Page last updated: 2024-08-26

cp 96345 and sr 48968

cp 96345 has been researched along with sr 48968 in 56 studies

Research

Studies (56)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's50 (89.29)18.2507
2000's6 (10.71)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Advenier, C; Bakdach, H; Brelière, JC; Emonds-Alt, X; Le Fur, G; Naline, E; Toty, L; Vilain, P1
Advenier, C; Emonds-Alt, X; Martin, CA; Naline, E1
Hay, DW; Hubbard, WC; Undem, BJ1
Advenier, C; Hirsch, A; Martin, CA; Molimard, M; Naline, E1
Gerard, NP; Gether, U; Jensen, CJ; Schwartz, TW1
Buéno, L; Julia, V; Morteau, O1
Gether, U; Lowe, JA; Schwartz, TW1
Killingsworth, CR; Shore, SA1
Boucher, S; Couture, R; Gitter, BD; Howbert, JJ; Picard, P; Regoli, D1
Advenier, C; Emonds-Alt, X; Qian, Y1
Brelière, JC; Emonds-Alt, X; Gether, U; Lowe, JA; Nakanishi, S; Schwartz, TW; Snider, RM; Yokota, Y1
Bertrand, C; Bunnett, NW; Debas, HT; Geppetti, P; Huber, O; Nadel, JA; Pellegrini, CA1
Giachetti, A; Giuliani, S; Maggi, CA; Patacchini, R1
Bartho, L; Giuliani, S; Maggi, CA; Santicioli, P1
Boucher, S; Couture, R; Picard, P; Regoli, D1
Bertrand, C; Geppetti, P; Graf, PD; Nadel, JA1
Bertrand, C; Geppetti, P; Graf, PD; Nadel, JA; Ricciardolo, FL; Yoshihara, S1
Gertner, SB; Selig, WM; Tocker, JE; Welton, AF1
Håkanson, R; Strichartz, GR; Tung, SR; Wang, ZY1
Bannenberg, G; Kimland, M; Lundberg, JM; Moldéus, P; Ryrfeldt, A1
Couture, R; Picard, P; Prat, A; Regoli, D1
Bertrand, C; Bunnett, NW; Debas, HT; Geppetti, P; Huber, O; Nadel, JA; Nakazato, P; Pellegrini, CA1
Bertrand, C; Foresi, A; Geppetti, P; Graf, PD; Nadel, JA1
Buckner, CK; Campbell, J; Dea, D; Krell, RD; Lengel, D; Liberati, N; Miller, S; Shenvi, A; Stinson-Fisher, C1
Barnes, PJ; Chung, KF; Sakamoto, T; Tsukagoshi, H1
Alger, LE; Garland, A; Gitter, B; Howbert, JJ; Jordan, JE; Kao, BM; Leff, AR; Necheles, J; Rodger, IW; Solway, J1
Doerfler, DL; Sailstad, DM; Selgrade, M; Veronesi, B1
Gascón, P; Rameshwar, P1
Jafri, MS; Weinreich, D1
Chapman, RW; Danko, G; del Prado, M; Hey, JA1
Burcher, E; Nail, B; Yuan, L1
Ikemura, T; Ishii, H; Ohmori, K; Sasaki, Y1
Henry, JL; Hui-Chan, CW; Yashpal, K1
Advenier, C; Bellamy, JF; Emonds-Alt, X; Molimard, M; Naline, E; Regoli, D1
Chrétien, L; Gobeil, F; Jukic, D; Nguyen, QT; Nguyen-Le, XK; Regoli, D1
Astolfi, M; Barnes, PJ; Evangelista, S; Mak, JC; Manzini, S; Zhang, XL1
Boyer, V; Harf, A; Jarreau, PH; Macquin-Mavier, I1
Culman, J; Klee, S; Ohlendorf, C; Unger, T1
Cirillo, R; Conte, B; Manzini, S; Parlani, M1
Ikeda, H; Kaneko, T; Nishikawa, M; Nishiyama, H; Okubo, T; Yamakawa, H1
Henry, JL; Radhakrishnan, V1
Holst, JJ; Rasmussen, TN; Schmidt, PT1
Auberson, S; Kordestani, RK; Lacroix, JS; Lundberg, JM1
Burcher, E; Nail, BS; Yuan, L1
Hsu, TH; Kou, YR; Lai, YL1
Wei, EQ; Wu, RY1
Coudoré-Civiale, MA; Courteix, C; Eschalier, A; Fialip, J1
Kohno, S; Nabe, T; Ogawa, K; Yamamura, H1
Gascón, P; Hameed, M; Joshi, DD; Maloof, PB; Mosenthal, A; Qian, J; Rameshwar, P; Singh, D1
Leah, JD; Redburn, JL1
Kamiki, T; Kohno, S; Nabe, T; Tanpo, T; Yasui, K1
Doi, H; Narita, H1
Lu, ZY; Wei, EQ; Zhang, WP1
Chien, CT; Hsu, SM; Lai, MK; Lin, TB; Yu, HJ1
Chang, LC; Chen, WC; Li, PC; Lin, SC1
Chen, SS; Chien, CT; Yang, CC1

Reviews

1 review(s) available for cp 96345 and sr 48968

ArticleYear
Tachykinin non-peptide antagonists: binding domain and molecular mode of action.
    Biochemical Society transactions, 1995, Volume: 23, Issue:1

    Topics: Animals; Benzamides; Binding Sites; Binding, Competitive; Biphenyl Compounds; GTP-Binding Proteins; Humans; Kinetics; Mutagenesis, Site-Directed; Neurokinin A; Piperidines; Point Mutation; Protein Structure, Secondary; Receptors, Tachykinin; Recombinant Fusion Proteins; Substance P; Tachykinins

1995

Other Studies

55 other study(ies) available for cp 96345 and sr 48968

ArticleYear
Effects on the isolated human bronchus of SR 48968, a potent and selective nonpeptide antagonist of the neurokinin A (NK2) receptors.
    The American review of respiratory disease, 1992, Volume: 146, Issue:5 Pt 1

    Topics: Acetylcholine; Amino Acid Sequence; Animals; Benzamides; Biphenyl Compounds; Bronchi; Bronchoconstriction; Cricetinae; Dinoprost; Dose-Response Relationship, Drug; Drug Antagonism; Drug Evaluation, Preclinical; Female; Histamine; Humans; In Vitro Techniques; Male; Middle Aged; Molecular Sequence Data; Neurokinin A; Peptide Fragments; Piperidines; Potassium Chloride; Racemases and Epimerases; Receptors, Neurokinin-2; Receptors, Neurotransmitter

1992
Influence of (+/-)-CP-96,345 and SR 48968 on electrical field stimulation of the isolated guinea-pig main bronchus.
    European journal of pharmacology, 1992, Dec-02, Volume: 224, Issue:2-3

    Topics: Animals; Benzamides; Biphenyl Compounds; Bronchi; Bronchoconstriction; Electric Stimulation; Female; Guinea Pigs; In Vitro Techniques; Male; Neurokinin A; Piperidines; Receptors, Neurokinin-2; Receptors, Neurotransmitter

1992
Relative contributions of direct and indirect mechanisms mediating endothelin-induced contraction of guinea-pig trachea.
    British journal of pharmacology, 1993, Volume: 110, Issue:3

    Topics: Animals; Benzamides; Biphenyl Compounds; Capsaicin; Dicarboxylic Acids; Endothelins; Epithelium; Guinea Pigs; Histamine Release; In Vitro Techniques; Kinetics; Leukotriene Antagonists; Male; Muscle Contraction; Neurokinin A; Piperidines; Prostaglandins; Receptors, Tachykinin; SRS-A; Tetrodotoxin; Trachea

1993
Contractile effects of bradykinin on the isolated human small bronchus.
    American journal of respiratory and critical care medicine, 1994, Volume: 149, Issue:1

    Topics: Acetylcholine; Aged; Atropine; Benzamides; Biphenyl Compounds; Bradykinin; Bronchi; Bronchoconstriction; Capsaicin; Humans; In Vitro Techniques; Indomethacin; Middle Aged; Muscle, Smooth; Nerve Fibers; Neurokinin A; Neurons, Afferent; Piperidines; Receptors, Bradykinin; Ruthenium Red; Tetrodotoxin

1994
The species selectivity of chemically distinct tachykinin nonpeptide antagonists is dependent on common divergent residues of the rat and human neurokinin-1 receptors.
    Molecular pharmacology, 1994, Volume: 45, Issue:2

    Topics: Amino Acid Sequence; Animals; Benzamides; Biphenyl Compounds; Cell Line; Dipeptides; Humans; Indoles; Molecular Sequence Data; Mutation; Neurokinin-1 Receptor Antagonists; Piperidines; Rats; Receptors, Neurokinin-1; Recombinant Proteins; Substance P

1994
Involvement of neurokinin 1 and 2 receptors in viscerosensitive response to rectal distension in rats.
    Gastroenterology, 1994, Volume: 107, Issue:1

    Topics: Abdomen; Animals; Benzamides; Biphenyl Compounds; Colon; Colonic Diseases, Functional; Gastrointestinal Motility; Hypnotics and Sedatives; Indoles; Isoindoles; Male; Neurokinin A; Peptide Fragments; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Tachykinin; Rectum; Substance P; Tachykinins

1994
Tachykinin receptors mediating contraction of guinea pig lung strips.
    Regulatory peptides, 1995, May-30, Volume: 57, Issue:2

    Topics: Acetylcholine; Animals; Benzamides; Biphenyl Compounds; Dipeptides; Guinea Pigs; In Vitro Techniques; Lung; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin B; Peptide Fragments; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Tachykinin; Substance P; Trachea

1995
Use of non-peptide tachykinin receptor antagonists to substantiate the involvement of NK1 and NK2 receptors in a spinal nociceptive reflex in the rat.
    European journal of pharmacology, 1993, Mar-02, Volume: 232, Issue:2-3

    Topics: Animals; Benzamides; Biphenyl Compounds; Hypnotics and Sedatives; Injections, Spinal; Male; Neurokinin A; Nociceptors; Pain Measurement; Pain Threshold; Peptide Fragments; Piperidines; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Receptors, Tachykinin; Reflex; Spinal Cord; Substance P

1993
Effects of capsaicin, (+/-)-CP-96,345 and SR 48968 on the bradykinin-induced airways microvascular leakage in guinea-pigs.
    Pulmonary pharmacology, 1993, Volume: 6, Issue:1

    Topics: Animals; Autonomic Nervous System; Benzamides; Biphenyl Compounds; Bradykinin; Capillary Permeability; Capsaicin; Evans Blue; Guinea Pigs; Hypnotics and Sedatives; In Vitro Techniques; Nerve Endings; Neurokinin A; Piperidines; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P

1993
Two nonpeptide tachykinin antagonists act through epitopes on corresponding segments of the NK1 and NK2 receptors.
    Proceedings of the National Academy of Sciences of the United States of America, 1993, Jul-01, Volume: 90, Issue:13

    Topics: Animals; Benzamides; Binding Sites; Biphenyl Compounds; Cells, Cultured; Epitopes; Neurokinin A; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P

1993
Tachykinins contract the circular muscle of the human esophageal body in vitro via NK2 receptors.
    Gastroenterology, 1993, Volume: 105, Issue:4

    Topics: Adolescent; Adult; Aged; Atropine; Benzamides; Biphenyl Compounds; Carbachol; Dose-Response Relationship, Drug; Esophagus; Glycopeptides; Humans; Isometric Contraction; Middle Aged; Muscle Contraction; Muscle, Smooth; Neprilysin; Neurokinin A; Neurokinin B; Piperidines; Receptors, Tachykinin; Substance P; Tachykinins; Tetrodotoxin

1993
In vivo and in vitro activity of SR 48,968, a non-peptide tachykinin NK-2 receptor antagonist.
    Regulatory peptides, 1993, Jul-02, Volume: 46, Issue:1-2

    Topics: Animals; Benzamides; Biphenyl Compounds; Blood Pressure; Muscle Contraction; Muscle, Smooth; Neurokinin A; Peptide Fragments; Piperidines; Rats; Receptors, Neurokinin-2; Saliva; Substance P; Sulfones; Urinary Bladder

1993
Tachykinin NK-1 and NK-2 receptors in the circular muscle of the guinea-pig proximal colon.
    Regulatory peptides, 1993, Jul-02, Volume: 46, Issue:1-2

    Topics: Animals; Benzamides; Biphenyl Compounds; Colon; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Peptides, Cyclic; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Sulfones; Tetrodotoxin

1993
Receptor characterization of the spinal action of neurokinins on nociception: a three receptor hypothesis.
    Regulatory peptides, 1993, Jul-02, Volume: 46, Issue:1-2

    Topics: Animals; Benzamides; Biphenyl Compounds; Models, Neurological; Neurokinin A; Neurokinin-1 Receptor Antagonists; Oligopeptides; Pain; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Neurotransmitter; Spinal Cord; Substance P

1993
Capsaicin increases airflow resistance in guinea pigs in vivo by activating both NK2 and NK1 tachykinin receptors.
    The American review of respiratory disease, 1993, Volume: 148, Issue:4 Pt 1

    Topics: Airway Resistance; Animals; Atropine; Benzamides; Biphenyl Compounds; Capsaicin; Dose-Response Relationship, Drug; Drug Interactions; Guinea Pigs; Histamine; Male; Neurokinin A; Peptide Fragments; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P

1993
Role of kinins in anaphylactic-induced bronchoconstriction mediated by tachykinins in guinea-pigs.
    British journal of pharmacology, 1994, Volume: 113, Issue:2

    Topics: Adrenergic beta-Antagonists; Airway Resistance; Anaphylaxis; Animals; Benzamides; Biphenyl Compounds; Bradykinin; Bronchoconstriction; Glycopeptides; Guinea Pigs; Hypnotics and Sedatives; Kinins; Male; Neprilysin; Neurokinin-1 Receptor Antagonists; Piperidines; Receptors, Neurokinin-2; Tachykinins

1994
Vagal stimulation augments pulmonary anaphylaxis in the guinea pig lung.
    American journal of respiratory and critical care medicine, 1995, Volume: 151, Issue:2 Pt 1

    Topics: Anaphylaxis; Animals; Atropine; Benzamides; Biphenyl Compounds; Bronchoconstriction; Electric Stimulation; Guinea Pigs; Hypnotics and Sedatives; Lung; Male; Neurokinin A; Organ Size; Physostigmine; Piperidines; Trachea; Vagus Nerve; Vasoconstriction

1995
Non-specific actions of the non-peptide tachykinin receptor antagonists, CP-96,345, RP 67580 and SR 48968, on neurotransmission.
    British journal of pharmacology, 1994, Volume: 111, Issue:1

    Topics: Action Potentials; Anesthetics, Local; Animals; Benzamides; Biphenyl Compounds; Bupivacaine; Electric Stimulation; Female; Guinea Pigs; In Vitro Techniques; Indoles; Iris; Isoindoles; Male; Muscle Contraction; Muscle, Smooth; Piperidines; Procaine; Rabbits; Rana catesbeiana; Receptors, Tachykinin; Sciatic Nerve; Synaptic Transmission; Vas Deferens

1994
Sensory neuropeptide-mediated bronchoconstriction of the guinea pig lung by diamide; a comparison to hydrogen peroxide.
    European journal of pharmacology, 1994, Apr-04, Volume: 270, Issue:2-3

    Topics: Animals; Benzamides; Biphenyl Compounds; Bronchoconstriction; Calcitonin Gene-Related Peptide; Capsaicin; Carbazoles; Diamide; Guinea Pigs; Hydrogen Peroxide; In Vitro Techniques; Lung; Male; Neurokinin A; Neurons, Afferent; Neuropeptides; Piperidines; Thromboxanes

1994
Characterization of the cardiovascular and behavioral effects of centrally administered neuropeptide K in the conscious rat.
    Regulatory peptides, 1993, Jul-02, Volume: 46, Issue:1-2

    Topics: Amino Acid Sequence; Animals; Benzamides; Biphenyl Compounds; Blood Pressure; Cerebral Ventricles; Fenclonine; Heart Rate; Injections, Intraventricular; Male; Molecular Sequence Data; Motor Activity; Neurokinin A; Neuropeptides; Oligopeptides; Piperidines; Rats; Rats, Wistar; Stereotyped Behavior; Tachykinins

1993
Tachykinins mediate contraction of the human lower esophageal sphincter in vitro via activation of NK2 receptors.
    European journal of pharmacology, 1993, Aug-03, Volume: 239, Issue:1-3

    Topics: Benzamides; Biphenyl Compounds; Dose-Response Relationship, Drug; Esophagogastric Junction; Glycopeptides; Humans; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Neprilysin; Neurokinin A; Neurokinin B; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Tachykinins

1993
Involvement of neurogenic inflammation in antigen-induced bronchoconstriction in guinea pigs.
    The American journal of physiology, 1993, Volume: 265, Issue:5 Pt 1

    Topics: Aerosols; Animals; Atropine; Benzamides; Biphenyl Compounds; Bronchoconstriction; Capsaicin; Glycopeptides; Guinea Pigs; Histamine; Immunization; Inflammation; Lung; Male; Neurokinin-1 Receptor Antagonists; Ovalbumin; Piperidines; Pulmonary Circulation; Receptors, Neurokinin-2; Vascular Resistance

1993
Differential blockade by tachykinin NK1 and NK2 receptor antagonists of bronchoconstriction induced by direct-acting agonists and the indirect-acting mimetics capsaicin, serotonin and 2-methyl-serotonin in the anesthetized guinea pig.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 267, Issue:3

    Topics: Amino Acid Sequence; Anesthesia; Animals; Benzamides; Biphenyl Compounds; Bronchial Spasm; Bronchoconstriction; Capsaicin; Guinea Pigs; Hypnotics and Sedatives; Injections, Intravenous; Male; Molecular Sequence Data; Neurokinin A; Piperidines; Receptors, Tachykinin; Serotonin

1993
Involvement of tachykinin receptors (NK1 and NK2) in sodium metabisulfite-induced airway effects.
    American journal of respiratory and critical care medicine, 1994, Volume: 149, Issue:2 Pt 1

    Topics: Administration, Inhalation; Animals; Benzamides; Biphenyl Compounds; Bronchoconstriction; Capillary Permeability; Female; Guinea Pigs; Pharmaceutic Aids; Piperidines; Receptors, Tachykinin; Sulfites

1994
Tachykinin receptor antagonists inhibit hyperpnea-induced bronchoconstriction in guinea pigs.
    The Journal of clinical investigation, 1993, Volume: 92, Issue:1

    Topics: Airway Resistance; Animals; Benzamides; Biphenyl Compounds; Bronchoconstriction; Dose-Response Relationship, Drug; Guinea Pigs; Male; Piperidines; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Tachykinins

1993
Neuropeptide modulation of chemically induced skin irritation.
    Toxicology and applied pharmacology, 1995, Volume: 135, Issue:2

    Topics: Administration, Cutaneous; Animals; Benzamides; Biphenyl Compounds; Capsaicin; Dermatitis, Contact; Dinitrofluorobenzene; Disease Models, Animal; Dose-Response Relationship, Drug; Ear, External; Female; Irritants; Mice; Mice, Inbred BALB C; Neurokinin A; Neuropeptides; Piperidines; Skin; Substance P; Synaptic Transmission

1995
Induction of negative hematopoietic regulators by neurokinin-A in bone marrow stroma.
    Blood, 1996, Jul-01, Volume: 88, Issue:1

    Topics: Amino Acid Sequence; Benzamides; Biphenyl Compounds; Bone Marrow; Bone Marrow Cells; Cell Division; Cells, Cultured; Chemokine CCL4; Connective Tissue; Depression, Chemical; Erythroid Precursor Cells; Hematopoietic Stem Cells; Humans; Macrophage Inflammatory Proteins; Molecular Sequence Data; Monokines; Neurokinin A; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Transforming Growth Factor beta

1996
Substance P hyperpolarizes vagal sensory neurones of the ferret.
    The Journal of physiology, 1996, May-15, Volume: 493 ( Pt 1)

    Topics: 4-Aminopyridine; Animals; Anti-Inflammatory Agents, Non-Steroidal; Apamin; Benzamides; Biphenyl Compounds; Cations, Divalent; Cesium; Electrophysiology; Ferrets; In Vitro Techniques; Male; Neurons, Afferent; Nodose Ganglion; Patch-Clamp Techniques; Peptide Fragments; Piperidines; Potassium; Pyrrolidonecarboxylic Acid; Quaternary Ammonium Compounds; Receptors, Tachykinin; Substance P; Vagus Nerve

1996
Augmentation of neurally evoked cholinergic bronchoconstrictor responses by prejunctional NK2 receptors in the guinea-pig.
    Journal of autonomic pharmacology, 1996, Volume: 16, Issue:1

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzamides; Biphenyl Compounds; Bronchoconstriction; Bronchoconstrictor Agents; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Male; Medulla Oblongata; Methacholine Chloride; Muscle, Smooth; Neurokinin A; Neurokinin B; Piperidines; Substance P

1996
Tachykinin receptors and non-cholinergic bronchoconstriction in the anaesthetized guinea-pig.
    Clinical and experimental pharmacology & physiology, 1996, Volume: 23, Issue:2

    Topics: Animals; Benzamides; Biphenyl Compounds; Bronchoconstriction; Electric Stimulation; Female; Guinea Pigs; Lung; Male; Peptides, Cyclic; Piperidines; Receptors, Tachykinin; Vagus Nerve

1996
Inhibitory effect of KW-4679, an anti-allergic drug, on tachykinin-mediated airway response induced by electrical vagal stimulation in guinea pigs.
    Japanese journal of pharmacology, 1996, Volume: 71, Issue:2

    Topics: Animals; Anti-Allergic Agents; Benzamides; Biphenyl Compounds; Bronchoconstriction; Dibenzoxepins; Electric Stimulation; Guinea Pigs; Male; Olopatadine Hydrochloride; Piperidines; Receptors, Tachykinin; Vagus Nerve

1996
SR 48968 specifically depresses neurokinin A- vs. substance P-induced hyperalgesia in a nociceptive withdrawal reflex.
    European journal of pharmacology, 1996, Jul-11, Volume: 308, Issue:1

    Topics: Animals; Benzamides; Biphenyl Compounds; Dose-Response Relationship, Drug; Hyperalgesia; Injections, Spinal; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Pain Measurement; Pain Threshold; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P

1996
Evidence for functional tachykinin NK1 receptors on human isolated small bronchi.
    The American journal of physiology, 1996, Volume: 271, Issue:5 Pt 1

    Topics: Benzamides; Biphenyl Compounds; Bronchi; Female; Hormone Antagonists; Humans; In Vitro Techniques; Indomethacin; Lung Neoplasms; Male; Middle Aged; Neurokinin-1 Receptor Antagonists; Piperidines; Quinuclidines; Receptors, Neurokinin-1; Substance P

1996
Neurokinin receptors in the guinea pig ileum.
    Pharmacology, 1996, Volume: 52, Issue:1

    Topics: Acetylcholine; Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzamides; Biphenyl Compounds; Guinea Pigs; Ileum; Male; Myenteric Plexus; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Radioligand Assay; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Stereoisomerism; Structure-Activity Relationship; Substance P

1996
Autoradiographic mapping of pulmonary NK1 and NK2 tachykinin receptors and changes after repeated antigen challenge in guinea pigs.
    Peptides, 1996, Volume: 17, Issue:8

    Topics: Animals; Antigens; Autoradiography; Benzamides; Binding Sites; Biphenyl Compounds; Guinea Pigs; Inflammation; Lung; Male; Neurokinin-1 Receptor Antagonists; Ovalbumin; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Tissue Distribution

1996
Aerosolized tachykinin antagonists inhibit pentamidine-induce bronchoconstriction in guinea pigs.
    Fundamental & clinical pharmacology, 1996, Volume: 10, Issue:6

    Topics: Aerosols; Animals; Benzamides; Biphenyl Compounds; Bronchi; Bronchoconstriction; Capillary Permeability; Dose-Response Relationship, Drug; Guinea Pigs; Male; Pentamidine; Piperidines; Receptors, Neurokinin-2; Substance P

1996
Effect of tachykinin receptor inhibition in the brain on cardiovascular and behavioral responses to stress.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 280, Issue:1

    Topics: Animals; Behavior, Animal; Benzamides; Biphenyl Compounds; Blood Pressure; Brain; Heart Rate; Indoles; Isoindoles; Male; Neurokinin-1 Receptor Antagonists; Periaqueductal Gray; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-2; Stress, Physiological

1997
Characterization of tachykinin NK2 receptor on dog proximal colon. Antagonism by MEN 10,627 and SR 48,968.
    European journal of pharmacology, 1996, Dec-30, Volume: 318, Issue:2-3

    Topics: Animals; Benzamides; Biphenyl Compounds; Colon; Dogs; Dose-Response Relationship, Drug; Gastrointestinal Motility; In Vitro Techniques; Muscle Contraction; Peptides, Cyclic; Piperidines; Receptors, Neurokinin-2

1996
[Airway hyperresponsiveness and airway mucosal permeability].
    Nihon Kyobu Shikkan Gakkai zasshi, 1996, Volume: 34 Suppl

    Topics: Animals; Benzamides; Biphenyl Compounds; Bronchi; Bronchial Hyperreactivity; Capillary Permeability; Guinea Pigs; Male; Piperidines; Receptors, Neurokinin-2; Superoxide Dismutase; Tachykinins

1996
Electrophysiological evidence that neurokinin A acts via NK-1 receptors in the cat dorsal horn.
    The European journal of neuroscience, 1997, Volume: 9, Issue:9

    Topics: Animals; Benzamides; Biphenyl Compounds; Cats; Iontophoresis; Neurokinin A; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Spinal Cord; Stereoisomerism; Substance P; Synapses

1997
Tachykinins may mediate capsaicin-induced, but not vagally induced motility in porcine antrum.
    Peptides, 1997, Volume: 18, Issue:10

    Topics: Animals; Benzamides; Biphenyl Compounds; Capsaicin; Electric Stimulation; Gastrointestinal Motility; Muscle Contraction; Neurokinin A; Neurokinin-1 Receptor Antagonists; Piperidines; Pyloric Antrum; Receptors, Neurokinin-2; Substance P; Swine; Tachykinins; Vagus Nerve

1997
Prejunctional control of pH 6-induced bronchoconstriction by NK1, NK2, mu-opioid, alpha2-adrenoceptor and glucocorticoid receptors in guinea-pig isolated perfused lung.
    The Journal of pharmacy and pharmacology, 1998, Volume: 50, Issue:8

    Topics: Adrenergic alpha-2 Receptor Agonists; Animals; Benzamides; Betamethasone; Biphenyl Compounds; Brimonidine Tartrate; Bronchoconstriction; Calcitonin Gene-Related Peptide; Female; Guinea Pigs; Hydrogen-Ion Concentration; In Vitro Techniques; Lung; Male; Morphine; Neurokinin-1 Receptor Antagonists; Perfusion; Piperidines; Quinoxalines; Quinuclidines; Receptors, Adrenergic, alpha-2; Receptors, Cell Surface; Receptors, Glucocorticoid; Receptors, Neurokinin-2; Receptors, Opioid, mu

1998
Characterization of tachykinin receptors mediating bronchomotor and vasodepressor responses to neuropeptide gamma and substance P in the anaesthetized rabbit.
    Pulmonary pharmacology & therapeutics, 1998, Volume: 11, Issue:1

    Topics: Anesthesia; Animals; Benzamides; Biphenyl Compounds; Bronchoconstriction; Drug Interactions; Glycopeptides; Neprilysin; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Protease Inhibitors; Rabbits; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Tachykinins; Vagus Nerve; Vasoconstriction

1998
Smoke-induced airway hyperresponsiveness to inhaled wood smoke in guinea pigs: tachykininergic and cholinergic mechanisms.
    Life sciences, 1998, Volume: 63, Issue:17

    Topics: Airway Resistance; Animals; Atropine; Benzamides; Biphenyl Compounds; Bronchi; Bronchial Hyperreactivity; Cholinergic Antagonists; Drug Combinations; Glycopeptides; Guinea Pigs; Male; Neprilysin; Piperidines; Protease Inhibitors; Receptors, Cholinergic; Receptors, Tachykinin; Smoke; Wood

1998
[Inhibitory effects of tachykinin receptor antagonists on leukotriene C4-induced cardiovascular responses in guinea pigs].
    Yao xue xue bao = Acta pharmaceutica Sinica, 1996, Volume: 31, Issue:12

    Topics: Animals; Benzamides; Biphenyl Compounds; Blood Pressure; Female; Guinea Pigs; Leukotriene C4; Male; Neurokinin-1 Receptor Antagonists; Piperidines; Receptors, Neurokinin-2

1996
Effect of tachykinin receptor antagonists in experimental neuropathic pain.
    European journal of pharmacology, 1998, Nov-20, Volume: 361, Issue:2-3

    Topics: Analgesics; Animals; Benzamides; Biphenyl Compounds; Denervation; Diabetes Mellitus, Experimental; Indoles; Isoindoles; Male; Neurokinin-1 Receptor Antagonists; Pain; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Sciatic Nerve

1998
Nanomolar concentrations of neuropeptides induce histamine release from peritoneal mast cells of a substrain of Wistar rats.
    European journal of pharmacology, 1999, Jun-18, Volume: 374, Issue:2

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzamides; Biphenyl Compounds; Dose-Response Relationship, Drug; Histamine Release; Male; Mast Cells; Neurokinin A; Peritoneum; Piperidines; Rats; Rats, Sprague-Dawley; Rats, Wistar; Species Specificity; Substance P; Tachykinins

1999
Increased expression of preprotachykinin-I and neurokinin receptors in human breast cancer cells: implications for bone marrow metastasis.
    Proceedings of the National Academy of Sciences of the United States of America, 2000, Jan-04, Volume: 97, Issue:1

    Topics: Benzamides; Biphenyl Compounds; Bone Marrow Cells; Bone Marrow Neoplasms; Breast Neoplasms; Cell Division; Female; Gene Expression Regulation, Neoplastic; Humans; In Situ Hybridization; Neurokinin-1 Receptor Antagonists; Piperidines; Protein Precursors; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Tachykinins; Tumor Cells, Cultured

2000
The induction and potentiation of c-Jun and c-Fos expression in spinal neurons mediated by NK1 and NK2 receptors.
    Neuropeptides, 1999, Volume: 33, Issue:2

    Topics: Animals; Benzamides; Biphenyl Compounds; Male; Neurokinin-1 Receptor Antagonists; Neurons; Patch-Clamp Techniques; Peptides, Cyclic; Piperidines; Proto-Oncogene Proteins c-fos; Proto-Oncogene Proteins c-jun; Rats; Rats, Wistar; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Sciatic Nerve; Spinal Cord

1999
Participation of neuropeptides in antigen-induced contraction of guinea pig bronchi via NK(2) but not NK(1) receptor stimulation.
    Pharmacology, 2000, Volume: 60, Issue:4

    Topics: Animals; Benzamides; Benzeneacetamides; Biphenyl Compounds; Bronchi; Bronchoconstriction; Female; gamma-Globulins; Guinea Pigs; Histamine H1 Antagonists; Leukotriene Antagonists; Male; Neurokinin-1 Receptor Antagonists; Neuropeptides; Penicillin G; Piperidines; Pyrilamine; Receptors, Neurokinin-2; Substance P; Thiazoles; Trachea

2000
Comparison of the effect of imidaprilat and ramiprilat on broncho-constriction and hypotension induced by bradykinin in guinea pigs.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 2000, Volume: 49, Issue:10

    Topics: Angiotensin I; Angiotensin-Converting Enzyme Inhibitors; Animals; Benzamides; Biphenyl Compounds; Blood Pressure; Bradykinin; Bronchoconstriction; Guinea Pigs; Imidazoles; Imidazolidines; Male; NG-Nitroarginine Methyl Ester; Piperidines; Ramipril

2000
[Effects of tachykinin receptor antagonists on allergic asthma in guinea pigs].
    Yao xue xue bao = Acta pharmaceutica Sinica, 1997, Volume: 32, Issue:5

    Topics: Animals; Asthma; Benzamides; Biphenyl Compounds; Bronchi; Bronchoconstriction; Female; Guinea Pigs; Male; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Ovalbumin; Piperidines; Receptors, Neurokinin-2; Receptors, Tachykinin; Trachea

1997
Substance P via NK1 receptor facilitates hyperactive bladder afferent signaling via action of ROS.
    American journal of physiology. Renal physiology, 2003, Volume: 284, Issue:4

    Topics: Animals; Benzamides; Biphenyl Compounds; Cell Adhesion Molecules; Dose-Response Relationship, Drug; Drug Administration Routes; Electric Stimulation; Female; Free Radical Scavengers; Muscle Contraction; Neurokinin-1 Receptor Antagonists; Pelvis; Piperidines; Rats; Rats, Wistar; Reactive Oxygen Species; Receptors, Neurokinin-1; Reflex, Abnormal; Signal Transduction; Sodium Chloride; Substance P; Superoxide Dismutase; Urinary Bladder; Urinary Bladder, Neurogenic; Urination; Visceral Afferents

2003
Substance P acts via the neurokinin receptor 1 to elicit bronchoconstriction, oxidative stress, and upregulated ICAM-1 expression after oil smoke exposure.
    American journal of physiology. Lung cellular and molecular physiology, 2008, Volume: 294, Issue:5

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Antioxidants; Ascorbic Acid; Benzamides; Biphenyl Compounds; Blood Pressure; Bronchoalveolar Lavage Fluid; Bronchoconstriction; Catechin; Intercellular Adhesion Molecule-1; Male; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Oxidative Stress; Petroleum; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Respiratory Distress Syndrome; Smoke; Smoke Inhalation Injury; Substance P; Up-Regulation

2008
Colorectal distension enforce acute urinary bladder distension-induced hepatic vasoconstriction in the rat.
    Neuroscience letters, 2008, Oct-10, Volume: 443, Issue:3

    Topics: Afferent Pathways; Animals; Benzamides; Biphenyl Compounds; Blood Pressure; Colon; Female; Liver; Neurokinin-1 Receptor Antagonists; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-2; Sympathectomy; Urinary Bladder; Vasoconstriction

2008