cyclothiazide and aniracetam

cyclothiazide has been researched along with aniracetam in 25 studies

Research

Studies (25)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's9 (36.00)18.2507
2000's12 (48.00)29.6817
2010's4 (16.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
de Tullio, P; Delarge, J; Diouf, O; Dupont, L; Lebrun, P; Lepagnol, J; Lestage, P; Morain, P; Pirotte, B; Podona, T; Somers, F; Spedding, M1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
England, PM; Fleming, JJ1
Ahmed, AH; Oswald, RE1
Grove, SJ; Jamieson, C; Maclean, JK; Morrow, JA; Rankovic, Z1
Hampson, A; Harris, C; Li, YX; Marrs, C; Mueller, R; Nielsson, L; Rachwal, S; Rogers, G; Ulas, J; Zhong, S1
Chaudhary, A; Johansen, TH; Verdoorn, TA1
Camici, O; Corazzi, L; Fallarino, F; Fioretti, MC; Genazzani, AA; L'Episcopo, MR; Nicoletti, F; Silla, S1
Boxall, AR; Garthwaite, J1
Mayer, ML; Wong, LA1
Fleck, MW; Mayer, ML; Partin, KM1
Lu, T; Shen, Y; Yang, XL1
Arvigo, D; Bonfanti, A; Pittaluga, A; Raiteri, M1
Iino, M; Nakagawa, T; Ozawa, S; Sekiguchi, M; Wada, K1
Bódi, I; Gueritaud, J; Kapus, G; Pataki, A; Székely, JI; Tarnawa, I1
Closier, M; Iop, F; Lestage, P; Lockhart, B1
Bolshakov, KV; Buldakova, SL; Magazanik, LG; Tikhonov, DB1
Croucher, MJ; Patel, DR; Young, AM1
Lei, S; MacDonald, JF; Orser, BA; Reynolds, JN; Thatcher, GR1
Baumbarger, P; Muhlhauser, M; Nisenbaum, ES; Yang, CR1
Aoki, S; Nishikawa, K; Sekiguchi, M; Wada, K1
Benardo, LS; Ling, DS1
Clark, S; Dudman, JT; Gouaux, E; Jin, R; Partin, KM; Weeks, AM1
Gouliaev, AH; Harpsøe, K; Liljefors, T; Peters, D; Varming, T1
Xu-Friedman, MA; Yang, H1

Other Studies

25 other study(ies) available for cyclothiazide and aniracetam

ArticleYear
4H-1,2,4-Pyridothiadiazine 1,1-dioxides and 2,3-dihydro-4H-1,2, 4-pyridothiadiazine 1,1-dioxides chemically related to diazoxide and cyclothiazide as powerful positive allosteric modulators of (R/S)-2-amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic aci
    Journal of medicinal chemistry, 1998, Jul-30, Volume: 41, Issue:16

    Topics: Adenosine Triphosphate; Allosteric Regulation; Animals; Benzothiadiazines; Cerebral Cortex; Cyclic S-Oxides; Diazoxide; Drug Design; Excitatory Postsynaptic Potentials; Hippocampus; In Vitro Techniques; Insulin; Insulin Antagonists; Insulin Secretion; Islets of Langerhans; Male; Mice; Mice, Inbred DBA; Oocytes; Potassium Channels; Rats; Rats, Wistar; Receptors, AMPA; RNA, Messenger; Solubility; Stereoisomerism; Structure-Activity Relationship; Thiadiazines; Xenopus laevis

1998
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Developing a complete pharmacology for AMPA receptors: a perspective on subtype-selective ligands.
    Bioorganic & medicinal chemistry, 2010, Feb-15, Volume: 18, Issue:4

    Topics: Allosteric Regulation; Animals; Binding Sites; Ligands; Receptors, AMPA

2010
Piracetam defines a new binding site for allosteric modulators of alpha-amino-3-hydroxy-5-methyl-4-isoxazole-propionic acid (AMPA) receptors.
    Journal of medicinal chemistry, 2010, Mar-11, Volume: 53, Issue:5

    Topics: Allosteric Regulation; Binding Sites; Humans; Mutagenesis, Insertional; Nootropic Agents; Piracetam; Pyrrolidinones; Receptors, AMPA; X-Ray Diffraction

2010
Positive allosteric modulators of the α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) receptor.
    Journal of medicinal chemistry, 2010, Oct-28, Volume: 53, Issue:20

    Topics: Allosteric Regulation; Animals; Benzamides; Benzothiadiazines; Binding Sites; Excitatory Amino Acid Agents; Humans; Indazoles; Ligands; Models, Molecular; Protein Conformation; Receptors, AMPA; Sulfonamides

2010
Benzoxazinones as potent positive allosteric AMPA receptor modulators: part I.
    Bioorganic & medicinal chemistry letters, 2011, Jul-01, Volume: 21, Issue:13

    Topics: Allosteric Regulation; Animals; Benzoxazines; Molecular Structure; Nootropic Agents; Prosencephalon; Pyrrolidinones; Rats; Receptors, AMPA; Structure-Activity Relationship

2011
Interactions among GYKI-52466, cyclothiazide, and aniracetam at recombinant AMPA and kainate receptors.
    Molecular pharmacology, 1995, Volume: 48, Issue:5

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Excitatory Amino Acid Antagonists; Humans; Pyrrolidinones; Receptors, AMPA; Receptors, Kainic Acid; Recombinant Proteins; Xenopus laevis

1995
[3H]aniracetam binds to specific recognition sites in brain membranes.
    Journal of neurochemistry, 1995, Volume: 65, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Binding Sites; Brain; Cells, Cultured; Cerebellum; Glutamic Acid; Male; Membranes; Phorbol 12,13-Dibutyrate; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Tissue Distribution; Tritium

1995
Synaptic excitation mediated by AMPA receptors in rat cerebellar slices is selectively enhanced by aniracetam and cyclothiazide.
    Neurochemical research, 1995, Volume: 20, Issue:5

    Topics: Animals; Benzothiadiazines; Cerebellum; In Vitro Techniques; Pyrrolidinones; Rats; Rats, Wistar; Receptors, AMPA; Stimulation, Chemical; Synaptic Transmission

1995
Differential modulation by cyclothiazide and concanavalin A of desensitization at native alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid- and kainate-preferring glutamate receptors.
    Molecular pharmacology, 1993, Volume: 44, Issue:3

    Topics: Alanine; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Concanavalin A; Ganglia, Spinal; Hippocampus; Ibotenic Acid; In Vitro Techniques; Kainic Acid; Neurons; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Glutamate; Receptors, Kainic Acid

1993
AMPA receptor flip/flop mutants affecting deactivation, desensitization, and modulation by cyclothiazide, aniracetam, and thiocyanate.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1996, Nov-01, Volume: 16, Issue:21

    Topics: Alternative Splicing; Amino Acid Sequence; Antihypertensive Agents; Benzothiadiazines; Cell Line; Fetus; Fibroblasts; Humans; Ion Channel Gating; Kidney; Kinetics; Molecular Sequence Data; Mutagenesis, Site-Directed; Patch-Clamp Techniques; Pyrrolidinones; Receptors, AMPA; Sensitivity and Specificity; Thiocyanates

1996
Modulation of desensitization at glutamate receptors in isolated crucian carp horizontal cells by concanavalin A, cyclothiazide, aniracetam and PEPA.
    Neuroscience, 1999, Volume: 89, Issue:3

    Topics: Animals; Aspartic Acid Endopeptidases; Benzothiadiazines; Concanavalin A; Goldfish; Nootropic Agents; Patch-Clamp Techniques; Pyrrolidinones; Receptors, AMPA; Receptors, Glutamate; Receptors, Kainic Acid

1999
Aniracetam, 1-BCP and cyclothiazide differentially modulate the function of NMDA and AMPA receptors mediating enhancement of noradrenaline release in rat hippocampal slices.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 359, Issue:4

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Antihypertensive Agents; Benzothiadiazines; Dioxoles; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Heterocyclic Compounds; Hippocampus; In Vitro Techniques; Kynurenic Acid; Male; N-Methylaspartate; Nootropic Agents; Norepinephrine; Piperidines; Pyrrolidinones; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Tritium

1999
Potentiating effects of 4-[2-(phenylsulfonylamino)ethylthio]-2,6-difluoro-phenoxyaceta mide (PEPA) on excitatory synaptic transmission in dentate granule cells.
    Neuroscience research, 1999, Dec-01, Volume: 35, Issue:3

    Topics: Animals; Antihypertensive Agents; Aspartic Acid Endopeptidases; Benzothiadiazines; Dentate Gyrus; Excitatory Amino Acids; Male; Neurons; Nootropic Agents; Pyrrolidinones; Rats; Rats, Wistar; Synapses; Synaptic Transmission

1999
Differential modulation of the GYKI 53784-induced inhibition of AMPA currents by various AMPA-positive modulators in cerebellar Purkinje cells.
    European journal of pharmacology, 2000, May-26, Volume: 397, Issue:1

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Cells, Cultured; Cerebellum; Dioxoles; Dose-Response Relationship, Drug; Drug Synergism; Excitatory Amino Acid Antagonists; Membrane Potentials; Piperidines; Purkinje Cells; Pyrrolidinones; Rats; Receptors, AMPA

2000
(S)-2,3-dihydro-[3,4]cyclopentano-1,2,4-benzothiadiazine-1,1-dioxide: (S18986-1) a positive modulator of AMPA receptors enhances (S)-AMPA-mediated [3H]noradrenaline release from rat hippocampal and frontal cortex slices.
    European journal of pharmacology, 2000, Aug-04, Volume: 401, Issue:2

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Calcium; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Synergism; Excitatory Amino Acid Antagonists; Frontal Lobe; Hippocampus; In Vitro Techniques; Male; Norepinephrine; Pyrrolidinones; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Stereoisomerism; Tetrodotoxin; Tritium

2000
Ca2+-dependent desensitization of AMPA receptors.
    Neuroreport, 2000, Sep-11, Volume: 11, Issue:13

    Topics: Adamantane; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Alternative Splicing; Animals; Animals, Newborn; Antihypertensive Agents; Benzothiadiazines; Calcium; Calcium Signaling; Dose-Response Relationship, Drug; Glutamic Acid; Hippocampus; Kainic Acid; Neurons; Nootropic Agents; Pyrrolidinones; Rats; Receptors, AMPA

2000
Presynaptic alpha-amino-3-hydroxy-5-methyl-4-isoxazole propionate receptor-mediated stimulation of glutamate and GABA release in the rat striatum in vivo: a dual-label microdialysis study.
    Neuroscience, 2001, Volume: 102, Issue:1

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Anxiety Agents; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Calcium; Carbon Radioisotopes; Corpus Striatum; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Kynurenic Acid; Male; Microdialysis; Nootropic Agents; Potassium; Presynaptic Terminals; Pyrrolidinones; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Tritium

2001
Positive allosteric modulators of AMPA receptors reduce proton-induced receptor desensitization in rat hippocampal neurons.
    Journal of neurophysiology, 2001, Volume: 85, Issue:5

    Topics: Allosteric Regulation; Animals; Benzothiadiazines; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Hippocampus; Hydrogen-Ion Concentration; Ion Channel Gating; Nerve Tissue Proteins; Neurons; Nitrates; Patch-Clamp Techniques; Protons; Pyrrolidinones; Rats; Rats, Wistar; Receptors, AMPA; Wheat Germ Agglutinins

2001
LY392098, a novel AMPA receptor potentiator: electrophysiological studies in prefrontal cortical neurons.
    Neuropharmacology, 2001, Volume: 40, Issue:8

    Topics: Action Potentials; Animals; Benzothiadiazines; Diuretics; Dose-Response Relationship, Drug; Drug Synergism; Excitatory Amino Acid Agonists; Male; Neurons; Prefrontal Cortex; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Sodium Chloride Symporter Inhibitors; Sulfonamides; Thiophenes

2001
A desensitization-selective potentiator of AMPA-type glutamate receptors.
    British journal of pharmacology, 2002, Volume: 136, Issue:7

    Topics: Allosteric Regulation; Animals; Benzothiadiazines; In Vitro Techniques; Kinetics; Oocytes; Patch-Clamp Techniques; Phenoxyacetates; Pyrrolidinones; Rats; Receptors, AMPA; Xenopus

2002
Nootropic agents enhance the recruitment of fast GABAA inhibition in rat neocortex.
    Cerebral cortex (New York, N.Y. : 1991), 2005, Volume: 15, Issue:7

    Topics: Animals; Antihypertensive Agents; Benzothiadiazines; Cognition; Concanavalin A; Evoked Potentials; Neocortex; Neural Inhibition; Nootropic Agents; Pyramidal Cells; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Receptors, GABA-A

2005
Mechanism of positive allosteric modulators acting on AMPA receptors.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Sep-28, Volume: 25, Issue:39

    Topics: Allosteric Regulation; Benzothiadiazines; Binding Sites; Cell Line; Crystallography; Dimerization; Drug Synergism; Electric Conductivity; Humans; Ligands; Molecular Conformation; Oxazines; Patch-Clamp Techniques; Protein Structure, Tertiary; Pyrrolidinones; Receptors, AMPA; Time Factors

2005
Identification of a putative binding site for 5-alkyl-benzothiadiazides in the AMPA receptor dimer interface.
    Journal of molecular graphics & modelling, 2007, Volume: 26, Issue:1

    Topics: Allosteric Site; Animals; Benzothiadiazines; Computer Simulation; Dimerization; In Vitro Techniques; Mice; Models, Molecular; Oxazines; Protein Structure, Quaternary; Pyrrolidinones; Receptors, AMPA; Structure-Activity Relationship

2007
Relative roles of different mechanisms of depression at the mouse endbulb of Held.
    Journal of neurophysiology, 2008, Volume: 99, Issue:5

    Topics: Animals; Benzothiadiazines; Cochlear Nucleus; Diuretics; Excitatory Postsynaptic Potentials; In Vitro Techniques; Mice; Mice, Inbred CBA; Models, Neurological; Neuronal Plasticity; Neurons; Nootropic Agents; Pyrrolidinones; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission

2008