Page last updated: 2024-09-04

cyc 202 and cycloheximide

cyc 202 has been researched along with cycloheximide in 18 studies

Compound Research Comparison

Studies
(cyc 202)
Trials
(cyc 202)
Recent Studies (post-2010)
(cyc 202)
Studies
(cycloheximide)
Trials
(cycloheximide)
Recent Studies (post-2010) (cycloheximide)
979739319,1096861

Protein Interaction Comparison

ProteinTaxonomycyc 202 (IC50)cycloheximide (IC50)
COUP transcription factor 2 isoform aHomo sapiens (human)1.315
Glucose transporterLeishmania mexicana0.242
Hexose transporter 1 Plasmodium falciparum (malaria parasite P. falciparum)0.31
Solute carrier family 2, facilitated glucose transporter member 1Homo sapiens (human)0.228
Eukaryotic initiation factor 4A-IHomo sapiens (human)0.139
Peptidyl-prolyl cis-trans isomerase FKBP1AHomo sapiens (human)3.6
Hypoxia-inducible factor 1-alphaHomo sapiens (human)0.036
Endothelial PAS domain-containing protein 1Homo sapiens (human)0.036

Research

Studies (18)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (11.11)18.2507
2000's13 (72.22)29.6817
2010's3 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Krucher, NA; Meijer, L; Roberts, MH1
Rosenberg, A; Schaffer, PA; Schang, LM1
Faerge, I; Hyttel, P; Mayes, M; Sirard, MA1
Dekel, N; Galiani, D; Lazar, S1
Dong, YB; Elliott, MJ; McMasters, KM; Yang, HL1
Gilbert, DM; Keezer, SM1
Le Beux, G; Richard, FJ; Sirard, MA1
Akiyama, T; Aoki, F; Kim, JM; Nagata, M1
Aoki, F; Hara, KT; Nagata, M; Naito, K; Oda, S; Schultz, RM1
Endo, T; Kashima, K; Kume, S; Naito, K; Nishimura, Y; Tojo, H1
Choi, YH; Hinrichs, K; Love, LB; Varner, DD1
Choi, YH; Chung, YG; Hinrichs, K; Love, CC; Varner, DD1
Kellogg, DR; McCusker, D; Royou, A; Sullivan, W1
Hong, SG; Hossein, MS; Koo, OJ; Lee, BC; Martinez-Conejero, JA1
de Sá Lorena, SE; Landim-Alvarenga, Fda C; Martins, LR; Minto, BW; Rascado, Tda S1
Blanco, ID; da Cruz Landim-Alvarenga, F; de Lima Neto, JF; Devito, LG; Fernandes, CB; Gonçalves, CG; Martins, LR; Tsuribe, PM1
Berger, F; Higashiyama, T; Kawashima, T; Kinoshita, T; Maruyama, D; Motomura, K1

Other Studies

18 other study(ies) available for cyc 202 and cycloheximide

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
The cyclin-dependent kinase (cdk) inhibitors, olomoucine and roscovitine, alter the expression of a molluscan circadian pacemaker.
    Cellular and molecular neurobiology, 1997, Volume: 17, Issue:5

    Topics: Animals; Biological Clocks; Circadian Rhythm; Cyclin-Dependent Kinases; Cycloheximide; Darkness; Dichlororibofuranosylbenzimidazole; Dose-Response Relationship, Drug; Enzyme Inhibitors; Kinetin; Mollusca; Nucleic Acid Synthesis Inhibitors; Ocular Physiological Phenomena; Photoperiod; Protein Synthesis Inhibitors; Purines; Roscovitine

1997
Transcription of herpes simplex virus immediate-early and early genes is inhibited by roscovitine, an inhibitor specific for cellular cyclin-dependent kinases.
    Journal of virology, 1999, Volume: 73, Issue:3

    Topics: Animals; Chlorocebus aethiops; Cyclin-Dependent Kinases; Cycloheximide; DNA Replication; Enzyme Inhibitors; Genes, Immediate-Early; Genes, Viral; Purines; Roscovitine; Simplexvirus; Transcription, Genetic; Vero Cells; Virus Replication

1999
Nuclear ultrastructure in bovine oocytes after inhibition of meiosis by chemical and biological inhibitors.
    Molecular reproduction and development, 2001, Volume: 59, Issue:4

    Topics: 4-Butyrolactone; Adenine; Animals; Antineoplastic Agents; Cattle; Cell Nucleolus; Cell Nucleus; Cells, Cultured; Cycloheximide; Enzyme Inhibitors; Female; Meiosis; Microscopy, Electron; Nuclear Envelope; Oocytes; Protein Synthesis Inhibitors; Purines; Roscovitine

2001
cAMP-Dependent PKA negatively regulates polyadenylation of c-mos mRNA in rat oocytes.
    Molecular endocrinology (Baltimore, Md.), 2002, Volume: 16, Issue:2

    Topics: Animals; Blotting, Western; CDC2 Protein Kinase; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cycloheximide; Enzyme Activation; Female; Gene Expression Regulation; Meiosis; Mitogen-Activated Protein Kinases; Oocytes; Polyadenylation; Protein Biosynthesis; Proto-Oncogene Proteins c-mos; Purines; Rats; RNA, Messenger; Roscovitine; Signal Transduction; Time Factors

2002
Adenovirus-mediated E2F-1 gene transfer sensitizes melanoma cells to apoptosis induced by topoisomerase II inhibitors.
    Cancer research, 2002, Mar-15, Volume: 62, Issue:6

    Topics: Adenoviridae; Animals; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Apoptosis; Cell Cycle Proteins; Cisplatin; Combined Modality Therapy; Cyclin-Dependent Kinase Inhibitor p21; Cyclins; Cycloheximide; DNA-Binding Proteins; Doxorubicin; Drug Synergism; E2F Transcription Factors; E2F1 Transcription Factor; Enzyme Inhibitors; Etoposide; Fluorouracil; Genetic Therapy; Genetic Vectors; Humans; Male; Melanoma; Mice; Mice, Inbred BALB C; Mice, Nude; Proliferating Cell Nuclear Antigen; Purines; Roscovitine; Topoisomerase II Inhibitors; Transcription Factors; Tumor Cells, Cultured; Xenograft Model Antitumor Assays

2002
Evidence for a pre-restriction point Cdk3 activity.
    Journal of cellular biochemistry, 2002, Volume: 85, Issue:3

    Topics: Animals; Cells, Cultured; CHO Cells; Cricetinae; Cyclin-Dependent Kinases; Cycloheximide; Cysteine Endopeptidases; Enzyme Inhibitors; G1 Phase; Leupeptins; Multienzyme Complexes; Precipitin Tests; Proteasome Endopeptidase Complex; Protein Kinases; Protein Synthesis Inhibitors; Purines; Replication Origin; Roscovitine

2002
Effect of cycloheximide, 6-DMAP, roscovitine and butyrolactone I on resumption of meiosis in porcine oocytes.
    Theriogenology, 2003, Oct-01, Volume: 60, Issue:6

    Topics: 4-Butyrolactone; Adenine; Animals; Cells, Cultured; Cyclin-Dependent Kinases; Cycloheximide; Enzyme Inhibitors; Female; Meiosis; Oocytes; Protein Kinase Inhibitors; Protein Synthesis Inhibitors; Purines; Roscovitine; Swine

2003
Regulation of histone acetylation during meiotic maturation in mouse oocytes.
    Molecular reproduction and development, 2004, Volume: 69, Issue:2

    Topics: Acetylation; Acetyltransferases; Animals; CDC2 Protein Kinase; Cyclin-Dependent Kinase-Activating Kinase; Cyclin-Dependent Kinases; Cycloheximide; Female; Histone Acetyltransferases; Histone Deacetylase Inhibitors; Histone Deacetylases; Histones; In Vitro Techniques; Meiosis; Mice; Oocytes; Protein Kinase Inhibitors; Purines; Roscovitine; Signal Transduction

2004
Cyclin A2-CDK2 regulates embryonic gene activation in 1-cell mouse embryos.
    Developmental biology, 2005, Oct-01, Volume: 286, Issue:1

    Topics: Animals; Base Sequence; Cleavage Stage, Ovum; Cyclin A; Cyclin-Dependent Kinase 2; Cycloheximide; Deoxyadenosines; DNA, Complementary; Female; Gene Expression Regulation, Developmental; In Vitro Techniques; Mice; Mice, Inbred ICR; Pregnancy; Protein Kinase Inhibitors; Purines; RNA, Messenger; RNA, Small Interfering; Roscovitine; Transcriptional Activation

2005
Activities of maturation-promoting factor (MPF) and mitogen-activated protein kinase (MAPK) are not required for the global histone deacetylation observed after germinal vesicle breakdown (GVBD) in porcine oocytes.
    Reproduction (Cambridge, England), 2006, Volume: 131, Issue:3

    Topics: Acetylation; Animals; Chromatin; Cycloheximide; Enzyme Activation; Female; Histone Deacetylase Inhibitors; Histone Deacetylases; Histones; Hydroxamic Acids; Immunoblotting; Immunohistochemistry; Maturation-Promoting Factor; Meiosis; Mesothelin; Mice; Mitogen-Activated Protein Kinase 1; Oocytes; Protein Synthesis Inhibitors; Purines; Roscovitine

2006
Holding immature equine oocytes in the absence of meiotic inhibitors: effect on germinal vesicle chromatin and blastocyst development after intracytoplasmic sperm injection.
    Theriogenology, 2006, Sep-01, Volume: 66, Issue:4

    Topics: Animals; Cells, Cultured; Chromatin; Cycloheximide; Embryonic Development; Female; Horses; Male; Meiosis; Oocyte Retrieval; Oocytes; Oogenesis; Pregnancy; Protein Kinase Inhibitors; Protein Synthesis Inhibitors; Purines; Roscovitine; Sperm Injections, Intracytoplasmic; Tissue Preservation

2006
Production of horse foals via direct injection of roscovitine-treated donor cells and activation by injection of sperm extract.
    Reproduction (Cambridge, England), 2006, Volume: 131, Issue:6

    Topics: Adenine; Animals; Cell Extracts; Cells, Cultured; Cloning, Organism; Culture Media; Cycloheximide; Embryo Transfer; Female; Fibroblasts; Flow Cytometry; Horses; Hybrid Cells; Male; Microinjections; Nuclear Transfer Techniques; Oocytes; Purines; Roscovitine; Spermatozoa

2006
Grapes(Chk1) prevents nuclear CDK1 activation by delaying cyclin B nuclear accumulation.
    The Journal of cell biology, 2008, Oct-06, Volume: 183, Issue:1

    Topics: Active Transport, Cell Nucleus; Animals; Aphidicolin; CDC2 Protein Kinase; Cell Cycle; Cell Cycle Proteins; Cell Nucleus; Cell Nucleus Division; Checkpoint Kinase 1; Cyclin B; Cycloheximide; Cytokinesis; Cytoplasm; Drosophila melanogaster; Drosophila Proteins; Embryo, Nonmammalian; Kinetochores; Mitosis; Mutation; Nuclear Envelope; Nuclear Proteins; Protein Kinase Inhibitors; Protein Kinases; Protein-Tyrosine Kinases; Purines; Quinolines; Recombinant Proteins; Roscovitine; Spindle Apparatus; Thiazoles

2008
Cell cycle synchronization of canine ear fibroblasts for somatic cell nuclear transfer.
    Zygote (Cambridge, England), 2009, Volume: 17, Issue:1

    Topics: Animals; Antifungal Agents; Antineoplastic Agents; Contact Inhibition; Cycloheximide; Dimethyl Sulfoxide; Dogs; Ear; Female; Fibroblasts; Free Radical Scavengers; G1 Phase; Nuclear Transfer Techniques; Purines; Resting Phase, Cell Cycle; Roscovitine; Serum

2009
Parthenogenetic development of domestic cat oocytes treated with ionomycin, cycloheximide, roscovitine and strontium.
    Theriogenology, 2010, Sep-01, Volume: 74, Issue:4

    Topics: Animals; Cats; Culture Media; Cycloheximide; Embryo Culture Techniques; Female; Ionomycin; Oocytes; Parthenogenesis; Purines; Roscovitine; Strontium

2010
Artificial activation of bovine and equine oocytes with cycloheximide, roscovitine, strontium, or 6-dimethylaminopurine in low or high calcium concentrations.
    Zygote (Cambridge, England), 2014, Volume: 22, Issue:3

    Topics: Adenine; Animals; Calcium; Cattle; Cells, Cultured; Cycloheximide; Female; Horses; In Vitro Oocyte Maturation Techniques; Ionomycin; Oocytes; Parthenogenesis; Purines; Roscovitine; Strontium

2014
A pharmacological study of
    Journal of cell science, 2018, 01-29, Volume: 131, Issue:2

    Topics: Actins; Arabidopsis; Brefeldin A; Bridged Bicyclo Compounds, Heterocyclic; Cell Fusion; Cyclin-Dependent Kinases; Cycloheximide; Deoxyadenosines; Dinitrobenzenes; Endosperm; Fertilization; Gene Expression Regulation, Plant; Mitosis; Phenotype; Polymerization; Roscovitine; Sulfanilamides; Thiazolidines

2018