cy 208-243 has been researched along with sk&f-38393 in 17 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 4 (23.53) | 18.7374 |
1990's | 13 (76.47) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Floersheim, P; Markstein, R; Seiler, MP; Widmer, A | 1 |
O'Boyle, KM; Waddington, JL | 1 |
Abbott, B; Starr, BS; Starr, MS | 1 |
Baldessarini, RJ; Booth, RG; Evans, HK; Gallitano, AL; Gelbard, HA; Marsh, ER; Teicher, MH | 1 |
Murray, AM; Waddington, JL | 1 |
Berry, SA; Gudelsky, GA | 1 |
Damsma, G; Fibiger, HC; Robertson, GS; Tham, CS | 1 |
al-Tajir, G; Starr, MS | 1 |
Chandler, CJ; Starr, BS; Starr, MS; Wohab, W | 1 |
Murphy, K; Peterson, MR; Robertson, GS; Robertson, HA | 1 |
Weiss, B; Winkler, JD | 1 |
Edwards, SR; Jackson, DM; Ross, SB | 1 |
Edwards, SR; Jackson, DM; Ross, SB; Wallis, EM | 1 |
Bergman, J; Rosenzweig-Lipson, S; Spealman, RD | 1 |
Barber, DJ; Cooper, SJ; Francis, J | 1 |
Gessa, GL; Imperato, A; Obinu, MC | 1 |
Brewster, WK; Knoerzer, TA; Mailman, RB; Mottola, D; Nichols, DE; Watts, VJ | 1 |
17 other study(ies) available for cy 208-243 and sk&f-38393
Article | Year |
---|---|
Structure-activity relationships in the trans-hexahydroindolo[4,3-ab]phenanthridine ("benzergoline") series. 2. Resolution, absolute configuration, and dopaminergic activity of the selective D1 agonist CY 208-243 and its implication for an "extended rotam
Topics: Adenylyl Cyclases; Animals; Brain; Cattle; Dopamine Agents; Indoles; Models, Molecular; Molecular Conformation; Phenanthridines; Rats; Stereoisomerism; Structure-Activity Relationship | 1993 |
Agonist and antagonist interactions with D1 dopamine receptors: agonist-induced masking of D1 receptors depends on intrinsic activity.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Analgesics; Animals; Benzazepines; Binding, Competitive; Cell Membrane; Corpus Striatum; Guanylyl Imidodiphosphate; Indoles; Kinetics; Phenanthridines; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone | 1992 |
CY 208-243 behaves as a typical D-1 agonist in the reserpine-treated mouse.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Dopamine Agents; Dose-Response Relationship, Drug; Female; Grooming; Indoles; Male; Metoclopramide; Mice; Motor Activity; Phenanthridines; Phenethylamines; Reaction Time; Receptors, Dopamine; Receptors, Dopamine D1; Reserpine | 1991 |
Dopamine D1 autoreceptor function: possible expression in developing rat prefrontal cortex and striatum.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Cerebral Cortex; Corpus Striatum; Dihydroxyphenylalanine; Dopamine Agents; Ergolines; Female; Indoles; Male; Phenanthridines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1 | 1991 |
New putative selective agonists at the D-1 dopamine receptor: behavioural and neurochemical comparison of CY 208-243 with SK&F 101384 and SK&F 103243.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Benzazepines; Corpus Striatum; Dopamine Agents; Fluorenes; Indoles; Male; Naphthalenes; Phenanthridines; Phenethylamines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Stereotyped Behavior; Tetrahydronaphthalenes | 1990 |
D1 receptors function to inhibit the activation of tuberoinfundibular dopamine neurons.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antiparkinson Agents; Brain; Dopamine; Haloperidol; Indoles; Injections, Intraperitoneal; Male; Neurons; Phenanthridines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Tyrosine 3-Monooxygenase | 1990 |
Dopamine D1 receptor stimulation increases striatal acetylcholine release in the rat.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acetylcholine; Animals; Antiparkinson Agents; Behavior, Animal; Benzazepines; Corpus Striatum; Dialysis; Dopamine Agents; Grooming; Indoles; Phenanthridines; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1990 |
Anticonvulsant action of SCH 23390 in the striatum of the rat.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Anticonvulsants; Antiparkinson Agents; Benzazepines; Corpus Striatum; Dopamine Agents; Ergolines; Female; Indoles; Injections; Male; Nucleus Accumbens; Phenanthridines; Pilocarpine; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Seizures; Stereotaxic Techniques | 1990 |
Motor depression: a new role for D1 receptors?
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Dopamine Antagonists; Drug Synergism; Female; Habituation, Psychophysiologic; Indoles; Male; Metoclopramide; Mice; Mice, Inbred Strains; Motor Activity; Phenanthridines; Receptors, Dopamine; Receptors, Dopamine D1; Sulpiride | 1990 |
D1-dopamine receptor agonists selectively activate striatal c-fos independent of rotational behaviour.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Corpus Striatum; Hydroxydopamines; Indoles; Male; Oxidopamine; Phenanthridines; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-fos; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Stereotyped Behavior | 1989 |
Effect of continuous exposure to selective D1 and D2 dopaminergic agonists on rotational behavior in supersensitive mice.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Benzazepines; Dopamine Agents; Ergolines; Fenoldopam; Indoles; Male; Mice; Phenanthridines; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Rotation; Tetrahydronaphthalenes; Thiophenes | 1989 |
Dopamine D2 agonist-induced behavioural depression is reversed by dopamine D1 agonists.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Bromocriptine; Dose-Response Relationship, Drug; Ergolines; Indoles; Male; Mice; Motor Activity; Phenanthridines; Quinpirole; Receptors, Dopamine | 1989 |
Enhancement by a single dose of reserpine (plus alpha methyl-p-tyrosine) of the central stimulatory effects evoked by dopamine D-1 and D-2 agonists in the mouse.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; alpha-Methyltyrosine; Animals; Appetite Depressants; Benzazepines; Central Nervous System; Corpus Striatum; Ergolines; Indoles; Male; Methyltyrosines; Mice; Motor Activity; Phenanthridines; Quinpirole; Receptors, Dopamine; Reserpine; Stereotyped Behavior | 1988 |
Differential effects of dopamine D1 and D2 receptor agonists on schedule-controlled behavior of squirrel monkeys.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Conditioning, Psychological; Dopamine Agonists; Indoles; Male; Oxazines; Phenanthridines; Phenethylamines; Receptors, Dopamine D1; Receptors, Dopamine D2; Saimiri | 1995 |
Selective dopamine D-1 receptor agonists, SK&F 38393 and CY 208-243 reduce sucrose sham-feeding in the rat.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Appetite Depressants; Dopamine Agents; Dose-Response Relationship, Drug; Feeding Behavior; Indoles; Male; Phenanthridines; Rats; Receptors, Dopamine D1; Sucrose | 1993 |
Stimulation of both dopamine D1 and D2 receptors facilitates in vivo acetylcholine release in the hippocampus.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acetylcholine; Animals; Apomorphine; Dialysis; Dopamine Agents; Dose-Response Relationship, Drug; Ergolines; Hippocampus; Indoles; Male; Phenanthridines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2 | 1993 |
Dopaminergic benzo[a]phenanthridines: resolution and pharmacological evaluation of the enantiomers of dihydrexidine, the full efficacy D1 dopamine receptor agonist.
Topics: Animals; Benzazepines; Binding Sites; Corpus Striatum; Dopamine Agents; Humans; Male; Mice; Phenanthridines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Stereoisomerism; Transfection | 1994 |