cyclothiazide and kainic acid

cyclothiazide has been researched along with kainic acid in 78 studies

Research

Studies (78)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's43 (55.13)18.2507
2000's31 (39.74)29.6817
2010's4 (5.13)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Butini, S; Campiani, G; Christensen, JK; Coccone, SS; De Angelis, M; Fiorini, I; Gemma, S; Guarino, E; Morelli, E; Novellino, E; Pickering, DS; Schousboe, A; Trotta, F1
England, PM; Fleming, JJ1
Gallo, V; Mayer, ML; Patneau, DK; Winters, C; Wright, PW1
Burnett, JP; May, PC; Mayne, NG; Sharp, RL; Snyder, YM1
Burnett, JP; Desai, MA; Schoepp, DD1
Burnett, JP; Desai, MA; Ornstein, PL; Schoepp, DD1
Blanchard, JC; Doble, A; Petitet, F2
Fattman, CL; Hoyt, KR; Rajdev, S; Reynolds, IJ1
Desai, MA; Monn, JA; Schoepp, DD; Valli, MJ1
Balázs, R; Hack, N1
Geiger, JR; Jonas, P; Koh, DS; Sakmann, B1
Berger, T1
Lodge, D; Palmer, AJ1
May, PC; Robison, PM1
Mayer, ML; Patneau, DK; Vyklicky, L1
Mayer, ML; Wong, LA1
Huettner, JE; Wilding, TJ1
Bowie, D; Mayer, ML; Partin, KM1
Baraldi, M; Bertolino, M; Braghiroli, D; Costa, E; DiBella, M; Parenti, C; Vicini, S1
Mayer, ML; Partin, KM; Patneau, DK1
Tang, CM; Yamada, KA1
Olney, JW; Price, MT; Yamada, KA; Zorumski, CF1
Gallo, V; Holtzclaw, LA; Russell, JT1
Huganir, RL; Moshaver, A; Raymond, LA; Tingley, WG1
Pidoplichko, VI; Reymann, KG; Wilsch, VW1
Deitmer, JW; Löhrke, S1
Bacskai, B; Pleasure, D; Yoshioka, A1
Magazanik, LG; Usherwood, PN1
Bonfanti, A; Pittaluga, A; Raiteri, M1
Fontana, G; Gemignani, A; Marchese, S; Raiteri, M1
Clements, JD; Feltz, A; Sahara, Y; Westbrook, GL1
Ohno, K; Okada, M; Sakamoto, S; Tsutsumi, R; Yamaguchi, T1
Matsumoto, N; Ohno, K; Okada, M; Tsutsumi, R; Yamaguchi, T1
Dougherty, PM; Lenz, FA; Mittman, S1
Horiuchi, K; Itoh, A; Itoh, T; Pleasure, D1
Donevan, SD; Rogawski, MA1
Holmberg, L; Souverbie, F; Sundström, E1
Carvalho, AP; Duarte, CB; Ferreira, IL1
Akaike, N; Harata, N; Katayama, J1
Blank, T; Cepok, S; Grafelmann, B; Kügler, H; Nijholt, I; Spiess, J1
Geurtz, W; Hatt, H; Okada, T; Schultz, K; Weiler, R1
Karkanias, NB; Papke, RL1
Shen, Y; Yang, XL; Zhou, Y1
Akaike, N; Nabekura, J; Nakanishi, H; Noda, M1
Cooke, IM; Duan, S1
Trussell, LO; Turecek, R1
Bol'shakov, KB; Buldakova, SL1
Isaac, JT; Kidd, FL1
Kijima, H; Koike, M; Ozawa, S; Tsukada, S; Tsuzuki, K1
Kohda, K; Wang, Y; Yuzaki, M1
Cebers, G; Kovács, AD; Liljequist, S1
Durkin, JP; Gendron, TF; MacLean, S; Mealing, G; Morley, P; Small, DL; Tremblay, R1
Ambrósio, AF; Carvalho, AP; Carvalho, CM; Malva, JO; Mesquita, JF; Silva, AP1
Haas, HL; Sergeeva, OA; Sharonova, IN; Vorobjev, VS1
Bolshakov, KV; Buldakova, SL; Magazanik, LG; Tikhonov, DB1
Brorson, JR; Ihle, EC; Patneau, DK; Robberecht, W; Vandenberghe, W1
Chatton, JY; Magistretti, PJ; Marquet, P1
Morsette, DJ; Sidorowicz, H; Sladek, CD1
Hartveit, E; Mørkve, SH; Veruki, ML1
Carvalho, CM; Cristóvão, AJ1
Frye, GD; Hsiao, SH1
Korpi, ER; Lovinger, DM; Möykkynen, T1
Bachurin, SO; Dranyi, OA; Grigorev, VV1
Bruno, V; Caciagli, F; Caricasole, A; Caruso, A; Castiglione, M; Di Giorgi Gerevini, V; Marinelli, F; Melchiorri, D; Moretti, A; Nicoletti, F; Pozzilli, C; Tomassini, V1
Ambrósio, AF; Araújo, IM; Carvalho, CM; Verdasca, MJ1
Bennett, SA; Cheung, EC; Cregan, SP; Ferguson, KL; McIntosh, WC; Melanson-Drapeau, L; Park, DS; Slack, RS; Vanderluit, JL1
Cunha, RA; Oliveira, CR; Rebola, N; Rodrigues, RJ1
Barygin, OI; Dorofeeva, NA; Magazanik, LG; Salnikov, YI; Tikhonov, DB; Tikhonova, TB1
Chen, G; Jiang, M; Qi, J; Wang, Y; Warren, P1
Bräuner-Osborne, H; Jensen, AA; Strange, M1
Chen, G; Fang, C; Luscher, B; Qi, JS; Yao, J1
Bernareggi, A; Dueñas, Z; Miledi, R; Reyes-Ruiz, JM; Ruzzier, F1
Chen, JH; Nie, H; Pan, ZZ; Weng, HR1
Gong, HQ; Liang, PJ; Sun, Y; Zhang, YT1
Chen, L; Kong, S; Qian, B; Sun, Y; Wan, L; Wang, Y; Wang, ZY; Wu, Z; Zhang, B; Zhang, F1
Barygin, OI1

Other Studies

78 other study(ies) available for cyclothiazide and kainic acid

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
1H-cyclopentapyrimidine-2,4(1H,3H)-dione-related ionotropic glutamate receptors ligands. structure-activity relationships and identification of potent and Selective iGluR5 modulators.
    Journal of medicinal chemistry, 2008, Oct-23, Volume: 51, Issue:20

    Topics: Animals; Cell Line; Electrophysiology; Excitatory Amino Acid Antagonists; Female; Humans; Ligands; Molecular Structure; Oocytes; Pyrimidinones; Rats; Receptors, Glutamate; Spodoptera; Structure-Activity Relationship; Thiophenes; Xenopus laevis

2008
Developing a complete pharmacology for AMPA receptors: a perspective on subtype-selective ligands.
    Bioorganic & medicinal chemistry, 2010, Feb-15, Volume: 18, Issue:4

    Topics: Allosteric Regulation; Animals; Binding Sites; Ligands; Receptors, AMPA

2010
Glial cells of the oligodendrocyte lineage express both kainate- and AMPA-preferring subtypes of glutamate receptor.
    Neuron, 1994, Volume: 12, Issue:2

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Blotting, Northern; Cell Line; Kainic Acid; Oligodendroglia; Rats; Rats, Sprague-Dawley; Receptors, Glutamate; Transcription, Genetic

1994
Cyclothiazide potentiates agonist responses at human AMPA/kainate receptors expressed in oocytes.
    European journal of pharmacology, 1994, Jan-01, Volume: 266, Issue:1

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Cloning, Molecular; Humans; Kainic Acid; Oocytes; Receptors, AMPA; Receptors, Glutamate; Receptors, Kainic Acid; Xenopus laevis

1994
Cyclothiazide selectively potentiates AMPA- and kainate-induced [3H]norepinephrine release from rat hippocampal slices.
    Journal of neurochemistry, 1994, Volume: 63, Issue:1

    Topics: 4-Aminopyridine; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Antihypertensive Agents; Benzothiadiazines; Drug Synergism; Hippocampus; Kainic Acid; Male; N-Methylaspartate; Norepinephrine; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Kainic Acid; Tritium; Veratridine

1994
Cyclothiazide acts at a site on the alpha-amino-3-hydroxy-5-methyl-4-isoxazole propionic acid receptor complex that does not recognize competitive or noncompetitive AMPA receptor antagonists.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 272, Issue:1

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Binding Sites; Binding, Competitive; Hippocampus; In Vitro Techniques; Isoquinolines; Kainic Acid; Male; Norepinephrine; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Tetrazoles

1995
Effects of non-NMDA receptor modulators on [3H] dopamine release from rat mesencephalic cells in primary culture.
    Journal of neurochemistry, 1995, Volume: 64, Issue:3

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Cells, Cultured; Dopamine; Drug Synergism; In Vitro Techniques; Kainic Acid; Mesencephalon; Rats; Receptors, AMPA; Receptors, Glutamate; Receptors, N-Methyl-D-Aspartate

1995
Cyclothiazide modulates AMPA receptor-mediated increases in intracellular free Ca2+ and Mg2+ in cultured neurons from rat brain.
    Journal of neurochemistry, 1995, Volume: 64, Issue:5

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Calcium; Cells, Cultured; Drug Synergism; Glutamic Acid; Kainic Acid; Magnesium; Neurons; Prosencephalon; Rats; Receptors, AMPA

1995
1-BCP, a memory-enhancing agent, selectively potentiates AMPA-induced [3H]norepinephrine release in rat hippocampal slices.
    Neuropharmacology, 1995, Volume: 34, Issue:2

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Dioxoles; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Hippocampus; Kainic Acid; Male; Memory; N-Methylaspartate; Norepinephrine; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, AMPA

1995
Properties of AMPA receptors expressed in rat cerebellar granule cell cultures: Ca2+ influx studies.
    Journal of neurochemistry, 1995, Volume: 65, Issue:3

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Calcium; Calcium Radioisotopes; Cell Survival; Cells, Cultured; Cerebellum; Cobalt; Concanavalin A; Excitatory Amino Acids; Kainic Acid; N-Methylaspartate; Quinoxalines; Rats; Receptors, AMPA; Wheat Germ Agglutinins

1995
Ca(2+)-permeable AMPA and NMDA receptor channels in basket cells of rat hippocampal dentate gyrus.
    The Journal of physiology, 1995, Jun-01, Volume: 485 ( Pt 2)

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Calcium Channels; Dendrites; Diuretics; Glutamic Acid; Hippocampus; In Vitro Techniques; Kainic Acid; Kinetics; Magnesium; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Sodium; Sodium Chloride Symporter Inhibitors

1995
AMPA-type glutamate receptors in glial precursor cells of the rat corpus callosum: ionic and pharmacological properties.
    Glia, 1995, Volume: 14, Issue:2

    Topics: Animals; Benzothiadiazines; Calcium; Chlorides; Concanavalin A; Corpus Callosum; Diuretics; Evans Blue; Kainic Acid; Neuroglia; Patch-Clamp Techniques; Quinoxalines; Rats; Receptors, AMPA; Receptors, Kainic Acid; Sodium Chloride Symporter Inhibitors; Zinc Compounds

1995
Cyclothiazide reverses AMPA receptor antagonism of the 2,3-benzodiazepine, GYKI 53655.
    European journal of pharmacology, 1993, Jan-15, Volume: 244, Issue:2

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Cerebral Cortex; Diuretics; Excitatory Amino Acid Antagonists; Ibotenic Acid; In Vitro Techniques; Kainic Acid; N-Methylaspartate; Quinoxalines; Rats; Receptors, AMPA; Sodium Chloride Symporter Inhibitors

1993
Cyclothiazide treatment unmasks AMPA excitotoxicity in rat primary hippocampal cultures.
    Journal of neurochemistry, 1993, Volume: 60, Issue:3

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Cells, Cultured; Drug Synergism; Hippocampus; Ibotenic Acid; Kainic Acid; Neurotoxins; Rats

1993
Hippocampal neurons exhibit cyclothiazide-sensitive rapidly desensitizing responses to kainate.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1993, Volume: 13, Issue:8

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Animals, Newborn; Benzothiadiazines; Cells, Cultured; Dose-Response Relationship, Drug; Drug Synergism; Drug Tolerance; Electrophysiology; Evoked Potentials; Glutamates; Glutamic Acid; Hippocampus; Ibotenic Acid; Kainic Acid; Kinetics; Neurons; Quisqualic Acid; Rats; Rats, Sprague-Dawley

1993
Differential modulation by cyclothiazide and concanavalin A of desensitization at native alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid- and kainate-preferring glutamate receptors.
    Molecular pharmacology, 1993, Volume: 44, Issue:3

    Topics: Alanine; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Concanavalin A; Ganglia, Spinal; Hippocampus; Ibotenic Acid; In Vitro Techniques; Kainic Acid; Neurons; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Glutamate; Receptors, Kainic Acid

1993
Differential antagonism of alpha-amino-3-hydroxy-5-methyl-4- isoxazolepropionic acid-preferring and kainate-preferring receptors by 2,3-benzodiazepines.
    Molecular pharmacology, 1995, Volume: 47, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Binding, Competitive; Cerebral Cortex; Concanavalin A; Electrophysiology; Ganglia, Spinal; Kainic Acid; Membrane Potentials; Neurons; Rats; Rats, Inbred Strains; Receptors, AMPA; Receptors, Kainic Acid; Substrate Specificity

1995
Structural determinants of allosteric regulation in alternatively spliced AMPA receptors.
    Neuron, 1995, Volume: 14, Issue:4

    Topics: Allosteric Regulation; Alternative Splicing; Amino Acid Sequence; Animals; Benzothiadiazines; Embryo, Mammalian; Embryo, Nonmammalian; Glutamic Acid; Glutamine; Humans; Kainic Acid; Kidney; Macromolecular Substances; Molecular Sequence Data; Mutagenesis, Site-Directed; Oocytes; Point Mutation; Receptors, AMPA; Receptors, Kainic Acid; Serine; Transfection; Xenopus laevis

1995
Modulation of AMPA/kainate receptors by analogues of diazoxide and cyclothiazide in thin slices of rat hippocampus.
    Receptors & channels, 1993, Volume: 1, Issue:4

    Topics: Action Potentials; Animals; Benzothiadiazines; Diazoxide; Glutamates; Glutamic Acid; Hippocampus; In Vitro Techniques; Kainic Acid; Membrane Potentials; Molecular Structure; Rats; Receptors, AMPA; Receptors, Kainic Acid

1993
Cyclothiazide differentially modulates desensitization of alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptor splice variants.
    Molecular pharmacology, 1994, Volume: 46, Issue:1

    Topics: Animals; Benzothiadiazines; Cells, Cultured; Female; Kainic Acid; Kinetics; Membrane Potentials; Receptors, AMPA; Receptors, Glutamate; RNA Splicing; Xenopus

1994
Benzothiadiazides inhibit rapid glutamate receptor desensitization and enhance glutamatergic synaptic currents.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1993, Volume: 13, Issue:9

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Benzothiadiazines; Cell Line; Cells, Cultured; Diazoxide; Diuretics; Electric Stimulation; Evoked Potentials; Hippocampus; Humans; Kainic Acid; Membrane Potentials; Molecular Structure; N-Methylaspartate; Neurons; Quinoxalines; Quisqualic Acid; Rats; Receptors, Glutamate; Structure-Activity Relationship; Synapses; Time Factors

1993
A benzodiazepine recognition site associated with the non-NMDA glutamate receptor.
    Neuron, 1993, Volume: 10, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Binding Sites; Binding, Competitive; Cells, Cultured; Chick Embryo; Electric Conductivity; Excitatory Amino Acid Antagonists; Hippocampus; Kainic Acid; Nerve Degeneration; Neurons; Quisqualic Acid; Rats; Receptors, Glutamate; Retina

1993
AMPA receptors shape Ca2+ responses in cortical oligodendrocyte progenitors and CG-4 cells.
    Journal of neuroscience research, 1995, Sep-01, Volume: 42, Issue:1

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Calcium; Cell Line; Cells, Cultured; Dose-Response Relationship, Drug; Glutamic Acid; Kainic Acid; Oligodendroglia; Quinoxalines; Receptors, AMPA; Time Factors

1995
Effects of AMPA receptor modulators on the production of arachidonic acid from striatal neurons.
    European journal of pharmacology, 1995, Oct-15, Volume: 291, Issue:2

    Topics: Animals; Arachidonic Acid; Atropine; Benzothiadiazines; Carbachol; Corpus Striatum; Female; Kainic Acid; Neurons; Rats; Receptors, AMPA

1995
Glutamate receptor ion channel properties predict vulnerability to cytotoxicity in a transfected nonneuronal cell line.
    Molecular and cellular neurosciences, 1996, Volume: 7, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Animals; Base Sequence; Benzothiadiazines; Cell Line; Cell Survival; Concanavalin A; Dizocilpine Maleate; DNA Primers; Evoked Potentials; Glutamic Acid; Humans; Ion Channels; Kainic Acid; Kidney; Mice; Molecular Sequence Data; Mutagenesis, Site-Directed; N-Methylaspartate; Neurotoxins; Patch-Clamp Techniques; Receptors, Glutamate; Receptors, N-Methyl-D-Aspartate; Transfection

1996
Fast desensitizing kainate-gated current resolved in whole-cell experiments on isolated rat hippocampal neurons.
    European journal of pharmacology, 1996, May-06, Volume: 303, Issue:1-2

    Topics: Animals; Benzothiadiazines; Cells, Cultured; Concanavalin A; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Hippocampus; Kainic Acid; Male; Patch-Clamp Techniques; Rats

1996
Kainate responses of leech Retzius neurons in situ and in vitro.
    Journal of neurobiology, 1996, Volume: 31, Issue:3

    Topics: Animals; Benzothiadiazines; Calcium; Calcium Channels; Cell Membrane Permeability; Cells, Cultured; Concanavalin A; Drug Synergism; Excitatory Amino Acid Agonists; Ganglia, Invertebrate; Kainic Acid; Leeches; Neurons

1996
Pathophysiology of oligodendroglial excitotoxicity.
    Journal of neuroscience research, 1996, Nov-15, Volume: 46, Issue:4

    Topics: Acetylcysteine; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Aurintricarboxylic Acid; Benzothiadiazines; Biological Transport; Calcium; Cell Line; Cell Membrane; DNA Fragmentation; Endodeoxyribonucleases; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Glutamic Acid; Kainic Acid; Nerve Tissue Proteins; Oligodendroglia; Rats; Receptors, AMPA; RNA, Messenger

1996
Competitive antagonism of recombinant AMPA/kainate receptors by N-methyl-D-aspartate and analogues.
    Neuroreport, 1996, Dec-20, Volume: 8, Issue:1

    Topics: Animals; Benzothiadiazines; Binding, Competitive; Diuretics; Excitatory Amino Acid Antagonists; Glycine; Kainic Acid; N-Methylaspartate; Rats; Receptors, AMPA; Receptors, Kainic Acid; Recombinant Proteins; Sodium Chloride Symporter Inhibitors; Xenopus laevis

1996
Differential desensitization of ionotropic non-NMDA receptors having distinct neuronal location and function.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:1

    Topics: Acetylcholine; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Calcium; Cerebral Cortex; Choline; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Hippocampus; In Vitro Techniques; Kainic Acid; Male; Norepinephrine; Potassium; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Glutamate; Receptors, Kainic Acid; Serotonin; Synaptosomes

1997
Neuropeptide Y release from cultured hippocampal neurons: stimulation by glutamate acting at N-methyl-D-aspartate and AMPA receptors.
    Neuroscience, 1997, Volume: 81, Issue:1

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Anxiety Agents; Antibody Specificity; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Calcium; Cells, Cultured; Chromatography, High Pressure Liquid; Dizocilpine Maleate; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Hippocampus; Kainic Acid; Magnesium; Neurons; Neuropeptide Y; Quinoxalines; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Tetrodotoxin

1997
Activation kinetics of AMPA receptor channels reveal the number of functional agonist binding sites.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1998, Jan-01, Volume: 18, Issue:1

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Animals, Newborn; Antihypertensive Agents; Benzothiadiazines; Binding Sites; Cells, Cultured; Enzyme Activation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Hippocampus; Ion Channel Gating; Kainic Acid; Kinetics; Neuromuscular Depolarizing Agents; Neurons; Patch-Clamp Techniques; Quisqualic Acid; Rats; Rats, Sprague-Dawley; Receptors, AMPA

1998
The AMPA-receptor antagonist YM90K reduces AMPA receptor-mediated excitotoxicity in rat hippocampal cultures.
    Japanese journal of pharmacology, 1998, Volume: 76, Issue:1

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Cells, Cultured; Diuretics; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Hippocampus; Kainic Acid; Neurons; Neuroprotective Agents; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Sodium Chloride Symporter Inhibitors

1998
Characterization of cyclothiazide-enhanced kainate excitotoxicity in rat hippocampal cultures.
    Neurochemistry international, 1998, Volume: 32, Issue:3

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Cells, Cultured; Dose-Response Relationship, Drug; Drug Synergism; Embryo, Mammalian; Hippocampus; Kainic Acid; Rats; Rats, Wistar; Receptors, AMPA

1998
Facilitation of responses to AMPA but not kainate by cyclothiazide in primate somatosensory thalamus.
    Neuroscience letters, 1998, Apr-17, Volume: 246, Issue:1

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Drug Synergism; Excitatory Amino Acid Agonists; Glutamic Acid; Kainic Acid; Macaca fascicularis; Male; N-Methylaspartate; Thalamic Nuclei

1998
AMPA receptor-mediated excitotoxicity in human NT2-N neurons results from loss of intracellular Ca2+ homeostasis following marked elevation of intracellular Na+.
    Journal of neurochemistry, 1998, Volume: 71, Issue:1

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Antihypertensive Agents; Benzothiadiazines; Calcium; Calcium Channel Blockers; Cell Death; Cell Membrane; Dizocilpine Maleate; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Extracellular Space; Glutamic Acid; Homeostasis; Humans; Kainic Acid; Membrane Potentials; Neurons; Neurotoxins; Nimodipine; Potassium; Receptors, AMPA; Sodium; Sodium-Calcium Exchanger; Spider Venoms

1998
Allosteric regulation of alpha-amino-3-hydroxy-5-methyl-4-isoxazole-propionate receptors by thiocyanate and cyclothiazide at a common modulatory site distinct from that of 2,3-benzodiazepines.
    Neuroscience, 1998, Volume: 87, Issue:3

    Topics: Allosteric Regulation; Animals; Anti-Anxiety Agents; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Binding Sites; Cells, Cultured; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Hippocampus; Ion Channel Gating; Kainic Acid; Membrane Potentials; N-Methylaspartate; Neurons; Oocytes; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Thiocyanates; Xenopus

1998
NMDA and AMPA receptors evoke transmitter release from noradrenergic axon terminals in the rat spinal cord.
    Neurochemical research, 1998, Volume: 23, Issue:12

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Concanavalin A; Dizocilpine Maleate; In Vitro Techniques; Kainic Acid; Male; N-Methylaspartate; Norepinephrine; Presynaptic Terminals; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Spinal Cord; Tetrodotoxin

1998
Kainate-induced retina amacrine-like cell damage is mediated by AMPA receptors.
    Neuroreport, 1998, Oct-26, Volume: 9, Issue:15

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Calcium Radioisotopes; Cells, Cultured; Chickens; Dizocilpine Maleate; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Kainic Acid; Neuromuscular Depolarizing Agents; Receptors, AMPA; Receptors, Kainic Acid; Retina

1998
Excitatory amino acid responses in relay neurons of the rat lateral geniculate nucleus.
    Neuroscience, 1999, Volume: 89, Issue:1

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Antihypertensive Agents; Benzothiadiazines; Concanavalin A; Dipeptides; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Geniculate Bodies; Glutamic Acid; Glycine; Ionophores; Kainic Acid; Membrane Potentials; N-Methylaspartate; Neurons; Neuroprotective Agents; Nystatin; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission

1999
NS-257, a novel competitive AMPA receptor antagonist, interacts with kainate and NMDA receptors.
    Brain research, 1999, Mar-13, Volume: 821, Issue:2

    Topics: Animals; Antihypertensive Agents; Benzothiadiazines; Concanavalin A; Dose-Response Relationship, Drug; Electrophysiology; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Indoles; Kainic Acid; Membrane Potentials; Mice; Mice, Inbred C57BL; Microinjections; N-Methylaspartate; Oocytes; Patch-Clamp Techniques; Receptors, AMPA; Receptors, Kainic Acid; Receptors, N-Methyl-D-Aspartate; RNA, Complementary; RNA, Messenger; Sulfonamides; Xenopus

1999
AMPA-preferring receptors with high Ca2+ permeability mediate dendritic plasticity of retinal horizontal cells.
    The European journal of neuroscience, 1999, Volume: 11, Issue:3

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Calcium; Carps; Dark Adaptation; Dendrites; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Kainic Acid; Membrane Potentials; Microscopy, Electron; Neuronal Plasticity; Patch-Clamp Techniques; Receptors, AMPA; Receptors, Kainic Acid; Retina

1999
Subtype-specific effects of lithium on glutamate receptor function.
    Journal of neurophysiology, 1999, Volume: 81, Issue:4

    Topics: Animals; Antihypertensive Agents; Benzothiadiazines; Biological Transport; Dose-Response Relationship, Drug; Electric Conductivity; Excitatory Amino Acid Agonists; Female; GluK2 Kainate Receptor; Ion Channel Gating; Kainic Acid; Lithium; Membrane Potentials; Patch-Clamp Techniques; Receptors, AMPA; Receptors, Glutamate; Receptors, Kainic Acid; Receptors, N-Methyl-D-Aspartate; RNA, Messenger; Rubidium; Sodium; Xenopus laevis

1999
Characterization of AMPA receptors on isolated amacrine-like cells in carp retina.
    The European journal of neuroscience, 1999, Volume: 11, Issue:12

    Topics: Alternative Splicing; Animals; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Cell Separation; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Goldfish; Ion Channels; Kainic Acid; Membrane Potentials; N-Methylaspartate; Patch-Clamp Techniques; Phenoxyacetates; Receptors, AMPA; Retina

1999
AMPA-kainate subtypes of glutamate receptor in rat cerebral microglia.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2000, Jan-01, Volume: 20, Issue:1

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Antihypertensive Agents; Benzothiadiazines; Calcium; Cells, Cultured; Cerebral Cortex; Concanavalin A; Excitatory Amino Acid Agonists; Glutamic Acid; Kainic Acid; Membrane Potentials; Microglia; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, AMPA; Receptors, Kainic Acid; Reverse Transcriptase Polymerase Chain Reaction; Stimulation, Chemical; Tumor Necrosis Factor-alpha

2000
Glutamate and GABA activate different receptors and Cl(-) conductances in crab peptide-secretory neurons.
    Journal of neurophysiology, 2000, Volume: 83, Issue:1

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Brachyura; Cells, Cultured; Chloride Channels; Chlorides; Concanavalin A; gamma-Aminobutyric Acid; Glutamic Acid; Glycine; Kainic Acid; N-Methylaspartate; Neurons; Patch-Clamp Techniques; Quisqualic Acid; Receptors, AMPA; Receptors, GABA; Receptors, Glutamate

2000
Control of synaptic depression by glutamate transporters.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2000, Mar-01, Volume: 20, Issue:5

    Topics: Action Potentials; Alanine Transaminase; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amino Acid Transport System X-AG; Animals; Anti-Bacterial Agents; Antihypertensive Agents; Aspartic Acid; ATP-Binding Cassette Transporters; Benzothiadiazines; Chick Embryo; Cochlear Nucleus; Excitatory Amino Acid Agonists; Excitatory Postsynaptic Potentials; Glutamic Acid; In Vitro Techniques; Kainic Acid; N-Methylaspartate; Neural Inhibition; Neuronal Plasticity; Receptors, AMPA; Synaptic Transmission

2000
[Pharmacologic analysis of the subunit composition of AMPA-receptors in the hippocampal neurons].
    Rossiiskii fiziologicheskii zhurnal imeni I.M. Sechenova, 1999, Volume: 85, Issue:12

    Topics: Adamantane; Alternative Splicing; Animals; Benzothiadiazines; Dentate Gyrus; Excitatory Amino Acid Agonists; Hippocampus; In Vitro Techniques; Interneurons; Kainic Acid; Neurons; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, AMPA

1999
Glutamate transport blockade has a differential effect on AMPA and NMDA receptor-mediated synaptic transmission in the developing barrel cortex.
    Neuropharmacology, 2000, Mar-03, Volume: 39, Issue:5

    Topics: Amino Acid Transport System X-AG; Animals; Aspartic Acid; ATP-Binding Cassette Transporters; Benzothiadiazines; Biological Transport; Dicarboxylic Acids; Diuretics; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; Glutamic Acid; In Vitro Techniques; Kainic Acid; Neurotransmitter Uptake Inhibitors; Picrotoxin; Pyrrolidines; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Sodium Chloride Symporter Inhibitors; Somatosensory Cortex; Synaptic Transmission; Thalamus

2000
Regulation of kinetic properties of GluR2 AMPA receptor channels by alternative splicing.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2000, Mar-15, Volume: 20, Issue:6

    Topics: Alternative Splicing; Animals; Antihypertensive Agents; Benzothiadiazines; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Glutamic Acid; Ion Channel Gating; Kainic Acid; Kinetics; Mutagenesis; Oocytes; Patch-Clamp Techniques; Rats; Receptors, AMPA; Xenopus

2000
Mutation of a glutamate receptor motif reveals its role in gating and delta2 receptor channel properties.
    Nature neuroscience, 2000, Volume: 3, Issue:4

    Topics: Amino Acid Sequence; Amino Acid Substitution; Animals; Anti-Anxiety Agents; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Cell Line; Conserved Sequence; Dizocilpine Maleate; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Humans; Ion Channel Gating; Kainic Acid; Kidney; Mice; Mice, Neurologic Mutants; Molecular Sequence Data; Mutagenesis; Neuromuscular Depolarizing Agents; Patch-Clamp Techniques; Purkinje Cells; Quinoxalines; Receptors, Glutamate; Transfection

2000
Kainate receptor-mediated activation of the AP-1 transcription factor complex in cultured rat cerebellar granule cells.
    Brain research bulletin, 2000, May-15, Volume: 52, Issue:2

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Cells, Cultured; Cerebellum; Concanavalin A; Dimerization; Excitatory Amino Acid Antagonists; Isoquinolines; Kainic Acid; Neurons; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Kainic Acid; Tetrazoles; Transcription Factor AP-1

2000
Pharmacological and molecular characterization of glutamate receptors in the MIN6 pancreatic beta-cell line.
    Neurological research, 2000, Volume: 22, Issue:4

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Anxiety Agents; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Biological Transport; Calcium; Cell Survival; DNA Primers; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Islets of Langerhans; Kainic Acid; Protein Kinase C; Quinoxalines; Rats; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Spider Venoms; Tumor Cells, Cultured

2000
Role of desensitization of AMPA receptors on the neuronal viability and on the [Ca2+]i changes in cultured rat hippocampal neurons.
    The European journal of neuroscience, 2000, Volume: 12, Issue:6

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Calcium; Cell Survival; Cells, Cultured; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Fetus; Hippocampus; Kainic Acid; Neurons; Neuroprotective Agents; Rats; Rats, Wistar; Receptors, AMPA

2000
Differential modulation of AMPA receptors by cyclothiazide in two types of striatal neurons.
    The European journal of neuroscience, 2000, Volume: 12, Issue:8

    Topics: Alternative Splicing; Animals; Antihypertensive Agents; Benzothiadiazines; Cell Separation; Cell Size; Corpus Striatum; DNA Primers; Drug Synergism; Excitatory Amino Acid Agonists; Glutamic Acid; Ion Channel Gating; Kainic Acid; Kinetics; Male; Neurons; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, AMPA; Reverse Transcriptase Polymerase Chain Reaction

2000
Ca2+-dependent desensitization of AMPA receptors.
    Neuroreport, 2000, Sep-11, Volume: 11, Issue:13

    Topics: Adamantane; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Alternative Splicing; Animals; Animals, Newborn; Antihypertensive Agents; Benzothiadiazines; Calcium; Calcium Signaling; Dose-Response Relationship, Drug; Glutamic Acid; Hippocampus; Kainic Acid; Neurons; Nootropic Agents; Pyrrolidinones; Rats; Receptors, AMPA

2000
AMPA receptor current density, not desensitization, predicts selective motoneuron vulnerability.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2000, Oct-01, Volume: 20, Issue:19

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Astrocytes; Benzodiazepines; Benzothiadiazines; Cells, Cultured; Coculture Techniques; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Glutamic Acid; Kainic Acid; Membrane Potentials; Motor Neurons; Patch-Clamp Techniques; Posterior Horn Cells; Protein Isoforms; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Spinal Cord

2000
A quantitative analysis of L-glutamate-regulated Na+ dynamics in mouse cortical astrocytes: implications for cellular bioenergetics.
    The European journal of neuroscience, 2000, Volume: 12, Issue:11

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amino Acid Transport System X-AG; Animals; Animals, Newborn; Astrocytes; Benzothiadiazines; Biological Transport; Carrier Proteins; Cells, Cultured; Cerebral Cortex; Glutamate Plasma Membrane Transport Proteins; Glutamic Acid; Kainic Acid; Kinetics; Mice; Models, Theoretical; N-Methylaspartate; Sodium; Symporters

2000
Role of non-NMDA receptors in vasopressin and oxytocin release from rat hypothalamo-neurohypophysial explants.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2001, Volume: 280, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Glutamates; Hypothalamo-Hypophyseal System; Kainic Acid; Kinetics; Male; N-Methylaspartate; Organ Culture Techniques; Oxytocin; Rats; Rats, Sprague-Dawley; Receptor Cross-Talk; Receptors, AMPA; Receptors, Kainic Acid; Receptors, N-Methyl-D-Aspartate; Vasopressins

2001
Functional characteristics of non-NMDA-type ionotropic glutamate receptor channels in AII amacrine cells in rat retina.
    The Journal of physiology, 2002, Jul-01, Volume: 542, Issue:Pt 1

    Topics: Algorithms; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Calcium; Concanavalin A; Electric Stimulation; Electrophysiology; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; In Vitro Techniques; Kainic Acid; Membrane Potentials; Patch-Clamp Techniques; Rats; Receptors, AMPA; Receptors, Glutamate; Retina; Sodium

2002
Development of chick retina cells in culture: cobalt entry through AMPA receptors and expression of GluR4 AMPA receptor subunit.
    Brain research. Developmental brain research, 2003, Jan-10, Volume: 140, Issue:1

    Topics: Animals; Benzothiadiazines; Cells, Cultured; Chick Embryo; Cobalt; Gene Expression Regulation, Developmental; Kainic Acid; Kinetics; Protein Subunits; Receptors, AMPA; Retina

2003
AMPA receptors on developing medial septum/diagonal band neurons are sensitive to early postnatal binge-like ethanol exposure.
    Brain research. Developmental brain research, 2003, Apr-14, Volume: 142, Issue:1

    Topics: Alcohol-Induced Disorders, Nervous System; Alcoholic Intoxication; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Anxiety Agents; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Blotting, Western; Cells, Cultured; Central Nervous System Depressants; Diagonal Band of Broca; Ethanol; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Female; Kainic Acid; Male; Membrane Potentials; Models, Animal; Neurons; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, AMPA

2003
Ethanol inhibits alpha-amino-3-hydyroxy-5-methyl-4-isoxazolepropionic acid (AMPA) receptor function in central nervous system neurons by stabilizing desensitization.
    The Journal of pharmacology and experimental therapeutics, 2003, Volume: 306, Issue:2

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amino Acid Substitution; Animals; Benzothiadiazines; Cells, Cultured; Central Nervous System; Central Nervous System Depressants; Drug Interactions; Ethanol; Excitatory Amino Acid Agonists; Humans; Kainic Acid; Leucine; Membrane Potentials; Mice; Mice, Inbred C57BL; Mutation; Neurons; Pyramidal Cells; Receptors, AMPA; Tyrosine

2003
Comparative study of action mechanisms of dimebon and memantine on AMPA- and NMDA-subtypes glutamate receptors in rat cerebral neurons.
    Bulletin of experimental biology and medicine, 2003, Volume: 136, Issue:5

    Topics: Animals; Benzothiadiazines; Cerebral Cortex; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Indoles; Kainic Acid; Memantine; N-Methylaspartate; Neurons; Patch-Clamp Techniques; Purkinje Cells; Rats; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate

2003
Testosterone amplifies excitotoxic damage of cultured oligodendrocytes.
    Journal of neurochemistry, 2004, Volume: 88, Issue:5

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Calcium; Cells, Cultured; Drug Synergism; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Gene Expression; Kainic Acid; L-Lactate Dehydrogenase; Neurotoxins; Oligodendroglia; Quinoxalines; Rats; Receptors, AMPA; Receptors, Androgen; Receptors, Kainic Acid; Testosterone; Time Factors

2004
Nitric oxide inhibits complex I following AMPA receptor activation via peroxynitrite.
    Neuroreport, 2004, Sep-15, Volume: 15, Issue:13

    Topics: Analysis of Variance; Animals; Antihypertensive Agents; Benzothiadiazines; Cells, Cultured; Cyclic GMP; Drug Interactions; Embryo, Mammalian; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Hippocampus; Immunohistochemistry; Kainic Acid; Microtubule-Associated Proteins; Neurons; NG-Nitroarginine Methyl Ester; Nitric Oxide; Peroxynitrous Acid; Proton Pumps; Quinoxalines; Rats; Receptors, AMPA; Tyrosine

2004
Apoptosis-inducing factor is a key factor in neuronal cell death propagated by BAX-dependent and BAX-independent mechanisms.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Feb-09, Volume: 25, Issue:6

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Apoptosis; Apoptosis Inducing Factor; Apoptotic Protease-Activating Factor 1; bcl-2-Associated X Protein; Benzodiazepines; Benzothiadiazines; Camptothecin; Caspase Inhibitors; Cells, Cultured; Cerebellum; Cerebral Cortex; Convulsants; Dizocilpine Maleate; Drug Resistance; Flavoproteins; Glutamic Acid; Glycine; Hippocampus; Kainic Acid; Male; Membrane Proteins; Mice; Mice, Knockout; Mice, Mutant Strains; N-Methylaspartate; Neurons; Neurotoxins; Proteins; Proto-Oncogene Proteins c-bcl-2; Recombinant Fusion Proteins; Seizures

2005
Different roles of adenosine A1, A2A and A3 receptors in controlling kainate-induced toxicity in cortical cultured neurons.
    Neurochemistry international, 2005, Volume: 47, Issue:5

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Adenosine A3 Receptor Agonists; Adenosine A3 Receptor Antagonists; Animals; Benzothiadiazines; Cell Death; Cells, Cultured; Cerebral Cortex; Diuretics; Excitatory Amino Acid Agonists; Immunohistochemistry; Kainic Acid; Neurons; Neuroprotective Agents; Rats; Rats, Wistar; Receptor, Adenosine A1; Receptor, Adenosine A2A; Receptor, Adenosine A3

2005
Action of extracellular divalent cations on native alpha-amino-3-hydroxy-5-methylisoxazole-4-propionate (AMPA) receptors.
    Journal of neurochemistry, 2005, Volume: 95, Issue:6

    Topics: Algorithms; Animals; Benzothiadiazines; Binding, Competitive; Cations, Divalent; Excitatory Amino Acid Agonists; Extracellular Space; Hippocampus; Kainic Acid; Pyramidal Cells; Quinoxalines; Rats; Receptors, AMPA

2005
Cyclothiazide induces robust epileptiform activity in rat hippocampal neurons both in vitro and in vivo.
    The Journal of physiology, 2006, Mar-15, Volume: 571, Issue:Pt 3

    Topics: Animals; Animals, Newborn; Benzothiadiazines; Calcium; Cell Survival; Cells, Cultured; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Postsynaptic Potentials; Hippocampus; Injections, Intraventricular; Kainic Acid; Neurons; Rats; Rats, Sprague-Dawley

2006
Functional characterisation of homomeric ionotropic glutamate receptors GluR1-GluR6 in a fluorescence-based high throughput screening assay.
    Combinatorial chemistry & high throughput screening, 2006, Volume: 9, Issue:2

    Topics: Aniline Compounds; Benzothiadiazines; Calcium; Cell Line; Combinatorial Chemistry Techniques; Concanavalin A; Drug Evaluation, Preclinical; Electrophysiology; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Fluorescence; Glutamic Acid; Humans; Kainic Acid; Quinoxalines; Receptors, AMPA; Receptors, Glutamate; Signal Transduction; Xanthenes

2006
Downregulation of tonic GABA currents following epileptogenic stimulation of rat hippocampal cultures.
    The Journal of physiology, 2006, Dec-01, Volume: 577, Issue:Pt 2

    Topics: Animals; Animals, Newborn; Benzothiadiazines; Cells, Cultured; Epilepsy, Temporal Lobe; Excitatory Amino Acid Agonists; gamma-Aminobutyric Acid; Hippocampus; Inhibitory Postsynaptic Potentials; Kainic Acid; Membrane Potentials; Neural Inhibition; Neuronal Plasticity; Neurons; Patch-Clamp Techniques; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Synapses

2006
Properties of glutamate receptors of Alzheimer's disease brain transplanted to frog oocytes.
    Proceedings of the National Academy of Sciences of the United States of America, 2007, Feb-20, Volume: 104, Issue:8

    Topics: Alzheimer Disease; Animals; Anura; Benzothiadiazines; Blotting, Western; Brain Tissue Transplantation; Cell Membrane; Cerebral Cortex; Electric Conductivity; gamma-Aminobutyric Acid; Gene Expression Regulation; Glutamic Acid; Humans; Kainic Acid; Oocytes; Protein Subunits; Receptors, GABA; Receptors, Glutamate; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Time Factors

2007
Glial glutamate transporter 1 regulates the spatial and temporal coding of glutamatergic synaptic transmission in spinal lamina II neurons.
    Neuroscience, 2007, Nov-23, Volume: 149, Issue:4

    Topics: Animals; Benzothiadiazines; Dose-Response Relationship, Radiation; Drug Interactions; Electric Stimulation; Enzyme Inhibitors; Excitatory Amino Acid Transporter 2; Excitatory Postsynaptic Potentials; Glutamic Acid; In Vitro Techniques; Kainic Acid; Male; Neurons; Oligopeptides; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Spinal Cord; Synaptic Transmission

2007
The mechanisms of Zn2+ effects on Ca2+-permeable AMPA receptors on carp retinal horizontal cells.
    Brain research, 2010, Jul-23, Volume: 1345

    Topics: Animals; Benzothiadiazines; Calcium; Carps; Cells, Cultured; Extracellular Space; GABA Modulators; Glutamic Acid; Isotonic Solutions; Kainic Acid; Membrane Potentials; Neurotransmitter Agents; Patch-Clamp Techniques; Pentobarbital; Receptors, AMPA; Retinal Horizontal Cells; Ringer's Solution; Zinc

2010
Epileptiform response of CA1 neurones to convulsant stimulation by cyclothiazide, kainic acid and pentylenetetrazol in anaesthetized rats.
    Seizure, 2011, Volume: 20, Issue:4

    Topics: Animals; Benzothiadiazines; Convulsants; Electrophysiology; Excitatory Postsynaptic Potentials; Hippocampus; Injections, Intraventricular; Kainic Acid; Male; Neurons; Pentylenetetrazole; Rats; Rats, Sprague-Dawley; Seizures

2011
Inhibition of calcium-permeable and calcium-impermeable AMPA receptors by perampanel in rat brain neurons.
    Neuroscience letters, 2016, 10-28, Volume: 633

    Topics: Animals; Anticonvulsants; Benzodiazepines; Benzothiadiazines; Binding Sites; Brain; CA1 Region, Hippocampal; Calcium; Corpus Striatum; Drug Interactions; Glutamic Acid; Interneurons; Kainic Acid; Neurons; Nitriles; Pyramidal Cells; Pyridones; Rats, Wistar; Receptors, AMPA

2016