Page last updated: 2024-08-26

cyanopindolol and cgp 20712a

cyanopindolol has been researched along with cgp 20712a in 18 studies

Research

Studies (18)

TimeframeStudies, this research(%)All Research%
pre-19902 (11.11)18.7374
1990's12 (66.67)18.2507
2000's4 (22.22)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Duke, BJ; Jackman, GP; Louis, SN; Louis, WJ; Machida, CA; Nero, TL; Rezmann-Vitti, LA1
Fraeyman, N; Van de Velde, E; Van Ermen, A; Vanscheeuwijck, P1
Esbenshade, TA; Granneman, JG; Han, C; Minneman, KP; Theroux, TL1
Amenta, F; Coppola, L; Ferrante, F; Forlani, A; Gallo, P; Monopoli, A; Napoleone, P1
Kim, YS; Molenaar, P; Sainz, RD; Summers, RJ1
Molenaar, P; Summers, RJ1
Canale, E; Molenaar, P; Summers, RJ1
Elnatan, J; Molenaar, P; Rosenfeldt, FL; Summers, RJ1
Molenaar, P; Sarsero, D1
Esbenshade, TA; Guerrero, SW; Minneman, KP; Zhong, H1
Bernstein, D; Chruscinski, A; Desai, KH; Kobilka, BK; Rohrer, DK; Schauble, E1
Malinowska, B; Schlicker, E1
Atlan, G; Collet, F; Féve, B; Frisdal, E; Pavoine, C; Pecker, F1
Guerrero, SW; Minneman, KP1
Brawley, L; MacDonald, A; Shaw, AM1
Töneke, K1
Brahmadevara, N; MacDonald, A; Shaw, AM1
Baranowska, M; Kozłowska, H; Kozłowski, M; Malinowska, B; Schlicker, E1

Other Studies

18 other study(ies) available for cyanopindolol and cgp 20712a

ArticleYear
Role of Tyr(356(7.43)) and Ser(190(4.57)) in antagonist binding in the rat beta1-adrenergic receptor.
    Journal of medicinal chemistry, 2006, Jun-15, Volume: 49, Issue:12

    Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Binding Sites; Binding, Competitive; CHO Cells; Cricetinae; Cricetulus; Models, Molecular; Mutagenesis, Site-Directed; Propanolamines; Rats; Receptors, Adrenergic, beta-1; Serine; Stereoisomerism; Transfection; Tyrosine

2006
Influence of age on the beta 1- and beta 2-adrenergic receptors in rat liver.
    Molecular pharmacology, 1992, Volume: 42, Issue:4

    Topics: Adenylyl Cyclases; Aging; Animals; Binding, Competitive; Cell Membrane; Imidazoles; Liver; Liver Glycogen; Male; Pindolol; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta

1992
Coexisting beta 1- and atypical beta-adrenergic receptors cause redundant increases in cyclic AMP in human neuroblastoma cells.
    Molecular pharmacology, 1992, Volume: 42, Issue:5

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Cyclic AMP; Ethanolamines; Humans; Imidazoles; Isoproterenol; Neuroblastoma; Pindolol; Radioligand Assay; Receptors, Adrenergic, beta; RNA, Messenger; Tumor Cells, Cultured

1992
Autoradiographic localization of beta-adrenergic receptors in human large coronary arteries.
    Circulation research, 1991, Volume: 68, Issue:6

    Topics: Adolescent; Adrenergic beta-Antagonists; Adult; Autoradiography; Binding, Competitive; Coronary Vessels; Female; Humans; Imidazoles; Male; Pindolol; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta; Silver; Tissue Distribution

1991
Characterization of beta 1- and beta 2-adrenoceptors in rat skeletal muscles.
    Biochemical pharmacology, 1991, Oct-09, Volume: 42, Issue:9

    Topics: Adrenergic beta-Antagonists; Animals; Autoradiography; Binding Sites; Binding, Competitive; Imidazoles; Male; Membranes; Muscles; Pindolol; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta

1991
Characterization of beta-1 and beta-2 adrenoceptors in guinea pig atrium: functional and receptor binding studies.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:3

    Topics: Animals; Electric Stimulation; Ethanolamines; Female; Guinea Pigs; Heart Atria; Heart Rate; Imidazoles; Isoproterenol; Kinetics; Myocardial Contraction; Myocardium; Pindolol; Procaterol; Propanolamines; Receptors, Adrenergic, beta; Stimulation, Chemical; Uterine Contraction; Uterus

1987
Autoradiographic localization of beta-1 and beta-2 adrenoceptors in guinea pig atrium and regions of the conducting system.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:3

    Topics: Animals; Autoradiography; Binding, Competitive; Guinea Pigs; Heart Atria; Heart Conduction System; Imidazoles; Isomerism; Kinetics; Myocardium; Pindolol; Propanolamines; Receptors, Adrenergic, beta

1987
Autoradiographic localization and quantitation of beta 1- and beta 2-adrenoceptors in the human atrioventricular conducting system: a comparison of patients with idiopathic dilated cardiomyopathy and ischemic heart disease.
    Journal of molecular and cellular cardiology, 1994, Volume: 26, Issue:3

    Topics: Adrenergic beta-Antagonists; Adult; Aged; Atrioventricular Node; Binding, Competitive; Bundle of His; Cardiomyopathy, Dilated; Down-Regulation; Female; Heart Septum; Humans; Imidazoles; Male; Middle Aged; Muscle Proteins; Myocardial Ischemia; Pindolol; Propanolamines; Receptors, Adrenergic, beta

1994
Effects of chronic infusion of (-)-isoprenaline on rat cardiac muscarinic (M2)-cholinoceptors and beta 1- and beta 2-adrenoceptors.
    Journal of autonomic pharmacology, 1995, Volume: 15, Issue:4

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Binding, Competitive; Down-Regulation; Heart Ventricles; Imidazoles; Infusion Pumps, Implantable; Isoproterenol; Male; Myocardium; N-Methylscopolamine; Pindolol; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Muscarinic; Scopolamine Derivatives

1995
Inducible expression of beta 1- and beta 2-adrenergic receptors in rat C6 glioma cells: functional interactions between closely related subtypes.
    Molecular pharmacology, 1996, Volume: 50, Issue:1

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Colforsin; Cyclic AMP; Epinephrine; Gene Expression Regulation, Neoplastic; Genomic Library; Glioma; Imidazoles; Isopropyl Thiogalactoside; Isoproterenol; Kinetics; Norepinephrine; Pindolol; Radioligand Assay; Rats; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Recombinant Proteins; Transfection; Tumor Cells, Cultured

1996
The developmental and physiological consequences of disrupting genes encoding beta 1 and beta 2 adrenoceptors.
    Advances in pharmacology (San Diego, Calif.), 1998, Volume: 42

    Topics: Adrenergic beta-Antagonists; Animals; Crosses, Genetic; Homozygote; Imidazoles; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Mice, Knockout; Pindolol; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Stem Cells

1998
Further evidence for differences between cardiac atypical beta-adrenoceptors and brown adipose tissue beta3-adrenoceptors in the pithed rat.
    British journal of pharmacology, 1997, Volume: 122, Issue:7

    Topics: Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dioxoles; Dose-Response Relationship, Drug; Heart Rate; Imidazoles; Male; Pindolol; Propanolamines; Rats; Rats, Wistar; Temperature

1997
Pharmacological and molecular characterisation of beta-adrenoceptors in adult rat diaphragm muscle.
    Respiration physiology, 1998, Volume: 112, Issue:1

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aging; Animals; Dose-Response Relationship, Drug; Fenoterol; Imidazoles; Isoproterenol; Male; Muscle, Smooth; Pindolol; Prenalterol; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3

1998
Coupling efficiencies of beta 1- and beta 2-adrenergic receptors expressed alone or together in transfected GH3 pituitary cells.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 290, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cells, Cultured; Cyclic AMP; Imidazoles; Iodine Radioisotopes; Isopropyl Thiogalactoside; Isoproterenol; Kinetics; Pindolol; Pituitary Gland, Anterior; Propanolamines; Rats; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Transfection

1999
Beta 1-, beta 2- and atypical beta-adrenoceptor-mediated relaxation in rat isolated aorta.
    British journal of pharmacology, 2000, Volume: 129, Issue:4

    Topics: Acetylcholine; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Aorta, Thoracic; Bupranolol; Dose-Response Relationship, Drug; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Norepinephrine; Pindolol; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Substrate Specificity; Vasodilator Agents

2000
Beta-adrenoceptors in equine trachea and heart.
    Veterinary research communications, 1999, Volume: 23, Issue:1

    Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Female; Heart Atria; Heart Ventricles; Horses; Imidazoles; Iodine Radioisotopes; Ligands; Male; Muscle, Smooth; Myocardium; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Regression Analysis; Spectrometry, Gamma; Trachea

1999
ALpha1-adrenoceptor antagonist properties of CGP 12177A and other beta-adrenoceptor ligands: evidence against beta(3)- or atypical beta-adrenoceptors in rat aorta.
    British journal of pharmacology, 2004, Volume: 142, Issue:4

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-1 Receptor Antagonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Aorta, Thoracic; Binding Sites; Bupranolol; Cell Membrane; Cerebral Cortex; Dose-Response Relationship, Drug; Ethanolamines; Imidazoles; Male; Muscle, Smooth, Vascular; Phenylephrine; Pindolol; Prazosin; Propanolamines; Propranolol; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-3; Tritium; United Kingdom; Vasoconstriction

2004
Potential involvement of a propranolol-insensitive atypical beta-adrenoceptor the vasodilator effect of cyanopindolol in the human pulmonary artery.
    Journal of physiology and pharmacology : an official journal of the Polish Physiological Society, 2006, Volume: 57, Issue:3

    Topics: Adrenergic beta-Antagonists; Analysis of Variance; Bupranolol; Dose-Response Relationship, Drug; Female; Humans; Imidazoles; In Vitro Techniques; Male; Middle Aged; Pindolol; Pulmonary Artery; Receptor, Serotonin, 5-HT2A; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Serotonin 5-HT2 Receptor Antagonists; Vasoconstriction; Vasodilation; Vasodilator Agents

2006