cyclo(sulfoalanyl-prolyl-valyl-leucyl-tryptophyl) has been researched along with bq 123 in 3 studies
| Studies (cyclo(sulfoalanyl-prolyl-valyl-leucyl-tryptophyl)) | Trials (cyclo(sulfoalanyl-prolyl-valyl-leucyl-tryptophyl)) | Recent Studies (post-2010) (cyclo(sulfoalanyl-prolyl-valyl-leucyl-tryptophyl)) | Studies (bq 123) | Trials (bq 123) | Recent Studies (post-2010) (bq 123) |
|---|---|---|---|---|---|
| 9 | 0 | 0 | 1,391 | 63 | 152 |
| Protein | Taxonomy | cyclo(sulfoalanyl-prolyl-valyl-leucyl-tryptophyl) (IC50) | bq 123 (IC50) |
|---|---|---|---|
| Endothelin-1 receptor | Homo sapiens (human) | 0.017 | |
| Endothelin-1 receptor | Rattus norvegicus (Norway rat) | 0.014 |
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 3 (100.00) | 18.2507 |
| 2000's | 0 (0.00) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Fukami, T; Fukuroda, T; Ihara, M; Ishikawa, K; Kimura, S; Nishikibe, M; Noguchi, K; Saeki, T; Tsuchida, S; Yano, M | 1 |
| Fukami, T; Ihara, M; Ishikawa, K; Ohwaki, K; Ozaki, S; Towers, P; Yamanaka, R; Yano, M | 1 |
| Alves, K; Chan, CP; Hollis, GF; Jones, KL; Tung, JS; Williams, DL | 1 |
3 other study(ies) available for cyclo(sulfoalanyl-prolyl-valyl-leucyl-tryptophyl) and bq 123
| Article | Year |
|---|---|
Biological profiles of highly potent novel endothelin antagonists selective for the ETA receptor.
Topics: Amino Acid Sequence; Animals; Cell Membrane; Endothelins; In Vitro Techniques; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth, Vascular; Peptides, Cyclic; Rats; Rats, Inbred WKY; Receptors, Cell Surface; Receptors, Endothelin; Swine | 1992 |
[3H]BQ-123, a highly specific and reversible radioligand for the endothelin ETA receptor subtype.
Topics: Amino Acid Sequence; Azepines; Binding, Competitive; Endothelin Receptor Antagonists; Endothelins; Humans; Indoles; Isotope Labeling; Molecular Sequence Data; Neuroblastoma; Oligopeptides; Peptides, Cyclic; Radioligand Assay; Receptor, Endothelin A; Receptors, Endothelin; Structure-Activity Relationship; Tritium; Tumor Cells, Cultured | 1995 |
Characterization of cloned human endothelin receptors.
Topics: Animals; Base Sequence; Binding Sites; CHO Cells; Cloning, Molecular; Cricetinae; Endothelins; Female; Humans; Molecular Sequence Data; Peptides, Cyclic; Phosphatidylinositols; Receptors, Endothelin | 1993 |