Page last updated: 2024-08-22

cyclazocine and enkephalin, leucine

cyclazocine has been researched along with enkephalin, leucine in 141 studies

Research

Studies (141)

Timeframe	Studies, this research(%)	All Research%
pre-1990	132 (93.62)	18.7374
1990's	9 (6.38)	18.2507
2000's	0 (0.00)	29.6817
2010's	0 (0.00)	24.3611
2020's	0 (0.00)	2.80

Authors

Authors	Studies
Brown, B; Dettmar, PW; Dobson, PR; Lynn, AG; Metcalf, G; Morgan, BA	1
Coale, EH; Hein, DW; Herling, S; Valentino, RJ; Woods, JH	1
Casacci, F; Della Bella, D; Sassi, A	1
Downs, DA; Wiley, JN	1
Kuhar, MJ; Wamsley, JK; Zarbin, MA	1
Hoss, W; Periyasamy, S	1
Biswas, R; Maneckjee, R; Vonderhaar, BK	1
Balster, RL; Martin, BR; Todd, SL	1
Bettaney, J; Dray, A; James, IF; Ketchum, SB; Perkins, MN	1
Hanissian, SH; Tejwani, GA	1
LoPresti, D; Porreca, F; Ward, SJ	1
Magnan, J; Tiberi, M	1
Barnette, MS; Barone, FC; Callahan, JF; Grous, M; Manning, CD	1
deGroat, WC; Hisamitsu, T; Nagel, J; Roppolo, JR; Thor, KB; Tuttle, P	1
Fedynyshyn, JP; Kwiat, G; Lee, NM	1
Bueno, L; Gué, M; Junien, JL	1
Brantl, V; Liebmann, C; Schrader, U	1
Bhargava, HN; Gulati, A; Ramarao, P	2
Bhargava, HN; Ramarao, P	1
Garzon, J; Landahl, HD; Lee, NM	1
Rauch, RJ; Stephenson, JD; Stolerman, IP	1
Frey, EA; Jacobson, AE; Rice, KC; Tocque, B	1
De Souza, EB; Kuhar, MJ; Schmidt, WK	1
Imai, T; Kamikubo, K; Miura, K; Miura, Y; Miyashita, T; Murase, H; Nakamura, S; Niwa, M; Satoh, T; Tomita, A	1
Burks, TF; Fox, DA	1
Larson, DL; Lipkowski, AW; Nagase, H; Portoghese, PS; Takemori, AE	1
Ishizuka, Y; Oka, T	1
Bertelli, GM; Borea, PA; Gilli, G	1
Cicero, TJ; Nock, B; O'Connor, LH; Rajpara, A	1
Nagase, H; Portoghese, PS; Takemori, AE	1
Ho, BY; Naeseth, JS; Portoghese, PS; Takemori, AE	1
Dougall, IG; Leff, P	1
Dashwood, MR; Muddle, JR; Spyer, KM	1
Su, TP	1
Moises, HC; Walker, JM	1
Herz, A; Schiller, PW; Schulz, R; Shearman, GT	1
Bicknell, RJ; Chapman, C; Leng, G	1
Falke, NE; Fischer, EG; Martin, R	1
Illes, P; Ramme, D	1
Geppert, M; Illes, P; Jackisch, R	1
Buder, M; Fuder, H; Riers, HD; Rothacher, G	1
Brenner, AS; Geppert, M; Illes, P; Jackisch, R	1
Kirby, GC; McQueen, DS	1
Burks, TF; Deupree, D; Hruby, V; Hsiao, S; Mosberg, HI; Porreca, F; Spencer, RL	1
Lipkowski, AW; Portoghese, PS; Takemori, AE	1
Itoh, Y; Nishibori, M; Oishi, R; Saeki, K	1
Russell, NJ; Schaible, HG; Schmidt, RF	1
Benyhe, S; Borsodi, A; Hepp, J; Khan, A; Medzihradszky, K; Simon, J; Szücs, M; Wollemann, M	1
Belisle, S; Bellabarba, D; Gallo-Payet, N; Lehoux, JG; Lemaire, S; Petit, A	1
Cruciani, RA; Gainer, H; Lang, MA; Pesce, GO; Rodbard, D; Russell, JT	1
Alvinerie, M; Bueno, L; Gue, M; Honde, C; Junien, JL; Pascaud, X	1
Goodman, SR; McLaughlin, PJ; Zagon, IS	1
Coscia, CJ; Roth, BL; Spain, JW	1
Portoghese, PS; Takemori, AE	2
Boublik, J; Funder, JW; Jefferys, D	1
Hammonds, RG; Ho, CL; Li, CH	1
Ensinger, HA	1
Benyhe, S; Borsodi, A; Simon, J; Szücs, M; Wollemann, M	1
Neil, A	2
Brown, SR; Cox, BM; Werling, LL; Zarr, GD	2
Dewar, D; Jenner, P; Marsden, CD	2
Bunn, SJ; Hanley, MR; Wilkin, GP	1
Krall, S; Lynch, WC; Paden, CM; Watt, J	1
Boudouresque, F; Bourhim, N; Cantau, P; Castanas, E; Giraud, P; Oliver, C	1
Hirobe, M; Konno, F; Sato, Y; Takayanagi, I; Togashi, K	1
Bidlack, JM; Denton, RR	1
Bell, RD; Cicero, TJ	1
Bettermann, R; Illes, P	1
Itzhak, Y; Pasternak, GW	1
Glasel, JA; Myers, WE	1
Su, TP; Weissman, AD; Yeh, SY	1
Simon, EJ	1
Faden, AI; Krumins, SA	1
Brown, SR; Cote, TE; Cox, BM; Puttfarcken, P; Werling, LL	1
Brown, SR; Cox, BM; Puttfarcken, P; Werling, LL	1
Goldberg, S; Haertzen, C; Johnson, RE; Kumor, K; Su, TP; Vaupel, B	1
Liu-Chen, LY; Tam, SW	1
Bakalkin, GIa; Iarygin, KN; Kobylianskiĭ, AG; Nesterenko, PN; Pivovarov, AS	1
Bhargava, HN; Das, S	2
Gardner, EL; Vaysse, PJ; Zukin, RS	1
Portoghese, PS; Schoenecker, JW; Takemori, AE	1
Krumins, SA	1
Delay-Goyet, P; Roques, BP; Zajac, JM	1
Lovett, JA; Portoghese, PS	1
Bardon, T; Ruckebusch, Y	1
Bardon, T; Pairet, M; Ruckebusch, Y	1
Garzón, J; Lee, NM; Sánchez-Blázquez, P	1
Loh, HH; Stokes, KB	1
Corbett, AD; Gillan, MG; Kosterlitz, HW; McKnight, AT; Paterson, SJ; Robson, LE	1
Stotland, LM; Wood, PL	1
Dawson, G; McLawhon, RW; Miller, RJ; West, RE	2
Dickinson, SL; Slater, P	1
Chavkin, C; Goldstein, A; James, IF	1
Charleson, S; Wood, PL	1
Ben-Sreti, MM; Sewell, RD	1
Huidobro-Toro, JP; Lee, NM; Loh, HH; Way, EL; Yoshimura, K	1
Tung, AS; Yaksh, TL	1
Goodman, RR; Snyder, SH	1
Huidobro-Toro, JP; Way, EL; Yoshimura, K	1
Garzón, J; Jen, MF; Lee, NM	1
Herz, A	1
Fujibayashi, K; Iwama, T; Kubota, A; Satoh, M; Takagi, H; Wada, T; Yasui, M	1
Pairet, M; Ruckebusch, Y	1
Rezvani, A; Way, EL	1
Burkard, WP; Flück, N; Müller, PM	1
Livingston, A; Morris, B	1
Hylden, JL; Wilcox, GL	1
Terenius, L	1
Pasternak, GW	1
Chang, KJ; Cuatrecasas, P; Hazum, E	1
Gähwiler, BH; Maurer, R	1
Kosterlitz, HW; Paterson, SJ; Robson, LE	1
Lajtha, A; Reith, ME; Sershen, H; Vadasz, C	1
Herz, A; Shearman, GT	1
Nishimura, S; Pasternak, GW; Wolozin, BL	1
Ishizuka, Y; Kajiwara, M; Matsumiya, T; Negishi, K; Oka, T; Watanabe, Y	1
Bajusz, S; Berzétei, IP; Hársing, LG; Rónai, AZ; Vizi, ES	1
Itzhak, Y; Keren, O; Sarne, Y	1
Nishimura, S; Pasternak, GW	1
Guidotti, A; Saiani, L	1
Bearden, LJ; Snead, OC	1
Takemori, AE; Ward, SJ	1
Attali, B; Audigier, Y; Cros, J; Gouardères, C; Mazarguil, H	1
Kandasamy, SB; Williams, BA	1
Johnson, N; Pasternak, GW	1
Rothman, RB; Westfall, TC	1
Tam, SW	1
Boublik, JH; Clements, JA; Funder, JW; Herington, AC	1
Killian, A; Mack, KJ; Weyhenmeyer, JA	1
Goldstein, A; Han, JS; Xie, GX	1
Puig, MM; Vargas, ML	1
Chaillet, P; Costentin, J; Marçais-Collado, H	1
Isaacson, RL; Lanthorn, TH	1
McCarthy, PS; Sanger, DJ	1

Reviews

3 review(s) available for cyclazocine and enkephalin, leucine

Article	Year
Classification of opioid and 5-hydroxytryptamine receptors by means of discriminative drug effects. Neuropharmacology, 1987, Volume: 26, Issue:7B Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Conditioning, Classical; Cyclazocine; Discrimination Learning; Dose-Response Relationship, Drug; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Lysergic Acid Diethylamide; Narcotics; Nicotine; Piperazines; Pyrimidines; Receptors, Opioid; Receptors, Serotonin; Research Design; Tetrahydronaphthalenes	1987
Recent studies on opioid receptors: heterogeneity and purification. Annals of the New York Academy of Sciences, 1986, Volume: 463 Topics: Alcohols; Animals; Brain Chemistry; Centrifugation, Density Gradient; Chromatography, Affinity; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Ethylmaleimide; Humans; Lectins; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, Phencyclidine; Solubility; Tritium; Wheat Germ Agglutinins	1986
Multiple opiate receptors and their functional significance. Journal of neural transmission. Supplementum, 1983, Volume: 18 Topics: Animals; beta-Endorphin; Brain; Cyclazocine; Dynorphins; Endorphins; Enkephalins; Ethylketocyclazocine; Morphine; Receptors, Opioid; Tissue Distribution	1983

Other Studies

138 other study(ies) available for cyclazocine and enkephalin, leucine

Article	Year
Opiate analgesics: the effect of agonist-antagonist character on prolactin secretion. The Journal of pharmacy and pharmacology, 1978, Volume: 30, Issue:10 Topics: Analgesics, Opioid; Animals; Buprenorphine; Cyclazocine; Enkephalins; Male; Morphine; Naloxone; Narcotic Antagonists; Prolactin; Rats	1978
Narcotic drug discriminations by rhesus monkeys and pigeons. NIDA research monograph, 1979, Volume: 27 Topics: Animals; Columbidae; Cyclazocine; D-Ala(2),MePhe(4),Met(0)-ol-enkephalin; Discrimination Learning; Dose-Response Relationship, Drug; Enkephalins; Ethylketocyclazocine; Etorphine; Hormones; Macaca; Macaca mulatta; Naltrexone; Narcotics; Phenazocine	1979
Opiate receptors: different ligand affinity in various brain regions. Advances in biochemical psychopharmacology, 1978, Volume: 18 Topics: Animals; Binding, Competitive; Brain; Cyclazocine; Dogs; Enkephalins; Ethanolamines; Ligands; Morphine; Morphine Derivatives; Receptors, Opioid; Stereoisomerism; Time Factors	1978
Naloxone-precipitated jumping in mice pretreated with acute injections of opioids. Life sciences, 1979, Aug-27, Volume: 25, Issue:9 Topics: Animals; Behavior, Animal; Cyclazocine; Dose-Response Relationship, Drug; Enkephalins; Heroin; Male; Methadone; Methadyl Acetate; Mice; Morphine; Naloxone; Narcotics; Pentazocine	1979
Anterograde transport of opioid receptors in rat vagus nerves and dorsal roots of spinal nerves: pharmacology and sensitivity to sodium and guanine nucleotides. Experimental brain research, 1990, Volume: 81, Issue:2 Topics: Animals; Axonal Transport; Colchicine; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guanosine Triphosphate; Male; Rats; Rats, Inbred Strains; Receptors, Opioid; Sodium Chloride; Spinal Nerve Roots; Vagus Nerve	1990
Kappa opioid receptors stimulate phosphoinositide turnover in rat brain. Life sciences, 1990, Volume: 47, Issue:3 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Brain; Cyclazocine; Dynorphins; Enkephalins; Ethylketocyclazocine; Male; Phosphatidylinositols; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa	1990
Binding of opioids to human MCF-7 breast cancer cells and their effects on growth. Cancer research, 1990, Apr-15, Volume: 50, Issue:8 Topics: Breast Neoplasms; Cell Division; Cell Line; Cell Membrane; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Estradiol; Etorphine; Female; Humans; Kinetics; Morphinans; Morphine; Receptors, Opioid; Tumor Cells, Cultured	1990
Affinity of the enantiomers of alpha- and beta-cyclazocine for binding to the phencyclidine and mu opioid receptors. Life sciences, 1990, Volume: 46, Issue:12 Topics: Animals; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Male; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Stereoisomerism	1990
Opioid receptor ligands in the neonatal rat spinal cord: binding and in vitro depression of the nociceptive responses. British journal of pharmacology, 1990, Volume: 99, Issue:3 Topics: Animals; Animals, Newborn; Benzeneacetamides; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Ethylketocyclazocine; In Vitro Techniques; Kinetics; Ligands; Morphine; Muscle, Smooth, Vascular; Naloxone; Narcotics; Nociceptors; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Spinal Cord	1990
Modulation of mu, delta and kappa opioid receptors in rat brain by metal ions and histidine. Neuropharmacology, 1990, Volume: 29, Issue:5 Topics: Animals; Brain Chemistry; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalins; Ethylketocyclazocine; Histidine; Kinetics; Male; Membranes; Oligopeptides; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Sulfhydryl Reagents; Trace Elements; Zinc	1990
Opioid agonist affinity in the guinea-pig ileum and mouse vas deferens. European journal of pharmacology, 1990, Apr-10, Volume: 179, Issue:1-2 Topics: Animals; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; Ileum; Male; Methadone; Mice; Morphine; Morphine Derivatives; Naltrexone; Receptors, Opioid; Vas Deferens	1990
Demonstration of the heterogeneity of the kappa-opioid receptors in guinea-pig cerebellum using selective and nonselective drugs. European journal of pharmacology, 1990, Jun-12, Volume: 188, Issue:6 Topics: Animals; Benzeneacetamides; Benzomorphans; Binding, Competitive; Cerebellum; Computers; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Ethylketocyclazocine; Guinea Pigs; In Vitro Techniques; Kinetics; Male; Membranes; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu	1990
Inhibition of neuronally induced relaxation of canine lower esophageal sphincter by opioid peptides. European journal of pharmacology, 1990, Jul-03, Volume: 182, Issue:2 Topics: Animals; Autonomic Nervous System; Cyclazocine; D-Ala(2),MePhe(4),Met(0)-ol-enkephalin; Dogs; Electric Stimulation; Endorphins; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Esophagogastric Junction; Ethylketocyclazocine; In Vitro Techniques; Muscle Relaxation; Muscle, Smooth; Neurons; Phenazocine	1990
Selective inhibitory effects of ethylketocyclazocine on reflex pathways to the external urethral sphincter of the cat. The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:3 Topics: Animals; Cats; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Female; Morphine; Naloxone; Oligopeptides; Receptors, Opioid; Receptors, Opioid, kappa; Reflex; Urethra; Urinary Bladder; Urinary Incontinence	1989
Characterization of high affinity opioid binding sites in rat periaqueductal gray P2 membrane. European journal of pharmacology, 1989, Jan-02, Volume: 159, Issue:1 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Ethylketocyclazocine; In Vitro Techniques; Male; Membranes; Periaqueductal Gray; Pyrrolidines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Opioid	1989
Central and peripheral opioid modulation of gastric relaxation induced by feeding in dogs. The Journal of pharmacology and experimental therapeutics, 1989, Volume: 250, Issue:3 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Cyclazocine; Dogs; Dose-Response Relationship, Drug; Eating; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Ethylketocyclazocine; Morphine; Muscle Relaxation; Naloxone; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Stomach; Vagotomy; Vagus Nerve	1989
Opioid receptor affinities of the blood-derived tetrapeptides hemorphin and cytochrophin. European journal of pharmacology, 1989, Aug-03, Volume: 166, Issue:3 Topics: Animals; Brain Chemistry; Cyclazocine; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Female; Guinea Pigs; Hemoglobins; In Vitro Techniques; Male; Peptide Fragments; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu	1989
Changes in multiple opioid receptors in regions of the brain in rats treated chronically with thyroxine. Neuropharmacology, 1989, Volume: 28, Issue:9 Topics: Animals; Blood Pressure; Body Weight; Brain; Chromatography, High Pressure Liquid; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalins; Ethylketocyclazocine; Heart Rate; Hyperthyroidism; Male; Membranes; Oligopeptides; Rats; Rats, Inbred Strains; Receptors, Opioid; Thyroxine	1989
Antagonism of kappa opioid mediated effects in the rat by cyclo(Leu-Gly). Life sciences, 1989, Volume: 45, Issue:26 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Cerebral Cortex; Cyclazocine; Diuresis; Drug Tolerance; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Male; Neuropeptides; Peptides, Cyclic; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Spinal Cord	1989
Computer analysis of the effect of beta-endorphin and dynorphin and related compounds on opioid binding to mouse brain membrane. Computers in biology and medicine, 1989, Volume: 19, Issue:3 Topics: Animals; beta-Endorphin; Binding, Competitive; Brain; Cyclazocine; Dihydromorphine; Dynorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Mice; Models, Neurological; Receptors, Opioid	1989
The mu-opioid receptor in the 7315c tumor cell. European journal of pharmacology, 1987, Nov-03, Volume: 143, Issue:1 Topics: Cell Membrane; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Methionine; Enkephalins; Ethylketocyclazocine; Oligopeptides; Receptors, Opioid; Receptors, Opioid, mu; Tumor Cells, Cultured	1987
Nalbuphine: an autoradiographic opioid receptor binding profile in the central nervous system of an agonist/antagonist analgesic. The Journal of pharmacology and experimental therapeutics, 1988, Volume: 244, Issue:1 Topics: Analgesia; Animals; Autoradiography; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Haplorhini; Male; Morphinans; Nalbuphine; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Spinal Cord	1988
Varying expression of opioid receptors and GTP-binding proteins in human pheochromocytomas. NIDA research monograph, 1986, Volume: 75 Topics: Adrenal Gland Neoplasms; beta-Endorphin; Cell Membrane; Cyclazocine; Diprenorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; GTP-Binding Proteins; Humans; Pheochromocytoma; Receptors, Opioid	1986
Roles of central and peripheral mu, delta and kappa opioid receptors in the mediation of gastric acid secretory effects in the rat. The Journal of pharmacology and experimental therapeutics, 1988, Volume: 244, Issue:2 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Brain; Cyclazocine; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Ethylketocyclazocine; Gastric Acid; Male; Morphine; Naltrexone; Pyrrolidines; Quaternary Ammonium Compounds; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu	1988
Binaltorphimine-related bivalent ligands and their kappa opioid receptor antagonist selectivity. Journal of medicinal chemistry, 1988, Volume: 31, Issue:4 Topics: Animals; Chemical Phenomena; Chemistry; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Male; Mice; Models, Molecular; Morphine; Muscle, Smooth; Naltrexone; Receptors, Opioid; Receptors, Opioid, kappa; Structure-Activity Relationship	1988
Relation of diltiazem binding sites to opioid receptor subtypes in the guinea-pig brain. The Tokai journal of experimental and clinical medicine, 1987, Volume: 12, Issue:1 Topics: Animals; Binding, Competitive; Brain; Cyclazocine; Dihydromorphine; Diltiazem; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Naloxone; Radioligand Assay; Receptors, Opioid	1987
Temperature dependence of the binding of mu, delta and kappa agonists to the opiate receptors in guinea-pig brain. European journal of pharmacology, 1988, Feb-09, Volume: 146, Issue:2-3 Topics: Animals; Brain; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Temperature	1988
[3H]U-69593 labels a subtype of kappa opiate receptor with characteristics different from that labeled by [3H]ethylketocyclazocine. Life sciences, 1988, Volume: 42, Issue:23 Topics: Animals; Benzeneacetamides; Binding, Competitive; Brain; Cell Membrane; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Male; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Sodium Chloride; Temperature; Tritium	1988
Only one pharmacophore is required for the kappa opioid antagonist selectivity of norbinaltorphimine. Journal of medicinal chemistry, 1988, Volume: 31, Issue:7 Topics: Animals; Chemical Phenomena; Chemistry; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Ileum; Male; Mice; Morphine; Naltrexone; Receptors, Opioid; Receptors, Opioid, kappa; Stereoisomerism; Structure-Activity Relationship; Vas Deferens	1988
Nor-binaltorphimine, a highly selective kappa-opioid antagonist in analgesic and receptor binding assays. The Journal of pharmacology and experimental therapeutics, 1988, Volume: 246, Issue:1 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesia; Animals; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; Male; Mice; Morphine; Naltrexone; Oligopeptides; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa	1988
Estimation of opioid receptor agonist dissociation constants with beta-chlornaltrexamine, an irreversible ligand which also displays agonism. British journal of pharmacology, 1988, Volume: 95, Issue:1 Topics: Animals; Cyclazocine; Drug Interactions; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Morphinans; Muscle, Smooth; Naltrexone; Narcotic Antagonists; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu	1988
Opiate receptor subtypes in the nucleus tractus solitarii of the cat: the effect of vagal section. European journal of pharmacology, 1988, Oct-11, Volume: 155, Issue:1-2 Topics: Animals; Autoradiography; Cats; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Ethylketocyclazocine; Female; Male; Medulla Oblongata; Naloxone; Receptors, Opioid; Vagotomy	1988
Effect of methimazole-induced hypothyroidism on multiple opioid receptors in rat brain regions. Pharmacology, 1988, Volume: 37, Issue:6 Topics: Animals; Body Temperature; Body Weight; Brain Chemistry; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalins; Ethylketocyclazocine; Heart Rate; Hypothyroidism; Male; Methimazole; Oligopeptides; Rats; Rats, Inbred Strains; Receptors, Opioid; Triiodothyronine	1988
Further demonstration of kappa opioid binding sites in the brain: evidence for heterogeneity. The Journal of pharmacology and experimental therapeutics, 1985, Volume: 232, Issue:1 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Binding Sites; Brain; Cyclazocine; Dynorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Etorphine; Guinea Pigs; Levallorphan; Peptide Fragments; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Stereoisomerism	1985
Electrophysiological effects of dynorphin peptides on hippocampal pyramidal cells in rat. European journal of pharmacology, 1985, Jan-15, Volume: 108, Issue:1 Topics: Animals; Cyclazocine; Dynorphins; Electrophysiology; Endorphins; Enkephalin, Leucine; Ethylketocyclazocine; gamma-Aminobutyric Acid; Hippocampus; Male; Peptide Fragments; Rats; Rats, Inbred Strains; Receptors, Opioid	1985
Generalization tests with intraventricularly applied pro-enkephalin B-derived peptides in rats trained to discriminate the opioid kappa receptor agonist ethylketocyclazocine. Psychopharmacology, 1985, Volume: 85, Issue:4 Topics: Animals; beta-Endorphin; Cyclazocine; Discrimination Learning; Dynorphins; Endorphins; Enkephalins; Ethylketocyclazocine; Generalization, Stimulus; Injections, Intraventricular; Male; Protein Precursors; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa	1985
Effects of opioid agonists and antagonists on oxytocin and vasopressin release in vitro. Neuroendocrinology, 1985, Volume: 41, Issue:2 Topics: Animals; Arginine Vasopressin; Benzomorphans; beta-Endorphin; Cyclazocine; Dynorphins; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Male; Naloxone; Oxytocin; Peptide Fragments; Pituitary Gland, Posterior; Rats; Rats, Inbred Strains	1985
Stereospecific opiate binding in living human polymorphonuclear leucocytes. Cell biology international reports, 1985, Volume: 9, Issue:11 Topics: Analgesics, Opioid; Cyclazocine; Diprenorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Granulocytes; Humans; Kinetics; Naloxone; Neutrophils; Receptors, Opioid	1985
Differential effect of stimulation strength in mouse vas deferens on inhibition of neuroeffector transmission by receptor type selective opioids. Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 332, Issue:1 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Cyclazocine; Dynorphins; Electric Stimulation; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; In Vitro Techniques; Male; Mice; Morphine Derivatives; Muscle, Smooth; Neuromuscular Junction; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Synaptic Transmission	1986
Characterization of opioid receptors modulating noradrenaline release in the hippocampus of the rabbit. Journal of neurochemistry, 1986, Volume: 46, Issue:6 Topics: Animals; Benzomorphans; Clonidine; Cyclazocine; Dynorphins; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalin, Methionine; Enkephalins; Ethylketocyclazocine; Hippocampus; Morphine; Norepinephrine; Rabbits; Receptors, Opioid	1986
On the opioid receptor subtype inhibiting the evoked release of 3H-noradrenaline from guinea-pig atria in vitro. Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 332, Issue:2 Topics: Animals; Atropine; Benzomorphans; Binding, Competitive; Corticosterone; Cyclazocine; Desipramine; Dynorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Etorphine; Guinea Pigs; Heart Atria; In Vitro Techniques; Morphine; Myocardium; Naloxone; Norepinephrine; Peptide Fragments; Phentolamine; Receptors, Opioid; Receptors, Opioid, kappa; Synapses	1986
Presynaptic opioid receptors modulating acetylcholine release in the hippocampus of the rabbit. Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 332, Issue:2 Topics: Acetylcholine; Animals; Benzomorphans; Choline; Cyclazocine; Dose-Response Relationship, Drug; Dynorphins; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Hippocampus; Naloxone; Peptide Fragments; Rabbits; Receptors, Opioid; Receptors, Opioid, kappa; Synapses	1986
Characterization of opioid receptors in the cat carotid body involved in chemosensory depression in vivo. British journal of pharmacology, 1986, Volume: 88, Issue:4 Topics: Animals; Carotid Body; Cats; Chemoreceptor Cells; Cyclazocine; Dose-Response Relationship, Drug; Dynorphins; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalin, Methionine; Enkephalins; Ethylketocyclazocine; Hypercapnia; Hypoxia; Peptide Fragments; Receptors, Opioid	1986
Centrally-administered opioid selective agonists inhibit drinking in the rat. Pharmacology, biochemistry, and behavior, 1986, Volume: 25, Issue:1 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Brain; Cyclazocine; Drinking Behavior; Dynorphins; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Ethylketocyclazocine; Male; Morphine; Naloxone; Peptide Fragments; Pyrrolidines; Rats; Receptors, Opioid	1986
Binaltorphimine and nor-binaltorphimine, potent and selective kappa-opioid receptor antagonists. Life sciences, 1987, Mar-30, Volume: 40, Issue:13 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Chemical Phenomena; Chemistry; Cyclazocine; Dynorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Male; Mice; Morphine; Naloxone; Naltrexone; Pyrrolidines; Rabbits; Receptors, Opioid; Receptors, Opioid, kappa	1987
Involvement of opioid receptors in phencyclidine-induced enhancement of brain histamine turnover in mice. Naunyn-Schmiedeberg's archives of pharmacology, 1987, Volume: 335, Issue:3 Topics: Analgesics, Opioid; Animals; Brain; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Haloperidol; Histamine; Histidine Decarboxylase; Ketamine; Male; Methylhistidines; Mice; Naloxone; Pargyline; Phenazocine; Phencyclidine; Receptors, Opioid	1987
Opiates inhibit the discharges of fine afferent units from inflamed knee joint of the cat. Neuroscience letters, 1987, Apr-23, Volume: 76, Issue:1 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Opioid; Animals; Arthritis; Cats; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Ethylketocyclazocine; Morphine; Naloxone; Nociceptors; Pain; Peripheral Nerves; Pyrrolidines	1987
Purification of a kappa-opioid receptor subtype from frog brain. Neuropeptides, 1987, Volume: 10, Issue:1 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Brain Chemistry; Chromatography, Gel; Cyclazocine; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Membranes; Molecular Weight; Naloxone; Peptide Fragments; Pyrrolidines; Rana esculenta; Receptors, Opioid; Receptors, Opioid, kappa; Solubility	1987
Functional opioid receptor sites in human placentas. The Journal of clinical endocrinology and metabolism, 1988, Volume: 66, Issue:2 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Cyclazocine; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Ethylketocyclazocine; Gonadotropin-Releasing Hormone; Humans; Kinetics; Placenta; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Thyrotropin-Releasing Hormone	1988
Opioid receptors of bovine posterior pituitary neurosecretosomes are exclusively kappa. NIDA research monograph, 1986, Volume: 75 Topics: Analgesics, Opioid; Animals; Cattle; Cyclazocine; Cytoplasmic Granules; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Etorphine; Kinetics; Morphinans; Pituitary Gland, Posterior; Receptors, Opioid; Receptors, Opioid, kappa	1986
CNS blockade of acoustic stress-induced gastric motor inhibition by kappa-opiate agonists in dogs. The American journal of physiology, 1988, Volume: 254, Issue:6 Pt 1 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Acoustic Stimulation; Adrenocorticotropic Hormone; Analgesics; Animals; Cyclazocine; Dogs; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Ethylketocyclazocine; Gastrointestinal Motility; Hydrocortisone; Pyrrolidines; Stress, Physiological	1988
Characterization of opioid binding sites in murine neuroblastoma. Brain research, 1988, May-24, Volume: 449, Issue:1-2 Topics: Analgesics, Opioid; Animals; Binding, Competitive; Cell Line; Clone Cells; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Kinetics; Ligands; Mice; Neuroblastoma; Receptors, Opioid	1988
Differential ontogeny of multiple opioid receptors (mu, delta, and kappa). The Journal of neuroscience : the official journal of the Society for Neuroscience, 1985, Volume: 5, Issue:3 Topics: Animals; Animals, Newborn; Brain; Computers; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Tritium	1985
TENA, a selective kappa opioid receptor antagonist. Life sciences, 1985, Feb-25, Volume: 36, Issue:8 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Azocines; Benzomorphans; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Ileum; Male; Mice; Naloxone; Naltrexone; Narcotic Antagonists; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Vas Deferens	1985
A kappa-selective opioidergic pathway is involved in the reversal of a behavioural effect of adrenalectomy. European journal of pharmacology, 1985, Jan-08, Volume: 107, Issue:3 Topics: Adrenalectomy; Animals; Benzomorphans; Cyclazocine; Enkephalins; Ethylketocyclazocine; Immobilization; Male; Memory; Rats; Receptors, Opioid; Receptors, Opioid, kappa	1985
Opiate receptor binding profile in the rabbit cerebellum and brain membranes. Biochemical pharmacology, 1985, Apr-01, Volume: 34, Issue:7 Topics: Animals; beta-Endorphin; Binding Sites; Binding, Competitive; Brain; Cerebellum; Cold Temperature; Cyclazocine; Dihydromorphine; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; In Vitro Techniques; Male; Rabbits; Receptors, Opioid; Sodium; Tritium	1985
Differentiating aspects of opioid receptor binding by [3H](-) (1R,5R,9R,2''S)-5,9-dimethyl-2-tetrahydrofurfuryl-2'-hydroxy-6,7- benzomorphan hydrochloride ([3H]Mr 2034), a drug preferentially acting on kappa-receptors. Arzneimittel-Forschung, 1985, Volume: 35, Issue:1A Topics: Animals; Benzomorphans; Binding, Competitive; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; In Vitro Techniques; Kinetics; Male; Morphinans; Naloxone; Rats; Receptors, Opioid; Receptors, Opioid, kappa	1985
Separation of kappa-opioid receptor subtype from frog brain. FEBS letters, 1985, Apr-22, Volume: 183, Issue:2 Topics: Animals; Brain Chemistry; Centrifugation, Density Gradient; Chromatography, Gel; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Methionine; Enkephalins; Ethylketocyclazocine; Rana esculenta; Receptors, Opioid; Receptors, Opioid, kappa	1985
Detection and characterization of four binding sites for opioids in the mouse brain. Acta pharmacologica et toxicologica, 1985, Volume: 56, Issue:2 Topics: Animals; Binding Sites; Brain Chemistry; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Models, Biological; Naloxone; Receptors, Opioid; Software; Tritium	1985
Opioid binding to rat and guinea-pig neural membranes in the presence of physiological cations at 37 degrees C. The Journal of pharmacology and experimental therapeutics, 1985, Volume: 233, Issue:3 Topics: Animals; Brain; Cations; Cyclazocine; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Guanosine Triphosphate; Guinea Pigs; In Vitro Techniques; Male; Narcotics; Rats; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Temperature; Tritium	1985
Behavioural effects in rats of unilateral and bilateral injections of opiate receptor agonists into the globus pallidus. Neuroscience, 1985, Volume: 15, Issue:1 Topics: Animals; Cyclazocine; D-Ala(2),MePhe(4),Met(0)-ol-enkephalin; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Female; Globus Pallidus; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu	1985
Evidence for a kappa-opioid receptor on pituitary astrocytes: an autoradiographic study. Neuroscience letters, 1985, Apr-19, Volume: 55, Issue:3 Topics: Animals; Astrocytes; Autoradiography; Binding Sites; Binding, Competitive; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Etorphine; Pituitary Gland; Rats; Receptors, Opioid; Receptors, Opioid, kappa	1985
Autoradiographic localization of kappa opiate receptors in CNS taste and feeding areas. Pharmacology, biochemistry, and behavior, 1985, Volume: 22, Issue:5 Topics: Animals; Autoradiography; Binding, Competitive; Brain; Corpus Striatum; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Feeding Behavior; Limbic System; Male; Morphine; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Taste	1985
Interaction of opiates with opioid binding sites in the bovine adrenal medulla: II. Interaction with kappa sites. Journal of neurochemistry, 1985, Volume: 45, Issue:3 Topics: Adrenal Medulla; Animals; Benzomorphans; Binding Sites; Calcium; Cattle; Cyclazocine; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalin, Methionine; Ethylketocyclazocine; Ethylmaleimide; Etorphine; Guinea Pigs; Kinetics; Lithium; Manganese; Narcotics; Oligopeptides; Phospholipases A; Potassium; Receptors, Opioid; Receptors, Opioid, kappa; Sodium; Stereoisomerism	1985
Interactions of codeine-7,8-oxide (codeine-epoxide), as a new metabolite of codeine, with multiple opiate receptors. General pharmacology, 1985, Volume: 16, Issue:4 Topics: Animals; Brain; Cell Membrane; Codeine; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guanosine Triphosphate; Male; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Opioid; Sodium Chloride	1985
A monoclonal antibody capable of modulating opioid binding to rat neural membranes. The Journal of biological chemistry, 1985, Dec-15, Volume: 260, Issue:29 Topics: Animals; Antibodies, Monoclonal; Cell Line; Cyclazocine; Dihydromorphine; Diprenorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Flunitrazepam; Immunoglobulin M; Kinetics; Male; Mice; Mice, Inbred BALB C; Molecular Weight; Naloxone; Narcotics; Nerve Tissue; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Opioid	1985
A radiolabeled-ligand-binding technique for the characterization of opioid receptors in the intact mouse vas deferens. Analytical biochemistry, 1985, Volume: 150, Issue:1 Topics: Animals; Binding, Competitive; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; In Vitro Techniques; Kinetics; Male; Mice; Morphine; Naltrexone; Radioligand Assay; Receptors, Opioid; Vas Deferens	1985
Classification of presynaptic opioid receptors in the rabbit ear artery by competitive antagonists. European journal of pharmacology, 1986, Mar-11, Volume: 122, Issue:1 Topics: Animals; Arteries; Benzomorphans; Binding, Competitive; Biological Assay; Cyclazocine; Ear; Enkephalin, Leucine; Ethylketocyclazocine; In Vitro Techniques; Naloxone; Rabbits; Receptors, Opioid; Synaptic Membranes	1986
Kappa-opiate binding to rat brain and guinea pig cerebellum: sensitivity towards ions and nucleotides. Neuroscience letters, 1986, Feb-14, Volume: 64, Issue:1 Topics: Animals; Brain; Cerebellum; Cyclazocine; Electrolytes; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Guanine Nucleotides; Guinea Pigs; Rats; Receptors, Opioid; Receptors, Opioid, kappa	1986
Subclass specificity of anti-idiotypic anti-opiate receptor antibodies in rat brain, guinea pig cerebellum, & neuroblastoma x glioma (NG 108-15). Life sciences, 1986, May-12, Volume: 38, Issue:19 Topics: Animals; Antibodies, Anti-Idiotypic; Binding, Competitive; Cell Line; Cerebellum; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; Morphine; Neurilemma; Neurons; Rats; Receptors, Opioid	1986
Endogenous ligands for sigma opioid receptors in the brain ("sigmaphin"): evidence from binding assays. Life sciences, 1986, Jun-16, Volume: 38, Issue:24 Topics: Animals; Binding, Competitive; Brain; Chromatography, Gel; Cyclazocine; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Kinetics; Male; Naloxone; Phenazocine; Phencyclidine; Radioligand Assay; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, Phencyclidine; Receptors, sigma	1986
Traumatic injury alters opiate receptor binding in rat spinal cord. Annals of neurology, 1986, Volume: 19, Issue:5 Topics: Animals; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Male; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Spinal Cord; Spinal Cord Injuries	1986
Sodium regulation of agonist binding at opioid receptors. I. Effects of sodium replacement on binding at mu- and delta-type receptors in 7315c and NG108-15 cells and cell membranes. Molecular pharmacology, 1986, Volume: 30, Issue:2 Topics: Adenylyl Cyclase Inhibitors; Animals; Cell Line; Cell Membrane; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Etorphine; Glioma; Guinea Pigs; Monensin; Naloxone; Neuroblastoma; Pituitary Neoplasms; Rats; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu; Sodium	1986
Sodium regulation of agonist binding at opioid receptors. II. Effects of sodium replacement on opioid binding in guinea pig cortical membranes. Molecular pharmacology, 1986, Volume: 30, Issue:2 Topics: Animals; Cell Membrane; Cerebral Cortex; Cyclazocine; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Etorphine; Guinea Pigs; Male; Oligopeptides; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Sodium	1986
Opioid ligand binding sites in the spinal cord of the guinea-pig. Neuropharmacology, 1986, Volume: 25, Issue:5 Topics: Animals; Binding, Competitive; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; In Vitro Techniques; Kinetics; Male; Membranes; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Spinal Cord	1986
Studies of kappa agonist. NIDA research monograph, 1986, Volume: 67 Topics: Animals; Brain; Cyclazocine; Enkephalin, Methionine; Enkephalins; Ethylketocyclazocine; Humans; Morphine; Naloxone; Receptors, Opioid; Receptors, Opioid, kappa	1986
Reversible and irreversible binding of beta-funaltrexamine to mu, delta and kappa opioid receptors in guinea pig brain membranes. The Journal of pharmacology and experimental therapeutics, 1986, Volume: 239, Issue:2 Topics: Animals; Brain; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Ethylmaleimide; Guinea Pigs; Kinetics; Male; Membranes; Naloxone; Naltrexone; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Sodium Chloride	1986
[Differences in opioid binding in the left and right visual cortex of the turtle]. Doklady Akademii nauk SSSR, 1986, Volume: 291, Issue:2 Topics: Animals; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Functional Laterality; Receptors, Opioid; Turtles; Visual Cortex	1986
Selective proliferation of brain kappa opiate receptors in spontaneously hypertensive rats. Life sciences, 1986, Dec-29, Volume: 39, Issue:26 Topics: Animals; Binding, Competitive; Brain; Cyclazocine; Enkephalin, Leucine; Ethylketocyclazocine; Kinetics; Male; Naltrexone; Oligopeptides; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Rats, Inbred WKY; Receptors, Opioid; Receptors, Opioid, kappa	1986
Unidirectional interaction between thyrotropin releasing hormone and opiates at the level of their brain receptors. General pharmacology, 1987, Volume: 18, Issue:1 Topics: Animals; Brain; Cyclazocine; Enkephalin, Leucine; Ethylketocyclazocine; Male; Naltrexone; Oligopeptides; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Opioid; Thyrotropin-Releasing Hormone	1987
Modulation of rat brain opioid receptors by cannabinoids. The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:2 Topics: Animals; Cannabinoids; Cyclazocine; Dihydromorphine; Dose-Response Relationship, Drug; Dronabinol; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Ethylketocyclazocine; Etorphine; Male; Naloxone; Rats; Rats, Inbred Strains; Receptors, Opioid; Spiperone	1987
Nonequilibrium opioid antagonist activity of 6,14-dideoxynaltrexone derivatives. Journal of medicinal chemistry, 1987, Volume: 30, Issue:6 Topics: Animals; Cyclazocine; Dose-Response Relationship, Drug; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Mice; Naltrexone; Narcotic Antagonists; Receptors, Opioid; Structure-Activity Relationship	1987
Opioid receptor binding in rat spinal cord. Neurochemical research, 1987, Volume: 12, Issue:3 Topics: Animals; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Ligands; Male; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Spinal Cord	1987
Differences of binding characteristics of non-selective opiates towards mu and delta receptor types. Life sciences, 1987, Aug-10, Volume: 41, Issue:6 Topics: Animals; Binding, Competitive; Brain; Cell Membrane; Cerebellum; Cyclazocine; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Ethylketocyclazocine; Etorphine; Male; Oligopeptides; Rabbits; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu	1987
Synthesis and evaluation of melphalan-containing N,N-dialkylenkephalin analogues as irreversible antagonists of the delta opioid receptor. Journal of medicinal chemistry, 1987, Volume: 30, Issue:9 Topics: Alkylation; Animals; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Melphalan; Mice; Morphine; Muscle, Smooth; Receptors, Opioid; Receptors, Opioid, delta; Structure-Activity Relationship	1987
Effects of opioid agonist drugs on the in vitro release of 3H-GABA, 3H-dopamine and 3H-5HT from slices of rat globus pallidus. Biochemical pharmacology, 1987, May-15, Volume: 36, Issue:10 Topics: Animals; Cyclazocine; D-Ala(2),MePhe(4),Met(0)-ol-enkephalin; Dopamine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Female; gamma-Aminobutyric Acid; Globus Pallidus; Potassium Chloride; Rats; Rats, Inbred Strains; Serotonin	1987
Comparative effects of opiate agonists on proximal and distal colonic motility in dogs. European journal of pharmacology, 1985, Apr-16, Volume: 110, Issue:3 Topics: Animals; Colon; Cyclazocine; Dogs; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Fentanyl; Gastrointestinal Motility; Injections, Intravenous; Injections, Spinal; Narcotics; Time Factors	1985
Opioid control of the ruminant stomach motility: functional importance of mu, kappa and delta receptors. Life sciences, 1984, Oct-22, Volume: 35, Issue:17 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalin, Methionine; Ethylketocyclazocine; Fentanyl; Gastrointestinal Motility; Morphine; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Sheep; Stomach	1984
[3H]Ethylketocyclazocine binding to mouse brain membranes: evidence for a kappa opioid receptor type. The Journal of pharmacology and experimental therapeutics, 1984, Volume: 231, Issue:1 Topics: Animals; Brain; Cyclazocine; D-Ala(2),MePhe(4),Met(0)-ol-enkephalin; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; In Vitro Techniques; Ligands; Male; Mice; Mice, Inbred ICR; Receptors, Opioid; Receptors, Opioid, kappa; Tritium	1984
Altered opiate receptor binding in synaptosomes: implication of phosphorylation. Proceedings of the Western Pharmacology Society, 1984, Volume: 27 Topics: Animals; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; In Vitro Techniques; Male; Mice; Mice, Inbred ICR; Phosphorylation; Receptors, Opioid; Synaptosomes	1984
Comparative antagonism by naltrexone and naloxone of mu, kappa, and delta agonists. European journal of pharmacology, 1984, Sep-03, Volume: 104, Issue:1-2 Topics: Animals; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Morphine; Muscle, Smooth; Naloxone; Naltrexone; Narcotic Antagonists; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Vas Deferens	1984
Radioligands for probing opioid receptors. Journal of receptor research, 1984, Volume: 4, Issue:1-6 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Binding Sites; Brain; Cyclazocine; Diprenorphine; Enkephalin, Leucine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Mice; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Naloxone; Pro-Opiomelanocortin; Protein Precursors; Pyrrolidines; Radioligand Assay; Rats; Receptors, Opioid; Vas Deferens	1984
Actions of enkephalin, mu and partial agonist analgesics on acetylcholine turnover in rat brain. Neuropharmacology, 1980, Volume: 19, Issue:10 Topics: Acetylcholine; Analgesics, Opioid; Animals; Behavior, Animal; Brain; Butorphanol; Cyclazocine; Endorphins; Enkephalins; In Vitro Techniques; Male; Nerve Tissue Proteins; Pentazocine; Rats	1980
Distinct high-affinity binding sites for benzomorphan drugs and enkephalin in a neuroblastoma--brain hybrid cell line. Proceedings of the National Academy of Sciences of the United States of America, 1981, Volume: 78, Issue:7 Topics: Analgesics, Opioid; Animals; Benzomorphans; Binding Sites; Binding, Competitive; Brain; Cell Line; Cyclazocine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Hybrid Cells; Kinetics; Morphinans; Neuroblastoma; Phenazocine; Rats; Receptors, Opioid	1981
Opiate receptor antagonism by L-prolyl-L-leucyl-glycinamide, MIF-I. Peptides, 1980,Winter, Volume: 1, Issue:4 Topics: Animals; Cyclazocine; Enkephalin, Leucine; Enkephalins; Ethylketocyclazocine; Female; Ileum; In Vitro Techniques; Male; Mice; Morphine; Motor Activity; MSH Release-Inhibiting Hormone; Muscle Contraction; Pain; Rats; Rats, Inbred Strains; Receptors, Opioid; Vas Deferens	1980
Dynorphin is a specific endogenous ligand of the kappa opioid receptor. Science (New York, N.Y.), 1982, Jan-22, Volume: 215, Issue:4531 Topics: Analgesics, Opioid; Animals; Binding, Competitive; Brain; Cyclazocine; Dynorphins; Endorphins; Enkephalin, Leucine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; In Vitro Techniques; Ligands; Morphine Derivatives; Myenteric Plexus; Naloxone; Peptide Fragments; Receptors, Opioid	1982
High affinity [3H]ethylketazocine binding: evidence for specific kappa receptors. Neuropharmacology, 1982, Volume: 21, Issue:3 Topics: Analgesics, Opioid; Animals; Cyclazocine; Enkephalins; Ethylketocyclazocine; Ethylmaleimide; Rats; Receptors, Opioid; Tritium	1982
Stereospecific inhibition of oxotremorine-induced antinociception by (+)-isomers of opioid antagonists: comparison with opioid receptor agonists. The Journal of pharmacy and pharmacology, 1982, Volume: 34, Issue:8 Topics: Animals; Benzomorphans; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Male; Mice; Morphine; Narcotic Antagonists; Nociceptors; Oxotremorine; Receptors, Opioid; Stereoisomerism	1982
Activation of K-opiate sites by dynorphin in the myenteric plexus. Advances in biochemical psychopharmacology, 1982, Volume: 33 Topics: Animals; Cyclazocine; Drug Tolerance; Dynorphins; Electric Stimulation; Endorphins; Enkephalin, Leucine; Ethylketocyclazocine; Guinea Pigs; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Narcotics; Receptors, Opioid; Receptors, Opioid, kappa	1982
In vivo evidence for multiple opiate receptors mediating analgesia in the rat spinal cord. Brain research, 1982, Sep-09, Volume: 247, Issue:1 Topics: Animals; Cyclazocine; Dose-Response Relationship, Drug; Dynorphins; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Injections, Spinal; Male; Naloxone; Pain; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Spinal Cord	1982
Kappa opiate receptors localized by autoradiography to deep layers of cerebral cortex: relation to sedative effects. Proceedings of the National Academy of Sciences of the United States of America, 1982, Volume: 79, Issue:18 Topics: Analgesics; Analgesics, Opioid; Animals; Autoradiography; Benzomorphans; Brain Stem; Cerebral Cortex; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Male; Morphine; Organ Specificity; Receptors, Opioid; Receptors, Opioid, kappa; Tritium	1982
Potency of three opiate antagonists to reverse the inhibitory activity of dynorphin, enkephalins and opioid-like alkaloids on the guinea pig ileum. European journal of pharmacology, 1982, Oct-15, Volume: 84, Issue:1-2 Topics: Animals; Azocines; Benzomorphans; Cyclazocine; Dynorphins; Endorphins; Enkephalins; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Morphine Derivatives; Muscle, Smooth; Naloxone; Narcotic Antagonists	1982
Differential modification of opiate receptor activity by arylsulfatase treatment. Biochemical pharmacology, 1983, May-01, Volume: 32, Issue:9 Topics: Analgesia; Analgesics, Opioid; Animals; Arylsulfatases; beta-Endorphin; Cyclazocine; D-Ala(2),MePhe(4),Met(0)-ol-enkephalin; Drug Antagonism; Endorphins; Enkephalin, Methionine; Enkephalins; Ethylketocyclazocine; Hormones; Kinetics; Male; Mice; Mice, Inbred ICR; Morphine; Naloxone; Receptors, Opioid; Sulfatases	1983
Comparison of analgesic potencies of mu, delta and kappa agonists locally applied to various CNS regions relevant to analgesia in rats. Life sciences, 1983, Volume: 33 Suppl 1 Topics: Analgesics, Opioid; Animals; Brain Stem; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Male; Morphine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu	1983
Opioid receptor agonists in the rabbit colon: comparison of in vivo and in vitro studies. Life sciences, 1984, Oct-15, Volume: 35, Issue:16 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Colon; Cyclazocine; Dynorphins; Electric Conductivity; Enkephalins; Ethylketocyclazocine; Fentanyl; Male; Morphine; Naloxone; Narcotics; Pyrrolidines; Rabbits; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu	1984
Dynorphin-(1-13) restores the potency of morphine on the tolerant guinea pig ileum. European journal of pharmacology, 1984, Jul-20, Volume: 102, Issue:3-4 Topics: Animals; beta-Endorphin; Cyclazocine; Drug Interactions; Drug Tolerance; Dynorphins; Endorphins; Enkephalin, Leucine; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Morphine; Muscle Contraction; Muscle, Smooth; Naloxone; Peptide Fragments	1984
Affinities of some common opioid analgesics towards four binding sites in mouse brain. Naunyn-Schmiedeberg's archives of pharmacology, 1984, Volume: 328, Issue:1 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Opioid; Animals; Binding Sites; Brain; Codeine; Cyclazocine; Dextropropoxyphene; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Methionine; Ethylketocyclazocine; In Vitro Techniques; Membranes; Methadone; Mice; Models, Biological; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu	1984
Characteristics of 3H-tifluadom binding in guinea-pig brain membranes. Journal of receptor research, 1984, Volume: 4, Issue:1-6 Topics: Animals; Benzodiazepines; Benzomorphans; Binding Sites; Brain; Cyclazocine; Dihydromorphine; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; In Vitro Techniques; Male; Morphine; Receptors, Opioid	1984
Binding of [3H]clonidine to membranes from cow neurohypophysis and cerebral cortex of the rat. Neuropharmacology, 1984, Volume: 23, Issue:11 Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Cattle; Cerebral Cortex; Clonidine; Cyclazocine; Enkephalin, Leucine; Ethylketocyclazocine; In Vitro Techniques; Kinetics; Male; Membranes; Morphine; Naloxone; Narcotics; Pituitary Gland, Posterior; Rats	1984
Intrathecal opioids block a spinal action of substance P in mice: functional importance of both mu- and delta-receptors. European journal of pharmacology, 1982, Dec-17, Volume: 86, Issue:1 Topics: Animals; Cyclazocine; Enkephalins; Ethylketocyclazocine; Injections, Spinal; Male; Mice; Morphine; Narcotics; Reaction Time; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu; Spinal Cord; Substance P; Synaptic Transmission	1982
Opiate receptors: problems of definition and characterization. Advances in biochemical psychopharmacology, 1980, Volume: 21 Topics: Animals; Binding Sites; Brain; Caudate Nucleus; Cyclazocine; Endorphins; Enkephalins; Hippocampus; Humans; Morphine; Naloxone; Naltrexone; Receptors, Opioid	1980
Multiple opiate receptors: [3H]ethylketocyclazocine receptor binding and ketocyclazocine analgesia. Proceedings of the National Academy of Sciences of the United States of America, 1980, Volume: 77, Issue:6 Topics: Analgesics; Animals; Brain; Cyclazocine; Dihydromorphine; Dose-Response Relationship, Drug; Enkephalin, Methionine; Enkephalins; Ethylketocyclazocine; In Vitro Techniques; Mice; Morphine; Motor Activity; Naloxone; Rats; Receptors, Opioid; Receptors, Opioid, kappa	1980
Possible role of distinct morphine and enkephalin receptors in mediating actins of benzomorphan drugs (putative kappa and sigma agonists). Proceedings of the National Academy of Sciences of the United States of America, 1980, Volume: 77, Issue:8 Topics: Animals; Benzomorphans; Brain; Cyclazocine; Diprenorphine; Endorphins; Enkephalins; Ethylketocyclazocine; Guanosine Triphosphate; Morphinans; Morphine; Naloxone; Neuroblastoma; Rats; Receptors, Opioid; Sodium; Synaptic Membranes	1980
Involvement of mu-receptors in the opioid-induced generation of bursting discharges in hippocampal pyramidal cells. Regulatory peptides, 1981, Volume: 2, Issue:2 Topics: Animals; Benzomorphans; Culture Techniques; Cyclazocine; D-Ala(2),MePhe(4),Met(0)-ol-enkephalin; Dose-Response Relationship, Drug; Electrophysiology; Endorphins; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Hippocampus; Membrane Potentials; Morphinans; Rats; Receptors, Opioid; Receptors, Opioid, mu	1981
Characterization of the kappa-subtype of the opiate receptor in the guinea-pig brain. British journal of pharmacology, 1981, Volume: 73, Issue:4 Topics: Animals; Benzomorphans; Binding Sites; Binding, Competitive; Brain; Cyclazocine; Dihydromorphine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; Naloxone; Naltrexone; Narcotics; Phenoxybenzamine; Receptors, Opioid	1981
Strain differences in opiate receptors in mouse brain. European journal of pharmacology, 1981, Sep-24, Volume: 74, Issue:4 Topics: Animals; Brain; Cyclazocine; Dihydromorphine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; In Vitro Techniques; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Naloxone; Receptors, Opioid; Species Specificity	1981
D-Ala2,D-Leu5-enkephalin generalizes to a discriminative stimulus produced by fentanyl but not ethylketocyclazocine. Pharmacology, biochemistry, and behavior, 1982, Volume: 16, Issue:2 Topics: Animals; Cyclazocine; Discrimination, Psychological; Endorphins; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Fentanyl; Generalization, Stimulus; Male; Naloxone; Rats; Rats, Inbred Strains; Receptors, Opioid	1982
The binding of kappa- and sigma-opiates in rat brain. The Journal of neuroscience : the official journal of the Society for Neuroscience, 1982, Volume: 2, Issue:6 Topics: Animals; Binding Sites; Brain; Culture Techniques; Cyclazocine; Dihydromorphine; Enkephalins; Ethylketocyclazocine; Ligands; Male; Naloxone; Narcotics; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Tritium	1982
The choice of opiate receptor subtype by neo-endorphins. European journal of pharmacology, 1982, Apr-23, Volume: 79, Issue:3-4 Topics: Animals; Benzomorphans; beta-Endorphin; Cyclazocine; Drug Interactions; Endorphins; Enkephalins; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Naloxone; Protein Precursors; Rabbits; Receptors, Opioid	1982
[Met5]enkephalin-Arg-Phe ACTS on vascular opiate receptors. European journal of pharmacology, 1982, Apr-23, Volume: 79, Issue:3-4 Topics: Animals; Cyclazocine; Electric Stimulation; Endorphins; Enkephalin, Methionine; Enkephalins; Ethylketocyclazocine; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Rabbits; Receptors, Opioid	1982
Differential effect of humoral endorphin on the binding of opiate agonists and antagonists. European journal of pharmacology, 1982, Jul-09, Volume: 81, Issue:2 Topics: Animals; Binding Sites; Binding, Competitive; Cyclazocine; Endorphins; Enkephalins; Ethylketocyclazocine; In Vitro Techniques; Male; Morphine; Naloxone; Narcotic Antagonists; Narcotics; Quinuclidinyl Benzilate; Radioligand Assay; Rats; Receptors, Opioid; Sodium	1982
Opiate and opioid peptide binding in rat goldfish: further evidence for opiate receptor heterogeneity. Brain research, 1982, Sep-23, Volume: 248, Issue:1 Topics: Animals; Brain; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Goldfish; Male; Naloxone; Narcotics; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, sigma	1982
Opiate receptor-mediated inhibition of catecholamine release in primary cultures of bovine adrenal chromaffin cells. Journal of neurochemistry, 1982, Volume: 39, Issue:6 Topics: Acetylcholine; Adrenal Medulla; Animals; beta-Endorphin; Catecholamines; Cattle; Cells, Cultured; Chromaffin Granules; Chromaffin System; Cyclazocine; Dihydromorphine; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Etorphine; Phenazocine; Receptors, Opioid	1982
The epileptogenic spectrum of opiate agonists. Neuropharmacology, 1982, Volume: 21, Issue:11 Topics: Animals; Anticonvulsants; beta-Endorphin; Cyclazocine; Electroencephalography; Endorphins; Enkephalin, Leucine; Epilepsy; Ethylketocyclazocine; Injections, Intraventricular; Male; Naloxone; Narcotics; Phenazocine; Rats; Rats, Inbred Strains	1982
Relative involvement of receptor subtypes in opioid-induced inhibition of gastrointestinal transit in mice. The Journal of pharmacology and experimental therapeutics, 1983, Volume: 224, Issue:2 Topics: Animals; Charcoal; Cyclazocine; Drug Interactions; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Female; Gastrointestinal Motility; Male; Mice; Morphine; Nalorphine; Naltrexone; Receptors, Opioid	1983
Evidence for multiple "Kappa" binding sites by use of opioid peptides in the guinea-pig lumbo-sacral spinal cord. Neuropeptides, 1982, Volume: 3, Issue:1 Topics: Animals; Binding Sites; Cyclazocine; Dihydromorphine; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Etorphine; Guinea Pigs; Radioligand Assay; Receptors, Opioid; Receptors, Opioid, kappa; Spinal Cord	1982
Peptide and non-peptide opioid-induced hyperthermia in rabbits. Brain research, 1983, Apr-11, Volume: 265, Issue:1 Topics: Animals; beta-Endorphin; Body Temperature; Cyclazocine; Endorphins; Enkephalin, Methionine; Enkephalins; Ethylketocyclazocine; Male; Morphine; Naloxone; Peptides; Phenazocine; Rats	1983
The binding to rat brain homogenates of Mr2034, a universal opiate. Life sciences, 1983, Sep-05, Volume: 33, Issue:10 Topics: Animals; Benzomorphans; Brain; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Male; Morphinans; Naloxone; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid	1983
Interaction of leucine enkephalin with (3H)naloxone binding in rat brain: evidence for an opioid receptor complex. Neurochemical research, 1983, Volume: 8, Issue:7 Topics: Animals; Brain; Cyclazocine; Enkephalin, Leucine; Kinetics; Male; Naloxone; Osmolar Concentration; Protein Binding; Protein Conformation; Rats; Rats, Inbred Strains; Receptors, Opioid	1983
Naloxone-inaccessible sigma receptor in rat central nervous system. Proceedings of the National Academy of Sciences of the United States of America, 1983, Volume: 80, Issue:21 Topics: Animals; Binding, Competitive; Brain; Cyclazocine; Enkephalins; Ethylketocyclazocine; Kinetics; Naloxone; Phenazocine; Phencyclidine; Rats; Receptors, Opioid; Receptors, sigma; Spinal Cord; Tissue Distribution	1983
Opiate binding sites in bovine adrenal medulla. Journal of receptor research, 1983, Volume: 3, Issue:4 Topics: Adrenal Medulla; Animals; Binding Sites; Brain; Brain Chemistry; Cattle; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; In Vitro Techniques; Ligands; Male; Morphine; Naloxone; Rats; Rats, Inbred Strains; Receptors, Opioid	1983
Comparison of mu, delta, and kappa opiate binding sites in rat brain and spinal cord. Life sciences, 1984, Jan-16, Volume: 34, Issue:3 Topics: Animals; Binding Sites; Brain; Cell Membrane; Cyclazocine; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Receptors, Opioid; Spinal Cord	1984
[3H]ethylketocyclazocine binding to NCB-20 hybrid neurotumor cells. Molecular pharmacology, 1983, Volume: 23, Issue:2 Topics: Animals; Binding, Competitive; Brain; Cricetinae; Cricetulus; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Hybrid Cells; Kinetics; Neuroblastoma; Trypsin	1983
Analgesia induced by intrathecal injection of dynorphin B in the rat. Life sciences, 1984, Apr-16, Volume: 34, Issue:16 Topics: Analgesics; Animals; Cyclazocine; Dose-Response Relationship, Drug; Drug Tolerance; Dynorphins; Endorphins; Enkephalin, Leucine; Ethylketocyclazocine; Female; Injections, Spinal; Morphine; Naloxone; Rats	1984
[Effect of opiates on the rat vas deferens]. Archivos de farmacologia y toxicologia, 1983, Volume: 9, Issue:3 Topics: Animals; Cyclazocine; Enkephalins; Male; Morphine; Muscle Contraction; Naloxone; Narcotics; Rats; Rats, Inbred Strains; Vas Deferens	1983
Catatonic or hypotonic immobility induced in mice by intracerebroventricular injection of mu or kappa opioid receptor agonists as well as enkephalins or inhibitors of their degradation. Life sciences, 1983, Nov-21, Volume: 33, Issue:21 Topics: Animals; Benzomorphans; Catatonia; Cyclazocine; Enkephalins; Ethylketocyclazocine; Fentanyl; Humans; Immobilization; Injections, Intraventricular; Male; Mice; Morphine; Naloxone; Narcotic Antagonists; Narcotics	1983
Hippocampal involvement in the pharmacologic induction of withdrawal-like behaviors. Federation proceedings, 1981, Volume: 40, Issue:5 Topics: Animals; Cyclazocine; Endorphins; Enkephalin, Methionine; Enkephalins; Escape Reaction; Ethylketocyclazocine; Hippocampus; Humans; Injections, Intraventricular; Kainic Acid; Morphine Dependence; Pyrrolidines; Rats; Serotonin; Shivering; Substance Withdrawal Syndrome; Valproic Acid	1981
Increased food and water intake produced in rats by opiate receptor agonists. Psychopharmacology, 1981, Volume: 74, Issue:3 Topics: Animals; Cyclazocine; Drinking; Drug Interactions; Eating; Enkephalins; Ethylketocyclazocine; Male; Morphine; Naloxone; Narcotics; Rats	1981