cyproheptadine and pizotyline

cyproheptadine has been researched along with pizotyline in 38 studies

Research

Studies (38)

TimeframeStudies, this research(%)All Research%
pre-199029 (76.32)18.7374
1990's5 (13.16)18.2507
2000's2 (5.26)29.6817
2010's2 (5.26)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Andrews, PR; Craik, DJ; Martin, JL1
Buescher, HH; Ebnöther, AM; Gadient, F; Hauser, D; Hill, RC; Huegi, BS; Petcher, TJ; Rissi, E; Roemer, D1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Agnoli, A; Carolei, A; Casacchia, M; Fazio, C; Zamponi, A1
Barnett, A; Malick, JB1
Apperley, E; Humphrey, PP; Levy, GP1
Colpaert, FC; Janssen, PA; Kuyps, JJ; Niemegeers, CJ1
Fozard, JR2
Dlabac, A; Metys, J; Metysová, J; Valchár, M1
Bille, B; Ludvigsson, J; Sanner, G1
Joost, HG1
Edvinsson, L; Hardebo, JE; Owman, C; Svendgaard, NA1
Hackaday, J1
Agostoni, A; Brandi, G; Cottino, A; Gai, V; Gastaldi, L; Lisino, F; Nattero, G2
May, B1
Klimek, A; Prusiński, A1
Dry, J; Perrault, M1
Ollat, H1
Eltze, M; Lambrecht, G; Mutschler, E1
Richards, MH1
Ekong, R; Pan, XQ; Peters, W; Robinson, BL; Warhurst, DC1
Bourin, M1
Kiesel, U; Kolb, H; Kolb-Bachofen, V; Martin, S1
Jeske, W; Kasperlik-Załuska, A; Migdalska, B; Sek, S; Wiśniewska-Woźniak, T1
Frycová, H; Metys, J1
Gorzalka, BB; Mendelson, SD1
Hiner, BC; Peroutka, SJ; Roth, HL1
Pan, XQ; Tong, XM; Zhou, MX1
Frycová, H; Metys, J; Soucek, R1
Anthony, M1
Hendry, JS; Minnema, DJ; Rosecrans, JA1
Fink, H; Gold, R; Morgenstern, R1
Freedman, M; Hamel, L; Luttinger, D; Perrone, M; Ward, SJ1
Abu-Arafeh, I; Russell, G; Symon, DN1
Bondareva, T; Glennon, RA; Khorana, N; Young, R1
Espinosa, EV; Karim, ZA; Khasawneh, FT; Lin, OA; Vemana, HP1

Reviews

5 review(s) available for cyproheptadine and pizotyline

ArticleYear
The animal pharmacology of drugs used in the treatment of migraine.
    The Journal of pharmacy and pharmacology, 1975, Volume: 27, Issue:5

    Topics: Acetaminophen; Adrenergic alpha-Antagonists; Analgesics; Animals; Aspirin; Caffeine; Clonidine; Cyproheptadine; Dihydroergotamine; Ergotamine; Humans; Methysergide; Migraine Disorders; Monoamine Oxidase Inhibitors; Muscle, Smooth; Pizotyline; Serotonin Antagonists; Sympathetic Nervous System; Synaptic Transmission; Tryptamines; Vagus Nerve; Vasoconstrictor Agents; Vasodilator Agents

1975
[Carcinoid: diagnosis and therapy].
    Deutsche medizinische Wochenschrift (1946), 1975, Oct-17, Volume: 100, Issue:42

    Topics: Aprotinin; Bradykinin; Carcinoid Heart Disease; Carcinoid Tumor; Cyproheptadine; Diagnosis, Differential; Ergot Alkaloids; Humans; Hydroxyindoleacetic Acid; Kallidin; Malignant Carcinoid Syndrome; Methylprednisolone; Methysergide; Phentolamine; Pizotyline; Serotonin

1975
[Serotonin agonists and antagonists in migraine].
    Pathologie-biologie, 1992, Volume: 40, Issue:4

    Topics: Benzoxepins; Contraindications; Cyproheptadine; Dihydroergotamine; Ergotamine; Histamine H1 Antagonists; Humans; Indoles; Methysergide; Migraine Disorders; Phenothiazines; Pizotyline; Receptors, Serotonin; Sulfonamides; Sumatriptan; Vasoconstrictor Agents

1992
Serotonin antagonists.
    Australian and New Zealand journal of medicine, 1984, Volume: 14, Issue:6

    Topics: Cyproheptadine; Depression; Ergotamine; Humans; Hypertension; Ketanserin; Lisuride; Methysergide; Mianserin; Migraine Disorders; Piperidines; Pizotyline; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Vascular Diseases

1984
Abdominal migraine: evidence for existence and treatment options.
    Paediatric drugs, 2002, Volume: 4, Issue:1

    Topics: Abdominal Pain; Child; Cyproheptadine; Diet; Humans; Migraine Disorders; Pizotyline; Propranolol; Secondary Prevention

2002

Trials

3 trial(s) available for cyproheptadine and pizotyline

ArticleYear
Prophylaxis of migraine in children.
    Headache, 1977, Volume: 17, Issue:2

    Topics: Adolescent; Child; Clinical Trials as Topic; Cyproheptadine; Humans; Migraine Disorders; Pizotyline; Propranolol; Recurrence; Thiophenes

1977
[Therapeutic possibilities in idiopathic headaches. Analysis of 1000 cases (author's transl)].
    MMW, Munchener medizinische Wochenschrift, 1975, Sep-19, Volume: 117, Issue:38

    Topics: Aspirin; Caffeine; Cinnarizine; Clinical Trials as Topic; Clonidine; Cyproheptadine; Drug Therapy, Combination; Ergotamine; Headache; Histamine; Humans; Indomethacin; Metergoline; Methysergide; Migraine Disorders; Pizotyline; Prochlorperazine; Reserpine; Retrospective Studies; Urea

1975
Antiserotonin agents in the treatment of migraine.
    Polish journal of pharmacology and pharmacy, 1975, Volume: 27, Issue:Suppl

    Topics: Adult; Clinical Trials as Topic; Cyproheptadine; Female; Humans; Male; Middle Aged; Migraine Disorders; Pizotyline; Placebos; Serotonin Antagonists; Thiophenes

1975

Other Studies

30 other study(ies) available for cyproheptadine and pizotyline

ArticleYear
Functional group contributions to drug-receptor interactions.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:12

    Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship

1984
Synthesis and pharmacological studies of 4,4-disubstituted piperidines: a new class of compounds with potent analgesic properties.
    Journal of medicinal chemistry, 1983, Volume: 26, Issue:1

    Topics: 5-Hydroxytryptophan; Analgesics; Animals; Binding, Competitive; Chemical Phenomena; Chemistry; Guinea Pigs; In Vitro Techniques; Membranes; Mice; Naloxone; Piperidines; Rats; Reaction Time; Serotonin Antagonists; Structure-Activity Relationship

1983
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
[Therapy of Parkinson's disease. Practical criteria of treatment].
    Recenti progressi in medicina, 1976, Volume: 60, Issue:5

    Topics: Amantadine; Antiparkinson Agents; Benserazide; Carbidopa; Cyproheptadine; Drug Therapy, Combination; Histamine H1 Antagonists; Humans; Levodopa; Parasympatholytics; Parkinson Disease; Piribedil; Pizotyline; Propranolol

1976
The role of serotonergic pathways in isolation-induced aggression in mice.
    Pharmacology, biochemistry, and behavior, 1976, Volume: 5, Issue:1

    Topics: 5-Hydroxytryptophan; Aggression; Amidines; Animals; Cinanserin; Cyproheptadine; Depression, Chemical; Drug Interactions; Fenclonine; Humans; Male; Methiothepin; Methysergide; Mianserin; Mice; Motor Activity; Neural Pathways; Phenyl Ethers; Physostigmine; Pizotyline; Receptors, Serotonin; Scopolamine; Serotonin; Social Isolation

1976
Receptors for 5-hydroxytryptamine and noradrenaline in rabbit isolated ear artery and aorta.
    British journal of pharmacology, 1976, Volume: 58, Issue:2

    Topics: Animals; Aorta, Thoracic; Arteries; Cyproheptadine; Ear, External; Female; In Vitro Techniques; Male; Methysergide; Muscle Contraction; Muscle, Smooth; Norepinephrine; Phentolamine; Pizotyline; Potassium Chloride; Rabbits; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Serotonin; Reserpine; Serotonin; Vasomotor System

1976
Narcotic cue and narcotic state: differential involvement of brain 5-hydroxytryptamine.
    Neuropharmacology, 1977, Volume: 16, Issue:1

    Topics: Animals; Brain; Cinanserin; Cues; Cyproheptadine; Discrimination Learning; Drug Interactions; Fenclonine; Fentanyl; Male; Methysergide; Narcotics; Pizotyline; Rats; Serotonin; Synaptic Transmission; Time Factors; Tryptamines; Tryptophan

1977
Comparative studies of a new anti-migraine drugs. II. To the mode of their central action.
    Activitas nervosa superior, 1979, Volume: 21, Issue:3

    Topics: 5-Hydroxytryptophan; Animals; Antidepressive Agents, Tricyclic; Benzothiepins; Cyproheptadine; Hypothermia; Mice; Perphenazine; Pizotyline; Reserpine; Thiophenes

1979
Inhibition of insulin secretion from the perfused pancreas of the rat by pizotifen.
    British journal of pharmacology, 1979, Volume: 67, Issue:2

    Topics: Animals; Chlorpromazine; Cyproheptadine; Doxepin; Glucose; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Male; Pizotyline; Rats; Thiophenes

1979
Potentiation and antagonism of serotonin effects on intracranial and extracranial vessels. Possible implications in migraine.
    Neurology, 1978, Volume: 28, Issue:1

    Topics: Animals; Arteries; Cats; Cerebral Arteries; Cyproheptadine; Dihydroergotamine; Drug Synergism; Ergotamine; Humans; In Vitro Techniques; Methysergide; Migraine Disorders; Pizotyline; Serotonin; Serotonin Antagonists; Vasoconstriction; Vasomotor System

1978
Migraine. Prophylactic drugs.
    Nursing mirror, 1977, Aug-11, Volume: 145, Issue:6

    Topics: Anticonvulsants; Clonidine; Cyproheptadine; Dihydroergotamine; Humans; Methysergide; Migraine Disorders; Pizotyline; Propranolol; Tranquilizing Agents

1977
[Therapeutic possibilities in idiopathic headaches. Analysis of about 1000 cases].
    Minerva medica, 1976, Jun-23, Volume: 67, Issue:31

    Topics: Cinnarizine; Clonidine; Cyproheptadine; Headache; Histamine; Humans; Methysergide; Migraine Disorders; Monoamine Oxidase Inhibitors; Peptides; Pizotyline; Reserpine; Urea; Vascular Headaches

1976
[Anti-amine treatment of migraines].
    La Revue du praticien, 1975, Jan-21, Volume: 25, Issue:5

    Topics: Biogenic Amines; Cyproheptadine; Humans; Methysergide; Migraine Disorders; Phenothiazines; Pizotyline

1975
Comparative effects of four migraine prophylactic drugs on an isolated extracranial artery.
    European journal of pharmacology, 1976, Volume: 36, Issue:1

    Topics: Animals; Carotid Artery, External; Chlorides; Clonidine; Cyproheptadine; Drug Interactions; Histamine; Methysergide; Norepinephrine; Phentolamine; Pizotyline; Potassium; Pyrilamine; Rabbits; Serotonin; Thiophenes; Tryptamines; Tyramine; Vasoconstrictor Agents

1976
Affinity profiles of pizotifen, ketotifen and other tricyclic antimuscarinics at muscarinic receptor subtypes M1, M2 and M3.
    European journal of pharmacology, 1992, Feb-18, Volume: 211, Issue:3

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Cyproheptadine; Guinea Pigs; Ileum; Ketotifen; Kinetics; Male; Muscarinic Antagonists; Pizotyline; Promethazine; Rabbits; Receptors, Muscarinic; Structure-Activity Relationship; Trachea; Vas Deferens

1992
Effects of cyproheptadine and pizotifen on central muscarinic receptors.
    European journal of pharmacology, 1991, Apr-03, Volume: 195, Issue:3

    Topics: Animals; Central Nervous System; Cyproheptadine; Hippocampus; In Vitro Techniques; Inositol Phosphates; Male; Parasympatholytics; Pizotyline; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1991
The chemotherapy of rodent malaria. XLV. Reversal of chloroquine resistance in rodent and human Plasmodium by antihistaminic agents.
    Annals of tropical medicine and parasitology, 1990, Volume: 84, Issue:6

    Topics: Animals; Chloroquine; Cyproheptadine; Dose-Response Relationship, Drug; Drug Resistance; Histamine Antagonists; Histamine H1 Antagonists; Humans; In Vitro Techniques; Ketotifen; Loratadine; Pizotyline; Plasmodium berghei; Plasmodium yoelii; Rats

1990
[Serotonin and antiserotonergic agents].
    La Revue du praticien, 1990, Jun-21, Volume: 40, Issue:18

    Topics: Cyproheptadine; Dihydroergotamine; Ergotamine; Humans; Methysergide; Pizotyline; Serotonin; Serotonin Antagonists

1990
Pathogenesis of low dose streptozotocin induced diabetes in mice: requirement for alpha 1-adrenoceptor activation and vasoactive amine release.
    Diabetologia, 1989, Volume: 32, Issue:2

    Topics: Animals; Cromolyn Sodium; Cyproheptadine; Diabetes Mellitus, Experimental; Histamine Antagonists; Methysergide; Pizotyline; Prazosin; Receptors, Adrenergic, alpha

1989
The relationship between cortisol and ACTH in patients with Cushing's disease following neurosurgery or pharmacotherapy.
    Endokrynologia Polska, 1989, Volume: 40, Issue:2

    Topics: Adolescent; Adrenocorticotropic Hormone; Adult; Aminoglutethimide; Cushing Syndrome; Cyproheptadine; Female; Humans; Hydrocortisone; Hypophysectomy; Male; Middle Aged; Pizotyline; Valproic Acid

1989
[Anti-allergic properties of pipethiaden--a new preventive agent for migraine].
    Ceskoslovenska farmacie, 1989, Volume: 38, Issue:6

    Topics: Anaphylaxis; Animals; Cyproheptadine; Female; Guinea Pigs; Mice; Migraine Disorders; Passive Cutaneous Anaphylaxis; Piperidines; Pizotyline; Rats

1989
Serotonin type 2 antagonists inhibit lordosis behavior in the female rat: reversal with quipazine.
    Life sciences, 1986, Jan-06, Volume: 38, Issue:1

    Topics: Analysis of Variance; Animals; Butyrophenones; Cyproheptadine; Estradiol; Female; Ketanserin; Methiothepin; Piperidines; Pizotyline; Posture; Progesterone; Quinolines; Quipazine; Rats; Rats, Inbred Strains; Serotonin Antagonists; Sexual Behavior, Animal

1986
Antimigraine drug interactions with 5-hydroxytryptamine1A receptors.
    Annals of neurology, 1986, Volume: 19, Issue:5

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Brain; Cyproheptadine; Dihydroalprenolol; Drug Interactions; Methysergide; Pizotyline; Propranolol; Rats; Receptors, Serotonin; Tetrahydronaphthalenes; Thiophenes

1986
[Observation on the inhibitory effect of ketotifen, cyproheptadine and pizotifenum on Plasmodium falciparum in vitro].
    Zhongguo ji sheng chong xue yu ji sheng chong bing za zhi = Chinese journal of parasitology & parasitic diseases, 1988, Volume: 6, Issue:2

    Topics: Animals; Cyproheptadine; Ketotifen; Mice; Pizotyline; Plasmodium falciparum; Thiophenes

1988
Inhibition of passive cutaneous anaphylaxis by several histamine (H1) and serotonin antagonists in the rat.
    Agents and actions, 1988, Volume: 23, Issue:3-4

    Topics: Animals; Cyproheptadine; Female; Histamine Antagonists; p-Methoxy-N-methylphenethylamine; Passive Cutaneous Anaphylaxis; Piperidines; Pizotyline; Rats; Rats, Inbred Strains; Serotonin Antagonists

1988
Discriminative stimulus properties of pizotifen maleate (BC105): a putative serotonin antagonist.
    Psychopharmacology, 1984, Volume: 83, Issue:2

    Topics: Animals; Cyproheptadine; Discrimination Learning; Generalization, Response; Lysergic Acid Diethylamide; Pizotyline; Promethazine; Rats; Rats, Inbred Strains; Thiophenes

1984
Effects of atypical antidepressants on LSD potentiated apomorphine hypermotility in rats.
    Acta biologica et medica Germanica, 1980, Volume: 39, Issue:8-9

    Topics: Animals; Apomorphine; Cyproheptadine; Lysergic Acid Diethylamide; Male; Mianserin; Motor Activity; Piperidines; Pizotyline; Rats; Serotonin Antagonists

1980
The effects of serotonin antagonists in a behavioral despair procedure in mice.
    European journal of pharmacology, 1984, Dec-15, Volume: 107, Issue:1

    Topics: Animals; Behavior, Animal; Cyproheptadine; Guinea Pigs; Ketanserin; Male; Methysergide; Mice; Muscle, Smooth; Piperidines; Pizotyline; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone; Trazodone; Tritium

1984
Pizotyline effectively attenuates the stimulus effects of N-methyl-3,4-methylenedioxyamphetamine (MDMA).
    Pharmacology, biochemistry, and behavior, 2005, Volume: 82, Issue:2

    Topics: Animals; Central Nervous System Stimulants; Cyproheptadine; Discrimination, Psychological; Dose-Response Relationship, Drug; Generalization, Psychological; Hallucinogens; Male; Methamphetamine; N-Methyl-3,4-methylenedioxyamphetamine; Pizotyline; Rats; Rats, Sprague-Dawley; Receptors, Neurotransmitter; Receptors, Serotonin; Serotonin Antagonists

2005
The antidepressant 5-HT2A receptor antagonists pizotifen and cyproheptadine inhibit serotonin-enhanced platelet function.
    PloS one, 2014, Volume: 9, Issue:1

    Topics: Adenosine Diphosphate; Animals; Antidepressive Agents; Blotting, Western; Calcium; Carotid Artery Thrombosis; Clopidogrel; Cyproheptadine; Flow Cytometry; Hemorrhage; Humans; Immunoprecipitation; Indoles; Male; Mice; Mice, Inbred C57BL; Piperazines; Pizotyline; Platelet Activation; Platelet Aggregation; Platelet Aggregation Inhibitors; Platelet Function Tests; Receptor, Serotonin, 5-HT2A; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Ticlopidine

2014