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cy 208-243 and sk&f-38393

cy 208-243 has been researched along with sk&f-38393 in 17 studies

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-19904 (23.53)18.7374
1990's13 (76.47)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Floersheim, P; Markstein, R; Seiler, MP; Widmer, A1
O'Boyle, KM; Waddington, JL1
Abbott, B; Starr, BS; Starr, MS1
Baldessarini, RJ; Booth, RG; Evans, HK; Gallitano, AL; Gelbard, HA; Marsh, ER; Teicher, MH1
Murray, AM; Waddington, JL1
Berry, SA; Gudelsky, GA1
Damsma, G; Fibiger, HC; Robertson, GS; Tham, CS1
al-Tajir, G; Starr, MS1
Chandler, CJ; Starr, BS; Starr, MS; Wohab, W1
Murphy, K; Peterson, MR; Robertson, GS; Robertson, HA1
Weiss, B; Winkler, JD1
Edwards, SR; Jackson, DM; Ross, SB1
Edwards, SR; Jackson, DM; Ross, SB; Wallis, EM1
Bergman, J; Rosenzweig-Lipson, S; Spealman, RD1
Barber, DJ; Cooper, SJ; Francis, J1
Gessa, GL; Imperato, A; Obinu, MC1
Brewster, WK; Knoerzer, TA; Mailman, RB; Mottola, D; Nichols, DE; Watts, VJ1

Other Studies

17 other study(ies) available for cy 208-243 and sk&f-38393

ArticleYear
Structure-activity relationships in the trans-hexahydroindolo[4,3-ab]phenanthridine ("benzergoline") series. 2. Resolution, absolute configuration, and dopaminergic activity of the selective D1 agonist CY 208-243 and its implication for an "extended rotam
    Journal of medicinal chemistry, 1993, Apr-16, Volume: 36, Issue:8

    Topics: Adenylyl Cyclases; Animals; Brain; Cattle; Dopamine Agents; Indoles; Models, Molecular; Molecular Conformation; Phenanthridines; Rats; Stereoisomerism; Structure-Activity Relationship

1993
Agonist and antagonist interactions with D1 dopamine receptors: agonist-induced masking of D1 receptors depends on intrinsic activity.
    Neuropharmacology, 1992, Volume: 31, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Analgesics; Animals; Benzazepines; Binding, Competitive; Cell Membrane; Corpus Striatum; Guanylyl Imidodiphosphate; Indoles; Kinetics; Phenanthridines; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

1992
CY 208-243 behaves as a typical D-1 agonist in the reserpine-treated mouse.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 38, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Dopamine Agents; Dose-Response Relationship, Drug; Female; Grooming; Indoles; Male; Metoclopramide; Mice; Motor Activity; Phenanthridines; Phenethylamines; Reaction Time; Receptors, Dopamine; Receptors, Dopamine D1; Reserpine

1991
Dopamine D1 autoreceptor function: possible expression in developing rat prefrontal cortex and striatum.
    Brain research. Developmental brain research, 1991, Nov-19, Volume: 63, Issue:1-2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Cerebral Cortex; Corpus Striatum; Dihydroxyphenylalanine; Dopamine Agents; Ergolines; Female; Indoles; Male; Phenanthridines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1

1991
New putative selective agonists at the D-1 dopamine receptor: behavioural and neurochemical comparison of CY 208-243 with SK&F 101384 and SK&F 103243.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 35, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Benzazepines; Corpus Striatum; Dopamine Agents; Fluorenes; Indoles; Male; Naphthalenes; Phenanthridines; Phenethylamines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Stereotyped Behavior; Tetrahydronaphthalenes

1990
D1 receptors function to inhibit the activation of tuberoinfundibular dopamine neurons.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 254, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antiparkinson Agents; Brain; Dopamine; Haloperidol; Indoles; Injections, Intraperitoneal; Male; Neurons; Phenanthridines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Tyrosine 3-Monooxygenase

1990
Dopamine D1 receptor stimulation increases striatal acetylcholine release in the rat.
    European journal of pharmacology, 1990, Sep-21, Volume: 186, Issue:2-3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acetylcholine; Animals; Antiparkinson Agents; Behavior, Animal; Benzazepines; Corpus Striatum; Dialysis; Dopamine Agents; Grooming; Indoles; Phenanthridines; Rats; Rats, Inbred Strains; Receptors, Dopamine

1990
Anticonvulsant action of SCH 23390 in the striatum of the rat.
    European journal of pharmacology, 1990, Dec-04, Volume: 191, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Anticonvulsants; Antiparkinson Agents; Benzazepines; Corpus Striatum; Dopamine Agents; Ergolines; Female; Indoles; Injections; Male; Nucleus Accumbens; Phenanthridines; Pilocarpine; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Seizures; Stereotaxic Techniques

1990
Motor depression: a new role for D1 receptors?
    Neuroscience, 1990, Volume: 38, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Dopamine Antagonists; Drug Synergism; Female; Habituation, Psychophysiologic; Indoles; Male; Metoclopramide; Mice; Mice, Inbred Strains; Motor Activity; Phenanthridines; Receptors, Dopamine; Receptors, Dopamine D1; Sulpiride

1990
D1-dopamine receptor agonists selectively activate striatal c-fos independent of rotational behaviour.
    Brain research, 1989, Dec-04, Volume: 503, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Corpus Striatum; Hydroxydopamines; Indoles; Male; Oxidopamine; Phenanthridines; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-fos; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Stereotyped Behavior

1989
Effect of continuous exposure to selective D1 and D2 dopaminergic agonists on rotational behavior in supersensitive mice.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 249, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Benzazepines; Dopamine Agents; Ergolines; Fenoldopam; Indoles; Male; Mice; Phenanthridines; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Rotation; Tetrahydronaphthalenes; Thiophenes

1989
Dopamine D2 agonist-induced behavioural depression is reversed by dopamine D1 agonists.
    Journal of neural transmission, 1989, Volume: 75, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Bromocriptine; Dose-Response Relationship, Drug; Ergolines; Indoles; Male; Mice; Motor Activity; Phenanthridines; Quinpirole; Receptors, Dopamine

1989
Enhancement by a single dose of reserpine (plus alpha methyl-p-tyrosine) of the central stimulatory effects evoked by dopamine D-1 and D-2 agonists in the mouse.
    Naunyn-Schmiedeberg's archives of pharmacology, 1988, Volume: 337, Issue:5

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; alpha-Methyltyrosine; Animals; Appetite Depressants; Benzazepines; Central Nervous System; Corpus Striatum; Ergolines; Indoles; Male; Methyltyrosines; Mice; Motor Activity; Phenanthridines; Quinpirole; Receptors, Dopamine; Reserpine; Stereotyped Behavior

1988
Differential effects of dopamine D1 and D2 receptor agonists on schedule-controlled behavior of squirrel monkeys.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 273, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Conditioning, Psychological; Dopamine Agonists; Indoles; Male; Oxazines; Phenanthridines; Phenethylamines; Receptors, Dopamine D1; Receptors, Dopamine D2; Saimiri

1995
Selective dopamine D-1 receptor agonists, SK&F 38393 and CY 208-243 reduce sucrose sham-feeding in the rat.
    Neuropharmacology, 1993, Volume: 32, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Appetite Depressants; Dopamine Agents; Dose-Response Relationship, Drug; Feeding Behavior; Indoles; Male; Phenanthridines; Rats; Receptors, Dopamine D1; Sucrose

1993
Stimulation of both dopamine D1 and D2 receptors facilitates in vivo acetylcholine release in the hippocampus.
    Brain research, 1993, Aug-06, Volume: 618, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acetylcholine; Animals; Apomorphine; Dialysis; Dopamine Agents; Dose-Response Relationship, Drug; Ergolines; Hippocampus; Indoles; Male; Phenanthridines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2

1993
Dopaminergic benzo[a]phenanthridines: resolution and pharmacological evaluation of the enantiomers of dihydrexidine, the full efficacy D1 dopamine receptor agonist.
    Journal of medicinal chemistry, 1994, Jul-22, Volume: 37, Issue:15

    Topics: Animals; Benzazepines; Binding Sites; Corpus Striatum; Dopamine Agents; Humans; Male; Mice; Phenanthridines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Stereoisomerism; Transfection

1994