cyclohexanol has been researched along with colforsin in 31 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 14 (45.16) | 18.2507 |
2000's | 12 (38.71) | 29.6817 |
2010's | 5 (16.13) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Gérard, CM; Mollereau, C; Parmentier, M; Vassart, G | 1 |
De Costa, BR; Groen, BG; Herkenham, M; Lynn, AB; Richfield, EK | 1 |
Cook, SA; Lichtman, AH; Martin, BR; Welch, SP | 1 |
Elwing, H; Karlsson, JO; Lundström, KI; Mårtensson, LG; Odman, S; Svensson, SP | 1 |
Kaminski, NE | 1 |
Axelrod, J; Briley, EM; Devane, WA; Felder, CC; Mackie, K; Simpson, JT | 1 |
Abood, M; Fan, F; Martin, BR; Tao, Q | 1 |
Barth, F; Bouaboula, M; Calandra, B; Casellas, P; Ferrara, P; Le Fur, G; Oustric, D; Rinaldi-Carmona, M; Shire, D | 1 |
Hawksworth, GM; Joe-Adigwe, G; Pertwee, RG | 1 |
Berrendero, F; Cebeira, M; de Miguel, R; Fernández-Ruiz, JJ; García-Gil, L; Hernández, ML; Ramos, JA; Romero, J | 1 |
Bonhaus, DW; Chang, LK; Kwan, J; Martin, GR | 1 |
Howlett, AC; Meschler, JP | 1 |
Brockie, HC; Makriyannis, A; Murphy, VL; Pertwee, RG; Ross, RA; Stevenson, LA; Templeton, F | 1 |
Crocker, P; Gibson, TM; Pertwee, RG; Razdan, RK; Ross, RA; Saha, B; Stevenson, LA | 1 |
Bouaboula, M; Casellas, P; Dornand, J; Gross, A; Liautard, JP; Marchant, J; Ouahrani-Bettache, S; Terraza, A | 1 |
Fan, X; Gonsiorek, W; Hipkin, RW; Lundell, D; Lunn, C; Narula, S | 1 |
Banner, WK; Gibson, TM; Martin, BR; Pertwee, RG; Razdan, RK; Ross, RA; Saha, B; Stevenson, LA | 1 |
Grimaldi, M; Hampson, AJ | 1 |
Fowler, CJ; Jacobsson, SO; Nilsson, O | 1 |
Engler, C; Feuerstein, TJ; Steffens, M; Zentner, J | 1 |
Adams, M; Cassar, S; Daza, A; Kage, K; Meyer, M; Mukherjee, S; Whiteaker, K; Yao, BB | 1 |
Armstrong, H; Fong, TM; Hagmann, W; Shen, CP; Xiao, JC | 1 |
Feng, Y; Fong, TM; Francis, B; Goulet, MT; Guan, XM; Hagmann, WK; Jewell, JP; Lanza, TJ; Lao, J; Lin, LS; Liu, P; MacIntyre, DE; Marsh, DJ; Qi, H; Rosko, KM; Shah, SK; Shearman, LP; Shen, CP; Strack, AM; Stribling, DS; Tong, X; Van der Ploeg, LH; Wang, J; Xiao, JC; Xu, SS; Yu, H | 1 |
Bingham, B; Chlenov, M; Cummons, TA; Harrison, JE; He, Y; Jones, PG; Kennedy, JD; Kotnis, S; Lu, P; Piesla, MJ; Resnick, L; Smith, VA; Strassle, BW; Sun, SC; Uveges, AJ; Whiteside, GT | 1 |
Dekkers, BG; Dröge, MJ; Elzinga, CR; Gkoumassi, E; Meurs, H; Nelemans, SA; Schmidt, M; Zaagsma, J | 1 |
Bosier, B; Hermans, E; Lambert, DM | 1 |
Gertsch, J; Lazo, JS; Schreiter, B; Wang, L; Xie, XQ; Xie, Z; Zhang, Y | 1 |
Ahmad, S; Groblewski, T; Ndong, C; O'Donnell, D | 1 |
Abood, ME; Anavi-Goffer, S; Baillie, GL; Bolognini, D; Horswill, JG; McAllister, S; Pertwee, RG; Reggio, PH; Ross, RA; Stephens, GJ; Strange, PG | 1 |
Kumar, P; Song, ZH | 1 |
Ford, BM; Franks, LN; Prather, PL; Radominska-Pandya, A | 1 |
31 other study(ies) available for cyclohexanol and colforsin
Article | Year |
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Molecular cloning of a human cannabinoid receptor which is also expressed in testis.
Topics: Amino Acid Sequence; Animals; Base Sequence; Blotting, Northern; Brain Stem; Cannabinoids; Cell Line; Cloning, Molecular; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Cyclohexanols; DNA; Gene Expression; Humans; Male; Molecular Sequence Data; Receptors, Cannabinoid; Receptors, Drug; RNA; Testis; Transcription, Genetic | 1991 |
Neuronal localization of cannabinoid receptors and second messengers in mutant mouse cerebellum.
Topics: Adenylyl Cyclases; Animals; Autoradiography; Cannabinoids; Cerebellum; Colforsin; Cyclohexanols; Heterozygote; Homozygote; Mice; Mice, Neurologic Mutants; Neurons; Phorbol 12,13-Dibutyrate; Protein Kinase C; Receptors, Cannabinoid; Receptors, Drug; Second Messenger Systems; Tritium | 1991 |
Evaluation of cAMP involvement in cannabinoid-induced antinociception.
Topics: Analgesics; Animals; Colforsin; Cyclic AMP; Cyclohexanols; Dronabinol; Injections, Intraventricular; Injections, Spinal; Male; Mice; Mice, Inbred ICR; Rats; Rats, Sprague-Dawley | 1995 |
Effects of odorants on pigment aggregation and cAMP in fish melanophores.
Topics: 1-Octanol; Acrolein; Adaptation, Physiological; Adenylyl Cyclases; Animals; Benzaldehydes; Colforsin; Cyclic AMP; Cyclohexanols; Enzyme Activation; Eucalyptol; Fishes; Melanocytes; Melanophores; Menthol; Monoterpenes; Norepinephrine; Norisoprenoids; Octanols; Odorants; Receptors, Adrenergic, alpha; Second Messenger Systems; Skin Pigmentation; Smell; Terpenes | 1994 |
Evidence for a cannabinoid receptor in immunomodulation by cannabinoid compounds.
Topics: Adenylyl Cyclases; Animals; Cannabinoids; Cells, Cultured; Colforsin; Cyclohexanols; Dronabinol; Female; Immunity; Immunoglobulin M; Mice; Receptors, Cannabinoid; Receptors, Drug; Spleen; Stereoisomerism | 1993 |
Anandamide, an endogenous cannabimimetic eicosanoid, binds to the cloned human cannabinoid receptor and stimulates receptor-mediated signal transduction.
Topics: Amides; Animals; Arachidonic Acids; Binding, Competitive; Calcium Channels; Cannabinoids; Cell Membrane; CHO Cells; Cloning, Molecular; Colforsin; Cricetinae; Cyclic AMP; Cyclohexanols; Endocannabinoids; Fatty Acids, Unsaturated; Humans; Kinetics; Pertussis Toxin; Polyunsaturated Alkamides; Radioligand Assay; Receptors, Cannabinoid; Receptors, Drug; Signal Transduction; Structure-Activity Relationship; Transfection; Tritium; Virulence Factors, Bordetella | 1993 |
Cannabinoid receptor down-regulation without alteration of the inhibitory effect of CP 55,940 on adenylyl cyclase in the cerebellum of CP 55,940-tolerant mice.
Topics: Adenylyl Cyclase Inhibitors; Animals; Body Temperature Regulation; Cannabinoids; Cerebellum; Colforsin; Cyclohexanols; Down-Regulation; Drug Tolerance; Enzyme Inhibitors; Male; Mice; Mice, Inbred ICR; Motor Activity; Receptors, Cannabinoid; Receptors, Drug; RNA, Messenger; Species Specificity | 1996 |
Characterization of two cloned human CB1 cannabinoid receptor isoforms.
Topics: Analgesics; Animals; Binding, Competitive; Cell Membrane; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Cyclohexanols; Dose-Response Relationship, Drug; Humans; Receptors, Cannabinoid; Receptors, Drug | 1996 |
Further evidence for the presence of cannabinoid CB1 receptors in mouse vas deferens.
Topics: Animals; Cannabinoids; Colforsin; Cyclic AMP; Cyclohexanols; In Vitro Techniques; Male; Mice; Piperidines; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Stereoisomerism; Vas Deferens | 1996 |
Localization of mRNA expression and activation of signal transduction mechanisms for cannabinoid receptor in rat brain during fetal development.
Topics: Animals; Autoradiography; Benzoxazines; Brain; Colforsin; Cyclic AMP; Cyclohexanols; Dronabinol; Gene Expression Regulation, Developmental; Gestational Age; Guanosine 5'-O-(3-Thiotriphosphate); In Situ Hybridization; Morpholines; Naphthalenes; Neuroglia; Protein Binding; Rats; Rats, Wistar; Receptors, Cannabinoid; Receptors, Drug; RNA, Messenger; Signal Transduction | 1998 |
Dual activation and inhibition of adenylyl cyclase by cannabinoid receptor agonists: evidence for agonist-specific trafficking of intracellular responses.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Arachidonic Acids; Benzoxazines; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Cyclohexanols; Dronabinol; Endocannabinoids; Enzyme Activation; Humans; Morpholines; Naphthalenes; Polyunsaturated Alkamides; Receptors, Cannabinoid; Receptors, Drug; Signal Transduction; Transfection | 1998 |
Thujone exhibits low affinity for cannabinoid receptors but fails to evoke cannabimimetic responses.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Artemisia; Behavior, Animal; Bicyclic Monoterpenes; Binding, Competitive; Brain Chemistry; Cannabinoids; Colforsin; Cyclohexanols; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; In Vitro Techniques; Male; Monoterpenes; Palatine Tonsil; Plants, Medicinal; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB2; Receptors, Cannabinoid; Receptors, Drug; Signal Transduction; Terpenes | 1999 |
Agonist-inverse agonist characterization at CB1 and CB2 cannabinoid receptors of L759633, L759656, and AM630.
Topics: Animals; Benzoxazines; Binding, Competitive; Camphanes; Cannabinoids; CHO Cells; Chromans; Colforsin; Cricetinae; Cyclic AMP; Cyclohexanols; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Indoles; Morpholines; Naphthalenes; Pyrazoles; Radioligand Assay; Receptors, Cannabinoid; Receptors, Drug; Tritium | 1999 |
Structural determinants of the partial agonist-inverse agonist properties of 6'-azidohex-2'-yne-delta8-tetrahydrocannabinol at cannabinoid receptors.
Topics: Animals; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Cyclohexanols; Dronabinol; Electric Stimulation; In Vitro Techniques; Male; Mice; Muscle Contraction; Receptors, Cannabinoid; Receptors, Drug; Structure-Activity Relationship; Vas Deferens | 1999 |
A beneficial aspect of a CB1 cannabinoid receptor antagonist: SR141716A is a potent inhibitor of macrophage infection by the intracellular pathogen Brucella suis.
Topics: Animals; Anti-Bacterial Agents; Antigens, CD; Benzoxazines; Brucella; Calcitriol; Camphanes; Cell Differentiation; Cell Line; Colforsin; Cyclic AMP; Cyclohexanols; Dose-Response Relationship, Drug; Humans; Intercellular Adhesion Molecule-1; Macrophage Activation; Macrophages; Mice; Monocytes; Morpholines; Naphthalenes; Phagocytosis; Piperidines; Pyrazoles; Reactive Oxygen Species; Receptors, Cannabinoid; Receptors, Drug; Rimonabant | 2000 |
Endocannabinoid 2-arachidonyl glycerol is a full agonist through human type 2 cannabinoid receptor: antagonism by anandamide.
Topics: Animals; Arachidonic Acids; Binding, Competitive; Calcium Channel Blockers; Cannabinoid Receptor Modulators; Cannabinoids; Cell Membrane; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Cyclohexanols; Drug Antagonism; Endocannabinoids; Glycerides; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Immunosuppressive Agents; Insecta; Polyunsaturated Alkamides; Receptors, Cannabinoid; Receptors, Drug; Sulfur Radioisotopes; Transfection | 2000 |
O-1057, a potent water-soluble cannabinoid receptor agonist with antinociceptive properties.
Topics: Analgesics; Analgesics, Non-Narcotic; Animals; Binding, Competitive; Cannabinoids; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Cyclohexanols; Dronabinol; Drug Interactions; Guinea Pigs; Male; Mice; Mice, Inbred ICR; Muscle Contraction; Rats; Receptor, Cannabinoid, CB2; Receptors, Cannabinoid; Receptors, Drug; Solubility; Tritium; Vas Deferens; Water | 2000 |
Cannabinoid receptor activation and elevated cyclic AMP reduce glutamate neurotoxicity.
Topics: Animals; Bucladesine; Calcium; Calcium Channels; Cannabinoids; Colforsin; Cyclic AMP; Cyclohexanols; Glutamic Acid; Neurotoxins; Rats; Rats, Wistar; Receptors, Cannabinoid; Receptors, Drug | 2001 |
Cannabinoid CB1 receptor activation does not prevent the toxicity of glutamate towards embryonic chick telencephalon primary cultures.
Topics: Animals; Arachidonic Acids; Cannabinoids; Cells, Cultured; Chick Embryo; Colforsin; Cyclic AMP; Cyclohexanols; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Combinations; Endocannabinoids; Excitatory Amino Acid Antagonists; Glutamic Acid; L-Lactate Dehydrogenase; Models, Animal; Neurons; Pipecolic Acids; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptor, Cannabinoid, CB1; Telencephalon | 2003 |
Cannabinoid CB1 receptor-mediated modulation of evoked dopamine release and of adenylyl cyclase activity in the human neocortex.
Topics: Adenylyl Cyclases; Amygdala; Animals; Arachidonic Acids; Benzoxazines; Binding Sites; Colforsin; Cyclic AMP; Cyclohexanols; Dopamine; Dronabinol; Electric Stimulation; Endocannabinoids; Female; Humans; Ligands; Male; Morpholines; Naphthalenes; Neocortex; Piperidines; Polyunsaturated Alkamides; Potassium; Pyrazoles; Rats; Receptor, Cannabinoid, CB1; Synaptosomes; Tetrodotoxin; Tritium | 2004 |
Species comparison and pharmacological characterization of rat and human CB2 cannabinoid receptors.
Topics: Animals; Arachidonic Acids; Benzoxazines; Binding, Competitive; Calcium; Cell Line; Chromones; Colforsin; Cyclic AMP; Cyclohexanols; DNA, Complementary; Dose-Response Relationship, Drug; Endocannabinoids; Glycerides; Humans; Indoles; Morpholines; Naphthalenes; Polyunsaturated Alkamides; Radioligand Assay; Rats; Receptor, Cannabinoid, CB2; Species Specificity; Transfection; Tritium | 2004 |
F200A substitution in the third transmembrane helix of human cannabinoid CB1 receptor converts AM2233 from receptor agonist to inverse agonist.
Topics: Alanine; Amino Acid Substitution; Animals; Binding Sites; Binding, Competitive; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Cyclohexanols; Dose-Response Relationship, Drug; Gene Expression; Humans; Indoles; Molecular Structure; Pertussis Toxin; Phenylalanine; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Tritium | 2006 |
Antiobesity efficacy of a novel cannabinoid-1 receptor inverse agonist, N-[(1S,2S)-3-(4-chlorophenyl)-2-(3-cyanophenyl)-1-methylpropyl]-2-methyl-2-[[5-(trifluoromethyl)pyridin-2-yl]oxy]propanamide (MK-0364), in rodents.
Topics: Amides; Animals; Anti-Obesity Agents; Binding, Competitive; Body Temperature; Body Weight; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Cyclohexanols; Dose-Response Relationship, Drug; Eating; Humans; Indoles; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Molecular Structure; Obesity; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Transfection | 2007 |
Species-specific in vitro pharmacological effects of the cannabinoid receptor 2 (CB2) selective ligand AM1241 and its resolved enantiomers.
Topics: Analgesics; Animals; Benzoxazines; Calcium Channel Blockers; Camphanes; Cannabinoids; Carrageenan; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Cyclohexanols; Dose-Response Relationship, Drug; Humans; Hyperalgesia; Indoles; Mice; Morpholines; Naphthalenes; Protein Binding; Pyrazoles; Radioligand Assay; Rats; Receptor, Cannabinoid, CB2; Species Specificity; Stereoisomerism; Tritium | 2007 |
Virodhamine and CP55,940 modulate cAMP production and IL-8 release in human bronchial epithelial cells.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Analgesics; Arachidonic Acids; Blotting, Western; Bronchi; Camphanes; Cannabinoids; Cell Line; Colforsin; Cyclic AMP; Cyclohexanols; Dose-Response Relationship, Drug; Drug Antagonism; Epithelial Cells; Humans; Immunosuppressive Agents; Interleukin-8; Pertussis Toxin; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Reverse Transcriptase Polymerase Chain Reaction; Rimonabant; RNA, Messenger; Tumor Necrosis Factor-alpha | 2007 |
Concomitant activation of adenylyl cyclase suppresses the opposite influences of CB(1) cannabinoid receptor agonists on tyrosine hydroxylase expression.
Topics: Adenylyl Cyclases; Animals; Cannabinoid Receptor Modulators; Cannabinoids; Cell Line, Tumor; Colforsin; Cyclohexanols; DNA Primers; Dronabinol; Enzyme Activation; Excitatory Amino Acid Antagonists; Genes, Reporter; Luciferases; Mice; Neuroblastoma; Pertussis Toxin; Polymerase Chain Reaction; Receptor, Cannabinoid, CB1; Tetradecanoylphorbol Acetate; Transcription, Genetic; Transfection; Tyrosine 3-Monooxygenase | 2009 |
Mutagenesis and computer modeling studies of a GPCR conserved residue W5.43(194) in ligand recognition and signal transduction for CB2 receptor.
Topics: Adenylyl Cyclases; Amino Acid Substitution; Benzoxazines; Binding Sites; Binding, Competitive; Camphanes; Cell Line, Transformed; Cell Membrane; Colforsin; Computer Simulation; Cyclic AMP; Cyclohexanols; HEK293 Cells; Humans; Ligands; Models, Molecular; Morpholines; Mutagenesis, Site-Directed; Naphthalenes; Protein Binding; Pyrazoles; Receptor, Cannabinoid, CB2; Receptors, G-Protein-Coupled; Recombinant Proteins; Signal Transduction | 2011 |
Cloning and pharmacological characterization of the dog cannabinoid CB₂receptor.
Topics: Amino Acid Sequence; Animals; Arachidonic Acids; Base Sequence; Benzoxazines; Binding, Competitive; Camphanes; CHO Cells; Cloning, Molecular; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Cyclohexanols; Dogs; Dronabinol; Endocannabinoids; Humans; Mice; Molecular Sequence Data; Morpholines; Naphthalenes; Pan troglodytes; Polyunsaturated Alkamides; Pyrazoles; Rats; Receptor, Cannabinoid, CB2; Sequence Alignment | 2011 |
CB(1) receptor allosteric modulators display both agonist and signaling pathway specificity.
Topics: Allosteric Regulation; Animals; Arrestins; Benzoxazines; beta-Arrestins; Brain; Cell Line; Cell Membrane; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Cyclohexanols; Guanosine 5'-O-(3-Thiotriphosphate); HEK293 Cells; Humans; Indoles; Kinetics; Ligands; Male; MAP Kinase Signaling System; Mice; Morpholines; Naphthalenes; Phosphorylation; Piperidines; Protein Binding; Receptor, Cannabinoid, CB1; Signal Transduction | 2013 |
Identification of raloxifene as a novel CB2 inverse agonist.
Topics: Benzoxazines; Binding, Competitive; Bone Density Conservation Agents; Colforsin; Cyclic AMP; Cyclohexanols; Dose-Response Relationship, Drug; Dronabinol; Drug Approval; Drug Evaluation, Preclinical; HEK293 Cells; Humans; Morpholines; Naphthalenes; Raloxifene Hydrochloride; Receptor, Cannabinoid, CB2; Transfection; Tritium; United States; United States Food and Drug Administration | 2013 |
Tamoxifen Isomers and Metabolites Exhibit Distinct Affinity and Activity at Cannabinoid Receptors: Potential Scaffold for Drug Development.
Topics: Adenylyl Cyclases; Animals; Binding, Competitive; Breast Neoplasms; Cannabinoid Receptor Agonists; Cannabinoid Receptor Antagonists; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Cyclohexanols; Female; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Indoles; Isomerism; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Selective Estrogen Receptor Modulators; Tamoxifen | 2016 |