cp 96345 has been researched along with sr 48968 in 56 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 50 (89.29) | 18.2507 |
2000's | 6 (10.71) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Advenier, C; Bakdach, H; Brelière, JC; Emonds-Alt, X; Le Fur, G; Naline, E; Toty, L; Vilain, P | 1 |
Advenier, C; Emonds-Alt, X; Martin, CA; Naline, E | 1 |
Hay, DW; Hubbard, WC; Undem, BJ | 1 |
Advenier, C; Hirsch, A; Martin, CA; Molimard, M; Naline, E | 1 |
Gerard, NP; Gether, U; Jensen, CJ; Schwartz, TW | 1 |
Buéno, L; Julia, V; Morteau, O | 1 |
Gether, U; Lowe, JA; Schwartz, TW | 1 |
Killingsworth, CR; Shore, SA | 1 |
Boucher, S; Couture, R; Gitter, BD; Howbert, JJ; Picard, P; Regoli, D | 1 |
Advenier, C; Emonds-Alt, X; Qian, Y | 1 |
Brelière, JC; Emonds-Alt, X; Gether, U; Lowe, JA; Nakanishi, S; Schwartz, TW; Snider, RM; Yokota, Y | 1 |
Bertrand, C; Bunnett, NW; Debas, HT; Geppetti, P; Huber, O; Nadel, JA; Pellegrini, CA | 1 |
Giachetti, A; Giuliani, S; Maggi, CA; Patacchini, R | 1 |
Bartho, L; Giuliani, S; Maggi, CA; Santicioli, P | 1 |
Boucher, S; Couture, R; Picard, P; Regoli, D | 1 |
Bertrand, C; Geppetti, P; Graf, PD; Nadel, JA | 1 |
Bertrand, C; Geppetti, P; Graf, PD; Nadel, JA; Ricciardolo, FL; Yoshihara, S | 1 |
Gertner, SB; Selig, WM; Tocker, JE; Welton, AF | 1 |
Håkanson, R; Strichartz, GR; Tung, SR; Wang, ZY | 1 |
Bannenberg, G; Kimland, M; Lundberg, JM; Moldéus, P; Ryrfeldt, A | 1 |
Couture, R; Picard, P; Prat, A; Regoli, D | 1 |
Bertrand, C; Bunnett, NW; Debas, HT; Geppetti, P; Huber, O; Nadel, JA; Nakazato, P; Pellegrini, CA | 1 |
Bertrand, C; Foresi, A; Geppetti, P; Graf, PD; Nadel, JA | 1 |
Buckner, CK; Campbell, J; Dea, D; Krell, RD; Lengel, D; Liberati, N; Miller, S; Shenvi, A; Stinson-Fisher, C | 1 |
Barnes, PJ; Chung, KF; Sakamoto, T; Tsukagoshi, H | 1 |
Alger, LE; Garland, A; Gitter, B; Howbert, JJ; Jordan, JE; Kao, BM; Leff, AR; Necheles, J; Rodger, IW; Solway, J | 1 |
Doerfler, DL; Sailstad, DM; Selgrade, M; Veronesi, B | 1 |
Gascón, P; Rameshwar, P | 1 |
Jafri, MS; Weinreich, D | 1 |
Chapman, RW; Danko, G; del Prado, M; Hey, JA | 1 |
Burcher, E; Nail, B; Yuan, L | 1 |
Ikemura, T; Ishii, H; Ohmori, K; Sasaki, Y | 1 |
Henry, JL; Hui-Chan, CW; Yashpal, K | 1 |
Advenier, C; Bellamy, JF; Emonds-Alt, X; Molimard, M; Naline, E; Regoli, D | 1 |
Chrétien, L; Gobeil, F; Jukic, D; Nguyen, QT; Nguyen-Le, XK; Regoli, D | 1 |
Astolfi, M; Barnes, PJ; Evangelista, S; Mak, JC; Manzini, S; Zhang, XL | 1 |
Boyer, V; Harf, A; Jarreau, PH; Macquin-Mavier, I | 1 |
Culman, J; Klee, S; Ohlendorf, C; Unger, T | 1 |
Cirillo, R; Conte, B; Manzini, S; Parlani, M | 1 |
Ikeda, H; Kaneko, T; Nishikawa, M; Nishiyama, H; Okubo, T; Yamakawa, H | 1 |
Henry, JL; Radhakrishnan, V | 1 |
Holst, JJ; Rasmussen, TN; Schmidt, PT | 1 |
Auberson, S; Kordestani, RK; Lacroix, JS; Lundberg, JM | 1 |
Burcher, E; Nail, BS; Yuan, L | 1 |
Hsu, TH; Kou, YR; Lai, YL | 1 |
Wei, EQ; Wu, RY | 1 |
Coudoré-Civiale, MA; Courteix, C; Eschalier, A; Fialip, J | 1 |
Kohno, S; Nabe, T; Ogawa, K; Yamamura, H | 1 |
Gascón, P; Hameed, M; Joshi, DD; Maloof, PB; Mosenthal, A; Qian, J; Rameshwar, P; Singh, D | 1 |
Leah, JD; Redburn, JL | 1 |
Kamiki, T; Kohno, S; Nabe, T; Tanpo, T; Yasui, K | 1 |
Doi, H; Narita, H | 1 |
Lu, ZY; Wei, EQ; Zhang, WP | 1 |
Chien, CT; Hsu, SM; Lai, MK; Lin, TB; Yu, HJ | 1 |
Chang, LC; Chen, WC; Li, PC; Lin, SC | 1 |
Chen, SS; Chien, CT; Yang, CC | 1 |
1 review(s) available for cp 96345 and sr 48968
Article | Year |
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Tachykinin non-peptide antagonists: binding domain and molecular mode of action.
Topics: Animals; Benzamides; Binding Sites; Binding, Competitive; Biphenyl Compounds; GTP-Binding Proteins; Humans; Kinetics; Mutagenesis, Site-Directed; Neurokinin A; Piperidines; Point Mutation; Protein Structure, Secondary; Receptors, Tachykinin; Recombinant Fusion Proteins; Substance P; Tachykinins | 1995 |
55 other study(ies) available for cp 96345 and sr 48968
Article | Year |
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Effects on the isolated human bronchus of SR 48968, a potent and selective nonpeptide antagonist of the neurokinin A (NK2) receptors.
Topics: Acetylcholine; Amino Acid Sequence; Animals; Benzamides; Biphenyl Compounds; Bronchi; Bronchoconstriction; Cricetinae; Dinoprost; Dose-Response Relationship, Drug; Drug Antagonism; Drug Evaluation, Preclinical; Female; Histamine; Humans; In Vitro Techniques; Male; Middle Aged; Molecular Sequence Data; Neurokinin A; Peptide Fragments; Piperidines; Potassium Chloride; Racemases and Epimerases; Receptors, Neurokinin-2; Receptors, Neurotransmitter | 1992 |
Influence of (+/-)-CP-96,345 and SR 48968 on electrical field stimulation of the isolated guinea-pig main bronchus.
Topics: Animals; Benzamides; Biphenyl Compounds; Bronchi; Bronchoconstriction; Electric Stimulation; Female; Guinea Pigs; In Vitro Techniques; Male; Neurokinin A; Piperidines; Receptors, Neurokinin-2; Receptors, Neurotransmitter | 1992 |
Relative contributions of direct and indirect mechanisms mediating endothelin-induced contraction of guinea-pig trachea.
Topics: Animals; Benzamides; Biphenyl Compounds; Capsaicin; Dicarboxylic Acids; Endothelins; Epithelium; Guinea Pigs; Histamine Release; In Vitro Techniques; Kinetics; Leukotriene Antagonists; Male; Muscle Contraction; Neurokinin A; Piperidines; Prostaglandins; Receptors, Tachykinin; SRS-A; Tetrodotoxin; Trachea | 1993 |
Contractile effects of bradykinin on the isolated human small bronchus.
Topics: Acetylcholine; Aged; Atropine; Benzamides; Biphenyl Compounds; Bradykinin; Bronchi; Bronchoconstriction; Capsaicin; Humans; In Vitro Techniques; Indomethacin; Middle Aged; Muscle, Smooth; Nerve Fibers; Neurokinin A; Neurons, Afferent; Piperidines; Receptors, Bradykinin; Ruthenium Red; Tetrodotoxin | 1994 |
The species selectivity of chemically distinct tachykinin nonpeptide antagonists is dependent on common divergent residues of the rat and human neurokinin-1 receptors.
Topics: Amino Acid Sequence; Animals; Benzamides; Biphenyl Compounds; Cell Line; Dipeptides; Humans; Indoles; Molecular Sequence Data; Mutation; Neurokinin-1 Receptor Antagonists; Piperidines; Rats; Receptors, Neurokinin-1; Recombinant Proteins; Substance P | 1994 |
Involvement of neurokinin 1 and 2 receptors in viscerosensitive response to rectal distension in rats.
Topics: Abdomen; Animals; Benzamides; Biphenyl Compounds; Colon; Colonic Diseases, Functional; Gastrointestinal Motility; Hypnotics and Sedatives; Indoles; Isoindoles; Male; Neurokinin A; Peptide Fragments; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Tachykinin; Rectum; Substance P; Tachykinins | 1994 |
Tachykinin receptors mediating contraction of guinea pig lung strips.
Topics: Acetylcholine; Animals; Benzamides; Biphenyl Compounds; Dipeptides; Guinea Pigs; In Vitro Techniques; Lung; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin B; Peptide Fragments; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Tachykinin; Substance P; Trachea | 1995 |
Use of non-peptide tachykinin receptor antagonists to substantiate the involvement of NK1 and NK2 receptors in a spinal nociceptive reflex in the rat.
Topics: Animals; Benzamides; Biphenyl Compounds; Hypnotics and Sedatives; Injections, Spinal; Male; Neurokinin A; Nociceptors; Pain Measurement; Pain Threshold; Peptide Fragments; Piperidines; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Receptors, Tachykinin; Reflex; Spinal Cord; Substance P | 1993 |
Effects of capsaicin, (+/-)-CP-96,345 and SR 48968 on the bradykinin-induced airways microvascular leakage in guinea-pigs.
Topics: Animals; Autonomic Nervous System; Benzamides; Biphenyl Compounds; Bradykinin; Capillary Permeability; Capsaicin; Evans Blue; Guinea Pigs; Hypnotics and Sedatives; In Vitro Techniques; Nerve Endings; Neurokinin A; Piperidines; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P | 1993 |
Two nonpeptide tachykinin antagonists act through epitopes on corresponding segments of the NK1 and NK2 receptors.
Topics: Animals; Benzamides; Binding Sites; Biphenyl Compounds; Cells, Cultured; Epitopes; Neurokinin A; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P | 1993 |
Tachykinins contract the circular muscle of the human esophageal body in vitro via NK2 receptors.
Topics: Adolescent; Adult; Aged; Atropine; Benzamides; Biphenyl Compounds; Carbachol; Dose-Response Relationship, Drug; Esophagus; Glycopeptides; Humans; Isometric Contraction; Middle Aged; Muscle Contraction; Muscle, Smooth; Neprilysin; Neurokinin A; Neurokinin B; Piperidines; Receptors, Tachykinin; Substance P; Tachykinins; Tetrodotoxin | 1993 |
In vivo and in vitro activity of SR 48,968, a non-peptide tachykinin NK-2 receptor antagonist.
Topics: Animals; Benzamides; Biphenyl Compounds; Blood Pressure; Muscle Contraction; Muscle, Smooth; Neurokinin A; Peptide Fragments; Piperidines; Rats; Receptors, Neurokinin-2; Saliva; Substance P; Sulfones; Urinary Bladder | 1993 |
Tachykinin NK-1 and NK-2 receptors in the circular muscle of the guinea-pig proximal colon.
Topics: Animals; Benzamides; Biphenyl Compounds; Colon; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Peptides, Cyclic; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Sulfones; Tetrodotoxin | 1993 |
Receptor characterization of the spinal action of neurokinins on nociception: a three receptor hypothesis.
Topics: Animals; Benzamides; Biphenyl Compounds; Models, Neurological; Neurokinin A; Neurokinin-1 Receptor Antagonists; Oligopeptides; Pain; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Neurotransmitter; Spinal Cord; Substance P | 1993 |
Capsaicin increases airflow resistance in guinea pigs in vivo by activating both NK2 and NK1 tachykinin receptors.
Topics: Airway Resistance; Animals; Atropine; Benzamides; Biphenyl Compounds; Capsaicin; Dose-Response Relationship, Drug; Drug Interactions; Guinea Pigs; Histamine; Male; Neurokinin A; Peptide Fragments; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P | 1993 |
Role of kinins in anaphylactic-induced bronchoconstriction mediated by tachykinins in guinea-pigs.
Topics: Adrenergic beta-Antagonists; Airway Resistance; Anaphylaxis; Animals; Benzamides; Biphenyl Compounds; Bradykinin; Bronchoconstriction; Glycopeptides; Guinea Pigs; Hypnotics and Sedatives; Kinins; Male; Neprilysin; Neurokinin-1 Receptor Antagonists; Piperidines; Receptors, Neurokinin-2; Tachykinins | 1994 |
Vagal stimulation augments pulmonary anaphylaxis in the guinea pig lung.
Topics: Anaphylaxis; Animals; Atropine; Benzamides; Biphenyl Compounds; Bronchoconstriction; Electric Stimulation; Guinea Pigs; Hypnotics and Sedatives; Lung; Male; Neurokinin A; Organ Size; Physostigmine; Piperidines; Trachea; Vagus Nerve; Vasoconstriction | 1995 |
Non-specific actions of the non-peptide tachykinin receptor antagonists, CP-96,345, RP 67580 and SR 48968, on neurotransmission.
Topics: Action Potentials; Anesthetics, Local; Animals; Benzamides; Biphenyl Compounds; Bupivacaine; Electric Stimulation; Female; Guinea Pigs; In Vitro Techniques; Indoles; Iris; Isoindoles; Male; Muscle Contraction; Muscle, Smooth; Piperidines; Procaine; Rabbits; Rana catesbeiana; Receptors, Tachykinin; Sciatic Nerve; Synaptic Transmission; Vas Deferens | 1994 |
Sensory neuropeptide-mediated bronchoconstriction of the guinea pig lung by diamide; a comparison to hydrogen peroxide.
Topics: Animals; Benzamides; Biphenyl Compounds; Bronchoconstriction; Calcitonin Gene-Related Peptide; Capsaicin; Carbazoles; Diamide; Guinea Pigs; Hydrogen Peroxide; In Vitro Techniques; Lung; Male; Neurokinin A; Neurons, Afferent; Neuropeptides; Piperidines; Thromboxanes | 1994 |
Characterization of the cardiovascular and behavioral effects of centrally administered neuropeptide K in the conscious rat.
Topics: Amino Acid Sequence; Animals; Benzamides; Biphenyl Compounds; Blood Pressure; Cerebral Ventricles; Fenclonine; Heart Rate; Injections, Intraventricular; Male; Molecular Sequence Data; Motor Activity; Neurokinin A; Neuropeptides; Oligopeptides; Piperidines; Rats; Rats, Wistar; Stereotyped Behavior; Tachykinins | 1993 |
Tachykinins mediate contraction of the human lower esophageal sphincter in vitro via activation of NK2 receptors.
Topics: Benzamides; Biphenyl Compounds; Dose-Response Relationship, Drug; Esophagogastric Junction; Glycopeptides; Humans; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Neprilysin; Neurokinin A; Neurokinin B; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Tachykinins | 1993 |
Involvement of neurogenic inflammation in antigen-induced bronchoconstriction in guinea pigs.
Topics: Aerosols; Animals; Atropine; Benzamides; Biphenyl Compounds; Bronchoconstriction; Capsaicin; Glycopeptides; Guinea Pigs; Histamine; Immunization; Inflammation; Lung; Male; Neurokinin-1 Receptor Antagonists; Ovalbumin; Piperidines; Pulmonary Circulation; Receptors, Neurokinin-2; Vascular Resistance | 1993 |
Differential blockade by tachykinin NK1 and NK2 receptor antagonists of bronchoconstriction induced by direct-acting agonists and the indirect-acting mimetics capsaicin, serotonin and 2-methyl-serotonin in the anesthetized guinea pig.
Topics: Amino Acid Sequence; Anesthesia; Animals; Benzamides; Biphenyl Compounds; Bronchial Spasm; Bronchoconstriction; Capsaicin; Guinea Pigs; Hypnotics and Sedatives; Injections, Intravenous; Male; Molecular Sequence Data; Neurokinin A; Piperidines; Receptors, Tachykinin; Serotonin | 1993 |
Involvement of tachykinin receptors (NK1 and NK2) in sodium metabisulfite-induced airway effects.
Topics: Administration, Inhalation; Animals; Benzamides; Biphenyl Compounds; Bronchoconstriction; Capillary Permeability; Female; Guinea Pigs; Pharmaceutic Aids; Piperidines; Receptors, Tachykinin; Sulfites | 1994 |
Tachykinin receptor antagonists inhibit hyperpnea-induced bronchoconstriction in guinea pigs.
Topics: Airway Resistance; Animals; Benzamides; Biphenyl Compounds; Bronchoconstriction; Dose-Response Relationship, Drug; Guinea Pigs; Male; Piperidines; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Tachykinins | 1993 |
Neuropeptide modulation of chemically induced skin irritation.
Topics: Administration, Cutaneous; Animals; Benzamides; Biphenyl Compounds; Capsaicin; Dermatitis, Contact; Dinitrofluorobenzene; Disease Models, Animal; Dose-Response Relationship, Drug; Ear, External; Female; Irritants; Mice; Mice, Inbred BALB C; Neurokinin A; Neuropeptides; Piperidines; Skin; Substance P; Synaptic Transmission | 1995 |
Induction of negative hematopoietic regulators by neurokinin-A in bone marrow stroma.
Topics: Amino Acid Sequence; Benzamides; Biphenyl Compounds; Bone Marrow; Bone Marrow Cells; Cell Division; Cells, Cultured; Chemokine CCL4; Connective Tissue; Depression, Chemical; Erythroid Precursor Cells; Hematopoietic Stem Cells; Humans; Macrophage Inflammatory Proteins; Molecular Sequence Data; Monokines; Neurokinin A; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Transforming Growth Factor beta | 1996 |
Substance P hyperpolarizes vagal sensory neurones of the ferret.
Topics: 4-Aminopyridine; Animals; Anti-Inflammatory Agents, Non-Steroidal; Apamin; Benzamides; Biphenyl Compounds; Cations, Divalent; Cesium; Electrophysiology; Ferrets; In Vitro Techniques; Male; Neurons, Afferent; Nodose Ganglion; Patch-Clamp Techniques; Peptide Fragments; Piperidines; Potassium; Pyrrolidonecarboxylic Acid; Quaternary Ammonium Compounds; Receptors, Tachykinin; Substance P; Vagus Nerve | 1996 |
Augmentation of neurally evoked cholinergic bronchoconstrictor responses by prejunctional NK2 receptors in the guinea-pig.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzamides; Biphenyl Compounds; Bronchoconstriction; Bronchoconstrictor Agents; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Male; Medulla Oblongata; Methacholine Chloride; Muscle, Smooth; Neurokinin A; Neurokinin B; Piperidines; Substance P | 1996 |
Tachykinin receptors and non-cholinergic bronchoconstriction in the anaesthetized guinea-pig.
Topics: Animals; Benzamides; Biphenyl Compounds; Bronchoconstriction; Electric Stimulation; Female; Guinea Pigs; Lung; Male; Peptides, Cyclic; Piperidines; Receptors, Tachykinin; Vagus Nerve | 1996 |
Inhibitory effect of KW-4679, an anti-allergic drug, on tachykinin-mediated airway response induced by electrical vagal stimulation in guinea pigs.
Topics: Animals; Anti-Allergic Agents; Benzamides; Biphenyl Compounds; Bronchoconstriction; Dibenzoxepins; Electric Stimulation; Guinea Pigs; Male; Olopatadine Hydrochloride; Piperidines; Receptors, Tachykinin; Vagus Nerve | 1996 |
SR 48968 specifically depresses neurokinin A- vs. substance P-induced hyperalgesia in a nociceptive withdrawal reflex.
Topics: Animals; Benzamides; Biphenyl Compounds; Dose-Response Relationship, Drug; Hyperalgesia; Injections, Spinal; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Pain Measurement; Pain Threshold; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P | 1996 |
Evidence for functional tachykinin NK1 receptors on human isolated small bronchi.
Topics: Benzamides; Biphenyl Compounds; Bronchi; Female; Hormone Antagonists; Humans; In Vitro Techniques; Indomethacin; Lung Neoplasms; Male; Middle Aged; Neurokinin-1 Receptor Antagonists; Piperidines; Quinuclidines; Receptors, Neurokinin-1; Substance P | 1996 |
Neurokinin receptors in the guinea pig ileum.
Topics: Acetylcholine; Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzamides; Biphenyl Compounds; Guinea Pigs; Ileum; Male; Myenteric Plexus; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Radioligand Assay; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Stereoisomerism; Structure-Activity Relationship; Substance P | 1996 |
Autoradiographic mapping of pulmonary NK1 and NK2 tachykinin receptors and changes after repeated antigen challenge in guinea pigs.
Topics: Animals; Antigens; Autoradiography; Benzamides; Binding Sites; Biphenyl Compounds; Guinea Pigs; Inflammation; Lung; Male; Neurokinin-1 Receptor Antagonists; Ovalbumin; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Tissue Distribution | 1996 |
Aerosolized tachykinin antagonists inhibit pentamidine-induce bronchoconstriction in guinea pigs.
Topics: Aerosols; Animals; Benzamides; Biphenyl Compounds; Bronchi; Bronchoconstriction; Capillary Permeability; Dose-Response Relationship, Drug; Guinea Pigs; Male; Pentamidine; Piperidines; Receptors, Neurokinin-2; Substance P | 1996 |
Effect of tachykinin receptor inhibition in the brain on cardiovascular and behavioral responses to stress.
Topics: Animals; Behavior, Animal; Benzamides; Biphenyl Compounds; Blood Pressure; Brain; Heart Rate; Indoles; Isoindoles; Male; Neurokinin-1 Receptor Antagonists; Periaqueductal Gray; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-2; Stress, Physiological | 1997 |
Characterization of tachykinin NK2 receptor on dog proximal colon. Antagonism by MEN 10,627 and SR 48,968.
Topics: Animals; Benzamides; Biphenyl Compounds; Colon; Dogs; Dose-Response Relationship, Drug; Gastrointestinal Motility; In Vitro Techniques; Muscle Contraction; Peptides, Cyclic; Piperidines; Receptors, Neurokinin-2 | 1996 |
[Airway hyperresponsiveness and airway mucosal permeability].
Topics: Animals; Benzamides; Biphenyl Compounds; Bronchi; Bronchial Hyperreactivity; Capillary Permeability; Guinea Pigs; Male; Piperidines; Receptors, Neurokinin-2; Superoxide Dismutase; Tachykinins | 1996 |
Electrophysiological evidence that neurokinin A acts via NK-1 receptors in the cat dorsal horn.
Topics: Animals; Benzamides; Biphenyl Compounds; Cats; Iontophoresis; Neurokinin A; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Spinal Cord; Stereoisomerism; Substance P; Synapses | 1997 |
Tachykinins may mediate capsaicin-induced, but not vagally induced motility in porcine antrum.
Topics: Animals; Benzamides; Biphenyl Compounds; Capsaicin; Electric Stimulation; Gastrointestinal Motility; Muscle Contraction; Neurokinin A; Neurokinin-1 Receptor Antagonists; Piperidines; Pyloric Antrum; Receptors, Neurokinin-2; Substance P; Swine; Tachykinins; Vagus Nerve | 1997 |
Prejunctional control of pH 6-induced bronchoconstriction by NK1, NK2, mu-opioid, alpha2-adrenoceptor and glucocorticoid receptors in guinea-pig isolated perfused lung.
Topics: Adrenergic alpha-2 Receptor Agonists; Animals; Benzamides; Betamethasone; Biphenyl Compounds; Brimonidine Tartrate; Bronchoconstriction; Calcitonin Gene-Related Peptide; Female; Guinea Pigs; Hydrogen-Ion Concentration; In Vitro Techniques; Lung; Male; Morphine; Neurokinin-1 Receptor Antagonists; Perfusion; Piperidines; Quinoxalines; Quinuclidines; Receptors, Adrenergic, alpha-2; Receptors, Cell Surface; Receptors, Glucocorticoid; Receptors, Neurokinin-2; Receptors, Opioid, mu | 1998 |
Characterization of tachykinin receptors mediating bronchomotor and vasodepressor responses to neuropeptide gamma and substance P in the anaesthetized rabbit.
Topics: Anesthesia; Animals; Benzamides; Biphenyl Compounds; Bronchoconstriction; Drug Interactions; Glycopeptides; Neprilysin; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Protease Inhibitors; Rabbits; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Tachykinins; Vagus Nerve; Vasoconstriction | 1998 |
Smoke-induced airway hyperresponsiveness to inhaled wood smoke in guinea pigs: tachykininergic and cholinergic mechanisms.
Topics: Airway Resistance; Animals; Atropine; Benzamides; Biphenyl Compounds; Bronchi; Bronchial Hyperreactivity; Cholinergic Antagonists; Drug Combinations; Glycopeptides; Guinea Pigs; Male; Neprilysin; Piperidines; Protease Inhibitors; Receptors, Cholinergic; Receptors, Tachykinin; Smoke; Wood | 1998 |
[Inhibitory effects of tachykinin receptor antagonists on leukotriene C4-induced cardiovascular responses in guinea pigs].
Topics: Animals; Benzamides; Biphenyl Compounds; Blood Pressure; Female; Guinea Pigs; Leukotriene C4; Male; Neurokinin-1 Receptor Antagonists; Piperidines; Receptors, Neurokinin-2 | 1996 |
Effect of tachykinin receptor antagonists in experimental neuropathic pain.
Topics: Analgesics; Animals; Benzamides; Biphenyl Compounds; Denervation; Diabetes Mellitus, Experimental; Indoles; Isoindoles; Male; Neurokinin-1 Receptor Antagonists; Pain; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Sciatic Nerve | 1998 |
Nanomolar concentrations of neuropeptides induce histamine release from peritoneal mast cells of a substrain of Wistar rats.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzamides; Biphenyl Compounds; Dose-Response Relationship, Drug; Histamine Release; Male; Mast Cells; Neurokinin A; Peritoneum; Piperidines; Rats; Rats, Sprague-Dawley; Rats, Wistar; Species Specificity; Substance P; Tachykinins | 1999 |
Increased expression of preprotachykinin-I and neurokinin receptors in human breast cancer cells: implications for bone marrow metastasis.
Topics: Benzamides; Biphenyl Compounds; Bone Marrow Cells; Bone Marrow Neoplasms; Breast Neoplasms; Cell Division; Female; Gene Expression Regulation, Neoplastic; Humans; In Situ Hybridization; Neurokinin-1 Receptor Antagonists; Piperidines; Protein Precursors; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Tachykinins; Tumor Cells, Cultured | 2000 |
The induction and potentiation of c-Jun and c-Fos expression in spinal neurons mediated by NK1 and NK2 receptors.
Topics: Animals; Benzamides; Biphenyl Compounds; Male; Neurokinin-1 Receptor Antagonists; Neurons; Patch-Clamp Techniques; Peptides, Cyclic; Piperidines; Proto-Oncogene Proteins c-fos; Proto-Oncogene Proteins c-jun; Rats; Rats, Wistar; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Sciatic Nerve; Spinal Cord | 1999 |
Participation of neuropeptides in antigen-induced contraction of guinea pig bronchi via NK(2) but not NK(1) receptor stimulation.
Topics: Animals; Benzamides; Benzeneacetamides; Biphenyl Compounds; Bronchi; Bronchoconstriction; Female; gamma-Globulins; Guinea Pigs; Histamine H1 Antagonists; Leukotriene Antagonists; Male; Neurokinin-1 Receptor Antagonists; Neuropeptides; Penicillin G; Piperidines; Pyrilamine; Receptors, Neurokinin-2; Substance P; Thiazoles; Trachea | 2000 |
Comparison of the effect of imidaprilat and ramiprilat on broncho-constriction and hypotension induced by bradykinin in guinea pigs.
Topics: Angiotensin I; Angiotensin-Converting Enzyme Inhibitors; Animals; Benzamides; Biphenyl Compounds; Blood Pressure; Bradykinin; Bronchoconstriction; Guinea Pigs; Imidazoles; Imidazolidines; Male; NG-Nitroarginine Methyl Ester; Piperidines; Ramipril | 2000 |
[Effects of tachykinin receptor antagonists on allergic asthma in guinea pigs].
Topics: Animals; Asthma; Benzamides; Biphenyl Compounds; Bronchi; Bronchoconstriction; Female; Guinea Pigs; Male; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Ovalbumin; Piperidines; Receptors, Neurokinin-2; Receptors, Tachykinin; Trachea | 1997 |
Substance P via NK1 receptor facilitates hyperactive bladder afferent signaling via action of ROS.
Topics: Animals; Benzamides; Biphenyl Compounds; Cell Adhesion Molecules; Dose-Response Relationship, Drug; Drug Administration Routes; Electric Stimulation; Female; Free Radical Scavengers; Muscle Contraction; Neurokinin-1 Receptor Antagonists; Pelvis; Piperidines; Rats; Rats, Wistar; Reactive Oxygen Species; Receptors, Neurokinin-1; Reflex, Abnormal; Signal Transduction; Sodium Chloride; Substance P; Superoxide Dismutase; Urinary Bladder; Urinary Bladder, Neurogenic; Urination; Visceral Afferents | 2003 |
Substance P acts via the neurokinin receptor 1 to elicit bronchoconstriction, oxidative stress, and upregulated ICAM-1 expression after oil smoke exposure.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Antioxidants; Ascorbic Acid; Benzamides; Biphenyl Compounds; Blood Pressure; Bronchoalveolar Lavage Fluid; Bronchoconstriction; Catechin; Intercellular Adhesion Molecule-1; Male; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Oxidative Stress; Petroleum; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Respiratory Distress Syndrome; Smoke; Smoke Inhalation Injury; Substance P; Up-Regulation | 2008 |
Colorectal distension enforce acute urinary bladder distension-induced hepatic vasoconstriction in the rat.
Topics: Afferent Pathways; Animals; Benzamides; Biphenyl Compounds; Blood Pressure; Colon; Female; Liver; Neurokinin-1 Receptor Antagonists; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-2; Sympathectomy; Urinary Bladder; Vasoconstriction | 2008 |