cyclothiazide and cx 614

cyclothiazide has been researched along with cx 614 in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's5 (50.00)29.6817
2010's5 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ahmed, AH; Oswald, RE1
Grove, SJ; Jamieson, C; Maclean, JK; Morrow, JA; Rankovic, Z1
Hampson, A; Harris, C; Li, YX; Marrs, C; Mueller, R; Nielsson, L; Rachwal, S; Rogers, G; Ulas, J; Zhong, S1
Arai, AC; Kessler, M; Lynch, G; Rogers, G1
Scriabine, A1
Clark, S; Dudman, JT; Gouaux, E; Jin, R; Partin, KM; Weeks, AM1
Gouliaev, AH; Harpsøe, K; Liljefors, T; Peters, D; Varming, T1
Fleck, MW; Mitchell, NA1
Benveniste, M; Harms, JE; Partin, KM; Weeks, AM1
Li, YX; Lippa, A; Purcell, R; Radin, DP; Rogers, G1

Other Studies

10 other study(ies) available for cyclothiazide and cx 614

ArticleYear
Piracetam defines a new binding site for allosteric modulators of alpha-amino-3-hydroxy-5-methyl-4-isoxazole-propionic acid (AMPA) receptors.
    Journal of medicinal chemistry, 2010, Mar-11, Volume: 53, Issue:5

    Topics: Allosteric Regulation; Binding Sites; Humans; Mutagenesis, Insertional; Nootropic Agents; Piracetam; Pyrrolidinones; Receptors, AMPA; X-Ray Diffraction

2010
Positive allosteric modulators of the α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) receptor.
    Journal of medicinal chemistry, 2010, Oct-28, Volume: 53, Issue:20

    Topics: Allosteric Regulation; Animals; Benzamides; Benzothiadiazines; Binding Sites; Excitatory Amino Acid Agents; Humans; Indazoles; Ligands; Models, Molecular; Protein Conformation; Receptors, AMPA; Sulfonamides

2010
Benzoxazinones as potent positive allosteric AMPA receptor modulators: part I.
    Bioorganic & medicinal chemistry letters, 2011, Jul-01, Volume: 21, Issue:13

    Topics: Allosteric Regulation; Animals; Benzoxazines; Molecular Structure; Nootropic Agents; Prosencephalon; Pyrrolidinones; Rats; Receptors, AMPA; Structure-Activity Relationship

2011
Effects of the potent ampakine CX614 on hippocampal and recombinant AMPA receptors: interactions with cyclothiazide and GYKI 52466.
    Molecular pharmacology, 2000, Volume: 58, Issue:4

    Topics: Alanine; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Cells, Cultured; Diuretics; Drug Interactions; Electrophysiology; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Hippocampus; Humans; In Vitro Techniques; Male; Oxazines; Pyrimidinones; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Recombinant Proteins; Sodium Chloride Symporter Inhibitors; Tritium; Uracil

2000
The Neurobiology and Neuropharmacology of Alzheimer's Disease. The ASPET - Ray Fuller Symposium. New Orleans, LA, USA, April 19-20, 2002.
    CNS drug reviews, 2002,Fall, Volume: 8, Issue:3

    Topics: Alzheimer Disease; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Humans; Neurobiology; Neuropharmacology; Neuroprotective Agents; Oxazines

2002
Mechanism of positive allosteric modulators acting on AMPA receptors.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Sep-28, Volume: 25, Issue:39

    Topics: Allosteric Regulation; Benzothiadiazines; Binding Sites; Cell Line; Crystallography; Dimerization; Drug Synergism; Electric Conductivity; Humans; Ligands; Molecular Conformation; Oxazines; Patch-Clamp Techniques; Protein Structure, Tertiary; Pyrrolidinones; Receptors, AMPA; Time Factors

2005
Identification of a putative binding site for 5-alkyl-benzothiadiazides in the AMPA receptor dimer interface.
    Journal of molecular graphics & modelling, 2007, Volume: 26, Issue:1

    Topics: Allosteric Site; Animals; Benzothiadiazines; Computer Simulation; Dimerization; In Vitro Techniques; Mice; Models, Molecular; Oxazines; Protein Structure, Quaternary; Pyrrolidinones; Receptors, AMPA; Structure-Activity Relationship

2007
Targeting AMPA receptor gating processes with allosteric modulators and mutations.
    Biophysical journal, 2007, Apr-01, Volume: 92, Issue:7

    Topics: Amino Acid Substitution; Benzothiadiazines; Cell Line; Dose-Response Relationship, Drug; Drug Delivery Systems; Humans; Ion Channel Gating; Kidney; Mutagenesis, Site-Directed; Oxazines; Receptors, AMPA; Structure-Activity Relationship; Trichlormethiazide

2007
Functional insight into development of positive allosteric modulators of AMPA receptors.
    Neuropharmacology, 2014, Volume: 85

    Topics: Benzothiadiazines; Binding Sites; Computer Simulation; Drug Discovery; Excitatory Amino Acid Agents; HEK293 Cells; Humans; Kinetics; Membrane Potentials; Models, Molecular; Mutation; Oxazines; Patch-Clamp Techniques; Receptors, AMPA; Transfection

2014
Stargazin differentially modulates ampakine gating kinetics and pharmacology.
    Biochemical pharmacology, 2018, Volume: 148

    Topics: Benzothiadiazines; Calcium Channels; Gene Expression Regulation; Glutamic Acid; HEK293 Cells; Humans; Membrane Potentials; Oxazines; Receptors, AMPA

2018