Compounds > cp 96345

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cp 96345 and 3,5-bis(trifluoromethyl)benzyl n-acetyltryptophan

cp 96345 has been researched along with 3,5-bis(trifluoromethyl)benzyl n-acetyltryptophan in 5 studies

Research

Studies (5)

Timeframe	Studies, this research(%)	All Research%
pre-1990	0 (0.00)	18.7374
1990's	5 (100.00)	18.2507
2000's	0 (0.00)	29.6817
2010's	0 (0.00)	24.3611
2020's	0 (0.00)	2.80

Authors

Authors	Studies
Ber, E; Brookfield, F; Casiceri, MA; Kelleher, F; MacLeod, AM; Merchant, KJ; Owens, AP; Sadowski, S; Stevenson, G; Swain, CJ	1
Cascieri, MA; Fong, TM; Hardwicke, S; Lewis, RT; MacIntyre, DE; MacLeod, AM; Merchant, KJ; Metzger, JM; Sadowski, S; Shepheard, S	1
Baker, R; Ber, E; Cascieri, MA; MacLeod, AM; Merchant, KJ; Sadowski, S; Swain, CJ	1
Beusen, DD; Marshall, GR; Shands, EF; Takeuchi, Y	1
Boudon, A; Fauchère, JL; Jacoby, E; Kucharczyk, N; Michel, A	1

Other Studies

5 other study(ies) available for cp 96345 and 3,5-bis(trifluoromethyl)benzyl n-acetyltryptophan

Article	Year
Identification of L-tryptophan derivatives with potent and selective antagonist activity at the NK1 receptor. Journal of medicinal chemistry, 1994, Apr-29, Volume: 37, Issue:9 Topics: Acylation; Amino Acid Sequence; Animals; CHO Cells; Computer Simulation; Cricetinae; Dermatitis, Contact; Guinea Pigs; Humans; Male; Models, Molecular; Molecular Conformation; Molecular Sequence Data; Molecular Structure; Neurokinin-1 Receptor Antagonists; Receptors, Neurokinin-1; Recombinant Proteins; Structure-Activity Relationship; Substance P; Tryptophan	1994
Synthesis and biological evaluation of NK1 antagonists derived from L-tryptophan. Journal of medicinal chemistry, 1995, Mar-17, Volume: 38, Issue:6 Topics: Amines; Amino Acid Sequence; Animals; Binding Sites; Biphenyl Compounds; Cardiovascular System; CHO Cells; Cricetinae; Esters; Extravasation of Diagnostic and Therapeutic Materials; Female; Ferrets; Guinea Pigs; Heterocyclic Compounds; Humans; Hypnotics and Sedatives; Male; Molecular Sequence Data; Neurokinin-1 Receptor Antagonists; Piperidines; Receptors, Neurokinin-1; Solubility; Structure-Activity Relationship; Substance P; Tryptophan	1995
N-acyl-L-tryptophan benzyl esters: potent substance P receptor antagonists. Journal of medicinal chemistry, 1993, Jul-09, Volume: 36, Issue:14 Topics: Benzyl Compounds; Esters; Humans; Receptors, Neurokinin-1; Receptors, Neurotransmitter; Structure-Activity Relationship; Tryptophan	1993
Derivation of a three-dimensional pharmacophore model of substance P antagonists bound to the neurokinin-1 receptor. Journal of medicinal chemistry, 1998, Sep-10, Volume: 41, Issue:19 Topics: Binding Sites; Biphenyl Compounds; Crystallography, X-Ray; Ligands; Models, Molecular; Molecular Conformation; Neurokinin-1 Receptor Antagonists; Receptors, Neurokinin-1; Structure-Activity Relationship; Substance P	1998
A structural rationale for the design of water soluble peptide-derived neurokinin-1 antagonists. Journal of receptor and signal transduction research, 1997, Volume: 17, Issue:6 Topics: Animals; Biphenyl Compounds; Dipeptides; Drug Design; Humans; In Vitro Techniques; Indoles; Models, Chemical; Models, Molecular; Molecular Mimicry; Neurokinin-1 Receptor Antagonists; Peptides; Rats; Solubility; Substance P; Tetrazoles; Tryptophan; Water	1997