cyc 202 has been researched along with 4,5,6,7-tetrabromo-2-azabenzimidazole in 2 studies
Studies (cyc 202) | Trials (cyc 202) | Recent Studies (post-2010) (cyc 202) | Studies (4,5,6,7-tetrabromo-2-azabenzimidazole) | Trials (4,5,6,7-tetrabromo-2-azabenzimidazole) | Recent Studies (post-2010) (4,5,6,7-tetrabromo-2-azabenzimidazole) |
---|---|---|---|---|---|
979 | 7 | 393 | 115 | 0 | 57 |
Protein | Taxonomy | cyc 202 (IC50) | 4,5,6,7-tetrabromo-2-azabenzimidazole (IC50) |
---|---|---|---|
Chain A, Cell division protein kinase 2 | Homo sapiens (human) | 15.6 | |
Casein kinase II subunit alpha' | Homo sapiens (human) | 0.7325 | |
Casein kinase II subunit beta | Homo sapiens (human) | 0.7325 | |
Casein kinase II subunit alpha | Homo sapiens (human) | 0.7354 | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A | Homo sapiens (human) | 2.68 | |
Casein kinase II subunit alpha 3 | Homo sapiens (human) | 0.8667 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 1 (50.00) | 29.6817 |
2010's | 1 (50.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bullock, AN; Fedorov, O; Knapp, S; Marsden, B; Müller, S; Pogacic, V; Rellos, P; Schwaller, J; Sundström, M | 1 |
Jarhad, DB; Jeong, LS; Kim, HR; Mashelkar, KK; Noh, M | 1 |
1 review(s) available for cyc 202 and 4,5,6,7-tetrabromo-2-azabenzimidazole
Article | Year |
---|---|
Dual-Specificity Tyrosine Phosphorylation-Regulated Kinase 1A (DYRK1A) Inhibitors as Potential Therapeutics.
Topics: Animals; Biological Products; Disease; Dyrk Kinases; Enzyme Activation; Humans; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases | 2018 |
1 other study(ies) available for cyc 202 and 4,5,6,7-tetrabromo-2-azabenzimidazole
Article | Year |
---|---|
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
Topics: Amino Acid Sequence; Binding Sites; Clinical Trials as Topic; Drug Evaluation, Preclinical; Enzyme Stability; Humans; Molecular Sequence Data; Phylogeny; Protein Array Analysis; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases | 2007 |