Page last updated: 2024-08-25

cromakalim and tolbutamide

cromakalim has been researched along with tolbutamide in 25 studies

Research

Studies (25)

TimeframeStudies, this research(%)All Research%
pre-19905 (20.00)18.7374
1990's18 (72.00)18.2507
2000's1 (4.00)29.6817
2010's1 (4.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
de Hemptinne, A; Vanheel, B1
Kozlowski, RZ; Nye, PC; Robertson, BE1
Henderson, G; Hicks, GA1
Chang, CC; Hong, SJ1
Pilsudski, R; Rougier, O; Tourneur, Y1
Antoine, MH; Berkenboom, G; Fang, ZY; Fontaine, J; Herchuelz, A; Hermann, M; Lebrun, P1
Dunne, MJ; Gallacher, DV; Petersen, OH; Yule, DI1
Wilson, C1
Brayden, JE; Davies, NW; Huang, Y; Nelson, MT; Quayle, JM; Standen, NB1
Sanguinetti, MC; Siegl, PK; Wolleben, CD1
Grafe, P; Lehmann-Horn, F; Spuler, A1
Grafe, P; Lehmann-Horn, F; Quasthoff, S; Spuler, A1
Do, ML; Halterman, TJ; Howe, BB; Kau, ST; Li, JH; McConville, MW; Trivedi, S; Yochim, CL; Zografos, P1
Nakaya, H1
Finta, EP; Fischer, HD; Harms, L; Illes, P; Sevcik, J1
Fleck, E; Henning, B; Hildebrandt, AG; Ott, T; Zünkler, BJ1
Fullerton, DA; McIntyre, RC; Meldrum, DR; Sheridan, BC1
Hosseinzadeh, H; Stone, TW1
Frey, G; Lucht, M; Schlue, WR1
Aguilar-Bryan, L; Babenko, AP; Bryan, J; Gonzalez, G1
Chagneau, C; De Gottardi, A; Fléjou, JF; Fouassier, L; Housset, C; Lahaye, P; Lebrec, D; Moreau, R; Reichen, J; Rona, JP; Tazi, KA1
Carpenter, E; Peers, C; Roberts, ML; Taylor, SC1
Smoak, IW1
Conte Camerino, D; Desai, RR; George, AL; Lundquist, AL; Mele, A; Tricarico, D1
Breschi, MC; Calderone, V; Cecchetti, V; Martelli, A; Sabatini, S; Testai, L1

Reviews

1 review(s) available for cromakalim and tolbutamide

ArticleYear
[Potential role of ATP-sensitive K+ channels in ischemia- and reperfusion-induced arrhythmias].
    Kokyu to junkan. Respiration & circulation, 1993, Volume: 41, Issue:6

    Topics: Action Potentials; Adenosine Triphosphate; Animals; Arrhythmias, Cardiac; Benzopyrans; Cromakalim; Glyburide; Guanidines; Humans; Myocardial Ischemia; Myocardial Reperfusion Injury; Myocardium; Niacinamide; Nicorandil; Pinacidil; Potassium; Potassium Channels; Pyrroles; Tolbutamide

1993

Other Studies

24 other study(ies) available for cromakalim and tolbutamide

ArticleYear
Influence of KATP channel modulation on net potassium efflux from ischaemic mammalian cardiac tissue.
    Cardiovascular research, 1992, Volume: 26, Issue:11

    Topics: Action Potentials; Animals; Barium; Benzopyrans; Cromakalim; Glyburide; Guinea Pigs; Hydrogen-Ion Concentration; Muscles; Myocardial Ischemia; Oxygen; Papillary Muscles; Potassium; Potassium Channels; Pyrroles; Tolbutamide; Vasodilator Agents

1992
Opposing actions of tolbutamide and glibenclamide on hypoxic pulmonary vasoconstriction.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1992, Volume: 102, Issue:3

    Topics: Animals; Benzopyrans; Cromakalim; Diazoxide; Glyburide; Hypoxia; In Vitro Techniques; Lung; Male; Potassium Channels; Pyrroles; Rats; Tolbutamide; Vasoconstriction

1992
Lack of evidence for coupling of the dopamine D2 receptor to an adenosine triphosphate-sensitive potassium (ATP-K+) channel in dopaminergic neurones of the rat substantia nigra.
    Neuroscience letters, 1992, Jul-20, Volume: 141, Issue:2

    Topics: Adenosine Triphosphate; Animals; Benzopyrans; Cromakalim; Dopamine; Electrophysiology; Glyburide; Male; Neurons; Potassium Channels; Pyrroles; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Dopamine D2; Substantia Nigra; Tolbutamide

1992
Hyperpolarization of denervated skeletal muscle by lemakalim and its antagonism by glybenclamide and tolbutamide.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 259, Issue:2

    Topics: Animals; Benzopyrans; Calcium Channel Blockers; Cesium; Cromakalim; Female; Glyburide; Male; Membrane Potentials; Mice; Muscle Denervation; Muscles; Pyrroles; Tolbutamide

1991
Action of cromakalim on potassium membrane conductance in isolated heart myocytes of frog.
    British journal of pharmacology, 1990, Volume: 100, Issue:3

    Topics: Adenosine Triphosphate; Animals; Barium; Benzopyrans; Cesium; Cromakalim; Glyburide; In Vitro Techniques; Membranes; Myocardium; Potassium Channels; Pyrroles; Rana esculenta; Sulfonylurea Compounds; Tolbutamide

1990
Hypoglycemic sulfonylureas antagonize the effects of cromakalim and pinacidil on 86Rb fluxes and contractile activity in the rat aorta.
    Pharmacology, 1990, Volume: 41, Issue:1

    Topics: Animals; Aorta, Thoracic; Benzopyrans; Cromakalim; Glyburide; Guanidines; Hypoglycemic Agents; In Vitro Techniques; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nitroprusside; Parasympatholytics; Pinacidil; Potassium Channels; Pyrroles; Rats; Rats, Inbred Strains; Rubidium Radioisotopes; Sulfonylurea Compounds; Tetraethylammonium Compounds; Tolbutamide; Vasodilator Agents

1990
Comparative study of the effects of cromakalim (BRL 34915) and diazoxide on membrane potential, [Ca2+]i and ATP-sensitive potassium currents in insulin-secreting cells.
    The Journal of membrane biology, 1990, Volume: 114, Issue:1

    Topics: Adenosine Triphosphate; Animals; Benzopyrans; Calcium; Cell Line; Cromakalim; Diazoxide; Glucose; Islets of Langerhans; Kinetics; Membrane Potentials; Potassium Channels; Pyrroles; Tolbutamide

1990
Inhibition by sulphonylureas of vasorelaxation induced by K+ channel activators in vitro.
    Journal of autonomic pharmacology, 1989, Volume: 9, Issue:1

    Topics: Animals; Antihypertensive Agents; Benzopyrans; Cromakalim; Drug Interactions; Glipizide; Glyburide; Guanidines; In Vitro Techniques; Male; Nifedipine; Norepinephrine; Pinacidil; Potassium Channels; Potassium Chloride; Pyrroles; Rabbits; Sulfonylurea Compounds; Tolbutamide; Vasodilator Agents

1989
Hyperpolarizing vasodilators activate ATP-sensitive K+ channels in arterial smooth muscle.
    Science (New York, N.Y.), 1989, Jul-14, Volume: 245, Issue:4914

    Topics: Acetylcholine; Adenosine Triphosphate; Animals; Benzopyrans; Cerebral Arteries; Cromakalim; Diazoxide; Glyburide; Guanidines; Mesenteric Arteries; Muscle, Smooth, Vascular; Pinacidil; Potassium Channels; Pyrroles; Rabbits; Rats; Tolbutamide; Vasoactive Intestinal Peptide; Vasodilator Agents

1989
Influence of ATP-sensitive potassium channel modulators on ischemia-induced fibrillation in isolated rat hearts.
    Journal of molecular and cellular cardiology, 1989, Volume: 21, Issue:8

    Topics: Adenosine Triphosphate; Animals; Antihypertensive Agents; Arrhythmias, Cardiac; Benzopyrans; Coronary Circulation; Coronary Disease; Cromakalim; Glyburide; Guanidines; Heart; Heart Rate; In Vitro Techniques; Male; Perfusion; Pinacidil; Potassium Channels; Pyrroles; Rats; Rats, Inbred Strains; Tolbutamide; Vascular Resistance

1989
Cromakalim (BRL 34915) restores in vitro the membrane potential of depolarized human skeletal muscle fibres.
    Naunyn-Schmiedeberg's archives of pharmacology, 1989, Volume: 339, Issue:3

    Topics: Barium; Benzopyrans; Cromakalim; Humans; Hyperkalemia; In Vitro Techniques; Membrane Potentials; Muscles; Paralysis; Pyrroles; Tolbutamide

1989
Cromakalim, pinacidil and RP 49356 activate a tolbutamide-sensitive K+ conductance in human skeletal muscle fibres.
    Pflugers Archiv : European journal of physiology, 1989, Volume: 414 Suppl 1

    Topics: Benzopyrans; Cromakalim; Guanidines; Humans; In Vitro Techniques; Membrane Potentials; Muscles; Picolines; Pinacidil; Potassium Channels; Pyrans; Pyrroles; Tolbutamide; Vasodilator Agents

1989
Characterization of ATP-sensitive potassium channel-blocking activity of ZENECA ZM181,037, a eukalemic diuretic.
    Pharmacology, 1994, Volume: 49, Issue:4

    Topics: Acetamides; Adenosine Triphosphate; Administration, Oral; Animals; Benzopyrans; Blood Glucose; Blood Pressure; Cromakalim; Diuretics; Dogs; Dose-Response Relationship, Drug; Electrophysiology; Glyburide; Guinea Pigs; Hypertension; In Vitro Techniques; Injections, Intravenous; Male; Muscle Relaxation; Muscle, Smooth; Muscle, Smooth, Vascular; Potassium Channel Blockers; Pyrroles; Rats; Rats, Inbred SHR; Rats, Sprague-Dawley; Stereoisomerism; Tolbutamide

1994
Effects of potassium channel openers and their antagonists on rat locus coeruleus neurones.
    British journal of pharmacology, 1993, Volume: 109, Issue:2

    Topics: Action Potentials; Adenosine Triphosphate; Animals; Barium; Benzopyrans; Cromakalim; Electrophysiology; Glyburide; In Vitro Techniques; Kynurenic Acid; Locus Coeruleus; Male; Membrane Potentials; Neurons; Parasympatholytics; Potassium Channels; Pyridines; Pyrroles; Rats; Rats, Wistar; Substantia Nigra; Tetrodotoxin; Tolbutamide

1993
Effects of tolbutamide on ATP-sensitive K+ channels from human right atrial cardiac myocytes.
    Pharmacology & toxicology, 1997, Volume: 80, Issue:2

    Topics: Adenosine Triphosphate; Adolescent; Adult; Aged; Atrial Function, Right; Benzopyrans; Child; Cromakalim; Drug Interactions; Female; Heart Atria; Humans; Hypoglycemic Agents; Kinetics; Male; Membrane Potentials; Middle Aged; Myocardial Ischemia; Myocardium; Potassium Channels; Pyrroles; Sensitivity and Specificity; Tolbutamide

1997
KATP channels contribute to beta- and adenosine receptor-mediated pulmonary vasorelaxation.
    The American journal of physiology, 1997, Volume: 273, Issue:5

    Topics: Acetylcholine; Adenosine; Adenylyl Cyclases; Animals; ATP-Binding Cassette Transporters; Colforsin; Cromakalim; Cyclic AMP; Cyclic GMP; Glyburide; In Vitro Techniques; Isoproterenol; KATP Channels; Kinetics; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Nitroprusside; Potassium Channels; Potassium Channels, Inwardly Rectifying; Pulmonary Artery; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Purinergic P1; Tolbutamide; Vasodilation

1997
Tolbutamide blocks postsynaptic but not presynaptic effects of adenosine on hippocampal CA1 neurones.
    Journal of neural transmission (Vienna, Austria : 1996), 1998, Volume: 105, Issue:2-3

    Topics: Adenosine; Animals; Baclofen; Calcium; Cardiovascular Agents; Cromakalim; Electric Stimulation; GABA Agonists; Hippocampus; Hypoglycemic Agents; Male; Neurons; Potassium Channel Blockers; Potassium Channels; Pyramidal Cells; Rats; Rats, Wistar; Receptors, Presynaptic; Synapses; Tolbutamide

1998
ATP-inhibited K+ channels and membrane potential of identified leech neurons.
    Brain research, 1998, Jul-06, Volume: 798, Issue:1-2

    Topics: Animal Nutritional Physiological Phenomena; Animals; Antimetabolites; ATP-Binding Cassette Transporters; Chromans; Cromakalim; Electrophysiology; Food Deprivation; KATP Channels; Leeches; Membrane Potentials; Microelectrodes; Neurons; Potassium Channels; Potassium Channels, Inwardly Rectifying; Pyrrolidines; Tolbutamide

1998
Reconstituted human cardiac KATP channels: functional identity with the native channels from the sarcolemma of human ventricular cells.
    Circulation research, 1998, Nov-30, Volume: 83, Issue:11

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Adolescent; Adult; Animals; ATP-Binding Cassette Transporters; Child; CHO Cells; Cloning, Molecular; COS Cells; Cricetinae; Cromakalim; Diazoxide; DNA, Complementary; Gene Library; Glyburide; Heart Ventricles; Humans; Magnesium; Middle Aged; Myocardium; Patch-Clamp Techniques; Pinacidil; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Receptors, Drug; Sarcolemma; Sulfonylurea Receptors; Tolbutamide; Transfection

1998
Endothelium-dependent blunted membrane potential responses to ATP-sensitive K+ channel modulators in aortae from rats with cirrhosis.
    Journal of hepatology, 1999, Volume: 30, Issue:1

    Topics: Adenosine Triphosphate; Animals; Aorta; Bosentan; Cromakalim; Diazoxide; Endothelin-1; Endothelium, Vascular; Glyburide; Liver Cirrhosis, Experimental; Male; Membrane Potentials; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Sprague-Dawley; Sulfonamides; Tolbutamide

1999
Potentiation of quantal catecholamine secretion by glibenclamide: evidence for a novel role of sulphonylurea receptors in regulating the Ca(2+) sensitivity of exocytosis.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1999, Jul-15, Volume: 19, Issue:14

    Topics: Animals; ATP-Binding Cassette Transporters; Caffeine; Calcium; Catecholamines; Cromakalim; Egtazic Acid; Electrochemistry; Exocytosis; Glyburide; Kinetics; Membrane Potentials; Patch-Clamp Techniques; PC12 Cells; Pinacidil; Potassium; Potassium Channels; Potassium Channels, Inwardly Rectifying; Quantum Theory; Rats; Receptors, Drug; Sulfonylurea Receptors; Tolbutamide

1999
Cromakalim: embryonic effects and reduction of tolbutamide-induced dysmorphogenesis in vitro.
    Teratology, 1999, Volume: 60, Issue:5

    Topics: Abnormalities, Multiple; Animals; Cromakalim; Embryonic and Fetal Development; Female; Hypoglycemic Agents; In Vitro Techniques; Male; Mice; Potassium Channels; Pregnancy; Somites; Tolbutamide; Vasodilator Agents

1999
Hybrid assemblies of ATP-sensitive K+ channels determine their muscle-type-dependent biophysical and pharmacological properties.
    Proceedings of the National Academy of Sciences of the United States of America, 2006, Jan-24, Volume: 103, Issue:4

    Topics: Adenosine Triphosphate; Animals; Anti-Arrhythmia Agents; Antihypertensive Agents; ATP-Binding Cassette Transporters; Biophysics; Cromakalim; Diazoxide; DNA Primers; Dose-Response Relationship, Drug; Gene Expression Regulation; Glyburide; Hypoglycemic Agents; KATP Channels; Kinetics; Male; Models, Statistical; Muscle Fibers, Skeletal; Muscle, Skeletal; Muscles; Patch-Clamp Techniques; Phenotype; Potassium; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Rats, Wistar; Receptors, Drug; Recombinant Fusion Proteins; Reverse Transcriptase Polymerase Chain Reaction; Sulfonylurea Receptors; Tolbutamide

2006
Effects of K openers on the QT prolongation induced by HERG-blocking drugs in guinea-pigs.
    The Journal of pharmacy and pharmacology, 2010, Volume: 62, Issue:7

    Topics: Animals; Benzothiadiazines; Cromakalim; Decanoic Acids; Ether-A-Go-Go Potassium Channels; Glyburide; Guinea Pigs; Heart; Humans; Hydroxy Acids; Intracellular Membranes; KATP Channels; Long QT Syndrome; Male; Membrane Transport Modulators; Mitochondrial Membranes; Picolines; Pinacidil; Potassium Channel Blockers; Pyrans; Sarcolemma; Tolbutamide

2010