgen Antagonists; Androgen Receptor Antagonists; Androgens; Animals; Antineoplastic Agents; Cell Line, Tumor; CHO Cells; Cricetinae; Cyproterone Acetate; Dimerization; Humans; Ligands; Male; Mifepristone; Nandrolone; Prostatic Neoplasms; Receptors, Androgen; Structure-Activity Relationship

2004
Ligand-specific dynamics of the androgen receptor at its response element in living cells.
    Molecular and cellular biology, 2007, Volume: 27, Issue:5

    Topics: Adenocarcinoma; Androgen Antagonists; Androgens; Anilides; Animals; Cell Line, Tumor; Chromatin Assembly and Disassembly; Cyproterone Acetate; Dihydrotestosterone; Female; Fluorescence Recovery After Photobleaching; Flutamide; Genes, Reporter; Green Fluorescent Proteins; In Situ Hybridization, Fluorescence; Ligands; Luciferases; Mammary Neoplasms, Animal; Mammary Tumor Virus, Mouse; Metribolone; Mice; Microscopy, Video; Mifepristone; Models, Biological; Nitriles; Plasmids; Promoter Regions, Genetic; Receptors, Androgen; Response Elements; Testosterone; Tosyl Compounds; Transcription, Genetic

2007
The androgen receptor T877A mutant recruits LXXLL and FXXLF peptides differently than wild-type androgen receptor in a time-resolved fluorescence resonance energy transfer assay.
    Biochemistry, 2007, Jan-23, Volume: 46, Issue:3

    Topics: Amino Acid Sequence; Amino Acid Substitution; Androgen Antagonists; Anilides; Animals; Cyproterone Acetate; Dihydrotestosterone; Fluoresceins; Fluorescence Resonance Energy Transfer; Flutamide; Ligands; Mifepristone; Nitriles; Oligopeptides; Rats; Receptors, Androgen; Tosyl Compounds

2007
Glucocorticoid receptor antagonism reverts docetaxel resistance in human prostate cancer.
    Endocrine-related cancer, 2016, Volume: 23, Issue:1

    Topics: Apoptosis; Cyproterone Acetate; Docetaxel; Drug Resistance, Neoplasm; Drug Synergism; Gene Expression Regulation, Neoplastic; Hormone Antagonists; Humans; Male; Mifepristone; Prostatic Neoplasms; Receptors, Glucocorticoid; Taxoids; Tumor Cells, Cultured

2016
Rapid Screening of Glucocorticoid Receptor (GR) Effectors Using Cortisol-Detecting Sensor Cells.
    International journal of molecular sciences, 2021, Apr-29, Volume: 22, Issue:9

    Topics: Atrophy; Biosensing Techniques; Cyproterone Acetate; Dexamethasone; Drug Evaluation, Preclinical; Estradiol; Fluorescence Polarization; Fluorometry; HeLa Cells; Humans; Hydrocortisone; Inteins; Limonene; Luminescent Proteins; Mentha piperita; Menthol; Mifepristone; Molecular Structure; Muscle, Skeletal; Myoblasts; Oils, Volatile; Plant Oils; Protein Splicing; Protein Transport; Receptors, Glucocorticoid; Recombinant Fusion Proteins; Red Fluorescent Protein

2021