Page last updated: 2024-09-04

cyc 202 and belinostat

cyc 202 has been researched along with belinostat in 2 studies

Compound Research Comparison

Studies
(cyc 202)
Trials
(cyc 202)
Recent Studies (post-2010)
(cyc 202)
Studies
(belinostat)
Trials
(belinostat)
Recent Studies (post-2010) (belinostat)
979739320830167
9797393807

Protein Interaction Comparison

ProteinTaxonomycyc 202 (IC50)belinostat (IC50)
Histone deacetylase 3Homo sapiens (human)0.1942
Bromodomain-containing protein 4Homo sapiens (human)0.027
Cytochrome P450 3A5Homo sapiens (human)0.2147
Histone deacetylase 4Homo sapiens (human)1.1602
Aspartyl/asparaginyl beta-hydroxylaseHomo sapiens (human)5.12
Histone deacetylase 1Homo sapiens (human)0.816
Histone deacetylase 7Homo sapiens (human)0.0357
Histone deacetylase 2Homo sapiens (human)0.2401
Polyamine deacetylase HDAC10Homo sapiens (human)0.0357
Histone deacetylase 11 Homo sapiens (human)1.5966
Histone deacetylase 8Homo sapiens (human)1.2526
Histone deacetylase 6Homo sapiens (human)1.1946
Histone deacetylase 9Homo sapiens (human)0.0357
Histone deacetylase 5Homo sapiens (human)0.0357
Histone deacetylase Plasmodium falciparum (malaria parasite P. falciparum)0.2147

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chia, DM; Chinnathambi, A; Goh, BC; Ho, PC; Kong, LR; Lau, JY; Ong, PS; Seah, JY; Sethi, G; Thuya, WL; Wang, L; Wong, AL; Yang, D; Yong, WP1
Davis, MI; Khan, J; Li, SQ; Patel, PR; Shen, M; Sun, H; Thomas, CJ1

Other Studies

2 other study(ies) available for cyc 202 and belinostat

ArticleYear
A novel combinatorial strategy using Seliciclib(®) and Belinostat(®) for eradication of non-small cell lung cancer via apoptosis induction and BID activation.
    Cancer letters, 2016, 10-10, Volume: 381, Issue:1

    Topics: A549 Cells; Antineoplastic Combined Chemotherapy Protocols; Apoptosis; BH3 Interacting Domain Death Agonist Protein; Carcinoma, Non-Small-Cell Lung; Caspase 3; Caspase 8; Caspase Inhibitors; Cell Proliferation; Dose-Response Relationship, Drug; Histone Deacetylase Inhibitors; Humans; Hydroxamic Acids; Inhibitory Concentration 50; Lung Neoplasms; Myeloid Cell Leukemia Sequence 1 Protein; Poly(ADP-ribose) Polymerases; Protein Kinase Inhibitors; Purines; RNA Interference; Roscovitine; Signal Transduction; Sulfonamides; Time Factors; Transfection; Tumor Suppressor Protein p53; X-Linked Inhibitor of Apoptosis Protein

2016
Identification of potent Yes1 kinase inhibitors using a library screening approach.
    Bioorganic & medicinal chemistry letters, 2013, Aug-01, Volume: 23, Issue:15

    Topics: Binding Sites; Cell Line; Cell Survival; Drug Design; Humans; Hydrogen Bonding; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-yes; Small Molecule Libraries; Structure-Activity Relationship

2013