Page last updated: 2024-08-26

cyanopindolol and isoproterenol

cyanopindolol has been researched along with isoproterenol in 65 studies

Research

Studies (65)

TimeframeStudies, this research(%)All Research%
pre-199014 (21.54)18.7374
1990's36 (55.38)18.2507
2000's14 (21.54)29.6817
2010's1 (1.54)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Charlton, SJ; Dickson, CJ; Duca, JS; Fairhurst, RA; Hornak, V; McKay, DJ; Pearlstein, RA; Reilly, J; Sandham, DA; Shaw, D; Sykes, DA; Velez-Vega, C1
Kompa, AR; Molenaar, P; Pak, HS; Roberts, SJ; Summers, RJ1
Tran, VT1
Liggett, SB1
Houslay, MD; Milligan, G; Strassheim, D1
Esbenshade, TA; Granneman, JG; Han, C; Minneman, KP; Theroux, TL1
Emmerich, B; Göhly, U; Haen, E; Hallek, M; Kamp, T; Remien, J1
MacDonald, A; McLaughlin, DP1
Lafontan, M; Langin, D; Portillo, MP; Saulnier-Blache, JS1
Carpéné, C; Dauzats, M; Lafontan, M; Larrouy, D; Quideau, N; Saulnier-Blache, JS1
Borst, SE; Conolly, ME; Hui, KK1
Caron, MG; Hausdorff, WP; Hnatowich, M; Lefkowitz, RJ; O'Dowd, BF1
Hintze, TH; Homcy, CJ; Nejima, J; Susanni, EE; Uemura, N; Vatner, DE; Vatner, SF1
Korichneva, IL; Krasnikova, TL; Radiukhin, VA1
Cardone, F; Cignarelli, M; Corso, M; De Pergola, G; Di Paolo, S; Garruti, G; Giorgino, R; Nardelli, G1
Grogan, DM; Hatjis, CG; Koritnik, DR1
Grogan, DM; Hatjis, CG1
Chung, MK; Gulick, T; Lange, LG; Pieper, SJ; Schreiner, GF1
Crews, A; Hatjis, CG1
Göthert, M; Hillenbrand, K; Schlicker, E1
Malta, E; Molenaar, P1
Gagne, B; Labrie, F; Lavoie, M; Poyet, P1
Levitzki, A; Marbach, I; Shiloach, J1
Engel, G; Göthert, M; Hillenbrand, K; Hoyer, D; Schlicker, E1
Crooke, ST; Heckman, GD; Nambi, P; Schmidt, DB; Stassen, FL; Whitman, MH1
Molenaar, P; Summers, RJ1
Blankesteijn, WM; de Pont, JJ; Graafsma, SJ; Thien, T; Willems, PH1
Bejarano, P; Green, SA; Hall, IP; Liggett, SB; Turki, J1
Hirsch, DJ; Morgunov, NS; You, YD1
Kompa, AR; Molenaar, P; Russell, FD; Summers, RJ1
Chiyotani, A; Konno, K; Takeuchi, S; Tamaoki, J; Yamauchi, F; Yamawaki, I1
Dombrowski, MP; Gauvin, JM; Hayashi, RH; Hurd, WW1
Clark, CJ; Connell, JM; Milligan, G1
Molenaar, P; Sarsero, D1
Molenaar, P; Roberts, SJ; Russell, FD; Summers, RJ1
Oriowo, MA1
Esbenshade, TA; Guerrero, SW; Minneman, KP; Zhong, H1
Cui, Y; Iwase, M; Kalthof, B; Sato, N; Shen, YT; Uechi, M; Vatner, DE; Vatner, SF1
Abraini, JH; Kriem, B; Rostain, JC1
Bouanani, NE; Crozatier, B; Su, JB; Xiong, L1
Gabilondo, AM; Krasel, C; Lohse, MJ1
Díaz-Laviada, I; Guillén, A; Haro, A; Nieto, JL1
Björntorp, P; Edén, S; Liu, X; Yang, S1
Houston, G; Kelly, J1
Cohen-Tannoudji, J; Coudouel, N; Lécrivain, JL; Legrand, C; Maltier, JP; Robin, MT1
Atlan, G; Collet, F; Féve, B; Frisdal, E; Pavoine, C; Pecker, F1
Isono, K; Nagai, A; Tagaya, E; Tamaoki, J1
Dhalla, NS; Elimban, V; Persad, S; Siddiqui, F1
Baranski, TJ; Bourne, HR; Iiri, T; Lichtarge, O; Meng, EC; Nissenson, RA; Sheikh, SP; Vilardarga, JP1
Guerrero, SW; Minneman, KP1
MacDonald, A; Watt, K1
Brawley, L; MacDonald, A; Shaw, AM2
Brink, CB; Neubig, RR; Wade, SM1
Evans, BA; Hutchinson, DS; Summers, RJ1
Engelhardt, S; Hein, L; Kaumann, AJ; Lohse, M; Molenaar, P1
Green, SA; Liggett, SB; Rathz, DA; Schuster, AJ1
Hussein, SM; Khan, I; Oriowo, M1
Barakat, H; Christian, B; Davis, J; Hickner, R; McConnaughey, MM; Privette, J; Sheets, KA1
Ishii, K; Karikomi, Y; Kubota, Y; Nakahara, T; Sakamoto, K1
Brown, MJ; O'Shaughnessy, KM; Sandilands, A; Yeo, G1
Chandrasekhar, B; Fatinikun, T; Kadavil, EA; Khan, I; Omu, AE; Oriowo, MA1
Desfontis, JC; Gogny, M; Holopherne, D; Le Coz, O; Mallem, Y; Reculeau, O1
Clark, RB; Dai, W; Friedman, J; Godines, V; Knoll, BJ; Millman, EE; Moore, RH; Tran, TM; Vaughan, DJ1
Amour, J; Birenbaum, A; Heymes, C; Loyer, X; Michelet, P; Riou, B1

Trials

1 trial(s) available for cyanopindolol and isoproterenol

ArticleYear
Differences in beta-adrenergic receptor densities in omental and subcutaneous adipose tissue from obese African American and Caucasian women.
    Metabolism: clinical and experimental, 2004, Volume: 53, Issue:2

    Topics: Adipose Tissue; Adrenergic beta-Agonists; Adult; Black or African American; Cell Membrane; Female; Humans; Immunoblotting; Isoproterenol; Kinetics; Lipolysis; Obesity, Morbid; Omentum; Pindolol; Radioligand Assay; Receptors, Adrenergic, beta; White People

2004

Other Studies

64 other study(ies) available for cyanopindolol and isoproterenol

ArticleYear
Uncoupling the Structure-Activity Relationships of β2 Adrenergic Receptor Ligands from Membrane Binding.
    Journal of medicinal chemistry, 2016, 06-23, Volume: 59, Issue:12

    Topics: Binding Sites; Cell Membrane; Dose-Response Relationship, Drug; Humans; Ligands; Models, Molecular; Molecular Structure; Receptors, Adrenergic, beta-2; Structure-Activity Relationship

2016
Localization of (-)-[125I]cyanopindolol binding in guinea-pig heart: characteristics of non-beta-adrenoceptor related binding in cardiac pacemaker and conducting regions.
    Neuroscience letters, 1992, Feb-17, Volume: 136, Issue:1

    Topics: Alprenolol; Animals; Ascorbic Acid; Binding Sites; Ethanolamines; Female; Guinea Pigs; Haloperidol; Heart Conduction System; Isoproterenol; Male; Myocardium; Peroxidase; Phentolamine; Pindolol; Propanolamines; Propranolol; Protein Binding; Receptors, Adrenergic, beta; Serotonin; Thiophenes; Trachea

1992
Human retinal pigment epithelial cells possess beta 2-adrenergic receptors.
    Experimental eye research, 1992, Volume: 55, Issue:3

    Topics: Adenylyl Cyclases; Betaxolol; Cells, Cultured; Cyclic AMP; Epinephrine; Humans; Isoproterenol; Norepinephrine; Pigment Epithelium of Eye; Pindolol; Propanolamines; Receptors, Adrenergic, beta

1992
Functional properties of the rat and human beta 3-adrenergic receptors: differential agonist activation of recombinant receptors in Chinese hamster ovary cells.
    Molecular pharmacology, 1992, Volume: 42, Issue:4

    Topics: Adenylyl Cyclases; Animals; Binding, Competitive; Cell Membrane; CHO Cells; Cricetinae; Enzyme Activation; Humans; Isoproterenol; Pindolol; Rats; Receptors, Adrenergic, beta; Recombinant Proteins

1992
Regulation of cardiac adenylate cyclase activity in rodent models of obesity.
    The Biochemical journal, 1992, Apr-01, Volume: 283 ( Pt 1)

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Binding, Competitive; Disease Models, Animal; GTP-Binding Proteins; Iodine Radioisotopes; Isoproterenol; Kinetics; Male; Membranes; Mice; Mice, Obese; Myocardium; Obesity; Pindolol; Rats; Rats, Zucker; Receptors, Adrenergic, beta; Stimulation, Chemical

1992
Coexisting beta 1- and atypical beta-adrenergic receptors cause redundant increases in cyclic AMP in human neuroblastoma cells.
    Molecular pharmacology, 1992, Volume: 42, Issue:5

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Cyclic AMP; Ethanolamines; Humans; Imidazoles; Isoproterenol; Neuroblastoma; Pindolol; Radioligand Assay; Receptors, Adrenergic, beta; RNA, Messenger; Tumor Cells, Cultured

1992
Reduced responsiveness of adenylate cyclase to forskolin in human lymphoma cells.
    Biochemical pharmacology, 1991, Sep-12, Volume: 42, Issue:7

    Topics: Adenylyl Cyclase Inhibitors; Aged; B-Lymphocytes; Binding Sites; Cholera Toxin; Colforsin; Cyclic AMP; Female; Humans; Isoproterenol; Lymphoma, Non-Hodgkin; Male; Middle Aged; Pindolol; Receptors, Adrenergic, beta; Signal Transduction; Tumor Cells, Cultured

1991
Characterization of catecholamine-mediated relaxations in rat isolated gastric fundus: evidence for an atypical beta-adrenoceptor.
    British journal of pharmacology, 1991, Volume: 103, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Animals; Catecholamines; Ethanolamines; Gastric Fundus; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle Tonus; Muscle, Smooth; Norepinephrine; Pindolol; Prazosin; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta

1991
Coexistence of three beta-adrenoceptor subtypes in white fat cells of various mammalian species.
    European journal of pharmacology, 1991, Jul-09, Volume: 199, Issue:3

    Topics: Adipose Tissue; Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cell Membrane; Cricetinae; Dogs; Ethanolamines; Humans; Iodine Radioisotopes; Isoproterenol; Kinetics; Lipolysis; Male; Mesocricetus; Muscle, Smooth; Pindolol; Propanolamines; Rabbits; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta

1991
Photoperiodic control of adipocyte alpha 2-adrenoceptors in Syrian hamsters: role of testosterone.
    Endocrinology, 1990, Volume: 127, Issue:3

    Topics: Adipose Tissue; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brain; Brimonidine Tartrate; Cricetinae; Dioxanes; Idazoxan; Isoproterenol; Kidney; Light; Lipolysis; Male; Mesocricetus; Periodicity; Pindolol; Quinoxalines; Receptors, Adrenergic, alpha; Testosterone

1990
Beta-adrenergic receptors on human lymphocytes: comparison of down-regulation in vivo and in vitro.
    Pharmacology, 1990, Volume: 40, Issue:6

    Topics: Adrenergic beta-Antagonists; Down-Regulation; Humans; Isoproterenol; Lymphocytes; Pindolol; Receptors, Adrenergic, beta; Terbutaline; Time Factors

1990
A mutation of the beta 2-adrenergic receptor impairs agonist activation of adenylyl cyclase without affecting high affinity agonist binding. Distinct molecular determinants of the receptor are involved in physical coupling to and functional activation of
    The Journal of biological chemistry, 1990, Jan-25, Volume: 265, Issue:3

    Topics: Adenylyl Cyclases; Amino Acid Sequence; Cell Compartmentation; DNA Mutational Analysis; Endocytosis; Enzyme Activation; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Humans; In Vitro Techniques; Isoproterenol; Macromolecular Substances; Molecular Sequence Data; Mutation; Pindolol; Radioligand Assay; Receptors, Adrenergic, beta; Structure-Activity Relationship

1990
Chronic norepinephrine elicits desensitization by uncoupling the beta-receptor.
    The Journal of clinical investigation, 1989, Volume: 84, Issue:6

    Topics: Adenylyl Cyclases; Animals; Colforsin; Dogs; Drug Tolerance; GTP-Binding Proteins; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Heart Ventricles; Hemodynamics; Isoproterenol; Norepinephrine; Organ Size; Pindolol; Receptors, Adrenergic, beta; Sodium Fluoride; Sodium-Potassium-Exchanging ATPase; Ventricular Function

1989
[Dependence of kinetic constants of intact human lymphocyte beta2-adrenoreceptors on the nature of the radioligands used].
    Biokhimiia (Moscow, Russia), 1989, Volume: 54, Issue:2

    Topics: Adrenergic beta-Antagonists; Alprenolol; Binding, Competitive; Ethylmaleimide; Humans; Isoproterenol; Kinetics; Lymphocytes; Pindolol; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta; Temperature

1989
Influence of lactate on isoproterenol-induced lipolysis and beta-adrenoceptors distribution in human fat cells.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 1989, Volume: 21, Issue:4

    Topics: Adipose Tissue; Adrenergic beta-Antagonists; Adult; Cell Membrane; Cells, Cultured; Humans; Isoproterenol; Lactates; Lipolysis; Middle Aged; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Serotonin Antagonists

1989
Treatment of oophorectomized guinea pigs with intrauterine 17 beta-estradiol pellets may modulate myometrial beta-adrenergic receptor binding properties.
    American journal of obstetrics and gynecology, 1989, Volume: 161, Issue:6 Pt 1

    Topics: Adrenergic beta-Antagonists; Animals; Estradiol; Female; Guanosine Triphosphate; Guinea Pigs; Isoproterenol; Myometrium; Ovariectomy; Pindolol; Progesterone; Receptors, Adrenergic, beta

1989
Pregnancy-induced changes in the interaction of guinea pig myometrial beta-adrenergic receptors with l-isoproterenol.
    American journal of obstetrics and gynecology, 1989, Volume: 161, Issue:6 Pt 1

    Topics: Adrenergic beta-Antagonists; Animals; Female; Guanosine Triphosphate; Guinea Pigs; Isoproterenol; Myometrium; Pindolol; Pregnancy; Pregnancy, Animal; Receptors, Adrenergic, beta

1989
Immune cytokine inhibition of beta-adrenergic agonist stimulated cyclic AMP generation in cardiac myocytes.
    Biochemical and biophysical research communications, 1988, Jan-15, Volume: 150, Issue:1

    Topics: Animals; Animals, Newborn; Biological Products; Cells, Cultured; Culture Media; Cyclic AMP; Cytokines; Isoproterenol; Lymphocyte Activation; Lymphocytes; Macrophages; Myocardium; Pindolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Spleen

1988
Regulation of guinea pig myometrial beta-adrenoreceptors by guanosine triphosphate and magnesium ion.
    Biology of reproduction, 1988, Volume: 38, Issue:3

    Topics: Animals; Female; Guanosine Triphosphate; Guinea Pigs; Iodine Radioisotopes; Isoproterenol; Magnesium; Myometrium; Pindolol; Pregnancy; Propranolol; Radioimmunoassay; Receptors, Adrenergic, beta

1988
Cyanopindolol is a highly potent and selective antagonist at the presynaptic serotonin autoreceptor in the rat brain cortex.
    Naunyn-Schmiedeberg's archives of pharmacology, 1985, Volume: 331, Issue:4

    Topics: Adrenergic beta-Antagonists; Animals; Cerebral Cortex; Isoproterenol; Male; Pindolol; Propanolamines; Rats; Receptors, Serotonin; Stereoisomerism

1985
Analysis of agonist dissociation constants as assessed by functional antagonism in guinea pig left atria.
    Journal of pharmacological methods, 1986, Volume: 15, Issue:2

    Topics: Adenosine; Adrenergic beta-Antagonists; Angiotensin-Converting Enzyme Inhibitors; Animals; Benzofurans; Carbachol; Catechols; Gallopamil; Guinea Pigs; Heart; In Vitro Techniques; Iodine Radioisotopes; Isoproterenol; Kinetics; Male; Myocardial Contraction; Nifedipine; Pindolol; Propanolamines

1986
Characteristics of the beta-adrenergic receptor in the rat ventral prostate using [125I]cyanopindolol.
    Molecular and cellular endocrinology, 1986, Volume: 48, Issue:1

    Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Chemical Precipitation; Epinephrine; Isoproterenol; Male; Norepinephrine; Pindolol; Polyethylene Glycols; Prostate; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta

1986
Gi affects the agonist-binding properties of beta-adrenoceptors in the presence of Gs.
    European journal of biochemistry, 1988, Feb-15, Volume: 172, Issue:1

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Catalysis; Cholera Toxin; Erythrocyte Membrane; GTP-Binding Proteins; Isoproterenol; Lymphoma; Pertussis Toxin; Pindolol; Receptors, Adrenergic, beta; Turkeys; Virulence Factors, Bordetella

1988
Identity of inhibitory presynaptic 5-hydroxytryptamine (5-HT) autoreceptors in the rat brain cortex with 5-HT1B binding sites.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 332, Issue:1

    Topics: Animals; Cerebral Cortex; In Vitro Techniques; Isoproterenol; Ketanserin; Kinetics; Male; Pindolol; Piperidines; Rats; Receptors, Serotonin; Serotonin Antagonists; Subcellular Fractions; Swine

1986
Induction of functional beta-adrenergic receptors in rat aortic smooth muscle cells by sodium butyrate.
    Biochemical pharmacology, 1986, Nov-01, Volume: 35, Issue:21

    Topics: Adenylyl Cyclases; Animals; Butyrates; Butyric Acid; Cell Membrane; Cells, Cultured; Isoproterenol; Kinetics; Muscle, Smooth, Vascular; Pindolol; Rats; Receptors, Adrenergic, beta

1986
Characterization of beta-1 and beta-2 adrenoceptors in guinea pig atrium: functional and receptor binding studies.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:3

    Topics: Animals; Electric Stimulation; Ethanolamines; Female; Guinea Pigs; Heart Atria; Heart Rate; Imidazoles; Isoproterenol; Kinetics; Myocardial Contraction; Myocardium; Pindolol; Procaterol; Propanolamines; Receptors, Adrenergic, beta; Stimulation, Chemical; Uterine Contraction; Uterus

1987
Forskolin-stimulated adenylyl cyclase activity is decreased but beta 2-adrenoceptor function is unchanged in primary hypertension.
    Journal of cardiovascular pharmacology, 1993, Volume: 22, Issue:5

    Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Adult; Binding, Competitive; Cell Membrane; Colforsin; Female; Hemodynamics; Humans; Hypertension; Isoproterenol; Leukocytes, Mononuclear; Male; Middle Aged; Pindolol; Receptors, Adrenergic, beta; Sex Factors

1993
Influence of beta 2-adrenergic receptor genotypes on signal transduction in human airway smooth muscle cells.
    American journal of respiratory cell and molecular biology, 1995, Volume: 13, Issue:1

    Topics: Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Cells, Cultured; Cyclic AMP; Dose-Response Relationship, Drug; Down-Regulation; Genotype; Humans; Isoproterenol; Muscle, Smooth; Pindolol; Radioligand Assay; Receptors, Adrenergic, beta-2; Second Messenger Systems; Signal Transduction; Trachea

1995
Response of mouse proximal straight tubule and medullary thick ascending limb to beta-agonist.
    Journal of the American Society of Nephrology : JASN, 1993, Volume: 4, Issue:5

    Topics: Adrenergic beta-Antagonists; Animals; Electrophysiology; Furosemide; In Vitro Techniques; Isoproterenol; Kidney Medulla; Kidney Tubules; Kidney Tubules, Proximal; Kinetics; Membrane Potentials; Mice; Perfusion; Pindolol; Propanolamines; Propranolol; Radioligand Assay; Receptors, Adrenergic, beta

1993
Regulation of beta-adrenoceptors in the guinea-pig sinoatrial node.
    Naunyn-Schmiedeberg's archives of pharmacology, 1994, Volume: 349, Issue:5

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Autoradiography; Binding Sites; Catechols; Chromatography, High Pressure Liquid; Densitometry; Down-Regulation; Drug Interactions; Female; Guinea Pigs; Heart Atria; Isoproterenol; Male; Myocardial Contraction; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Sinoatrial Node

1994
Atypical beta-adrenoceptor- (beta 3-adrenoceptor) mediated relaxation of canine isolated bronchial smooth muscle.
    Journal of applied physiology (Bethesda, Md. : 1985), 1993, Volume: 74, Issue:1

    Topics: Acetylcholine; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Bronchi; Cyclic AMP; Dogs; Ethanolamines; Female; In Vitro Techniques; Isometric Contraction; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Phentolamine; Pindolol; Propanolamines; Receptors, Adrenergic, beta

1993
Cocaine selectively inhibits beta-adrenergic receptor binding in pregnant human myometrium.
    American journal of obstetrics and gynecology, 1993, Volume: 169, Issue:3

    Topics: Adrenergic beta-Antagonists; Binding, Competitive; Cocaine; Dihydroergotoxine; Dose-Response Relationship, Drug; Female; Humans; In Vitro Techniques; Isoproterenol; Least-Squares Analysis; Molecular Structure; Myometrium; Pindolol; Pregnancy; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta

1993
Guanine nucleotide regulatory protein alterations in young Milan hypertensive strain rats.
    Biochimica et biophysica acta, 1994, Jan-11, Volume: 1225, Issue:2

    Topics: Adenylyl Cyclases; Alprostadil; Amino Acid Sequence; Animals; Cell Membrane; Cells, Cultured; Colforsin; GTP-Binding Proteins; Hypertension; Immune Sera; Isoproterenol; Molecular Sequence Data; Muscle, Smooth, Vascular; Pindolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Signal Transduction

1994
Effects of chronic infusion of (-)-isoprenaline on rat cardiac muscarinic (M2)-cholinoceptors and beta 1- and beta 2-adrenoceptors.
    Journal of autonomic pharmacology, 1995, Volume: 15, Issue:4

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Binding, Competitive; Down-Regulation; Heart Ventricles; Imidazoles; Infusion Pumps, Implantable; Isoproterenol; Male; Myocardium; N-Methylscopolamine; Pindolol; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Muscarinic; Scopolamine Derivatives

1995
Characterization and localization of atypical beta-adrenoceptors in rat ileum.
    British journal of pharmacology, 1995, Volume: 116, Issue:6

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Autoradiography; Binding Sites; Binding, Competitive; Female; Ileum; Iodine Radioisotopes; Isoproterenol; Kinetics; Male; Pindolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2

1995
Different atypical beta-adrenoceptors mediate isoprenaline-induced relaxation in vascular and non-vascular smooth muscles.
    Life sciences, 1995, Mar-03, Volume: 56, Issue:15

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Ethanolamines; Female; In Vitro Techniques; Isoproterenol; Muscle Relaxation; Muscle, Smooth; Muscle, Smooth, Vascular; Pindolol; Rats; Receptors, Adrenergic, beta

1995
Inducible expression of beta 1- and beta 2-adrenergic receptors in rat C6 glioma cells: functional interactions between closely related subtypes.
    Molecular pharmacology, 1996, Volume: 50, Issue:1

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Colforsin; Cyclic AMP; Epinephrine; Gene Expression Regulation, Neoplastic; Genomic Library; Glioma; Imidazoles; Isopropyl Thiogalactoside; Isoproterenol; Kinetics; Norepinephrine; Pindolol; Radioligand Assay; Rats; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Recombinant Proteins; Transfection; Tumor Cells, Cultured

1996
Identification and functional role of beta-adrenergic receptor subtypes in primate and rodent: in vivo versus isolated myocytes.
    Journal of molecular and cellular cardiology, 1996, Volume: 28, Issue:6

    Topics: Adrenergic beta-Antagonists; Animals; Betaxolol; Blood Pressure; Cells, Cultured; Coronary Vessels; Heart; Heart Rate; In Vitro Techniques; Isoproterenol; Kinetics; Male; Myocardium; Papio; Pindolol; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Vascular Resistance; Ventricular Function, Left; Ventricular Function, Right

1996
Role of 5-HT1b receptor in the pressure-induced behavioral and neurochemical disorders in rats.
    Pharmacology, biochemistry, and behavior, 1996, Volume: 53, Issue:2

    Topics: Adrenergic beta-Agonists; Animals; Atmospheric Pressure; Behavior, Animal; Brain Chemistry; Calibration; Dopamine; Electrochemistry; Electrodes; High Pressure Neurological Syndrome; Isoproterenol; Male; Motor Activity; Neostriatum; Pindolol; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1996
Propranolol therapy in experimental heart failure in rabbits improves cardiac response to catecholamines without beta-adrenoceptor up-regulation.
    Fundamental & clinical pharmacology, 1995, Volume: 9, Issue:6

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-Antagonists; Animals; Cardiac Output, Low; Catecholamines; Female; Heart; Heart Function Tests; Heart Rate; Hemodynamics; Isoproterenol; Male; Myocardium; Norepinephrine; Pindolol; Propranolol; Rabbits; Receptors, Adrenergic, beta; Up-Regulation; Ventricular Function

1995
Mutations of Tyr326 in the beta 2-adrenoceptor disrupt multiple receptor functions.
    European journal of pharmacology, 1996, Jun-27, Volume: 307, Issue:2

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alanine; Animals; Cell Membrane; CHO Cells; Cloning, Molecular; Cricetinae; Gene Expression; Humans; Iodine Radioisotopes; Isoproterenol; Mutagenesis, Site-Directed; Mutation; Phenylalanine; Pindolol; Protein Binding; Radioligand Assay; Receptors, Adrenergic, beta-2; Transfection; Tyrosine

1996
Effect of endurance physical training on rat liver adenylyl cyclase system.
    Cellular signalling, 1996, Volume: 8, Issue:4

    Topics: Adaptation, Physiological; Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Colforsin; Enzyme Activation; Fluorides; Glucagon; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Isoproterenol; Liver; Male; Manganese; Physical Conditioning, Animal; Physical Endurance; Pindolol; Random Allocation; Rats; Rats, Wistar; Receptors, Adrenergic, beta

1996
Growth hormone treatment of hypophysectomized rats increases catecholamine-induced lipolysis and the number of beta-adrenergic receptors in adipocytes: no differences in the effects of growth hormone on different fat depots.
    Obesity research, 1996, Volume: 4, Issue:5

    Topics: Adipocytes; Adrenergic beta-Agonists; Animals; Female; Growth Hormone; Hypophysectomy; Iodine Radioisotopes; Isoproterenol; Lipolysis; Male; Norepinephrine; Pindolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta

1996
Beta 3-adrenoceptors mediating relaxation of the oesophageal tunica muscularis mucosae and distal colon in the rat: comparative pharmacology and their desensitization by BRL 37344.
    Journal of autonomic pharmacology, 1996, Volume: 16, Issue:4

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Colon; Dose-Response Relationship, Drug; Esophagus; Ethanolamines; Isoproterenol; Male; Muscle Relaxation; Pindolol; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3

1996
Molecular mechanisms of adenylyl cyclase desensitization in pregnant rat myometrium following in vivo administration of the beta-adrenergic agonist, isoproterenol.
    Biology of reproduction, 1998, Volume: 59, Issue:1

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Colforsin; Drug Tolerance; Female; GTP-Binding Proteins; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Isoproterenol; Myometrium; Pindolol; Pregnancy; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; RNA, Messenger

1998
Pharmacological and molecular characterisation of beta-adrenoceptors in adult rat diaphragm muscle.
    Respiration physiology, 1998, Volume: 112, Issue:1

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aging; Animals; Dose-Response Relationship, Drug; Fenoterol; Imidazoles; Isoproterenol; Male; Muscle, Smooth; Pindolol; Prenalterol; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3

1998
Atypical adrenoceptor-mediated relaxation of canine pulmonary artery through a cAMP-dependent pathway.
    Biochemical and biophysical research communications, 1998, Jul-30, Volume: 248, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Cyclic AMP; Dioxoles; Dogs; Ethanolamines; Female; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Pindolol; Propanolamines; Pulmonary Artery; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3

1998
Alterations in cardiac membrane beta-adrenoceptors and adenylyl cyclase due to hypochlorous acid.
    Journal of molecular and cellular cardiology, 1999, Volume: 31, Issue:1

    Topics: Adenosine Diphosphate; Adenylate Cyclase Toxin; Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Ascorbic Acid; Cholera Toxin; Colforsin; Dose-Response Relationship, Drug; Ethylmaleimide; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Hypochlorous Acid; Immunoblotting; Isoproterenol; Lipid Peroxidation; Methionine; Myocardium; Pertussis Toxin; Pindolol; Propane; Rats; Receptors, Adrenergic; Sodium Fluoride; Virulence Factors, Bordetella

1999
Similar structures and shared switch mechanisms of the beta2-adrenoceptor and the parathyroid hormone receptor. Zn(II) bridges between helices III and VI block activation.
    The Journal of biological chemistry, 1999, Jun-11, Volume: 274, Issue:24

    Topics: Animals; Binding, Competitive; Evolution, Molecular; GTP-Binding Protein alpha Subunits, Gs; Guanosine 5'-O-(3-Thiotriphosphate); Histidine; Humans; Isoproterenol; Models, Molecular; Mutation; Pindolol; Protein Engineering; Protein Structure, Secondary; Receptors, Adrenergic, beta-2; Receptors, Parathyroid Hormone; Rod Opsins; Secretin; Sequence Alignment; Signal Transduction; Zinc

1999
Coupling efficiencies of beta 1- and beta 2-adrenergic receptors expressed alone or together in transfected GH3 pituitary cells.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 290, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cells, Cultured; Cyclic AMP; Imidazoles; Iodine Radioisotopes; Isopropyl Thiogalactoside; Isoproterenol; Kinetics; Pindolol; Pituitary Gland, Anterior; Propanolamines; Rats; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Transfection

1999
Characterisation of the atypical beta-adrenoceptor in rabbit isolated jejunum using BRL 37344, cyanopindolol and SR 59230A.
    Journal of autonomic pharmacology, 1999, Volume: 19, Issue:2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; Drug Interactions; Ethanolamines; Female; In Vitro Techniques; Isoproterenol; Jejunum; Male; Pindolol; Propanolamines; Propranolol; Rabbits; Receptors, Adrenergic, beta

1999
Beta 1-, beta 2- and atypical beta-adrenoceptor-mediated relaxation in rat isolated aorta.
    British journal of pharmacology, 2000, Volume: 129, Issue:4

    Topics: Acetylcholine; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Aorta, Thoracic; Bupranolol; Dose-Response Relationship, Drug; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Norepinephrine; Pindolol; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Substrate Specificity; Vasodilator Agents

2000
Role of endothelium/nitric oxide in atypical beta-adrenoceptor-mediated relaxation in rat isolated aorta.
    European journal of pharmacology, 2000, Jun-16, Volume: 398, Issue:2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Aorta, Thoracic; Dose-Response Relationship, Drug; Endothelium, Vascular; In Vitro Techniques; Isoproterenol; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitroprusside; Norepinephrine; Oxadiazoles; Phenoxyacetates; Phenoxypropanolamines; Phenylacetates; Pindolol; Propanolamines; Propranolol; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Vasodilation

2000
Agonist-directed trafficking of porcine alpha(2A)-adrenergic receptor signaling in Chinese hamster ovary cells: l-isoproterenol selectively activates G(s).
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 294, Issue:2

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Animals; Binding Sites; Brimonidine Tartrate; CHO Cells; Cricetinae; Drug Interactions; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; Isoproterenol; Kinetics; Oxymetazoline; Pindolol; Protein Binding; Quinoxalines; Receptors, Adrenergic, alpha-2; Serotonin Antagonists; Signal Transduction; Swine; Yohimbine

2000
beta(1)-Adrenoceptors compensate for beta(3)-adrenoceptors in ileum from beta(3)-adrenoceptor knock-out mice.
    British journal of pharmacology, 2001, Volume: 132, Issue:2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dioxoles; Genotype; Ileum; In Vitro Techniques; Isoproterenol; Mice; Mice, Knockout; Muscle Relaxation; Muscle, Smooth; Pindolol; Propranolol; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger

2001
Abolition of (-)-CGP 12177-evoked cardiostimulation in double beta1/beta2-adrenoceptor knockout mice. Obligatory role of beta1-adrenoceptors for putative beta4-adrenoceptor pharmacology.
    Naunyn-Schmiedeberg's archives of pharmacology, 2001, Volume: 363, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Atrial Function; Binding, Competitive; Bucladesine; Dose-Response Relationship, Drug; Female; Genotype; Heart Atria; In Vitro Techniques; Isoproterenol; Male; Membranes; Mice; Mice, Knockout; Myocardial Contraction; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Sinoatrial Node; Tritium

2001
The Ile164 beta(2)-adrenoceptor polymorphism alters salmeterol exosite binding and conventional agonist coupling to G(s).
    European journal of pharmacology, 2001, Jun-15, Volume: 421, Issue:3

    Topics: Adrenergic beta-Agonists; Albuterol; Amino Acid Substitution; Animals; Binding Sites; Binding, Competitive; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; Genotype; Humans; Iodine Radioisotopes; Isoproterenol; Metaproterenol; Pindolol; Polymorphism, Genetic; Radioligand Assay; Receptors, Adrenergic, beta-2; Salmeterol Xinafoate; Terbutaline

2001
Studies on the expression and function of beta-3-adrenoceptors in the colon of rats with acetic acid-induced colitis.
    Pharmacology, 2002, Volume: 64, Issue:2

    Topics: Acetic Acid; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Colitis, Ulcerative; Colon; Dose-Response Relationship, Drug; Ethanolamines; Female; Isoproterenol; Muscle Relaxation; Muscle, Smooth; Peroxidase; Pindolol; Potassium Chloride; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-3; RNA, Messenger

2002
Characterization of mexiletine as an antagonist of beta-adrenoceptor in Chinese hamster ovary cells expressing cloned human beta-adrenoceptors.
    Biochemical pharmacology, 2004, Mar-01, Volume: 67, Issue:5

    Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Antagonists; Animals; Anti-Arrhythmia Agents; Binding, Competitive; Cell Membrane; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Drug Interactions; Female; Humans; Iodine Radioisotopes; Isoproterenol; Kinetics; Lidocaine; Mexiletine; Pindolol; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Transfection

2004
Functional responses of human beta1 adrenoceptors with defined haplotypes for the common 389R>G and 49S>G polymorphisms.
    Pharmacogenetics, 2004, Volume: 14, Issue:6

    Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Cells, Cultured; Cyclic AMP; DNA, Complementary; Down-Regulation; Genotype; Haplotypes; Humans; Iodine Radioisotopes; Isoproterenol; Kidney; Ligands; Pindolol; Polymorphism, Genetic; Receptors, Adrenergic, beta-1

2004
Evidence for the presence of beta-3-adrenoceptors mediating relaxation in the human oviduct.
    Pharmacology, 2005, Volume: 74, Issue:3

    Topics: Adrenergic beta-3 Receptor Agonists; Adrenergic beta-3 Receptor Antagonists; Adult; Dose-Response Relationship, Drug; Ethanolamines; Fallopian Tubes; Female; Humans; In Vitro Techniques; Isoproterenol; Middle Aged; Muscle Relaxation; Pindolol; Propranolol; Receptors, Adrenergic, beta-3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger

2005
Beta-adrenoceptor-mediated vascular relaxation in spontaneously hypertensive rats.
    Autonomic neuroscience : basic & clinical, 2005, Mar-31, Volume: 118, Issue:1-2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Aorta, Thoracic; Dose-Response Relationship, Drug; Endothelium, Vascular; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Pindolol; Propanolamines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta; Tetrahydronaphthalenes

2005
Role of the G protein-coupled receptor kinase site serine cluster in beta2-adrenergic receptor internalization, desensitization, and beta-arrestin translocation.
    The Journal of biological chemistry, 2006, Mar-17, Volume: 281, Issue:11

    Topics: Adenylyl Cyclases; Alanine; Arrestins; Aspartic Acid; beta-Arrestin 1; beta-Arrestin 2; beta-Arrestins; Binding Sites; Blotting, Western; Cell Line; Cell Membrane; Cyclic AMP-Dependent Protein Kinases; DNA, Complementary; Epinephrine; G-Protein-Coupled Receptor Kinase 1; Green Fluorescent Proteins; Humans; Isoproterenol; Kinetics; Mutation; Phosphorylation; Pindolol; Protein Structure, Tertiary; Protein Transport; Receptors, Adrenergic, beta-2; Serine; Time Factors; Transfection

2006
Preservation of the positive lusitropic effect of beta-adrenoceptors stimulation in diabetic cardiomyopathy.
    Anesthesia and analgesia, 2008, Volume: 107, Issue:4

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cardiomyopathies; Colforsin; Diabetes Complications; Diabetes Mellitus, Experimental; Echocardiography; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; NG-Nitroarginine Methyl Ester; Nitric Oxide; Papillary Muscles; Phentolamine; Pindolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta

2008