Page last updated: 2024-09-04

cyc 202 and tg 003

cyc 202 has been researched along with tg 003 in 5 studies

Compound Research Comparison

Studies
(cyc 202)
Trials
(cyc 202)
Recent Studies (post-2010)
(cyc 202)
Studies
(tg 003)
Trials
(tg 003)
Recent Studies (post-2010) (tg 003)
979739345033

Protein Interaction Comparison

ProteinTaxonomycyc 202 (IC50)tg 003 (IC50)
Dual specificity protein kinase CLK2Mus musculus (house mouse)0.2
Dual specificity protein kinase CLK4Mus musculus (house mouse)0.015
Dual specificity protein kinase CLK1Mus musculus (house mouse)0.02
Dual specificity protein kinase CLK1Homo sapiens (human)0.064
Dual specificity tyrosine-phosphorylation-regulated kinase 1AHomo sapiens (human)0.6172
Dual specificity tyrosine-phosphorylation-regulated kinase 1AMus musculus (house mouse)0.012

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (40.00)29.6817
2010's3 (60.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bullock, AN; Fedorov, O; Knapp, S; Marsden, B; Müller, S; Pogacic, V; Rellos, P; Schwaller, J; Sundström, M1
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1
Babault, L; Baratte, B; Bazureau, JP; Carreaux, F; Debdab, M; Eisenreich, A; Fedorov, O; Filippakopoulos, P; Hagiwara, M; Knapp, S; Lozach, O; Meijer, L; Ogawa, Y; Rauch, U; Renault, S; Soundararajan, M; Tahtouh, T1
Bui, LC; Cariou, K; Dairou, J; Delabar, JM; Denhez, C; Dodd, RH; Gourdain, S; Janel, N; Rodrigues-Lima, F1
Jarhad, DB; Jeong, LS; Kim, HR; Mashelkar, KK; Noh, M1

Reviews

1 review(s) available for cyc 202 and tg 003

ArticleYear
Dual-Specificity Tyrosine Phosphorylation-Regulated Kinase 1A (DYRK1A) Inhibitors as Potential Therapeutics.
    Journal of medicinal chemistry, 2018, 11-21, Volume: 61, Issue:22

    Topics: Animals; Biological Products; Disease; Dyrk Kinases; Enzyme Activation; Humans; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases

2018

Other Studies

4 other study(ies) available for cyc 202 and tg 003

ArticleYear
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
    Proceedings of the National Academy of Sciences of the United States of America, 2007, Dec-18, Volume: 104, Issue:51

    Topics: Amino Acid Sequence; Binding Sites; Clinical Trials as Topic; Drug Evaluation, Preclinical; Enzyme Stability; Humans; Molecular Sequence Data; Phylogeny; Protein Array Analysis; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases

2007
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009
Leucettines, a class of potent inhibitors of cdc2-like kinases and dual specificity, tyrosine phosphorylation regulated kinases derived from the marine sponge leucettamine B: modulation of alternative pre-RNA splicing.
    Journal of medicinal chemistry, 2011, Jun-23, Volume: 54, Issue:12

    Topics: Alternative Splicing; Animals; Aquatic Organisms; Benzodioxoles; Crystallography, X-Ray; Cyclin-Dependent Kinases; Dyrk Kinases; Endothelial Cells; Humans; Imidazolines; Microvessels; Models, Molecular; Nuclear Proteins; Phosphorylation; Porifera; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Quantitative Structure-Activity Relationship; RNA Precursors; RNA-Binding Proteins; Serine-Arginine Splicing Factors; Stereoisomerism

2011
Development of DANDYs, new 3,5-diaryl-7-azaindoles demonstrating potent DYRK1A kinase inhibitory activity.
    Journal of medicinal chemistry, 2013, Dec-12, Volume: 56, Issue:23

    Topics: Dyrk Kinases; Enzyme Inhibitors; Humans; Hydrogen Bonding; Indoles; KB Cells; Molecular Docking Simulation; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Pyridines

2013