Page last updated: 2024-08-26

cp 96345 and aprepitant

cp 96345 has been researched along with aprepitant in 2 studies

Research

Studies (2)

Timeframe	Studies, this research(%)	All Research%
pre-1990	0 (0.00)	18.7374
1990's	0 (0.00)	18.2507
2000's	0 (0.00)	29.6817
2010's	2 (100.00)	24.3611
2020's	0 (0.00)	2.80

Authors

Authors	Studies
Bissantz, C; Bohnert, C; Hoffmann, T; Malherbe, P; Marcuz, A; Schnider, P	1
Alvaro, G; Braggio, S; Carletti, R; Corsi, M; Di Fabio, R; Gerrard, PA; Griffante, C; Marchioro, C; Melotto, S; Piccoli, L; Poffe, A; Pozzan, A; Ratti, E; Spada, S; Tranquillini, E; Trower, M	1

Other Studies

2 other study(ies) available for cp 96345 and aprepitant

Article	Year
Identification of a crucial amino acid in the helix position 6.51 of human tachykinin neurokinin 1 and 3 receptors contributing to the insurmountable mode of antagonism by dual NK₁/NK₃ antagonists. Journal of medicinal chemistry, 2012, Jun-14, Volume: 55, Issue:11 Topics: Amino Acids; Aminopyridines; Benzeneacetamides; HEK293 Cells; Humans; Inositol Phosphates; Models, Molecular; Mutagenesis, Site-Directed; Mutation; Neurokinin-1 Receptor Antagonists; Protein Structure, Secondary; Radioligand Assay; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Stereoisomerism	2012
Identification, biological characterization and pharmacophoric analysis of a new potent and selective NK1 receptor antagonist clinical candidate. Bioorganic & medicinal chemistry, 2013, Nov-01, Volume: 21, Issue:21 Topics: Animals; Antidepressive Agents; Behavior, Animal; Bridged Bicyclo Compounds, Heterocyclic; CHO Cells; Cricetinae; Cricetulus; Dogs; Female; Gerbillinae; Half-Life; Humans; Male; Models, Molecular; Molecular Conformation; Neurokinin-1 Receptor Antagonists; Piperazines; Piperidines; Protein Binding; Rats; Receptors, Neurokinin-1	2013

Article

Year

Identification of a crucial amino acid in the helix position 6.51 of human tachykinin neurokinin 1 and 3 receptors contributing to the insurmountable mode of antagonism by dual NK₁/NK₃ antagonists.

Journal of medicinal chemistry, 2012, Jun-14, Volume: 55, Issue:11

Topics: Amino Acids; Aminopyridines; Benzeneacetamides; HEK293 Cells; Humans; Inositol Phosphates; Models, Molecular; Mutagenesis, Site-Directed; Mutation; Neurokinin-1 Receptor Antagonists; Protein Structure, Secondary; Radioligand Assay; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Stereoisomerism

2012

Identification, biological characterization and pharmacophoric analysis of a new potent and selective NK1 receptor antagonist clinical candidate.

Bioorganic & medicinal chemistry, 2013, Nov-01, Volume: 21, Issue:21

Topics: Animals; Antidepressive Agents; Behavior, Animal; Bridged Bicyclo Compounds, Heterocyclic; CHO Cells; Cricetinae; Cricetulus; Dogs; Female; Gerbillinae; Half-Life; Humans; Male; Models, Molecular; Molecular Conformation; Neurokinin-1 Receptor Antagonists; Piperazines; Piperidines; Protein Binding; Rats; Receptors, Neurokinin-1

2013