Compounds > cyclothiazide

cyclothiazide and ly 404187

cyclothiazide has been researched along with ly 404187 in 6 studies

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's5 (83.33)29.6817
2010's1 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Arnold, MB; Baker, SR; Bleakman, D; Bleisch, TJ; Cantrell, B; Deverill, M; Gates, M; Ho, K; Jarvie, KR; Kamboj, RK; Mandelzys, A; Ornstein, PL; Simon, R; Tizzano, JP; Zarrinmayeh, H; Zimmerman, DM1
Bleakman, D; Gates, MR; Grabell, J; Gupta, A; Ho, K; Jarvie, KR; Miu, P; Ogden, A; Ornstein, PL; Peters, D; Radhakrishnan, V; Zarrinmayeh, H; Zimmerman, DM1
Castaño, A; Dominguez, E; Escribano, A; Fernandez, MC; Hong, E; Hornback, WJ; Jiang, D; Jimenez, A; Nisenbaum, ES; Rankl, N; Tromiczak, E; Vaught, G; Zarrinmayeh, H; Zimmerman, DM1
Grove, SJ; Jamieson, C; Maclean, JK; Morrow, JA; Rankovic, Z1
Bleakman, D; Gates, M; Ogden, A1
Nisenbaum, ES; Quirk, JC1

Other Studies

6 other study(ies) available for cyclothiazide and ly 404187

ArticleYear
Biarylpropylsulfonamides as novel, potent potentiators of 2-amino-3- (5-methyl-3-hydroxyisoxazol-4-yl)- propanoic acid (AMPA) receptors.
    Journal of medicinal chemistry, 2000, Nov-16, Volume: 43, Issue:23

    Topics: Cell Line; Humans; Receptors, AMPA; Structure-Activity Relationship; Sulfonamides

2000
Novel AMPA receptor potentiators LY392098 and LY404187: effects on recombinant human AMPA receptors in vitro.
    Neuropharmacology, 2001, Volume: 40, Issue:8

    Topics: Allosteric Regulation; Antihypertensive Agents; Benzothiadiazines; Calcium; Cell Line; Dioxoles; Dose-Response Relationship, Drug; Drug Synergism; Electrophysiology; Excitatory Amino Acid Agonists; Humans; Piperidines; Receptors, AMPA; Receptors, Glutamate; Recombinant Proteins; Sulfonamides; Thiophenes

2001
A novel class of AMPA receptor allosteric modulators. Part 1: design, synthesis, and SAR of 3-aryl-4-cyano-5-substituted-heteroaryl-2-carboxylic acid derivatives.
    Bioorganic & medicinal chemistry letters, 2006, Oct-01, Volume: 16, Issue:19

    Topics: Allosteric Regulation; Carboxylic Acids; Drug Design; Excitatory Amino Acid Agents; Heterocyclic Compounds; Humans; Receptors, AMPA; Structure-Activity Relationship; Sulfides

2006
Positive allosteric modulators of the α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) receptor.
    Journal of medicinal chemistry, 2010, Oct-28, Volume: 53, Issue:20

    Topics: Allosteric Regulation; Animals; Benzamides; Benzothiadiazines; Binding Sites; Excitatory Amino Acid Agents; Humans; Indazoles; Ligands; Models, Molecular; Protein Conformation; Receptors, AMPA; Sulfonamides

2010
Pharmacological effects of AMPA receptor potentiators LY392098 and LY404187 on rat neuronal AMPA receptors in vitro.
    Neuropharmacology, 2001, Volume: 40, Issue:8

    Topics: Allosteric Regulation; Animals; Antihypertensive Agents; Benzothiadiazines; Cells, Cultured; Drug Synergism; Excitatory Amino Acid Agonists; Hippocampus; Neurons; Purkinje Cells; Rats; Receptors, AMPA; Receptors, Kainic Acid; Sulfonamides; Thiophenes

2001
Multiple molecular determinants for allosteric modulation of alternatively spliced AMPA receptors.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2003, Nov-26, Volume: 23, Issue:34

    Topics: Allosteric Regulation; Alternative Splicing; Benzothiadiazines; Cell Line; Dose-Response Relationship, Drug; Humans; Kidney; Mutagenesis, Site-Directed; Receptors, AMPA; Recombinant Proteins; Sulfonamides

2003