Page last updated: 2024-09-04

cyc 202 and glutamic acid

cyc 202 has been researched along with glutamic acid in 13 studies

Compound Research Comparison

Studies
(cyc 202)
Trials
(cyc 202)
Recent Studies (post-2010)
(cyc 202)
Studies
(glutamic acid)
Trials
(glutamic acid)
Recent Studies (post-2010) (glutamic acid)
979739341,75745212,876

Protein Interaction Comparison

ProteinTaxonomycyc 202 (IC50)glutamic acid (IC50)
Chain A, GLUTAMATE RECEPTOR SUBUNIT 2Rattus norvegicus (Norway rat)0.821
Chain A, Glutamate Receptor Subunit 2Rattus norvegicus (Norway rat)0.821
Chain B, Glutamate Receptor Subunit 2Rattus norvegicus (Norway rat)0.821
Metabotropic glutamate receptor 8Homo sapiens (human)0.0057
Glutamate receptor ionotropic, NMDA 2DHomo sapiens (human)0.07
Glutamate receptor ionotropic, NMDA 3BHomo sapiens (human)0.07
Glutamate receptor 1Rattus norvegicus (Norway rat)0.5885
Glutamate receptor 2Rattus norvegicus (Norway rat)0.5885
Glutamate receptor 3Rattus norvegicus (Norway rat)0.5885
Glutamate receptor 4Rattus norvegicus (Norway rat)0.5885
Glutamate receptor ionotropic, kainate 1Rattus norvegicus (Norway rat)0.38
Glutamate receptor ionotropic, NMDA 1 Rattus norvegicus (Norway rat)0.1533
Glutamate receptor ionotropic, kainate 2Rattus norvegicus (Norway rat)0.38
Glutamate receptor 1Homo sapiens (human)0.613
Glutamate receptor 2Homo sapiens (human)0.613
Glutamate receptor 3Homo sapiens (human)0.613
Glutamate receptor ionotropic, kainate 3Rattus norvegicus (Norway rat)0.38
Excitatory amino acid transporter 1Homo sapiens (human)207
Glutamate receptor 4Homo sapiens (human)0.613
Glutamate receptor ionotropic, NMDA 2A Rattus norvegicus (Norway rat)0.1533
Glutamate receptor ionotropic, NMDA 2BRattus norvegicus (Norway rat)0.1533
Glutamate receptor ionotropic, NMDA 2CRattus norvegicus (Norway rat)0.1533
Glutamate receptor ionotropic, kainate 4Rattus norvegicus (Norway rat)0.38
Glutamate receptor ionotropic, NMDA 1Homo sapiens (human)0.07
Glutamate receptor ionotropic, NMDA 2AHomo sapiens (human)0.07
Glutamate receptor ionotropic, NMDA 2BHomo sapiens (human)0.07
Glutamate receptor ionotropic, NMDA 2CHomo sapiens (human)0.07
Glutamate receptor ionotropic, NMDA 2DRattus norvegicus (Norway rat)0.1533
Glutamate receptor ionotropic, kainate 5Rattus norvegicus (Norway rat)0.38
Glutamate receptor ionotropic, NMDA 3AHomo sapiens (human)0.07
Glutamate receptor ionotropic, NMDA 3BRattus norvegicus (Norway rat)0.1533
Glutamate receptor ionotropic, NMDA 3ARattus norvegicus (Norway rat)0.1533

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's7 (53.85)29.6817
2010's4 (30.77)24.3611
2020's2 (15.38)2.80

Authors

AuthorsStudies
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Li, ST; Matsui, H; Matsushita, M; Moriwaki, A; Ohta, J; Takei, K; Tomizawa, K1
Hyman, SE; Minassian, R; Nairn, AC; Sgambato, V1
Chergui, K; Greengard, P; Svenningsson, P1
Gong, X; Mao, Z; Park, D; Tang, X; Tong, M; Wang, X; Xia, Z1
Monaco, EA; Vallano, ML1
Asada, A; Fukunaga, K; Hisanaga, S; Hosokawa, T; Itakura, M; Ohshima, T; Saito, T; Takahashi, M1
Chen, GD; Chiu, CH; Hsien, MC; Lai, CY; Lee, SD; Liao, JM; Lin, TB; Lu, HT; Peng, HY; Tung, KC1
Antonucci, L; Edwards, J; Hunce, R; Krucher, NA; Lentine, B; Marallano, V1
Hernández-Echeagaray, E; Miranda-Barrientos, J; Nieto-Mendoza, E1
Cardona-Gómez, GP; Palacio-Castañeda, V; Posada-Duque, RA1
Ai, LQ; Chen, C; Gao, L; Lin, S; Liu, W; Xiao, H; Ye, J; Zhou, Y1
Konishi, S; Satake, SI1

Other Studies

13 other study(ies) available for cyc 202 and glutamic acid

ArticleYear
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Cdk5/p35 regulates neurotransmitter release through phosphorylation and downregulation of P/Q-type voltage-dependent calcium channel activity.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2002, Apr-01, Volume: 22, Issue:7

    Topics: Animals; Calcium; Calcium Channel Blockers; Calcium Channels, P-Type; Calcium Channels, Q-Type; Cyclin-Dependent Kinase 5; Cyclin-Dependent Kinases; Down-Regulation; Electric Stimulation; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; Exocytosis; Glutamic Acid; Hippocampus; In Vitro Techniques; Kinetin; Male; Nerve Tissue Proteins; Neurons; Neurotransmitter Agents; Phosphorylation; Protein Isoforms; Purines; Rats; Rats, Wistar; Roscovitine; Synaptosomes

2002
Regulation of ania-6 splice variants by distinct signaling pathways in striatal neurons.
    Journal of neurochemistry, 2003, Volume: 86, Issue:1

    Topics: Alternative Splicing; Animals; Binding Sites; Calcium; Cells, Cultured; Corpus Striatum; Cyclins; Enzyme Inhibitors; Glutamic Acid; Macromolecular Substances; Mitogen-Activated Protein Kinases; Neurons; PC12 Cells; Phosphorylation; Potassium Chloride; Promoter Regions, Genetic; Purines; Rats; Rats, Sprague-Dawley; Response Elements; Roscovitine; Signal Transduction; Transcription Factor AP-1

2003
Cyclin-dependent kinase 5 regulates dopaminergic and glutamatergic transmission in the striatum.
    Proceedings of the National Academy of Sciences of the United States of America, 2004, Feb-17, Volume: 101, Issue:7

    Topics: Animals; Cyclin-Dependent Kinase 5; Cyclin-Dependent Kinases; Dopamine; Dopamine and cAMP-Regulated Phosphoprotein 32; Enzyme Inhibitors; Glutamic Acid; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Neostriatum; Nerve Tissue Proteins; Phosphoproteins; Phosphorylation; Purines; Receptors, AMPA; Receptors, Dopamine D1; Receptors, N-Methyl-D-Aspartate; RNA, Messenger; Roscovitine; Synapses; Synaptic Transmission

2004
Cyclin-dependent kinase 5 mediates neurotoxin-induced degradation of the transcription factor myocyte enhancer factor 2.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, May-11, Volume: 25, Issue:19

    Topics: Amino Acid Chloromethyl Ketones; Animals; Animals, Newborn; Blotting, Western; Caspase Inhibitors; Caspases; Cell Count; Cell Death; Cells, Cultured; Cerebellum; Chromatin; Cyclin-Dependent Kinase 5; Drug Interactions; Glutamic Acid; Green Fluorescent Proteins; Luciferases; MEF2 Transcription Factors; Myogenic Regulatory Factors; Neurons; Neurotoxins; Oligopeptides; Protein Kinase Inhibitors; Purines; Rats; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Roscovitine; Subcellular Fractions; Time Factors; Transfection

2005
Roscovitine triggers excitotoxicity in cultured granule neurons by enhancing glutamate release.
    Molecular pharmacology, 2005, Volume: 68, Issue:5

    Topics: Action Potentials; Animals; Calcium; Calcium Channels, L-Type; Calcium Channels, N-Type; Cells, Cultured; Cerebellum; Cytoplasmic Granules; Glutamic Acid; Necrosis; Neurons; Potassium Channel Blockers; Potassium Chloride; Protein Kinase Inhibitors; Purines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Roscovitine; Synaptic Transmission

2005
Enhanced activation of Ca2+/calmodulin-dependent protein kinase II upon downregulation of cyclin-dependent kinase 5-p35.
    Journal of neuroscience research, 2006, Volume: 84, Issue:4

    Topics: Animals; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Cells, Cultured; Cerebral Cortex; Cyclin-Dependent Kinase 5; Down-Regulation; Embryo, Mammalian; Enzyme Activation; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Fluorescent Antibody Technique; Glutamic Acid; Immunoprecipitation; In Vitro Techniques; N-Methylaspartate; Neurons; Phosphorylation; Phosphotransferases; Protein Kinases; Purines; Rats; Roscovitine

2006
Colon mustard oil instillation induced cross-organ reflex sensitization on the pelvic-urethra reflex activity in rats.
    Pain, 2009, Volume: 142, Issue:1-2

    Topics: Animals; Colon; Cyclin-Dependent Kinase 5; Electric Stimulation; Excitatory Amino Acid Agents; Glutamic Acid; Inflammation; Male; Mustard Plant; Pelvis; Piperidines; Plant Oils; Protein Kinase Inhibitors; Purines; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Reflex; RNA, Small Interfering; Roscovitine; TRPV Cation Channels; Urethra

2009
Dephosphorylation of threonine-821 of the retinoblastoma tumor suppressor protein (Rb) is required for apoptosis induced by UV and Cdk inhibition.
    Cell cycle (Georgetown, Tex.), 2012, Sep-01, Volume: 11, Issue:17

    Topics: Apoptosis; Blotting, Western; Cell Line, Tumor; Cyclin-Dependent Kinases; Enzyme-Linked Immunosorbent Assay; Glutamic Acid; Humans; Mutagenesis; Mutation, Missense; Phosphorylation; Purines; Retinoblastoma Protein; Roscovitine; S Phase Cell Cycle Checkpoints; Ultraviolet Rays

2012
The Cdk5 inhibitor Roscovitine increases LTP induction in corticostriatal synapses.
    ASN neuro, 2014, Mar-19, Volume: 6, Issue:2

    Topics: Animals; Calcium Channels, L-Type; Cerebral Cortex; Corpus Striatum; Cyclic AMP-Dependent Protein Kinases; Cyclin-Dependent Kinase 5; Excitatory Postsynaptic Potentials; Glutamic Acid; Long-Term Potentiation; Long-Term Synaptic Depression; Male; Mice; Mice, Inbred C57BL; Neural Pathways; Protein Kinase Inhibitors; Purines; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, N-Methyl-D-Aspartate; Roscovitine; Synaptic Transmission

2014
CDK5 knockdown in astrocytes provide neuroprotection as a trophic source via Rac1.
    Molecular and cellular neurosciences, 2015, Volume: 68

    Topics: Animals; Animals, Newborn; Astrocytes; Cells, Cultured; Cerebral Cortex; Coculture Techniques; Cyclin-Dependent Kinase 5; Embryo, Mammalian; Excitatory Amino Acid Agonists; Glioma; Glutamic Acid; Mutation; Nerve Tissue Proteins; Neurons; Neuroprotection; Protein Kinase Inhibitors; Purines; rac1 GTP-Binding Protein; Rats; Rats, Wistar; rhoA GTP-Binding Protein; Roscovitine; Time Factors

2015
Vps35 Deficiency Impairs Cdk5/p35 Degradation and Promotes the Hyperphosphorylation of Tau Protein in Retinal Ganglion Cells.
    Investigative ophthalmology & visual science, 2020, Jan-23, Volume: 61, Issue:1

    Topics: Animals; Blotting, Western; Cells, Cultured; Cyclin-Dependent Kinase 5; Down-Regulation; Fluorescent Antibody Technique, Indirect; Glutamic Acid; Lysosomal Membrane Proteins; Male; Mice; Phosphorylation; Phosphotransferases; Protein Kinase Inhibitors; Rats; Rats, Sprague-Dawley; Real-Time Polymerase Chain Reaction; Retinal Degeneration; Retinal Ganglion Cells; Roscovitine; tau Proteins; Transfection; Ubiquitin-Activating Enzymes; Vesicular Transport Proteins

2020
Topographical distance between presynaptic Ca
    The European journal of neuroscience, 2021, Volume: 54, Issue:9

    Topics: Animals; Calcium Channels, N-Type; Cerebellum; Glutamic Acid; Neurotransmitter Agents; Presynaptic Terminals; Rats; Roscovitine; Synapses; Synaptic Transmission

2021