Page last updated: 2024-09-04

cyc 202 and eliprodil

cyc 202 has been researched along with eliprodil in 2 studies

Compound Research Comparison

Studies
(cyc 202)
Trials
(cyc 202)
Recent Studies (post-2010)
(cyc 202)
Studies
(eliprodil)
Trials
(eliprodil)
Recent Studies (post-2010) (eliprodil)
9797393104323

Protein Interaction Comparison

ProteinTaxonomycyc 202 (IC50)eliprodil (IC50)
N-methyl-D-aspartate receptor Sus scrofa (pig)0.0826
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)3.3
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)3.3
Glutamate receptor ionotropic, NMDA 1 Rattus norvegicus (Norway rat)1.4
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)3.3
Glutamate receptor ionotropic, NMDA 2BRattus norvegicus (Norway rat)1.4

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's1 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1
Davis, MI; Khan, J; Li, SQ; Patel, PR; Shen, M; Sun, H; Thomas, CJ1

Other Studies

2 other study(ies) available for cyc 202 and eliprodil

ArticleYear
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009
Identification of potent Yes1 kinase inhibitors using a library screening approach.
    Bioorganic & medicinal chemistry letters, 2013, Aug-01, Volume: 23, Issue:15

    Topics: Binding Sites; Cell Line; Cell Survival; Drug Design; Humans; Hydrogen Bonding; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-yes; Small Molecule Libraries; Structure-Activity Relationship

2013